Lista de obras - Wim M De Borggraeve - Dominio Público Uruguay

2-(4-Meth-oxy-benz-yl)-4,6-diphenyl-2,5-diaza-bicyclo-[2.2.2]oct-5-en-3-one.

artículo científico publicado en 2011

8-HaloBODIPYs and their 8-(C, N, O, S) substituted analogues: solvent dependent UV-vis spectroscopy, variable temperature NMR, crystal structure determination, and quantum chemical calculations.

artículo científico publicado en 2014

A Tripodal Ruthenium–Gadolinium Metallostar as a Potential αvβ3 Integrin Specific Bimodal Imaging Contrast Agent

article

A heterobimetallic ruthenium-gadolinium complex as a potential agent for bimodal imaging

artículo científico publicado en 2011

Active Principles of Tetradenia riparia. IV. Anthelmintic Activity of 8(14),15-Sandaracopimaradiene-7α,18-diol.

artículo científico publicado en 2018

Acylated sulfonamide adenosines as potent inhibitors of the adenylate-forming enzyme superfamily

artículo científico publicado en 2019

Alpha-helical destabilization of the Bcl-2-BH4-domain peptide abolishes its ability to inhibit the IP3 receptor

artículo científico publicado en 2013

An integrated fragment based screening approach for the discovery of small molecule modulators of the VWF-GPIbα interaction.

artículo científico publicado en 2012

Anticonvulsant activity of bisabolene sesquiterpenoids of Curcuma longa in zebrafish and mouse seizure models.

artículo científico publicado en 2012

BODIPY-based hydroxyaryl derivatives as fluorescent pH probes.

artículo científico publicado en 2005

Bioassay-guided isolation of active substances from Semen Torreyae identifies two new anthelmintic compounds with novel mechanism of action

artículo científico publicado en 2018

Bioassay-guided isolation of three anthelmintic compounds from Warburgia ugandensis Sprague subspecies ugandensis, and the mechanism of action of polygodial

artículo científico publicado en 2018

Biofilm inhibiting properties of compounds from the leaves of Warburgia ugandensis Sprague subsp ugandensis against Candida and staphylococcal biofilms

scientific article published on 30 October 2019

Carbonylation as a novel method for the assembly of pyrazine based oligoamide alpha-helix mimetics

artículo científico publicado en 2016

Chemical structure and biological properties of sulfated fucan from the sequential extraction of subAntarctic Lessonia sp (Phaeophyceae)

artículo científico publicado en 2018

Concomitant positive patch test reactions in FreeStyle®-allergic patients sensitized to isobornyl acrylate

scientific article published on 23 September 2020

Conformational Analysis of TOAC-Labelled Alamethicin F50/5 Analogues

article

Crystal structure of 5-benzyl-8-bromo-2-meth-yl-1,3-oxazolo[4,5-c][1,8]naphthyridin-4(5H)-one.

artículo científico publicado en 2017

Design, Synthesis, and Preferred Conformation of Peptides Based on a Highly Constrained, β,β′-Diphenyl Substituted Cyclopropane α-Amino Acid

scholarly article published 2006

Direct Access to Aryl Bis(trifluoromethyl)carbinols from Aryl Bromides or Fluorosulfates: Palladium-Catalyzed Carbonylation

artículo científico publicado en 2018

Direct functionalization of BODIPY dyes by oxidative nucleophilic hydrogen substitution at the 3- or 3,5-positions

artículo científico publicado en 2010

Discovery of a potent protein kinase D inhibitor: insights in the binding mode of pyrazolo[3,4-d]pyrimidine analogues.

artículo científico publicado en 2017

Electrochemistry and Photoredox Catalysis: A Comparative Evaluation in Organic Synthesis

scientific article published on 05 June 2019

Ex Situ Generation of Sulfuryl Fluoride for the Synthesis of Aryl Fluorosulfates

artículo científico publicado en 2017

Exploring polyoxometalates as non-destructive staining agents for contrast-enhanced microfocus computed tomography of biological tissues

scientific article published on 26 January 2020

Generalized solvent scales as a tool for investigating solvent dependence of spectroscopic and kinetic parameters. Application to fluorescent BODIPY dyes

artículo científico publicado en 2010

High-speed microwave-promoted hetero-Diels-Alder reactions of 2(1H)-pyrazinones in ionic liquid doped solvents

artículo científico publicado en 2002

Identification of a small molecule that modulates platelet glycoprotein Ib-von Willebrand factor interaction

artículo científico publicado en 2012

Identification of fukinolic acid from Cimicifuga heracleifolia and its derivatives as novel antiviral compounds against enterovirus A71 infection

scientific article published on 29 July 2018

Improved detection of β-N-methylamino-L-alanine using N-hydroxysuccinimide ester of N-butylnicotinic acid for the localization of BMAA in blue mussels (Mytilus edulis).

artículo científico publicado en 2015

Introduction of Aryl Fluorosulfates into the Realm of Catellani Reaction Substrates

scientific article published on 12 November 2019

Ketone Synthesis by a Nickel-Catalyzed Dehydrogenative Cross-Coupling of Primary Alcohols

scientific article published on 18 April 2019

Measuring cooperative Rev protein-protein interactions on Rev responsive RNA by fluorescence resonance energy transfer

artículo científico publicado en 2011

Mechanism and related kinetics of 5-methyltetrahydrofolic acid degradation during combined high hydrostatic pressure-thermal treatments.

artículo científico publicado en 2009

Methylated flavonoids as anti-seizure agents: Naringenin 4',7-dimethyl ether attenuates epileptic seizures in zebrafish and mouse models.

artículo científico publicado en 2017

Nanocellulosic materials as bioinks for 3D bioprinting

artículo científico publicado en 2017

Nematicidal Activity of Holigarna caustica (Dennst.) Oken Fruit Is Due to Linoleic Acid

artículo científico publicado en 2020

Non-innocent probes in direct sonication: Metal assistance in oxidative radical CH functionalization.

artículo científico publicado en 2017

Photophysics and stability of cyano-substituted boradiazaindacene dyes.

artículo científico publicado en 2009

Photophysics of 3,5-diphenoxy substituted BODIPY dyes in solution

artículo científico publicado en 2007

Practical preparation of challenging amides from non-nucleophilic amines and esters under flow conditions

artículo científico publicado en 2014

Preferred 3D-structure of peptides rich in a severely conformationally restricted cyclopropane analogue of phenylalanine.

artículo científico publicado en 2005

Preparation and characterization of hydrogels based on homopolymeric fractions of sodium alginate and PNIPAAm

article

Ratiometric, fluorescent BODIPY dye with aza crown ether functionality: synthesis, solvatochromism, and metal ion complex formation.

artículo científico publicado en 2008

Rational design, synthesis, and spectroscopic and photophysical properties of a visible-light-excitable, ratiometric, fluorescent near-neutral pH indicator based on BODIPY.

artículo científico publicado en 2011

Rationalising Supramolecular Hydrogelation of Bis-Urea-Based Gelators through a Multiscale Approach

artículo científico publicado en 2019

Rationalising Supramolecular Hydrogelation of Bis-Urea-Based Gelators through a Multiscale Approach

artículo científico publicado en 2019

Robust scalable synthesis of a bis-urea derivative forming thixotropic and cytocompatible supramolecular hydrogels

artículo científico publicado en 2019

Scaffold hopping via a transannular rearrangement-encompassing cascade

artículo científico publicado en 2013

Selective LC-MS/MS method for the identification of BMAA from its isomers in biological samples.

artículo científico publicado en 2012

Solvent and pH dependent fluorescent properties of a dimethylaminostyryl borondipyrromethene dye in solution.

artículo científico publicado en 2006

Synthesis and in vitro evaluation of a PDT active BODIPY-NLS conjugate

artículo científico publicado en 2013

Synthesis of 2(1H)-pyrazinone phosphonates via an Arbuzov-type reaction

artículo científico publicado en 2007

Synthesis of N-Acyl Sulfamates from Fluorosulfates and Amides

artículo científico publicado en 2019

Synthesis of highly functionalized 2(1H)-pyrazinone 3-carboxamide scaffolds

artículo científico publicado en 2008

Synthesis of the orthogonally protected amino alcohol Phaol and analogs

artículo científico publicado en 2011

Synthesis of triterpenoid triazine derivatives from allobetulone and betulonic acid with biological activities.

artículo científico publicado en 2014

Synthetic protocol toward fused pyrazolone derivatives via a Michael addition and reductive ring closing strategy

artículo científico publicado en 2014

Tanshinone IIA exhibits anticonvulsant activity in zebrafish and mouse seizure models.

artículo científico publicado en 2013

The C terminus of Bax inhibitor-1 forms a Ca2+-permeable channel pore.

artículo científico publicado en 2011

The orthorhombic pseudopolymorph of tacrine hydrochloride

artículo científico publicado en 2016

The zeamine antibiotics affect the integrity of bacterial membranes.

artículo científico publicado en 2014

Total synthesis of Septocylindrin B and C-terminus modified analogues

artículo científico publicado en 2012

Triple Hyp→Pro replacement in integramide A, a peptaib inhibitor of HIV-1 integrase: Effect on conformation and bioactivity

artículo científico publicado en 2011

Turn and helical peptide handedness governed exclusively by side-chain chiral centers.

artículo científico publicado en 2005

trans-Chlorido[6-chloro-4-(4-methoxy-benz-yl)-3-oxo-3,4-dihydro-pyrazin-2-yl]-bis-(triphenyl-phosphine)palladium(II).

artículo científico publicado en 2007

Lista de obras de Wim M De Borggraeve

2-(4-Meth-oxy-benz-yl)-4,6-diphenyl-2,5-diaza-bicyclo-[2.2.2]oct-5-en-3-one.

8-HaloBODIPYs and their 8-(C, N, O, S) substituted analogues: solvent dependent UV-vis spectroscopy, variable temperature NMR, crystal structure determination, and quantum chemical calculations.

A Tripodal Ruthenium–Gadolinium Metallostar as a Potential αvβ3 Integrin Specific Bimodal Imaging Contrast Agent

A heterobimetallic ruthenium-gadolinium complex as a potential agent for bimodal imaging

Active Principles of Tetradenia riparia. IV. Anthelmintic Activity of 8(14),15-Sandaracopimaradiene-7α,18-diol.

Acylated sulfonamide adenosines as potent inhibitors of the adenylate-forming enzyme superfamily

Alpha-helical destabilization of the Bcl-2-BH4-domain peptide abolishes its ability to inhibit the IP3 receptor

An integrated fragment based screening approach for the discovery of small molecule modulators of the VWF-GPIbα interaction.

Anticonvulsant activity of bisabolene sesquiterpenoids of Curcuma longa in zebrafish and mouse seizure models.

BODIPY-based hydroxyaryl derivatives as fluorescent pH probes.

Bioassay-guided isolation of active substances from Semen Torreyae identifies two new anthelmintic compounds with novel mechanism of action

Bioassay-guided isolation of three anthelmintic compounds from Warburgia ugandensis Sprague subspecies ugandensis, and the mechanism of action of polygodial

Biofilm inhibiting properties of compounds from the leaves of Warburgia ugandensis Sprague subsp ugandensis against Candida and staphylococcal biofilms

Carbonylation as a novel method for the assembly of pyrazine based oligoamide alpha-helix mimetics

Chemical structure and biological properties of sulfated fucan from the sequential extraction of subAntarctic Lessonia sp (Phaeophyceae)

Concomitant positive patch test reactions in FreeStyle®-allergic patients sensitized to isobornyl acrylate

Conformational Analysis of TOAC-Labelled Alamethicin F50/5 Analogues

Crystal structure of 5-benzyl-8-bromo-2-meth-yl-1,3-oxazolo[4,5-c][1,8]naphthyridin-4(5H)-one.

Design, Synthesis, and Preferred Conformation of Peptides Based on a Highly Constrained, β,β′-Diphenyl Substituted Cyclopropane α-Amino Acid

Direct Access to Aryl Bis(trifluoromethyl)carbinols from Aryl Bromides or Fluorosulfates: Palladium-Catalyzed Carbonylation

Direct functionalization of BODIPY dyes by oxidative nucleophilic hydrogen substitution at the 3- or 3,5-positions

Discovery of a potent protein kinase D inhibitor: insights in the binding mode of pyrazolo[3,4-d]pyrimidine analogues.

Electrochemistry and Photoredox Catalysis: A Comparative Evaluation in Organic Synthesis

Ex Situ Generation of Sulfuryl Fluoride for the Synthesis of Aryl Fluorosulfates

Exploring polyoxometalates as non-destructive staining agents for contrast-enhanced microfocus computed tomography of biological tissues

Generalized solvent scales as a tool for investigating solvent dependence of spectroscopic and kinetic parameters. Application to fluorescent BODIPY dyes

High-speed microwave-promoted hetero-Diels-Alder reactions of 2(1H)-pyrazinones in ionic liquid doped solvents

Identification of a small molecule that modulates platelet glycoprotein Ib-von Willebrand factor interaction

Identification of fukinolic acid from Cimicifuga heracleifolia and its derivatives as novel antiviral compounds against enterovirus A71 infection

Improved detection of β-N-methylamino-L-alanine using N-hydroxysuccinimide ester of N-butylnicotinic acid for the localization of BMAA in blue mussels (Mytilus edulis).

Introduction of Aryl Fluorosulfates into the Realm of Catellani Reaction Substrates

Ketone Synthesis by a Nickel-Catalyzed Dehydrogenative Cross-Coupling of Primary Alcohols

Measuring cooperative Rev protein-protein interactions on Rev responsive RNA by fluorescence resonance energy transfer

Mechanism and related kinetics of 5-methyltetrahydrofolic acid degradation during combined high hydrostatic pressure-thermal treatments.

Methylated flavonoids as anti-seizure agents: Naringenin 4',7-dimethyl ether attenuates epileptic seizures in zebrafish and mouse models.

Nanocellulosic materials as bioinks for 3D bioprinting

Nematicidal Activity of Holigarna caustica (Dennst.) Oken Fruit Is Due to Linoleic Acid

Non-innocent probes in direct sonication: Metal assistance in oxidative radical CH functionalization.

Photophysics and stability of cyano-substituted boradiazaindacene dyes.

Photophysics of 3,5-diphenoxy substituted BODIPY dyes in solution

Practical preparation of challenging amides from non-nucleophilic amines and esters under flow conditions

Preferred 3D-structure of peptides rich in a severely conformationally restricted cyclopropane analogue of phenylalanine.

Preparation and characterization of hydrogels based on homopolymeric fractions of sodium alginate and PNIPAAm

Ratiometric, fluorescent BODIPY dye with aza crown ether functionality: synthesis, solvatochromism, and metal ion complex formation.

Rational design, synthesis, and spectroscopic and photophysical properties of a visible-light-excitable, ratiometric, fluorescent near-neutral pH indicator based on BODIPY.

Rationalising Supramolecular Hydrogelation of Bis-Urea-Based Gelators through a Multiscale Approach

Rationalising Supramolecular Hydrogelation of Bis-Urea-Based Gelators through a Multiscale Approach

Robust scalable synthesis of a bis-urea derivative forming thixotropic and cytocompatible supramolecular hydrogels

Scaffold hopping via a transannular rearrangement-encompassing cascade

Selective LC-MS/MS method for the identification of BMAA from its isomers in biological samples.

Solvent and pH dependent fluorescent properties of a dimethylaminostyryl borondipyrromethene dye in solution.

Synthesis and in vitro evaluation of a PDT active BODIPY-NLS conjugate

Synthesis of 2(1H)-pyrazinone phosphonates via an Arbuzov-type reaction

Synthesis of N-Acyl Sulfamates from Fluorosulfates and Amides

Synthesis of highly functionalized 2(1H)-pyrazinone 3-carboxamide scaffolds

Synthesis of the orthogonally protected amino alcohol Phaol and analogs

Synthesis of triterpenoid triazine derivatives from allobetulone and betulonic acid with biological activities.

Synthetic protocol toward fused pyrazolone derivatives via a Michael addition and reductive ring closing strategy

Tanshinone IIA exhibits anticonvulsant activity in zebrafish and mouse seizure models.

The C terminus of Bax inhibitor-1 forms a Ca2+-permeable channel pore.

The orthorhombic pseudopolymorph of tacrine hydrochloride

The zeamine antibiotics affect the integrity of bacterial membranes.

Total synthesis of Septocylindrin B and C-terminus modified analogues

Triple Hyp→Pro replacement in integramide A, a peptaib inhibitor of HIV-1 integrase: Effect on conformation and bioactivity

Turn and helical peptide handedness governed exclusively by side-chain chiral centers.

trans-Chlorido[6-chloro-4-(4-methoxy-benz-yl)-3-oxo-3,4-dihydro-pyrazin-2-yl]-bis-(triphenyl-phosphine)palladium(II).