Lista de obras -

A Sample-Centric and Knowledge-Driven Computational Framework for Natural Products Drug Discovery ⬇️

Absolute configuration of a tetrahydrophenanthrene from Heliotropium ovalifolium by LC-NMR of its Mosher esters.

artículo científico publicado en 2003

Addressing the Most Neglected Diseases through an Open Research Model: the Discovery of Fenarimols as Novel Drug Candidates for Eumycetoma

Addressing the most neglected diseases through an open research model: The discovery of fenarimols as novel drug candidates for eumycetoma.

artículo científico publicado en 2018

An LC/DAD-UV/MS method for the rapid detection of aristolochic acid in plant preparations

artículo científico publicado en 2002

Antileishmanial activities associated with plants used in the Malian traditional medicine

artículo científico publicado en 2006

Antileishmanial and antifungal acridone derivatives from the roots of Thamnosma rhodesica

artículo científico publicado en 2004

Antiprotozoal Activity Profiling of Approved Drugs: A Starting Point toward Drug Repositioning

artículo científico publicado en 2015

Assessing anti-T. cruzi candidates in vitro for sterile cidality

artículo científico publicado en 2016

Bio-guided isolation of cholinesterase inhibitors from the bulbs of Crinum x powellii

artículo científico publicado en 2005

Catechol pyrazolinones as trypanocidals: fragment-based design, synthesis, and pharmacological evaluation of nanomolar inhibitors of trypanosomal phosphodiesterase B1

article

Complete LC/MS analysis of a Tinnevelli senna pod extract and subsequent isolation and identification of two new benzophenone glucosides

artículo científico publicado en 2002

Correction: Identification of Compounds with Anti-Proliferative Activity against Strain 427 by a Whole Cell Viability Based HTS Campaign

Development and Validation of a Novel Leishmania donovani Screening Cascade for High-Throughput Screening Using a Novel Axenic Assay with High Predictivity of Leishmanicidal Intracellular Activity.

artículo científico publicado en 2015

Discovery of potent nitrotriazole-based antitrypanosomal agents: In vitro and in vivo evaluation

artículo científico publicado en 2015

Drug discovery and development for neglected diseases: the DNDi model

artículo científico publicado en 2011

Drugs for Neglected Diseases initiative model of drug development for neglected diseases: current status and future challenges

artículo científico publicado en 2011

Ellagic acid derivatives from Syzygium cumini stem bark: investigation of their antiplasmodial activity.

artículo científico publicado en 2009

Evaluation of Parameters Impacting Drug Susceptibility in Intracellular Trypanosoma cruzi Assay Protocols

artículo científico publicado en 2016

Flavonoid profiling among wild type and related GM wheat varieties

article

Four new sesquiterpenoid derivatives from the heartwood of Mansonia gagei

artículo científico publicado en 2002

Identification of compounds with anti-proliferative activity against Trypanosoma brucei brucei strain 427 by a whole cell viability based HTS campaign

artículo científico publicado en 2012

Identification of two isomeric meroterpenoid naphthoquinones fromCordia linnaei by liquid chromatography-mass spectrometry and liquid chromatography-nuclear magnetic resonance spectroscopy

article

Limonoid orthoacetates and antiprotozoal compounds from the roots of Pseudocedrela kotschyi

artículo científico publicado en 2007

Novel 3-nitro-1H-1,2,4-triazole-based amides and sulfonamides as potential antitrypanosomal agents

artículo científico publicado en 2012

Novel 3-nitro-1H-1,2,4-triazole-based piperazines and 2-amino-1,3-benzothiazoles as antichagasic agents

artículo científico publicado en 2013

Novel 3-nitrotriazole-based amides and carbinols as bifunctional antichagasic agents

artículo científico publicado en 2015

Novel benzoxaborole, nitroimidazole and aminopyrazoles with activity against experimental cutaneous leishmaniasis

scientific article published on 26 February 2019

On-line characterisation of apple polyphenols by liquid chromatography coupled with mass spectrometry and ultraviolet absorbance detection

artículo científico publicado en 2004

Phenotypic screening approaches for Chagas disease drug discovery

artículo científico publicado en 2017

Qualitative and quantitative determination of yohimbine in authentic yohimbe bark and in commercial aphrodisiacs by HPLC-UV-API/ MS methods

artículo científico publicado en 2003

Repurposing of the Open Access Malaria Box for Kinetoplastid Diseases Identifies Novel Active Scaffolds against Trypanosomatids

artículo científico publicado en 2015

Screening strategies to identify new chemical diversity for drug development to treat kinetoplastid infections

artículo científico publicado en 2013

Selection and optimization of hits from a high-throughput phenotypic screen against Trypanosoma cruzi.

artículo científico publicado en 2013

Simple field assays to check quality of current artemisinin-based antimalarial combination formulations

artículo científico publicado en 2009

Synthesis and evaluation of analogs of the phenylpyridazinone NPD-001 as potent trypanosomal TbrPDEB1 phosphodiesterase inhibitors and in vitro trypanocidals

artículo científico publicado en 2016

Lista de obras de

A Sample-Centric and Knowledge-Driven Computational Framework for Natural Products Drug Discovery ⬇️

Absolute configuration of a tetrahydrophenanthrene from Heliotropium ovalifolium by LC-NMR of its Mosher esters.

Addressing the Most Neglected Diseases through an Open Research Model: the Discovery of Fenarimols as Novel Drug Candidates for Eumycetoma

Addressing the most neglected diseases through an open research model: The discovery of fenarimols as novel drug candidates for eumycetoma.

An LC/DAD-UV/MS method for the rapid detection of aristolochic acid in plant preparations

Antileishmanial activities associated with plants used in the Malian traditional medicine

Antileishmanial and antifungal acridone derivatives from the roots of Thamnosma rhodesica

Antiprotozoal Activity Profiling of Approved Drugs: A Starting Point toward Drug Repositioning

Assessing anti-T. cruzi candidates in vitro for sterile cidality

Bio-guided isolation of cholinesterase inhibitors from the bulbs of Crinum x powellii

Catechol pyrazolinones as trypanocidals: fragment-based design, synthesis, and pharmacological evaluation of nanomolar inhibitors of trypanosomal phosphodiesterase B1

Complete LC/MS analysis of a Tinnevelli senna pod extract and subsequent isolation and identification of two new benzophenone glucosides

Correction: Identification of Compounds with Anti-Proliferative Activity against Strain 427 by a Whole Cell Viability Based HTS Campaign

Development and Validation of a Novel Leishmania donovani Screening Cascade for High-Throughput Screening Using a Novel Axenic Assay with High Predictivity of Leishmanicidal Intracellular Activity.

Discovery of potent nitrotriazole-based antitrypanosomal agents: In vitro and in vivo evaluation

Drug discovery and development for neglected diseases: the DNDi model

Drugs for Neglected Diseases initiative model of drug development for neglected diseases: current status and future challenges

Ellagic acid derivatives from Syzygium cumini stem bark: investigation of their antiplasmodial activity.

Evaluation of Parameters Impacting Drug Susceptibility in Intracellular Trypanosoma cruzi Assay Protocols

Flavonoid profiling among wild type and related GM wheat varieties

Four new sesquiterpenoid derivatives from the heartwood of Mansonia gagei

Identification of compounds with anti-proliferative activity against Trypanosoma brucei brucei strain 427 by a whole cell viability based HTS campaign

Identification of two isomeric meroterpenoid naphthoquinones fromCordia linnaei by liquid chromatography-mass spectrometry and liquid chromatography-nuclear magnetic resonance spectroscopy

Limonoid orthoacetates and antiprotozoal compounds from the roots of Pseudocedrela kotschyi

Novel 3-nitro-1H-1,2,4-triazole-based amides and sulfonamides as potential antitrypanosomal agents

Novel 3-nitro-1H-1,2,4-triazole-based piperazines and 2-amino-1,3-benzothiazoles as antichagasic agents

Novel 3-nitrotriazole-based amides and carbinols as bifunctional antichagasic agents

Novel benzoxaborole, nitroimidazole and aminopyrazoles with activity against experimental cutaneous leishmaniasis

On-line characterisation of apple polyphenols by liquid chromatography coupled with mass spectrometry and ultraviolet absorbance detection

Phenotypic screening approaches for Chagas disease drug discovery

Qualitative and quantitative determination of yohimbine in authentic yohimbe bark and in commercial aphrodisiacs by HPLC-UV-API/ MS methods

Repurposing of the Open Access Malaria Box for Kinetoplastid Diseases Identifies Novel Active Scaffolds against Trypanosomatids

Screening strategies to identify new chemical diversity for drug development to treat kinetoplastid infections

Selection and optimization of hits from a high-throughput phenotypic screen against Trypanosoma cruzi.

Simple field assays to check quality of current artemisinin-based antimalarial combination formulations

Synthesis and evaluation of analogs of the phenylpyridazinone NPD-001 as potent trypanosomal TbrPDEB1 phosphodiesterase inhibitors and in vitro trypanocidals