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2,3-Dihydro-1H-cyclopenta[b]quinoline Derivatives as Acetylcholinesterase Inhibitors—Synthesis, Radiolabeling and Biodistribution

artículo científico publicado el 13 de agosto de 2012

Adaptation of high-throughput screening in drug discovery-toxicological screening tests.

artículo científico publicado en 2011

An investigation into the pleiotropic activity of metformin. A glimpse of haemostasis

artículo científico publicado en 2020

Antiproliferative activity of new benzimidazole derivatives

artículo científico publicado el 25 de julio de 2013

Aronia melanocarpa Elliot reduces the activity of angiotensin i-converting enzyme-in vitro and ex vivo studies

artículo científico publicado en 2014

Biocompatibility Studies of Gadolinium Complexes with Iminodiacetic Acid Derivatives

artículo científico publicado en 2018

Biocompatible sulfenamide and sulfonamide derivatives of metformin can exert beneficial effects on plasma haemostasis

artículo científico publicado en 2017

Biological approach of anticancer activity of new benzimidazole derivatives

artículo científico publicado en 2014

Biological evaluation of the activity of some benzimidazole-4,7-dione derivatives

artículo científico publicado en 2014

Biological evaluation of the toxicity and the cell cycle interruption by some benzimidazole derivatives

artículo científico publicado en 2016

Determination of stability constants and acute toxicity of potential hepatotropic gadolinium complexes.

artículo científico publicado en 2010

Development of copper based drugs, radiopharmaceuticals and medical materials.

artículo científico publicado en 2012

Diagnostics and therapy of Alzheimer's disease.

artículo científico publicado en 2007

Erratum to: Biological evaluation of the toxicity and the cell cycle interruption by some benzimidazole derivatives

artículo científico publicado en 2016

Evaluation of poly(amidoamine) dendrimers as potential carriers of iminodiacetic derivatives using solubility studies and 2D-NOESY NMR spectroscopy.

artículo científico publicado en 2012

Extract of Aronia melanocarpa-modified hemostasis: in vitro studies

artículo científico publicado en 2014

Gadolinium Gd(III) complexes with derivatives of nitriloacetic acid: synthesis and biological properties.

artículo científico publicado en 2008

Generation 2 (G2) - Generation 4 (G4) PAMAM dendrimers disrupt key plasma coagulation parameters

scientific article published on 11 April 2019

Is Metformin a Perfect Drug? Updates in Pharmacokinetics and Pharmacodynamics

artículo científico publicado en 2016

Metabolite Profiling of Eastern Teaberry (Gaultheria procumbens L.) Lipophilic Leaf Extracts with Hyaluronidase and Lipoxygenase Inhibitory Activity.

artículo científico publicado en 2017

Metformin - a Future Therapy for Neurodegenerative Diseases : Theme: Drug Discovery, Development and Delivery in Alzheimer's Disease Guest Editor: Davide Brambilla

artículo científico

Metformin and Its Sulfenamide Prodrugs Inhibit Human Cholinesterase Activity

artículo científico publicado en 2017

Neuroimaging diagnosis in neurodegenerative diseases

artículo científico publicado el 1 de enero de 2010

New Perspectives of Alzheimer Disease Diagnosis - the Most Popular and Future Methods.

artículo científico publicado en 2017

New benzimidazole derivatives with potential cytotoxic activity--study of their stability by RP-HPLC

artículo científico publicado el 11 de junio de 2012

New cyclopentaquinoline derivatives with fluorobenzoic acid induce G1 arrest and apoptosis in human lung adenocarcinoma cells

artículo científico publicado en 2014

New derivatives of quinazoline and 1, 2-dihydroquinazoline n3-oxide with expected antitumor activity

artículo científico publicado en 2004

New prodrugs of metformin do not influence the overall haemostasis potential and integrity of the erythrocyte membrane

artículo científico publicado en 2017

New tacrine analogs as acetylcholinesterase inhibitors - theoretical study with chemometric analysis.

artículo científico publicado en 2013

Novel tetrahydroacridine and cyclopentaquinoline derivatives with fluorobenzoic acid moiety induce cell cycle arrest and apoptosis in lung cancer cells by activation of DNA damage signaling.

artículo científico publicado en 2017

Novel tetrahydroacridine derivatives inhibit human lung adenocarcinoma cell growth by inducing G1 phase cell cycle arrest and apoptosis

artículo científico publicado en 2014

Novel tetrahydroacridine derivatives with iodobenzoic acid moiety as multifunctional acetylcholinesterase inhibitors.

artículo científico publicado en 2017

PAMAM Dendrimers as Potential Carriers of Gadolinium Complexes of Iminodiacetic Acid Derivatives for Magnetic Resonance Imaging

Radiolabeled Peptides and Antibodies in Medicine

artículo científico publicado en 2020

Re-evaluation of the retention time prediction "polarity" model in the context of the development of a stationary phase variable.

artículo científico publicado en 2014

Short-term supplementation with Aronia melanocarpa extract improves platelet aggregation, clotting, and fibrinolysis in patients with metabolic syndrome

artículo científico publicado en 2011

Some characteristics of activity of potential chemotherapeutics--benzimidazole derivatives

artículo científico

Stability of erythrocyte membrane and overall hemostasis potential - A biocompatibility study of mebrofenin and other iminodiacetic acid derivatives

scientific article published on 04 June 2015

Studies towards biocompatibility of PAMAM dendrimers--overall hemostasis potential and integrity of the human aortic endothelial barrier

artículo científico publicado en 2014

Sulfenamide and sulfonamide derivatives of metformin can exert anti-coagulant and pro-fibrinolytic properties

artículo científico publicado en 2018

Synthesis and Biocompatibility Studies of New Iminodiacetic Acid Derivatives

artículo científico publicado en 2017

Synthesis and biological activity of derivatives of tetrahydroacridine as acetylcholinesterase inhibitors

artículo científico publicado el 12 de mayo de 2011

Synthesis, biological activity and HPLC validation of 1,2,3,4-tetrahydroacridine derivatives as acetylcholinesterase inhibitors.

artículo científico publicado en 2011

Synthesis, biological evaluation and molecular modeling of new tetrahydroacridine derivatives as potential multifunctional agents for the treatment of Alzheimer's disease.

artículo científico publicado en 2015

Synthesis, physicochemical and biological studies of technetium-99m labeled tacrine derivative as a diagnostic tool for evaluation of cholinesterase level

artículo científico publicado en 2016

Taxodione and Extracts from Salvia austriaca Roots as Human Cholinesterase Inhibitors.

artículo científico publicado en 2015

Tetrahydroacridine derivatives with fluorobenzoic acid moiety as multifunctional agents for Alzheimer's disease treatment

artículo científico publicado en 2017

The Associations between Central Nervous System Diseases and Haemostatic Disorders

artículo científico publicado en 2019