Lista de obras -

1,2,4-Triazolidine-3-thiones Have Specific Activity against Acinetobacter baumannii among Common Nosocomial Pathogens.

artículo científico publicado en 2016

1,2,4-Triazolidine-3-thiones as Narrow Spectrum Antibiotics against Multidrug-Resistant Acinetobacter baumannii.

artículo científico publicado en 2016

2-Aminobenzimidazoles as antibiofilm agents against serovar Typhimurium

scientific article published on 02 August 2018

2-aminoimidazoles collapse mycobacterial proton motive force and block the electron transport chain

artículo científico publicado en 2019

2-aminoimidazoles potentiate ß-lactam antimicrobial activity against Mycobacterium tuberculosis by reducing ß-lactamase secretion and increasing cell envelope permeability.

artículo científico publicado en 2017

A Clerodane Diterpene from Callicarpa americana Resensitizes Methicillin-Resistant Staphylococcus aureus to ß-Lactam Antibiotics

artículo científico publicado en 2020

A bifurcated proteoglycan binding small molecule carrier for siRNA delivery.

artículo científico publicado en 2014

Augmenting the Activity of Macrolide Adjuvants against Acinetobacter baumannii

scientific article published on 12 August 2020

Controlling bacterial behavior with indole-containing natural products and derivatives

artículo científico publicado en 2014

Disruption of heterotypic community development by Porphyromonas gingivalis with small molecule inhibitors

artículo científico publicado en 2014

Eukaryotic phosphatase inhibitors enhance colistin efficacy in gram-negative bacteria

scientific article published on 19 June 2020

From worms to targeting virulence factors

artículo científico publicado en 2015

Identification of Anti-Mycobacterial Biofilm Agents Based on the 2-Aminoimidazole Scaffold

artículo científico publicado en 2019

Inhibition and breaking of advanced glycation end-products (AGEs) with bis-2-aminoimidazole derivatives

artículo científico publicado en 2015

Innovative strategies for combating biofilm-based infections

artículo científico publicado en 2015

Marine sponge alkaloids as a source of anti-bacterial adjuvants.

artículo científico publicado en 2016

Meridianin D Analogues Display Antibiofilm Activity against MRSA and Increase Colistin Efficacy in Gram-Negative Bacteria

artículo científico publicado en 2018

Narrow-Spectrum Antibacterial Agents.

artículo científico publicado en 2017

Natural products as inspiration for the development of bacterial antibiofilm agents

artículo científico publicado en 2020

New Class of Adjuvants Enables Lower Dosing of Colistin Against Acinetobacter baumannii

artículo científico publicado en 2018

Potentiation of Francisella Resistance to Conventional Antibiotics through Small Molecule Adjuvants

artículo científico publicado en 2015

Probing the Mechanism of LAL-32, a Gold Nanoparticle-Based Antibiotic Discovered through Small Molecule Variable Ligand Display.

artículo científico publicado en 2017

Re-sensitizing Multidrug Resistant Bacteria to Antibiotics by Targeting Bacterial Response Regulators: Characterization and Comparison of Interactions between 2-Aminoimidazoles and the Response Regulators BfmR from Acinetobacter baumannii and QseB f

artículo científico publicado en 2018

Repurposing Eukaryotic Kinase Inhibitors as Colistin Adjuvants in Gram-Negative Bacteria

scientific article published on 04 September 2019

Reversal of Mycobacterium tuberculosis phenotypic drug resistance by 2-aminoimidazole-based small molecules

artículo científico publicado en 2014

Screening an established natural product library identifies secondary metabolites that potentiate conventional antibiotics

scientific article published on 18 August 2020

Second Generation Meridianin Analogs Inhibit the Formation of Mycobacterium smegmatis Biofilms and Sensitize Polymyxin-Resistant Gram-Negative Bacteria to Colistin

artículo científico publicado en 2020

Second Generation Modifiers of Colistin Resistance Show Enhanced Activity and Lower Inherent Toxicity

artículo científico publicado en 2016

Second generation 2-aminoimidazole based advanced glycation end product inhibitors and breakers

artículo científico publicado en 2015

Second-Generation Tryptamine Derivatives Potently Sensitize Colistin Resistant Bacteria to Colistin

artículo científico publicado en 2019

Small Molecule Potentiation of Gram-Positive Selective Antibiotics against Acinetobacter baumannii

artículo científico publicado en 2019

Small molecule adjuvants that suppress both chromosomal and mcr-1 encoded colistin-resistance and amplify colistin efficacy in polymyxin-susceptible bacteria.

artículo científico publicado en 2017

Small steps to new drugs for bugs

artículo científico publicado en 2015

Small-molecule suppression of β-lactam resistance in multidrug-resistant gram-negative pathogens

artículo científico publicado en 2014

Structure of the Francisella response regulator QseB receiver domain, and characterization of QseB inhibition by antibiofilm 2-aminoimidazole-based compounds

artículo científico publicado en 2017

Synthesis and Biofilm Inhibition Studies of 2-(2-amino-6-arylpyrimidin-4-yl)quinazolin-4(3H)-ones

artículo científico publicado en 2020

The Challenge of Overcoming Antibiotic Resistance: An Adjuvant Approach?

artículo científico publicado en 2017

The Discovery of 2-Aminobenzimidazoles That Sensitize Mycobacterium smegmatis and M. tuberculosis to β-Lactam Antibiotics in a Pattern Distinct from β-Lactamase Inhibitors.

artículo científico publicado en 2017

Thiol-modified gold nanoparticles for the inhibition of Mycobacterium smegmatis

artículo científico publicado en 2014

Tryptamine derivatives disarm colistin resistance in polymyxin-resistant gram-negative bacteria

artículo científico publicado en 2019

Using 2-aminobenzimidazole derivatives to inhibit Mycobacterium smegmatis biofilm formation

Using Small-Molecule Adjuvants to Repurpose Azithromycin for Use against Pseudomonas aeruginosa

scientific article published on 29 November 2018

Lista de obras de

1,2,4-Triazolidine-3-thiones Have Specific Activity against Acinetobacter baumannii among Common Nosocomial Pathogens.

1,2,4-Triazolidine-3-thiones as Narrow Spectrum Antibiotics against Multidrug-Resistant Acinetobacter baumannii.

2-Aminobenzimidazoles as antibiofilm agents against serovar Typhimurium

2-aminoimidazoles collapse mycobacterial proton motive force and block the electron transport chain

2-aminoimidazoles potentiate ß-lactam antimicrobial activity against Mycobacterium tuberculosis by reducing ß-lactamase secretion and increasing cell envelope permeability.

A Clerodane Diterpene from Callicarpa americana Resensitizes Methicillin-Resistant Staphylococcus aureus to ß-Lactam Antibiotics

A bifurcated proteoglycan binding small molecule carrier for siRNA delivery.

Augmenting the Activity of Macrolide Adjuvants against Acinetobacter baumannii

Controlling bacterial behavior with indole-containing natural products and derivatives

Disruption of heterotypic community development by Porphyromonas gingivalis with small molecule inhibitors

Eukaryotic phosphatase inhibitors enhance colistin efficacy in gram-negative bacteria

From worms to targeting virulence factors

Identification of Anti-Mycobacterial Biofilm Agents Based on the 2-Aminoimidazole Scaffold

Inhibition and breaking of advanced glycation end-products (AGEs) with bis-2-aminoimidazole derivatives

Innovative strategies for combating biofilm-based infections

Marine sponge alkaloids as a source of anti-bacterial adjuvants.

Meridianin D Analogues Display Antibiofilm Activity against MRSA and Increase Colistin Efficacy in Gram-Negative Bacteria

Narrow-Spectrum Antibacterial Agents.

Natural products as inspiration for the development of bacterial antibiofilm agents

New Class of Adjuvants Enables Lower Dosing of Colistin Against Acinetobacter baumannii

Potentiation of Francisella Resistance to Conventional Antibiotics through Small Molecule Adjuvants

Probing the Mechanism of LAL-32, a Gold Nanoparticle-Based Antibiotic Discovered through Small Molecule Variable Ligand Display.

Re-sensitizing Multidrug Resistant Bacteria to Antibiotics by Targeting Bacterial Response Regulators: Characterization and Comparison of Interactions between 2-Aminoimidazoles and the Response Regulators BfmR from Acinetobacter baumannii and QseB f

Repurposing Eukaryotic Kinase Inhibitors as Colistin Adjuvants in Gram-Negative Bacteria

Reversal of Mycobacterium tuberculosis phenotypic drug resistance by 2-aminoimidazole-based small molecules

Screening an established natural product library identifies secondary metabolites that potentiate conventional antibiotics

Second Generation Meridianin Analogs Inhibit the Formation of Mycobacterium smegmatis Biofilms and Sensitize Polymyxin-Resistant Gram-Negative Bacteria to Colistin

Second Generation Modifiers of Colistin Resistance Show Enhanced Activity and Lower Inherent Toxicity

Second generation 2-aminoimidazole based advanced glycation end product inhibitors and breakers

Second-Generation Tryptamine Derivatives Potently Sensitize Colistin Resistant Bacteria to Colistin

Small Molecule Potentiation of Gram-Positive Selective Antibiotics against Acinetobacter baumannii

Small molecule adjuvants that suppress both chromosomal and mcr-1 encoded colistin-resistance and amplify colistin efficacy in polymyxin-susceptible bacteria.

Small steps to new drugs for bugs

Small-molecule suppression of β-lactam resistance in multidrug-resistant gram-negative pathogens

Structure of the Francisella response regulator QseB receiver domain, and characterization of QseB inhibition by antibiofilm 2-aminoimidazole-based compounds

Synthesis and Biofilm Inhibition Studies of 2-(2-amino-6-arylpyrimidin-4-yl)quinazolin-4(3H)-ones

The Challenge of Overcoming Antibiotic Resistance: An Adjuvant Approach?

The Discovery of 2-Aminobenzimidazoles That Sensitize Mycobacterium smegmatis and M. tuberculosis to β-Lactam Antibiotics in a Pattern Distinct from β-Lactamase Inhibitors.

Thiol-modified gold nanoparticles for the inhibition of Mycobacterium smegmatis

Tryptamine derivatives disarm colistin resistance in polymyxin-resistant gram-negative bacteria

Using 2-aminobenzimidazole derivatives to inhibit Mycobacterium smegmatis biofilm formation

Using Small-Molecule Adjuvants to Repurpose Azithromycin for Use against Pseudomonas aeruginosa