Lista de obras -

A Novel Allosteric Activator of Free Fatty Acid 2 Receptor Displays Unique Gi-functional Bias

artículo científico publicado en 2016

A single extracellular amino acid in Free Fatty Acid Receptor 2 defines antagonist species selectivity and G protein selection bias

artículo científico publicado en 2017

AM630 behaves as a protean ligand at the human cannabinoid CB2 receptor.

artículo científico publicado en 2012

CB(1) receptor allosteric modulators display both agonist and signaling pathway specificity.

artículo científico publicado en 2012

CB2 cannabinoid receptor agonist enantiomers HU-433 and HU-308: An inverse relationship between binding affinity and biological potency

artículo científico publicado en 2015

Cannabidiol, a non-psychoactive cannabinoid compound, inhibits proliferation and invasion in U87-MG and T98G glioma cells through a multitarget effect

artículo científico publicado en 2013

Chemogenetics defines receptor-mediated functions of short chain free fatty acids

artículo científico publicado en 2019

Discovery of a Potent Thiazolidine Free Fatty Acid Receptor 2 Agonist with Favorable Pharmacokinetic Properties

scientific article published on 12 October 2018

Expression and function of the endocannabinoid system in glial cells

artículo científico publicado en 2008

In vitro and in vivo pharmacological characterization of two novel selective cannabinoid CB(2) receptor inverse agonists

artículo científico publicado en 2009

Investigations on the 4-quinolone-3-carboxylic acid motif part 5: modulation of the physicochemical profile of a set of potent and selective cannabinoid-2 receptor ligands through a bioisosteric approach.

artículo científico publicado en 2012

Investigations on the 4-quinolone-3-carboxylic acid motif. 3. Synthesis, structure-affinity relationships, and pharmacological characterization of 6-substituted 4-quinolone-3-carboxamides as highly selective cannabinoid-2 receptor ligands

artículo científico publicado en 2010

Investigations on the 4-quinolone-3-carboxylic acid motif. 6. Synthesis and pharmacological evaluation of 7-substituted quinolone-3-carboxamide derivatives as high affinity ligands for cannabinoid receptors

artículo científico publicado en 2012

Ligands at the Free Fatty Acid Receptors 2/3 (GPR43/GPR41).

artículo científico publicado en 2016

Metabolic and inflammatory functions of short-chain fatty acid receptors

artículo científico publicado en 2020

On-target and off-target effects of novel orthosteric and allosteric activators of GPR84

artículo científico publicado en 2019

Structural and pharmacological analysis of O-2050, a putative neutral cannabinoid CB(1) receptor antagonist.

artículo científico publicado en 2010

The Pharmacology and Function of Receptors for Short-Chain Fatty Acids.

artículo científico

The plant cannabinoid Delta9-tetrahydrocannabivarin can decrease signs of inflammation and inflammatory pain in mice

artículo científico publicado en 2010

Treatment of Active Crohn’s Disease With an Ordinary Food-based Diet That Replicates Exclusive Enteral Nutrition

artículo científico publicado en 2018

Lista de obras de

A Novel Allosteric Activator of Free Fatty Acid 2 Receptor Displays Unique Gi-functional Bias

A single extracellular amino acid in Free Fatty Acid Receptor 2 defines antagonist species selectivity and G protein selection bias

AM630 behaves as a protean ligand at the human cannabinoid CB2 receptor.

CB(1) receptor allosteric modulators display both agonist and signaling pathway specificity.

CB2 cannabinoid receptor agonist enantiomers HU-433 and HU-308: An inverse relationship between binding affinity and biological potency

Cannabidiol, a non-psychoactive cannabinoid compound, inhibits proliferation and invasion in U87-MG and T98G glioma cells through a multitarget effect

Chemogenetics defines receptor-mediated functions of short chain free fatty acids

Discovery of a Potent Thiazolidine Free Fatty Acid Receptor 2 Agonist with Favorable Pharmacokinetic Properties

Expression and function of the endocannabinoid system in glial cells

In vitro and in vivo pharmacological characterization of two novel selective cannabinoid CB(2) receptor inverse agonists

Investigations on the 4-quinolone-3-carboxylic acid motif part 5: modulation of the physicochemical profile of a set of potent and selective cannabinoid-2 receptor ligands through a bioisosteric approach.

Investigations on the 4-quinolone-3-carboxylic acid motif. 3. Synthesis, structure-affinity relationships, and pharmacological characterization of 6-substituted 4-quinolone-3-carboxamides as highly selective cannabinoid-2 receptor ligands

Investigations on the 4-quinolone-3-carboxylic acid motif. 6. Synthesis and pharmacological evaluation of 7-substituted quinolone-3-carboxamide derivatives as high affinity ligands for cannabinoid receptors

Ligands at the Free Fatty Acid Receptors 2/3 (GPR43/GPR41).

Metabolic and inflammatory functions of short-chain fatty acid receptors

On-target and off-target effects of novel orthosteric and allosteric activators of GPR84

Structural and pharmacological analysis of O-2050, a putative neutral cannabinoid CB(1) receptor antagonist.

The Pharmacology and Function of Receptors for Short-Chain Fatty Acids.

The plant cannabinoid Delta9-tetrahydrocannabivarin can decrease signs of inflammation and inflammatory pain in mice

Treatment of Active Crohn’s Disease With an Ordinary Food-based Diet That Replicates Exclusive Enteral Nutrition