Lista de obras -

18F-labeling and evaluation of novel MDL 100907 derivatives as potential 5-HT2A antagonists for molecular imaging

artículo científico publicado en 2010

72/74As-labeling of HPMA based polymers for long-term in vivo PET imaging

artículo científico publicado en 2010

AAZTA5/AAZTA5-TOC: synthesis and radiochemical evaluation with 68Ga, 44Sc and 177Lu

scientific article published on 01 August 2019

Activation of P-glycoprotein (Pgp)-mediated drug efflux by extracellular acidosis: in vivo imaging with 68Ga-labelled PET tracer

artículo científico publicado en 2010

An approach to the evaluation of the activity of the DNA repair enzyme O6-methylguanine-DNA-methyl-transferase in tumor tissue in vivo: syntheses of 6-benzyloxy-9-(2-[18F]fluoroethyl)-9H-purin-2-yl-amine and 6-benzyloxy-7-(2-[18F]fluoroethyl)-7H-pur

artículo científico publicado en 2002

Assessing p-Glycoprotein (Pgp) Activity In Vivo Utilizing 68Ga–Schiff Base Complexes ⬇️

artículo científico publicado el 1 de octubre de 2011

Association of low striatal dopamine d2 receptor availability with nicotine dependence similar to that seen with other drugs of abuse

artículo científico publicado en 2008

Asymmetry in dopamine D(2/3) receptors of caudate nucleus is lost with age.

artículo científico publicado en 2006

Automated synthesis and purification of [18F]fluoro-[di-deutero]methyl tosylate

artículo científico publicado en 2013

Brain and plasma pharmacokinetics of aripiprazole in patients with schizophrenia: an [18F]fallypride PET study

artículo científico publicado en 2008

Characterization of the serotonin 2A receptor selective PET tracer (R)-[18F]MH.MZ in the human brain

artículo científico publicado en 2019

Clinical Translation and First In-Human Use of [44Sc]Sc-PSMA-617 for PET Imaging of Metastasized Castrate-Resistant Prostate Cancer

artículo científico publicado en 2017

Comparison Study of Two Differently Clicked 18F-Folates-Lipophilicity Plays a Key Role

artículo científico publicado en 2018

Comparison of Linear and Hyperbranched Polyether Lipids for Liposome Shielding by 18F-Radiolabeling and Positron Emission Tomography

artículo científico publicado en 2018

Correlation between dopamine D(2) receptors in the ventral striatum and central processing of alcohol cues and craving

artículo científico publicado en 2004

Correlation of alcohol craving with striatal dopamine synthesis capacity and D2/3 receptor availability: a combined [18F]DOPA and [18F]DMFP PET study in detoxified alcoholic patients.

artículo científico publicado en 2005

Decreased dopamine D2/D3-receptor binding in temporal lobe epilepsy: an [18F]fallypride PET study

artículo científico publicado en 2006

Direct radiofluorination of [18F]MH.MZ for 5-HT2A receptor molecular imaging with PET

scholarly article by Matthias M. Herth et al published July 2012 in Journal of Labelled Compounds and Radiopharmaceuticals

Dopamine D2/3 receptor occupancy by quetiapine in striatal and extrastriatal areas

artículo científico publicado en 2010

Electron- and positron-emitting radiolanthanides for therapy: aspects of dosimetry and production

article

Equilibrium, Kinetic and Structural Properties of Gallium(III) and Some Divalent Metal Complexes Formed with the New DATAm and DATA5m Ligands.

artículo científico publicado en 2017

Ethanol-Based Post-processing of Generator-Derived ⁶⁸Ga Toward Kit-Type Preparation of ⁶⁸Ga-Radiopharmaceuticals

artículo científico publicado en 2014

Evaluation of P-glycoprotein (abcb1a/b) modulation of [(18)F]fallypride in MicroPET imaging studies

artículo científico publicado en 2013

Evaluation of safety and dosimetry of <sup>177</sup>Lu DOTA-ZOL for therapy of bone metastases

artículo científico publicado en 2021

Evaluation of the inverse electron demand Diels-Alder reaction in rats using a scandium-44-labelled tetrazine for pretargeted PET imaging

artículo científico publicado en 2019

Fate of linear and branched polyether-lipids in vivo in comparison to their liposomal formulations by 18F-radiolabeling and positron emission tomography

artículo científico publicado en 2015

Ga[Ga]-, In[In]-oxine: a novel strategy of radiolabeling of HPMA-based micelles

HPMA Based Amphiphilic Copolymers Mediate Central Nervous Effects of Domperidone

artículo científico publicado en 2011

HPMA-LMA copolymer drug carriers in oncology: an in vivo PET study to assess the tumor line-specific polymer uptake and body distribution

artículo científico publicado en 2013

High opiate receptor binding potential in the human lateral pain system

artículo científico publicado en 2005

High striatal occupancy of D2-like dopamine receptors by amisulpride in the brain of patients with schizophrenia

artículo científico publicado en 2004

Image quality analysis of 44Sc on two preclinical PET scanners: a comparison to 68Ga

artículo científico publicado en 2020

Imaging Nigrostriatal Dopaminergic Deficit in Holmes Tremor with 18F-PR04.MZ-PET/CT.

artículo científico publicado en 2015

Imaging of protein synthesis: in vitro and in vivo evaluation of (44)Sc-DOTA-puromycin.

artículo científico publicado en 2013

Improved Efficacy of Synthesizing *MIII-Labeled DOTA Complexes in Binary Mixtures of Water and Organic Solvents. A Combined Radio- and Physicochemical Study

artículo científico publicado en 2018

In vitro affinities of various halogenated benzamide derivatives as potential radioligands for non-invasive quantification of D(2)-like dopamine receptors

artículo científico publicado en 2007

In vitro and in vivo structure-property relationship of (68)Ga-labeled Schiff base derivatives for functional myocardial pet imaging

artículo científico publicado en 2014

In vivo Evaluation of [225Ac]Ac-DOTAZOL for α-Therapy of Bone Metastases

artículo científico publicado en 2018

Inhibition of O6-methylguanine-DNA methyltransferase by glucose-conjugated inhibitors: comparison with nonconjugated inhibitors and effect on fotemustine and temozolomide-induced cell death

artículo científico publicado en 2004

Labeling of DOTA-conjugated HPMA-based polymers with trivalent metallic radionuclides for molecular imaging.

artículo científico publicado en 2018

Long-term biodistribution study of HPMA-ran-LMA copolymers in vivo by means of 131I-labeling

artículo científico publicado en 2017

Measurement of Protein Synthesis: In Vitro Comparison of 68Ga-DOTA-Puromycin, [3H]Tyrosine, and 2-Fluoro-[3H]tyrosine ⬇️

artículo científico publicado el 1 de enero de 2013

Modifying the body distribution of HPMA-based copolymers by molecular weight and aggregate formation

artículo científico publicado en 2011

NODAPA-OH and NODAPA-(NCS)n: synthesis, 68Ga-radiolabelling and in vitro characterisation of novel versatile bifunctional chelators for molecular imaging

artículo científico publicado en 2008

Net influx of plasma 6-[18F]fluoro-L-DOPA (FDOPA) to the ventral striatum correlates with prefrontal processing of affective stimuli

artículo científico publicado en 2006

On the consensus nomenclature rules for radiopharmaceutical chemistry - Reconsideration of radiochemical conversion

artículo científico publicado en 2020

Opiate-induced dopamine release is modulated by severity of alcohol dependence: an [(18)F]fallypride positron emission tomography study

artículo científico publicado en 2011

Optimization of Labeling PSMAHBED with Ethanol-Postprocessed 68Ga and Its Quality Control Systems

artículo científico publicado en 2017

PEGylation of HPMA-based block copolymers enhances tumor accumulation in vivo: a quantitative study using radiolabeling and positron emission tomography

artículo científico publicado en 2013

PET imaging of the impact of extracellular pH and MAP kinases on the p-glycoprotein (Pgp) activity

artículo científico publicado en 2013

Parametric mapping of binding in human brain of D2 receptor ligands of different affinities

artículo científico publicado en 2005

Pharmacokinetic evaluation of [18F]PR04.MZ for PET/CT imaging and quantification of dopamine transporters in the human brain

scientific article published on 01 December 2019

Positron emission tomography in CNS drug discovery and drug monitoring

artículo científico publicado en 2014

Predicting the in vivo release from a liposomal formulation by IVIVC and non-invasive positron emission tomography imaging

artículo científico publicado en 2010

Preliminary in vivo and ex vivo evaluation of the 5-HT2A imaging probe [(18)F]MH.MZ.

artículo científico publicado en 2009

Processing of generator-produced 68Ga for medical application.

artículo científico publicado en 2007

Quantification of D2-like dopamine receptors in the human brain with 18F-desmethoxyfallypride.

artículo científico publicado en 2003

Quantitative online isolation of 68Ge from 68Ge/68Ga generator eluates for purification and immediate quality control of breakthrough ⬇️

artículo científico publicado el 25 de julio de 2013

Radioactive labeling of defined HPMA-based polymeric structures using [18F]FETos for in vivo imaging by positron emission tomography.

artículo científico publicado en 2009

Radiolabelling and preliminary evaluation of 68Ga-tetrapyrrole derivatives as potential tracers for PET ⬇️

artículo científico publicado el 21 de diciembre de 2012

Radiolanthanides in nuclear medicine.

artículo científico publicado en 2004

Ratio of dopamine synthesis capacity to D2 receptor availability in ventral striatum correlates with central processing of affective stimuli

artículo científico publicado en 2008

Selective binding to monoamine oxidase A: in vitro and in vivo evaluation of (18)F-labeled β-carboline derivatives

artículo científico publicado en 2014

Striatal and extrastriatal D2/D3-receptor-binding properties of ziprasidone: a positron emission tomography study with [18F]Fallypride and [11C]raclopride (D2/D3-receptor occupancy of ziprasidone).

artículo científico publicado en 2008

Structural combination of established 5-HT(2A) receptor ligands: new aspects of the binding mode

artículo científico publicado en 2010

Structure-function evaluation of imidazopyridine derivatives selective for δ subunit containing γ-aminobutyric acid type A (GABAA) receptors

artículo científico publicado en 2018

Surrogate markers for cerebral blood flow correlate with [¹⁸F]-fallypride binding potential at dopamine D(2/3) receptors in human striatum.

artículo científico publicado en 2013

Synthesis and evaluation of 5,7-dichloro-4-(3-{4-[4-(2-[18F]fluoroethyl)-piperazin-1-yl]-phenyl}-ureido)-1,2,3,4-tetrahydroquinoline-2-carboxylic acid as a potential NMDA ligand to study glutamatergic neurotransmission in vivo

Synthesis and in vitro affinities of various MDL 100907 derivatives as potential 18F-radioligands for 5-HT2A receptor imaging with PET.

artículo científico publicado en 2009

Synthesis and in vitro evaluation of (S)-2-([11C]methoxy)-4-[3-methyl-1-(2-piperidine-1-yl-phenyl)-butyl-carbamoyl]-benzoic acid ([11C]methoxy-repaglinide): a potential beta-cell imaging agent

artículo científico publicado en 2004

Synthesis and preliminary evaluation of (R,R)(S,S) 5-(2-(2-[4-(2-[(18)F]fluoroethoxy)phenyl]-1-methylethylamino)-1-hydroxyethyl)-benzene-1,3-diol ([(18)F]FEFE) for the in vivo visualisation and quantification of the beta2-adrenergic receptor status

artículo científico publicado en 2003

Synthesis of 131I-labeled glucose-conjugated inhibitors of O6-methylguanine-DNA methyltransferase (MGMT) and comparison with nonconjugated inhibitors as potential tools for in vivo MGMT imaging

artículo científico publicado en 2006

Targeting fibroblast activation protein (FAP): next generation PET radiotracers using squaramide coupled bifunctional DOTA and DATA5m chelators

artículo científico publicado en 2020

The applicability of SRTM in [18F]fallypride PET investigations: Impact of scan durations ⬇️

artículo científico publicado el 18 de mayo de 2011

The dopamine D2 receptor ligand 18F-desmethoxyfallypride: an appropriate fluorinated PET tracer for the differential diagnosis of parkinsonism

artículo científico publicado en 2004

The striatal and extrastriatal D2/D3 receptor-binding profile of clozapine in patients with schizophrenia

artículo científico publicado en 2006

Total synthesis and evaluation of [18F]MHMZ.

artículo científico publicado en 2007

Vulnerability to psychotogenic effects of ketamine is associated with elevated D2/3-receptor availability

artículo científico publicado en 2012

[(11)C]PR04.MZ, a promising DAT ligand for low concentration imaging: Synthesis, efficient (11)C-O-methylation and initial small animal PET studies.

artículo científico publicado en 2009

[18F]PR04.MZ PET/CT Imaging for Evaluation of Nigrostriatal Neuron Integrity in Patients With Parkinson Disease

artículo científico publicado en 2020

[68Ga]Ga-DATA5m-LM4, a PET Radiotracer in the Diagnosis of SST2R-Positive Tumors: Preclinical and First Clinical Results

artículo científico publicado en 2022

⁶⁸Ge content quality control of ⁶⁸Ge/⁶⁸Ga-generator eluates and ⁶⁸Ga radiopharmaceuticals--a protocol for determining the ⁶⁸Ge content using thin-layer chromatography

artículo científico publicado en 2014

Lista de obras de

18F-labeling and evaluation of novel MDL 100907 derivatives as potential 5-HT2A antagonists for molecular imaging

72/74As-labeling of HPMA based polymers for long-term in vivo PET imaging

AAZTA5/AAZTA5-TOC: synthesis and radiochemical evaluation with 68Ga, 44Sc and 177Lu

Activation of P-glycoprotein (Pgp)-mediated drug efflux by extracellular acidosis: in vivo imaging with 68Ga-labelled PET tracer

An approach to the evaluation of the activity of the DNA repair enzyme O6-methylguanine-DNA-methyl-transferase in tumor tissue in vivo: syntheses of 6-benzyloxy-9-(2-[18F]fluoroethyl)-9H-purin-2-yl-amine and 6-benzyloxy-7-(2-[18F]fluoroethyl)-7H-pur

Assessing p-Glycoprotein (Pgp) Activity In Vivo Utilizing 68Ga–Schiff Base Complexes ⬇️

Association of low striatal dopamine d2 receptor availability with nicotine dependence similar to that seen with other drugs of abuse

Asymmetry in dopamine D(2/3) receptors of caudate nucleus is lost with age.

Automated synthesis and purification of [18F]fluoro-[di-deutero]methyl tosylate

Brain and plasma pharmacokinetics of aripiprazole in patients with schizophrenia: an [18F]fallypride PET study

Characterization of the serotonin 2A receptor selective PET tracer (R)-[18F]MH.MZ in the human brain

Clinical Translation and First In-Human Use of [44Sc]Sc-PSMA-617 for PET Imaging of Metastasized Castrate-Resistant Prostate Cancer

Comparison Study of Two Differently Clicked 18F-Folates-Lipophilicity Plays a Key Role

Comparison of Linear and Hyperbranched Polyether Lipids for Liposome Shielding by 18F-Radiolabeling and Positron Emission Tomography

Correlation between dopamine D(2) receptors in the ventral striatum and central processing of alcohol cues and craving

Correlation of alcohol craving with striatal dopamine synthesis capacity and D2/3 receptor availability: a combined [18F]DOPA and [18F]DMFP PET study in detoxified alcoholic patients.

Decreased dopamine D2/D3-receptor binding in temporal lobe epilepsy: an [18F]fallypride PET study

Direct radiofluorination of [18F]MH.MZ for 5-HT2A receptor molecular imaging with PET

Dopamine D2/3 receptor occupancy by quetiapine in striatal and extrastriatal areas

Electron- and positron-emitting radiolanthanides for therapy: aspects of dosimetry and production

Equilibrium, Kinetic and Structural Properties of Gallium(III) and Some Divalent Metal Complexes Formed with the New DATAm and DATA5m Ligands.

Ethanol-Based Post-processing of Generator-Derived ⁶⁸Ga Toward Kit-Type Preparation of ⁶⁸Ga-Radiopharmaceuticals

Evaluation of P-glycoprotein (abcb1a/b) modulation of [(18)F]fallypride in MicroPET imaging studies

Evaluation of safety and dosimetry of <sup>177</sup>Lu DOTA-ZOL for therapy of bone metastases

Evaluation of the inverse electron demand Diels-Alder reaction in rats using a scandium-44-labelled tetrazine for pretargeted PET imaging

Fate of linear and branched polyether-lipids in vivo in comparison to their liposomal formulations by 18F-radiolabeling and positron emission tomography

Ga[Ga]-, In[In]-oxine: a novel strategy of radiolabeling of HPMA-based micelles

HPMA Based Amphiphilic Copolymers Mediate Central Nervous Effects of Domperidone

HPMA-LMA copolymer drug carriers in oncology: an in vivo PET study to assess the tumor line-specific polymer uptake and body distribution

High opiate receptor binding potential in the human lateral pain system

High striatal occupancy of D2-like dopamine receptors by amisulpride in the brain of patients with schizophrenia

Image quality analysis of 44Sc on two preclinical PET scanners: a comparison to 68Ga

Imaging Nigrostriatal Dopaminergic Deficit in Holmes Tremor with 18F-PR04.MZ-PET/CT.

Imaging of protein synthesis: in vitro and in vivo evaluation of (44)Sc-DOTA-puromycin.

Improved Efficacy of Synthesizing *MIII-Labeled DOTA Complexes in Binary Mixtures of Water and Organic Solvents. A Combined Radio- and Physicochemical Study

In vitro affinities of various halogenated benzamide derivatives as potential radioligands for non-invasive quantification of D(2)-like dopamine receptors

In vitro and in vivo structure-property relationship of (68)Ga-labeled Schiff base derivatives for functional myocardial pet imaging

In vivo Evaluation of [225Ac]Ac-DOTAZOL for α-Therapy of Bone Metastases

Inhibition of O6-methylguanine-DNA methyltransferase by glucose-conjugated inhibitors: comparison with nonconjugated inhibitors and effect on fotemustine and temozolomide-induced cell death

Labeling of DOTA-conjugated HPMA-based polymers with trivalent metallic radionuclides for molecular imaging.

Long-term biodistribution study of HPMA-ran-LMA copolymers in vivo by means of 131I-labeling

Measurement of Protein Synthesis: In Vitro Comparison of 68Ga-DOTA-Puromycin, [3H]Tyrosine, and 2-Fluoro-[3H]tyrosine ⬇️

Modifying the body distribution of HPMA-based copolymers by molecular weight and aggregate formation

NODAPA-OH and NODAPA-(NCS)n: synthesis, 68Ga-radiolabelling and in vitro characterisation of novel versatile bifunctional chelators for molecular imaging

Net influx of plasma 6-[18F]fluoro-L-DOPA (FDOPA) to the ventral striatum correlates with prefrontal processing of affective stimuli

On the consensus nomenclature rules for radiopharmaceutical chemistry - Reconsideration of radiochemical conversion

Opiate-induced dopamine release is modulated by severity of alcohol dependence: an [(18)F]fallypride positron emission tomography study

Optimization of Labeling PSMAHBED with Ethanol-Postprocessed 68Ga and Its Quality Control Systems

PEGylation of HPMA-based block copolymers enhances tumor accumulation in vivo: a quantitative study using radiolabeling and positron emission tomography

PET imaging of the impact of extracellular pH and MAP kinases on the p-glycoprotein (Pgp) activity

Parametric mapping of binding in human brain of D2 receptor ligands of different affinities

Pharmacokinetic evaluation of [18F]PR04.MZ for PET/CT imaging and quantification of dopamine transporters in the human brain

Positron emission tomography in CNS drug discovery and drug monitoring

Predicting the in vivo release from a liposomal formulation by IVIVC and non-invasive positron emission tomography imaging

Preliminary in vivo and ex vivo evaluation of the 5-HT2A imaging probe [(18)F]MH.MZ.

Processing of generator-produced 68Ga for medical application.

Quantification of D2-like dopamine receptors in the human brain with 18F-desmethoxyfallypride.

Quantitative online isolation of 68Ge from 68Ge/68Ga generator eluates for purification and immediate quality control of breakthrough ⬇️

Radioactive labeling of defined HPMA-based polymeric structures using [18F]FETos for in vivo imaging by positron emission tomography.

Radiolabelling and preliminary evaluation of 68Ga-tetrapyrrole derivatives as potential tracers for PET ⬇️

Radiolanthanides in nuclear medicine.

Ratio of dopamine synthesis capacity to D2 receptor availability in ventral striatum correlates with central processing of affective stimuli

Selective binding to monoamine oxidase A: in vitro and in vivo evaluation of (18)F-labeled β-carboline derivatives

Striatal and extrastriatal D2/D3-receptor-binding properties of ziprasidone: a positron emission tomography study with [18F]Fallypride and [11C]raclopride (D2/D3-receptor occupancy of ziprasidone).

Structural combination of established 5-HT(2A) receptor ligands: new aspects of the binding mode

Structure-function evaluation of imidazopyridine derivatives selective for δ subunit containing γ-aminobutyric acid type A (GABAA) receptors

Surrogate markers for cerebral blood flow correlate with [¹⁸F]-fallypride binding potential at dopamine D(2/3) receptors in human striatum.

Synthesis and evaluation of 5,7-dichloro-4-(3-{4-[4-(2-[18F]fluoroethyl)-piperazin-1-yl]-phenyl}-ureido)-1,2,3,4-tetrahydroquinoline-2-carboxylic acid as a potential NMDA ligand to study glutamatergic neurotransmission in vivo

Synthesis and in vitro affinities of various MDL 100907 derivatives as potential 18F-radioligands for 5-HT2A receptor imaging with PET.

Synthesis and in vitro evaluation of (S)-2-([11C]methoxy)-4-[3-methyl-1-(2-piperidine-1-yl-phenyl)-butyl-carbamoyl]-benzoic acid ([11C]methoxy-repaglinide): a potential beta-cell imaging agent

Synthesis and preliminary evaluation of (R,R)(S,S) 5-(2-(2-[4-(2-[(18)F]fluoroethoxy)phenyl]-1-methylethylamino)-1-hydroxyethyl)-benzene-1,3-diol ([(18)F]FEFE) for the in vivo visualisation and quantification of the beta2-adrenergic receptor status

Synthesis of 131I-labeled glucose-conjugated inhibitors of O6-methylguanine-DNA methyltransferase (MGMT) and comparison with nonconjugated inhibitors as potential tools for in vivo MGMT imaging

Targeting fibroblast activation protein (FAP): next generation PET radiotracers using squaramide coupled bifunctional DOTA and DATA5m chelators

The applicability of SRTM in [18F]fallypride PET investigations: Impact of scan durations ⬇️

The dopamine D2 receptor ligand 18F-desmethoxyfallypride: an appropriate fluorinated PET tracer for the differential diagnosis of parkinsonism

The striatal and extrastriatal D2/D3 receptor-binding profile of clozapine in patients with schizophrenia

Total synthesis and evaluation of [18F]MHMZ.

Vulnerability to psychotogenic effects of ketamine is associated with elevated D2/3-receptor availability

[(11)C]PR04.MZ, a promising DAT ligand for low concentration imaging: Synthesis, efficient (11)C-O-methylation and initial small animal PET studies.