Lista de obras -

A Gold(I)-Catalyzed Hydroamination/Cycloisomerization Cascade: Concise Synthesis of (±)-seco-Antofine and (±)-Septicine

artículo científico publicado en 2020

A Gold-Catalyzed Domino Cyclization Enabling Rapid Construction of Diverse Polyheterocyclic Frameworks

artículo científico publicado en 2017

A Lewis Base Catalysis Approach for the Photoredox Activation of Boronic Acids and Esters.

artículo científico publicado en 2017

A chromone analog inhibits TNF-alpha induced expression of cell adhesion molecules on human endothelial cells via blocking NF-kappaB activation

artículo científico publicado en 2007

A divergent synthesis of substituted 2-aminoimidazoles from 2-aminopyrimidines

artículo científico publicado en 2008

A gold-triggered dearomative spirocarbocyclization/Diels-Alder reaction cascade towards diverse bridged N-heterocycles

scientific article published on 01 November 2019

A microwave-assisted diastereoselective multicomponent reaction to access dibenzo[c,e]azepinones: synthesis and biological evaluation.

artículo científico publicado en 2011

A new colorimetric test for solid-phase amines and thiols

artículo científico publicado en 2008

A novel and versatile entry to asymmetrically substituted pyrazines

artículo científico publicado en 2008

A walk around the A3-coupling

artículo científico

Access to Polycyclic Azepino[5,4,3-cd]indoles via a Gold-Catalyzed Post-Ugi Dearomatization Cascade

artículo científico publicado en 2020

Aldehydes: magnificent acyl equivalents for direct acylation

artículo científico publicado en 2020

An antibiofilm coating of 5-aryl-2-aminoimidazole covalently attached to a titanium surface

artículo científico publicado en 2018

Anti-inflammatory and antioxidant properties of Piper species: a perspective from screening to molecular mechanisms.

artículo científico publicado en 2015

C-N bond forming cross-coupling reactions: an overview

artículo científico

Chemo- and Regioselective Catalyst-Controlled Carbocyclization of Alkynyl Ketones: Rapid Synthesis of 1-Indanones and 1-Naphthols

scientific article published on 10 May 2019

Click chemistry under non-classical reaction conditions.

scientific article published on 27 July 2009

Combining the Ugi-azide multicomponent reaction and rhodium(III)-catalyzed annulation for the synthesis of tetrazole-isoquinolone/pyridone hybrids

scientific article published on 16 October 2019

Concise and diversity-oriented route toward polysubstituted 2-aminoimidazole alkaloids and their analogues.

artículo científico publicado en 2010

CuICuII and AgIp-isocyanobenzoates as novel 1D semiconducting coordination oligomers

artículo científico publicado en 2020

DBU-Catalyzed Alkyne-Imidate Cyclization toward 1-Alkoxypyrazino[1,2- a]indole Synthesis

artículo científico publicado en 2018

Development of a new microwave-assisted cleavable backbone amide linker (BAL): a comparative study

artículo científico publicado en 2009

Developments in direct C-H arylation of (hetero)arenes under microwave irradiation.

artículo científico publicado en 2013

Diversity oriented microwave-assisted synthesis of (-)-steganacin aza-analogues.

artículo científico publicado en 2008

Doebner-type pyrazolopyridine carboxylic acids in an Ugi four-component reaction

artículo científico publicado en 2019

Domino Carbopalladation/C-H Functionalization Sequence: An Expedient Synthesis of Bis-Heteroaryls through Transient Alkyl/Vinyl-Palladium Species Capture

artículo científico publicado en 2015

Enhancing the anti-biofilm activity of 5-aryl-2-aminoimidazoles through nature inspired dimerisation

artículo científico publicado en 2018

Evaluation of the antibacterial and antibiofilm activities of novel CRAMP-vancomycin conjugates with diverse linkers.

artículo científico publicado en 2015

Evaluation of the toxicity of 5-aryl-2-aminoimidazole-based biofilm inhibitors against eukaryotic cell lines, bone cells and the nematode Caenorhabditis elegans.

artículo científico publicado en 2014

Facile access to functionalized spiro[indoline-3,2'-pyrrole]-2,5'-diones via post-Ugi domino Buchwald-Hartwig/Michael reaction

artículo científico publicado en 2014

Facile construction of diverse polyheterocyclic scaffolds via gold-catalysed dearomative spirocyclization/1,6-addition cascade

scientific article published on 01 June 2019

Gold-Catalyzed Post-Ugi Ipso-Cyclization with Switchable Diastereoselectivity

artículo científico publicado en 2018

Gold-catalyzed diastereoselective domino dearomatization/ipso-cyclization/aza-Michael sequence: a facile access to diverse fused azaspiro tetracyclic scaffolds.

artículo científico publicado en 2017

Gold-catalyzed post-MCR transformations towards complex (poly)heterocycles

scientific article published on 28 August 2018

Gold-catalyzed post-Ugi alkyne hydroarylation for the synthesis of 2-quinolones

artículo científico publicado en 2018

Heck-Suzuki Tandem Reaction for the Synthesis of 3-Benzazepines

artículo científico publicado en 2015

High-speed microwave-promoted hetero-Diels-Alder reactions of 2(1H)-pyrazinones in ionic liquid doped solvents

artículo científico publicado en 2002

Hypervalent Iodine(III)-Mediated Cascade Cyclization of Propargylguanidines and Total Syntheses of Kealiinine B and C.

artículo científico publicado en 2017

Identification of small peptides inhibiting the integrase-LEDGF/p75 interaction through targeting the cellular co-factor

artículo científico publicado en 2013

Inhibiting bacterial cooperation is an evolutionarily robust anti-biofilm strategy

artículo científico publicado en 2020

Iron(II)-Catalyzed Heck-Type Coupling of Vinylarenes with Alkyl Iodides

artículo científico publicado en 2019

Iterative Chemical Engineering of Vancomycin Leads to Novel Vancomycin Analogs With a High in Vitro Therapeutic Index.

artículo científico publicado en 2018

Metal-Free Dearomatization: Direct Access to Spiroindol(en)ines in Batch and Continuous-Flow

artículo científico publicado en 2019

Metal-mediated post-Ugi transformations for the construction of diverse heterocyclic scaffolds

artículo científico

Microwave-Assisted Copper-Catalyzed Oxidative Cyclization of Acrylamides with Non-Activated Ketones

artículo científico publicado en 2016

Microwave-assisted Cu(I)-catalyzed, three-component synthesis of 2-(4-((1-phenyl-1H-1,2,3-triazol-4-yl)methoxy)phenyl)-1H-benzo[d]imidazoles

artículo científico publicado en 2014

Microwave-assisted C–C bond forming cross-coupling reactions: an overview ⬇️

artículo científico publicado el 30 de junio de 2011

Microwave-assisted cycloaddition reactions

artículo científico publicado en 2009

Microwave-assisted one-pot synthesis and anti-biofilm activity of 2-amino-1H-imidazole/triazole conjugates

artículo científico publicado en 2014

Microwave-assisted synthesis of a novel class of imidazolylthiazolidin-4-ones and evaluation of its biological activities.

artículo científico publicado en 2010

Microwave-assisted synthesis of medium-sized heterocycles

artículo científico publicado en 2011

Microwave-enhanced transition metal-catalyzed decoration of 2(1H)-pyrazinone scaffolds

artículo científico publicado en 2003

Modular Access to Diverse Bridged Indole Alkaloid Mimics via a Gold-Triggered Cascade Dearomative Spirocarbocyclization/[4 + 2] Cycloaddition Sequence

scientific article published on 05 June 2019

Modulation of the Substitution Pattern of 5-Aryl-2-Aminoimidazoles Allows Fine-Tuning of Their Antibiofilm Activity Spectrum and Toxicity.

artículo científico publicado en 2016

New tricks of well-known aminoazoles in isocyanide-based multicomponent reactions and antibacterial activity of the compounds synthesized.

artículo científico publicado en 2017

Novel (2-amino-4-arylimidazolyl)propanoic acids and pyrrolo[1,2-c]imidazoles via the domino reactions of 2-amino-4-arylimidazoles with carbonyl and methylene active compounds

scientific article published on 06 May 2019

One-pot microwave-assisted protocol for the synthesis of substituted 2-amino-1H-imidazoles ⬇️

artículo científico publicado el 26 de agosto de 2010

Pd-catalyzed Csp(2) -H functionalization of heteroarenes via isocyanide insertion: concise synthesis of di-(hetero)aryl ketones and di-(hetero)aryl alkylamines

artículo científico publicado en 2015

Peptide macrocyclization by transition metal catalysis

artículo científico publicado en 2020

Photoredox-Catalyzed Hydrosulfonylation of Arylallenes

artículo científico publicado en 2020

Polysubstituted 2-aminoimidazoles as anti-biofilm and antiproliferative agents: Discovery of potent lead.

artículo científico publicado en 2017

Post-Ugi Cyclization for the Construction of Diverse Heterocyclic Compounds: Recent Updates

artículo científico publicado en 2018

Post-Ugi gold-catalyzed diastereoselective domino cyclization for the synthesis of diversely substituted spiroindolines

artículo científico publicado en 2013

Reactions of secondary propargylamines with heteroallenes for the synthesis of diverse heterocycles.

artículo científico publicado en 2018

Recent Advances in Phthalan and Coumaran Chemistry

artículo científico publicado en 2018

Recent advances in spirocyclization of indole derivatives.

artículo científico publicado en 2018

Retraction of "Iron-Catalyzed Three-Component Reaction: Synthesis of Fluoroalkylated 2 H-Azirines"

scientific article published on 21 November 2018

Rhodium(iii)-catalyzed intramolecular annulation through C-H activation: concise synthesis of rosettacin and oxypalmatime.

artículo científico publicado en 2017

Ruthenium-catalysed one-pot regio- and diastereoselective synthesis of pyrrolo[1,2-a]indoles via cascade C-H functionalization/annulation

artículo científico publicado en 2017

Sequential and direct multicomponent reaction (MCR)-based dearomatization strategies

artículo científico publicado en 2020

Smart Metal-Organic Framework Coatings: Triggered Antibiofilm Compound Release

artículo científico publicado en 2017

Solid-phase synthesis of the 2(1H)-pyrazinone scaffold: a new approach toward diversely substituted heterocycles

artículo científico publicado en 2005

Structure-activity relationship of 2-hydroxy-2-aryl-2,3-dihydro-imidazo[1,2-a]pyrimidinium salts and 2N-substituted 4(5)-aryl-2-amino-1H-imidazoles as inhibitors of biofilm formation by Salmonella Typhimurium and Pseudomonas aeruginosa.

artículo científico publicado en 2011

Structure-activity relationship of 4(5)-aryl-2-amino-1H-imidazoles, N1-substituted 2-aminoimidazoles and imidazo[1,2-a]pyrimidinium salts as inhibitors of biofilm formation by Salmonella typhimurium and Pseudomonas aeruginosa.

artículo científico publicado en 2010

Suzuki-Miyaura and Stille reactions as key steps in the synthesis of diversely functionalized Amaryllidaceae alkaloid analogs bearing a 5,6,7,8-tetrahydrobenzo[c,e]azocine skeleton

artículo científico publicado en 2007

Switching the regioselectivity via indium(III) and gold(I) catalysis: a post-Ugi intramolecular hydroarylation to azepino- and azocino-[c,d]indolones.

artículo científico publicado en 2013

Synthesis and HIV-1 RT inhibitory action of novel (4/6-substituted benzo[d]thiazol -2-yl)thiazolidin-4-ones. Divergence from the non-competitive inhibition mechanism

artículo científico publicado en 2012

Synthesis and anti-inflammatory activity evaluation of novel chroman derivatives

artículo científico publicado en 2020

Synthesis and anti-inflammatory activity evaluation of novel triazolyl-isatin hybrids.

artículo científico publicado en 2016

Synthesis and fungicidal activity of 3,5-dichloropyrazin-2(1H)-one derivatives.

artículo científico publicado en 2009

Synthesis of 1-(-methoxyphenyl)tetrazolyl-Substituted 1,2,3,4-Tetrahydroisoquinolines and Their Transformations Involving Activated Alkynes

artículo científico publicado en 2018

Synthesis of Pyrrolo[1,2-b]isoquinolines via Gold(I)-Catalyzed Cyclization/Enyne Cycloisomerization/1,2-Migration Cascade

artículo científico publicado en 2020

Synthetic Access to Secondary Propargylamines via a Copper-Catalyzed Oxidative Deamination/Alkynylation Cascade

scientific article published on 07 August 2019

The application of "click chemistry" for the decoration of 2(1H)-pyrazinone scaffold: generation of templates.

artículo científico publicado en 2005

Three-Component Reaction of 3-Arylidene-3H-Indolium Salts, Isocyanides, and Alcohols

scientific article published on 16 May 2019

Three-component reaction of a 2-aminoazine, a 2-oxoaldehyde, and a cyclic 1,3-dicarbonyl compound for the synthesis of imidazo[1,2-a]azine derivatives

artículo científico publicado en 2014

Transition metal-catalyzed C-C bond formation via C-S bond cleavage: an overview

artículo científico

Transition metal-catalyzed orthogonal solid-phase decoration of the 2(1H)-pyrazinone scaffold using a sulfur linker

artículo científico publicado en 2007

Tunability of Size and Magnetic Moment of Iron Oxide Nanoparticles Synthesized by Forced Hydrolysis

artículo científico publicado en 2016

Unprecedented Cu(I)-catalyzed microwave-assisted three-component coupling of a ketone, an alkyne, and a primary amine.

artículo científico publicado en 2010

Validation of an ultra-high-performance liquid chromatography-mass spectrometry method for the quantification of cysteinylated aldehydes and application to malt and beer samples

scientific article published on 20 August 2019

Visible light-mediated chemistry of indoles and related heterocycles

artículo científico publicado en 2019

Lista de obras de

A Gold(I)-Catalyzed Hydroamination/Cycloisomerization Cascade: Concise Synthesis of (±)-seco-Antofine and (±)-Septicine

A Gold-Catalyzed Domino Cyclization Enabling Rapid Construction of Diverse Polyheterocyclic Frameworks

A Lewis Base Catalysis Approach for the Photoredox Activation of Boronic Acids and Esters.

A chromone analog inhibits TNF-alpha induced expression of cell adhesion molecules on human endothelial cells via blocking NF-kappaB activation

A divergent synthesis of substituted 2-aminoimidazoles from 2-aminopyrimidines

A gold-triggered dearomative spirocarbocyclization/Diels-Alder reaction cascade towards diverse bridged N-heterocycles

A microwave-assisted diastereoselective multicomponent reaction to access dibenzo[c,e]azepinones: synthesis and biological evaluation.

A new colorimetric test for solid-phase amines and thiols

A novel and versatile entry to asymmetrically substituted pyrazines

A walk around the A3-coupling

Access to Polycyclic Azepino[5,4,3-cd]indoles via a Gold-Catalyzed Post-Ugi Dearomatization Cascade

Aldehydes: magnificent acyl equivalents for direct acylation

An antibiofilm coating of 5-aryl-2-aminoimidazole covalently attached to a titanium surface

Anti-inflammatory and antioxidant properties of Piper species: a perspective from screening to molecular mechanisms.

C-N bond forming cross-coupling reactions: an overview

Chemo- and Regioselective Catalyst-Controlled Carbocyclization of Alkynyl Ketones: Rapid Synthesis of 1-Indanones and 1-Naphthols

Click chemistry under non-classical reaction conditions.

Combining the Ugi-azide multicomponent reaction and rhodium(III)-catalyzed annulation for the synthesis of tetrazole-isoquinolone/pyridone hybrids

Concise and diversity-oriented route toward polysubstituted 2-aminoimidazole alkaloids and their analogues.

CuICuII and AgIp-isocyanobenzoates as novel 1D semiconducting coordination oligomers

DBU-Catalyzed Alkyne-Imidate Cyclization toward 1-Alkoxypyrazino[1,2- a]indole Synthesis

Development of a new microwave-assisted cleavable backbone amide linker (BAL): a comparative study

Developments in direct C-H arylation of (hetero)arenes under microwave irradiation.

Diversity oriented microwave-assisted synthesis of (-)-steganacin aza-analogues.

Doebner-type pyrazolopyridine carboxylic acids in an Ugi four-component reaction

Domino Carbopalladation/C-H Functionalization Sequence: An Expedient Synthesis of Bis-Heteroaryls through Transient Alkyl/Vinyl-Palladium Species Capture

Enhancing the anti-biofilm activity of 5-aryl-2-aminoimidazoles through nature inspired dimerisation

Evaluation of the antibacterial and antibiofilm activities of novel CRAMP-vancomycin conjugates with diverse linkers.

Evaluation of the toxicity of 5-aryl-2-aminoimidazole-based biofilm inhibitors against eukaryotic cell lines, bone cells and the nematode Caenorhabditis elegans.

Facile access to functionalized spiro[indoline-3,2'-pyrrole]-2,5'-diones via post-Ugi domino Buchwald-Hartwig/Michael reaction

Facile construction of diverse polyheterocyclic scaffolds via gold-catalysed dearomative spirocyclization/1,6-addition cascade

Gold-Catalyzed Post-Ugi Ipso-Cyclization with Switchable Diastereoselectivity

Gold-catalyzed diastereoselective domino dearomatization/ipso-cyclization/aza-Michael sequence: a facile access to diverse fused azaspiro tetracyclic scaffolds.

Gold-catalyzed post-MCR transformations towards complex (poly)heterocycles

Gold-catalyzed post-Ugi alkyne hydroarylation for the synthesis of 2-quinolones

Heck-Suzuki Tandem Reaction for the Synthesis of 3-Benzazepines

High-speed microwave-promoted hetero-Diels-Alder reactions of 2(1H)-pyrazinones in ionic liquid doped solvents

Hypervalent Iodine(III)-Mediated Cascade Cyclization of Propargylguanidines and Total Syntheses of Kealiinine B and C.

Identification of small peptides inhibiting the integrase-LEDGF/p75 interaction through targeting the cellular co-factor

Inhibiting bacterial cooperation is an evolutionarily robust anti-biofilm strategy

Iron(II)-Catalyzed Heck-Type Coupling of Vinylarenes with Alkyl Iodides

Iterative Chemical Engineering of Vancomycin Leads to Novel Vancomycin Analogs With a High in Vitro Therapeutic Index.

Metal-Free Dearomatization: Direct Access to Spiroindol(en)ines in Batch and Continuous-Flow

Metal-mediated post-Ugi transformations for the construction of diverse heterocyclic scaffolds

Microwave-Assisted Copper-Catalyzed Oxidative Cyclization of Acrylamides with Non-Activated Ketones

Microwave-assisted Cu(I)-catalyzed, three-component synthesis of 2-(4-((1-phenyl-1H-1,2,3-triazol-4-yl)methoxy)phenyl)-1H-benzo[d]imidazoles

Microwave-assisted C–C bond forming cross-coupling reactions: an overview ⬇️

Microwave-assisted cycloaddition reactions

Microwave-assisted one-pot synthesis and anti-biofilm activity of 2-amino-1H-imidazole/triazole conjugates

Microwave-assisted synthesis of a novel class of imidazolylthiazolidin-4-ones and evaluation of its biological activities.

Microwave-assisted synthesis of medium-sized heterocycles

Microwave-enhanced transition metal-catalyzed decoration of 2(1H)-pyrazinone scaffolds

Modular Access to Diverse Bridged Indole Alkaloid Mimics via a Gold-Triggered Cascade Dearomative Spirocarbocyclization/[4 + 2] Cycloaddition Sequence

Modulation of the Substitution Pattern of 5-Aryl-2-Aminoimidazoles Allows Fine-Tuning of Their Antibiofilm Activity Spectrum and Toxicity.

New tricks of well-known aminoazoles in isocyanide-based multicomponent reactions and antibacterial activity of the compounds synthesized.

Novel (2-amino-4-arylimidazolyl)propanoic acids and pyrrolo[1,2-c]imidazoles via the domino reactions of 2-amino-4-arylimidazoles with carbonyl and methylene active compounds

One-pot microwave-assisted protocol for the synthesis of substituted 2-amino-1H-imidazoles ⬇️

Pd-catalyzed Csp(2) -H functionalization of heteroarenes via isocyanide insertion: concise synthesis of di-(hetero)aryl ketones and di-(hetero)aryl alkylamines

Peptide macrocyclization by transition metal catalysis

Photoredox-Catalyzed Hydrosulfonylation of Arylallenes

Polysubstituted 2-aminoimidazoles as anti-biofilm and antiproliferative agents: Discovery of potent lead.

Post-Ugi Cyclization for the Construction of Diverse Heterocyclic Compounds: Recent Updates

Post-Ugi gold-catalyzed diastereoselective domino cyclization for the synthesis of diversely substituted spiroindolines

Reactions of secondary propargylamines with heteroallenes for the synthesis of diverse heterocycles.

Recent Advances in Phthalan and Coumaran Chemistry

Recent advances in spirocyclization of indole derivatives.

Retraction of "Iron-Catalyzed Three-Component Reaction: Synthesis of Fluoroalkylated 2 H-Azirines"

Rhodium(iii)-catalyzed intramolecular annulation through C-H activation: concise synthesis of rosettacin and oxypalmatime.

Ruthenium-catalysed one-pot regio- and diastereoselective synthesis of pyrrolo[1,2-a]indoles via cascade C-H functionalization/annulation

Sequential and direct multicomponent reaction (MCR)-based dearomatization strategies

Smart Metal-Organic Framework Coatings: Triggered Antibiofilm Compound Release

Solid-phase synthesis of the 2(1H)-pyrazinone scaffold: a new approach toward diversely substituted heterocycles

Structure-activity relationship of 2-hydroxy-2-aryl-2,3-dihydro-imidazo[1,2-a]pyrimidinium salts and 2N-substituted 4(5)-aryl-2-amino-1H-imidazoles as inhibitors of biofilm formation by Salmonella Typhimurium and Pseudomonas aeruginosa.

Structure-activity relationship of 4(5)-aryl-2-amino-1H-imidazoles, N1-substituted 2-aminoimidazoles and imidazo[1,2-a]pyrimidinium salts as inhibitors of biofilm formation by Salmonella typhimurium and Pseudomonas aeruginosa.

Suzuki-Miyaura and Stille reactions as key steps in the synthesis of diversely functionalized Amaryllidaceae alkaloid analogs bearing a 5,6,7,8-tetrahydrobenzo[c,e]azocine skeleton

Switching the regioselectivity via indium(III) and gold(I) catalysis: a post-Ugi intramolecular hydroarylation to azepino- and azocino-[c,d]indolones.

Synthesis and HIV-1 RT inhibitory action of novel (4/6-substituted benzo[d]thiazol -2-yl)thiazolidin-4-ones. Divergence from the non-competitive inhibition mechanism

Synthesis and anti-inflammatory activity evaluation of novel chroman derivatives

Synthesis and anti-inflammatory activity evaluation of novel triazolyl-isatin hybrids.