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Addressing Structural Flexibility at the A-Ring on Salvinorin A: Discovery of a Potent Kappa-Opioid Agonist with Enhanced Metabolic Stability

artículo científico publicado en 2017

Assessment of rimonabant-like adverse effects of purported CB1R neutral antagonist / CB2R agonist aminoalkylindole derivatives in mice

artículo científico publicado en 2018

Azaphilones inhibit tau aggregation and dissolve tau aggregates in vitro

artículo científico publicado en 2015

Behavioral Effects and Central Nervous System Levels of the Broadly Available κ-Agonist Hallucinogen Salvinorin A Are Affected by P-Glycoprotein Modulation In Vivo

artículo científico publicado el 20 de marzo de 2012

Behavioral and Physiological Effects of a Novel Kappa-Opioid Receptor-Based DREADD in Rats

scientific article published on 28 May 2015

Behavioral evaluation of modafinil and the abuse-related effects of cocaine in rhesus monkeys

artículo científico publicado el 1 de octubre de 2010

Benzylimidazolines as h5-HT1B/1D Serotonin Receptor Ligands: A Structure−Affinity Investigation

artículo científico publicado el 18 de junio de 1998

Correction to "Structure-Activity Relationship Studies of Functionally Selective Kappa Opioid Receptor Agonists that Modulate ERK 1/2 Phosphorylation While Preserving G Protein Over βArrestin2 Signaling Bias".

artículo científico publicado en 2017

Development of functionally selective, small molecule agonists at kappa opioid receptors

artículo científico publicado en 2013

Discovery of Small-Molecule Inhibitors Targeting the E3 Ubiquitin Ligase Activity of the Herpes Simplex Virus 1 ICP0 Protein Using an In Vitro High-Throughput Screening Assay

scientific article published on 14 June 2019

Effects of mesyl salvinorin B alone and in combination with naltrexone on alcohol deprivation effect in male and female mice

artículo científico publicado en 2018

Further exploration of the structure-activity relationship of imidazoquinolines; identification of potent C7-substituted imidazoquinolines

artículo científico publicado en 2019

High‐dose fenfluramine administration decreases serotonin transporter binding, but not serotonin transporter protein levels, in rat forebrain

artículo científico publicado el 1 de diciembre de 2003

Holo Structure and Steady State Kinetics of the Thiazolinyl Imine Reductases for Siderophore Biosynthesis

artículo científico publicado en 2016

Impact of Pharmacological Manipulation of the κ-Opioid Receptor System on Self-grooming and Anhedonic-like Behaviors in Male Mice

scientific article published on 11 April 2019

Kappa Opioid Receptor Agonist Mesyl Sal B Attenuates Behavioral Sensitization to Cocaine with Fewer Aversive Side-Effects than Salvinorin A in Rodents

artículo científico publicado en 2018

Kappa opioid agonists reduce oxycodone self-administration in male rhesus monkeys

artículo científico publicado en 2020

Modular Approach to pseudo-Neoclerodanes as Designer κ-Opioid Ligands.

artículo científico publicado en 2017

N-acetyl-S-(N,N-diethylcarbamoyl) cysteine in rat nucleus accumbens, medial prefrontal cortex, and in rat and human plasma after disulfiram administration

artículo científico publicado en 2015

Nalfurafine promotes myelination <scp><i>in vitro</i></scp> and facilitates recovery from cuprizone + rapamycin‐induced demyelination in mice

NeuroChat with Professor Thomas E. Prisinzaro

artículo científico publicado en 2020

Neuropharmacology of the Naturally Occurring κ-Opioid Hallucinogen Salvinorin A

artículo científico publicado el 28 de marzo de 2011

Novel psychotherapeutics - a cautiously optimistic focus on Hallucinogens.

artículo científico publicado en 2017

Opioid Receptor Probes Derived from Cycloaddition of the Hallucinogen Natural Product Salvinorin A

artículo científico publicado el 21 de febrero de 2011

Permeation and metabolism of cocaine in the nasal mucosa

artículo científico publicado el 18 de febrero de 2012

Pharmacology and anti-addiction effects of the novel κ opioid receptor agonist Mesyl Sal B, a potent and long-acting analogue of salvinorin A

artículo científico publicado en 2014

Preclinical Testing of Nalfurafine as an Opioid-sparing Adjuvant that Potentiates Analgesia by the Mu Opioid Receptor-targeting Agonist Morphine

scientific article published on 06 September 2019

R-modafinil (armodafinil): a unique dopamine uptake inhibitor and potential medication for psychostimulant abuse

artículo científico publicado en 2012

Reinstatement of methamphetamine seeking in male and female rats treated with modafinil and allopregnanolone

artículo científico publicado el 5 de agosto de 2011

Role of Ventral Subiculum in Context-Induced Relapse to Alcohol Seeking after Punishment-Imposed Abstinence

artículo científico publicado en 2016

Scalable Regioselective and Stereoselective Synthesis of Functionalized (E)-4-Iodobut-3-en-1-ols: Gram-Scale Total Synthesis of Fungal Decanolides and Derivatives.

artículo científico publicado en 2017

Semisynthesis and Kappa-Opioid Receptor Activity of Derivatives of Columbin, a Furanolactone Diterpene.

artículo científico publicado en 2017

Semisynthetic neoclerodanes as kappa opioid receptor probes

artículo científico publicado el 1 de mayo de 2012

Strategies for developing kappa opioid receptor agonists for the treatment of pain with fewer side-effects

scientific article published on 10 September 2020

Structure-Activity Relationships at the Monoamine Transporters for a Novel Series of Modafinil (2-[(diphenylmethyl)sulfinyl]acetamide) Analogues

artículo científico publicado en 2010

Stuffed Methyltransferase Catalyzes the Penultimate Step of Pyochelin Biosynthesis

artículo científico publicado en 2018

Synergistic blockade of alcohol escalation drinking in mice by a combination of novel kappa opioid receptor agonist Mesyl Salvinorin B and naltrexone

artículo científico publicado en 2017

Synthesis and Opioid Activity of Tyr1 -ψ[(Z)CF=CH]-Gly2 and Tyr1 -ψ[(S)/(R)-CF3 CH-NH]-Gly2 Leu-enkephalin Fluorinated Peptidomimetics

artículo científico publicado en 2017

Synthesis and κ-opioid receptor activity of furan-substituted salvinorin A analogues

artículo científico publicado en 2014

Synthetic Studies of Neoclerodane Diterpenes from Salvia divinorum: Identification of a Potent and Centrally Acting μ Opioid Analgesic with Reduced Abuse Liability.

artículo científico publicado en 2016

Synthetic studies on neoclerodane diterpenes from Salvia splendens: oxidative modifications of ring A

artículo científico publicado el 21 de febrero de 2009

The Kappa Opioid Receptor Agonist 16-Bromo Salvinorin A Has Anti-Cocaine Effects without Significant Effects on Locomotion, Food Reward, Learning and Memory, or Anxiety and Depressive-like Behaviors

The analgesic and anti-inflammatory effects of Salvinorin A analogue β-tetrahydropyran Salvinorin B in mice.

artículo científico publicado en 2017

The unique psychostimulant profile of (±)-modafinil: investigation of behavioral and neurochemical effects in mice

artículo científico publicado en 2016

Time course of pharmacokinetic and hormonal effects of inhaled high-dose salvinorin A in humans

artículo científico publicado en 2016

Utilizing Nature as a Source of New Probes for Opioid Pharmacology

artículo científico publicado el 1 de mayo de 2009