Lista de obras -

'Atypical Ugi' tetrazoles

artículo científico publicado en 2020

2-Aminoimidazole-based antagonists of the 5-HT6 receptor - A new concept in aminergic GPCR ligand design

artículo científico publicado en 2019

A Simple Synthesis of New 2-Thioxoimidazolidine-4,5-dicarboxylates from Vicinal Diisothiocyanatocarboxylates

artículo científico publicado en 2008

A triclinic crystal form of Escherichia coli 4-diphosphocytidyl-2C-methyl-D-erythritol kinase and reassessment of the quaternary structure

artículo científico publicado en 2010

Acoustic Droplet Ejection Enabled Automated Reaction Scouting

artículo científico publicado en 2019

Ammonia-Promoted One-Pot Tetrazolopiperidinone Synthesis by Ugi Reaction

artículo científico publicado en 2017

An Approach to 2,3-Diaminosuccinic Acid Derivatives—Synthesis of 2-Thioxo-1,3-Imidazolidines by a Mannich Reaction

artículo científico publicado en 2012

Application of 2,4,6-trioxo-pyrimidin-5-ylidene alditols in the synthesis of pyrano[2,3-d]pyrimidines containing a sugar moiety by hetero-Diels–Alder reactions and by conjugate Michael addition–cyclizations

artículo científico publicado en 2013

Application of dimedone enamines as dienophiles: stereoselective synthesis of amino enols of fused uracils containing a sugar moiety by hetero-Diels–Alder reactions of barbituric acid 5-ylidene alditols with dimedone enamines

artículo científico publicado en 2015

Artificial Macrocycles by Ugi Reaction and Passerini Ring Closure.

artículo científico publicado en 2016

Arylpiperazinylalkyl derivatives of 8-amino-1,3-dimethylpurine-2,6-dione as novel multitarget 5-HT/D receptor agents with potential antipsychotic activity

artículo científico publicado en 2015

Bismuth triiodide complexes: structure, spectroscopy, electronic properties, and memristive properties

artículo científico publicado en 2020

Bitter sweeteners: tetrazole derivatives of arylsulfonylalcanoids--synthesis, structure and comparative study.

artículo científico publicado en 2008

Cerium(IV) based oxidative free radical cyclization of active methylene compounds with some cyclic alkenes: A useful annulation method for terpene functionalization

artículo científico publicado en 2019

Cleavable β-Cyanoethyl Isocyanide in the Ugi Tetrazole Reaction

artículo científico publicado en 2016

Concise Synthesis of Tetrazole Macrocycle

artículo científico publicado en 2017

Copper-Catalyzed Modular Assembly of Polyheterocycles

artículo científico publicado en 2020

Crystal structures of IspF from Plasmodium falciparum and Burkholderia cenocepacia: comparisons inform antimicrobial drug target assessment

artículo científico publicado en 2014

Cysteine Isocyanide in Multicomponent Reaction: Synthesis of Peptido-Mimetic 1,3-Azoles.

artículo científico publicado en 2017

De Novo Assembly of Highly Substituted Morpholines and Piperazines

artículo científico publicado en 2017

Diastereoselective One Pot Five-Component Reaction toward 4-(Tetrazole)-1,3-Oxazinanes.

artículo científico publicado en 2017

Dimethyl dl-2,3-dibenzyl-2,3-diisothio-cyanatosuccinate.

artículo científico publicado en 2012

Discovery of chromenes as inhibitors of macrophage migration inhibitory factor.

artículo científico publicado en 2017

Diverse Isoquinoline Scaffolds by Ugi/Pomeranz-Fritsch and Ugi/Schlittler-Müller Reactions

scientific article published on 29 April 2019

Electrostatic potential and non-covalent interactions analysis for the design of selective 5-HT7 ligands

artículo científico publicado en 2019

Flat or angular? The impact of the nitrogen atom hybridization on the docking results for arylpiperazine derivatives as an example

artículo científico publicado en 2019

Fourfold symmetric MCR's via the tetraisocyanide 1,3-diisocyano-2,2-bis(isocyanomethyl)propane

artículo científico publicado en 2020

Glycoconjugates via phosphorus ylides

scientific article published on 03 May 2019

Hitting on the move: Targeting intrinsically disordered protein states of the MDM2-p53 interaction

scientific article published on 06 August 2019

How can fluorine directly and indirectly affect the hydrogen bonding in molecular systems? – A case study for monofluoroanilines

artículo científico publicado en 2021

Hydrazine in the Ugi Tetrazole Reaction

artículo científico publicado en 2016

Influence of the position of the methyl substituent and N-oxide formation on the geometry and intermolecular interactions of 1-(phenoxyethyl)piperidin-4-ol derivatives

scientific article published on 01 January 2020

Isocyanide-Based Multicomponent Reactions of Free Phenylboronic Acids

artículo científico publicado en 2019

Library-to-Library Synthesis of Highly Substituted α-Aminomethyl Tetrazoles via Ugi Reaction.

artículo científico publicado en 2017

Multicomponent Reaction Based Synthesis of 1-Tetrazolylimidazo[1,5- a]pyridines

artículo científico publicado en 2018

Multifunctional arylsulfonamide derivatives with 5-HT/5-HT receptor antagonistic activity: a structural study

artículo científico publicado en 2018

New 7-arylpiperazinylalkyl-8-morpholin-4-yl-purine-2,6-dione derivatives with anxiolytic activity – Synthesis, crystal structure and structure–activity study

artículo científico publicado en 2014

Ratiometric fluorescent Zn 2+ and In 3+ receptors of fused pyrazine with an aminopropanol chain in acetonitrile

artículo científico publicado en 2014

Rational design of 5-HT 6 R ligands using a bioisosteric strategy: synthesis, biological evaluation and molecular modelling

artículo científico publicado en 2015

Room temperature bistability in an Ni-Fe chain: electron transfer controlled by temperature, pressure, light and humidity

artículo científico publicado en 2020

Scaffolding-induced property modulation of chemical space

scientific article published on 22 May 2020

Sequential Multicomponent Synthesis of 2-(Imidazo[1,5-α]pyridin-1-yl)-1,3,4-Oxadiazoles

artículo científico publicado en 2019

Structure and Reactivity of Glycosyl Isocyanides

artículo científico publicado en 2019

Succinonitrile Activated by Thiating Agents as Precursor of Bis-cyclic Amidines, Tectons for Molecular Engineering

artículo científico publicado en 2007

Synthesis and reactivity of bis(cycloamidinium-2-yl)alkane bromide tribromides, brominating agents and tectons for molecular engineering

artículo científico publicado en 2008

Synthesis of highly substituted imidazole Uracil containing molecules via Ugi-4CR and Passerini-3CR.

artículo científico publicado en 2018

The effect of the intramolecular C-H⋯O interactions on the conformational preferences of bis-arylsulfones - 5-HT receptor antagonists and beyond

artículo científico publicado en 2018

Titanium(IV) Enolates of 2-Nitrocarboxylic Esters and Their Oxidative Chlorination. A Convenient Route to α-Chloro-α-nitrocarboxylates

artículo científico publicado en 2012

Triiodide Organic Salts: Photoelectrochemistry at the Border between Insulators and Semiconductors

artículo científico publicado en 2018

Two-Step Macrocycle Synthesis by Classical Ugi Reaction.

artículo científico publicado en 2018

Two-Step Synthesis of Complex Artificial Macrocyclic Compounds

artículo científico publicado en 2017

Ugi Multicomponent Reaction Based Synthesis of Medium-Sized Rings

artículo científico publicado en 2017

Versatile Multicomponent Reaction Macrocycle Synthesis Using α-Isocyano-ω-carboxylic Acids

artículo científico publicado en 2015

Versatile Protecting-Group Free Tetrazolomethane Amine Synthesis by Ugi Reaction

artículo científico publicado en 2016

α-Amino Acid-Isosteric α-Amino Tetrazoles.

artículo científico

Lista de obras de

'Atypical Ugi' tetrazoles

2-Aminoimidazole-based antagonists of the 5-HT6 receptor - A new concept in aminergic GPCR ligand design

A Simple Synthesis of New 2-Thioxoimidazolidine-4,5-dicarboxylates from Vicinal Diisothiocyanatocarboxylates

A triclinic crystal form of Escherichia coli 4-diphosphocytidyl-2C-methyl-D-erythritol kinase and reassessment of the quaternary structure

Acoustic Droplet Ejection Enabled Automated Reaction Scouting

Ammonia-Promoted One-Pot Tetrazolopiperidinone Synthesis by Ugi Reaction

An Approach to 2,3-Diaminosuccinic Acid Derivatives—Synthesis of 2-Thioxo-1,3-Imidazolidines by a Mannich Reaction

Application of 2,4,6-trioxo-pyrimidin-5-ylidene alditols in the synthesis of pyrano[2,3-d]pyrimidines containing a sugar moiety by hetero-Diels–Alder reactions and by conjugate Michael addition–cyclizations

Application of dimedone enamines as dienophiles: stereoselective synthesis of amino enols of fused uracils containing a sugar moiety by hetero-Diels–Alder reactions of barbituric acid 5-ylidene alditols with dimedone enamines

Artificial Macrocycles by Ugi Reaction and Passerini Ring Closure.

Arylpiperazinylalkyl derivatives of 8-amino-1,3-dimethylpurine-2,6-dione as novel multitarget 5-HT/D receptor agents with potential antipsychotic activity

Bismuth triiodide complexes: structure, spectroscopy, electronic properties, and memristive properties

Bitter sweeteners: tetrazole derivatives of arylsulfonylalcanoids--synthesis, structure and comparative study.

Cerium(IV) based oxidative free radical cyclization of active methylene compounds with some cyclic alkenes: A useful annulation method for terpene functionalization

Cleavable β-Cyanoethyl Isocyanide in the Ugi Tetrazole Reaction

Concise Synthesis of Tetrazole Macrocycle

Copper-Catalyzed Modular Assembly of Polyheterocycles

Crystal structures of IspF from Plasmodium falciparum and Burkholderia cenocepacia: comparisons inform antimicrobial drug target assessment

Cysteine Isocyanide in Multicomponent Reaction: Synthesis of Peptido-Mimetic 1,3-Azoles.

De Novo Assembly of Highly Substituted Morpholines and Piperazines

Diastereoselective One Pot Five-Component Reaction toward 4-(Tetrazole)-1,3-Oxazinanes.

Dimethyl dl-2,3-dibenzyl-2,3-diisothio-cyanatosuccinate.

Discovery of chromenes as inhibitors of macrophage migration inhibitory factor.

Diverse Isoquinoline Scaffolds by Ugi/Pomeranz-Fritsch and Ugi/Schlittler-Müller Reactions

Electrostatic potential and non-covalent interactions analysis for the design of selective 5-HT7 ligands

Flat or angular? The impact of the nitrogen atom hybridization on the docking results for arylpiperazine derivatives as an example

Fourfold symmetric MCR's via the tetraisocyanide 1,3-diisocyano-2,2-bis(isocyanomethyl)propane

Glycoconjugates via phosphorus ylides

Hitting on the move: Targeting intrinsically disordered protein states of the MDM2-p53 interaction

How can fluorine directly and indirectly affect the hydrogen bonding in molecular systems? – A case study for monofluoroanilines

Hydrazine in the Ugi Tetrazole Reaction

Influence of the position of the methyl substituent and N-oxide formation on the geometry and intermolecular interactions of 1-(phenoxyethyl)piperidin-4-ol derivatives

Isocyanide-Based Multicomponent Reactions of Free Phenylboronic Acids

Library-to-Library Synthesis of Highly Substituted α-Aminomethyl Tetrazoles via Ugi Reaction.

Multicomponent Reaction Based Synthesis of 1-Tetrazolylimidazo[1,5- a]pyridines

Multifunctional arylsulfonamide derivatives with 5-HT/5-HT receptor antagonistic activity: a structural study

New 7-arylpiperazinylalkyl-8-morpholin-4-yl-purine-2,6-dione derivatives with anxiolytic activity – Synthesis, crystal structure and structure–activity study

Ratiometric fluorescent Zn 2+ and In 3+ receptors of fused pyrazine with an aminopropanol chain in acetonitrile

Rational design of 5-HT 6 R ligands using a bioisosteric strategy: synthesis, biological evaluation and molecular modelling

Room temperature bistability in an Ni-Fe chain: electron transfer controlled by temperature, pressure, light and humidity

Scaffolding-induced property modulation of chemical space

Sequential Multicomponent Synthesis of 2-(Imidazo[1,5-α]pyridin-1-yl)-1,3,4-Oxadiazoles

Structure and Reactivity of Glycosyl Isocyanides

Succinonitrile Activated by Thiating Agents as Precursor of Bis-cyclic Amidines, Tectons for Molecular Engineering

Synthesis and reactivity of bis(cycloamidinium-2-yl)alkane bromide tribromides, brominating agents and tectons for molecular engineering

Synthesis of highly substituted imidazole Uracil containing molecules via Ugi-4CR and Passerini-3CR.

The effect of the intramolecular C-H⋯O interactions on the conformational preferences of bis-arylsulfones - 5-HT receptor antagonists and beyond

Titanium(IV) Enolates of 2-Nitrocarboxylic Esters and Their Oxidative Chlorination. A Convenient Route to α-Chloro-α-nitrocarboxylates

Triiodide Organic Salts: Photoelectrochemistry at the Border between Insulators and Semiconductors

Two-Step Macrocycle Synthesis by Classical Ugi Reaction.

Two-Step Synthesis of Complex Artificial Macrocyclic Compounds

Ugi Multicomponent Reaction Based Synthesis of Medium-Sized Rings

Versatile Multicomponent Reaction Macrocycle Synthesis Using α-Isocyano-ω-carboxylic Acids

Versatile Protecting-Group Free Tetrazolomethane Amine Synthesis by Ugi Reaction

α-Amino Acid-Isosteric α-Amino Tetrazoles.