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A hybrid indoloquinolizidine peptide as allosteric modulator of dopamine D1 receptors

artículo científico publicado en 2009

A2A adenosine receptor ligand binding and signalling is allosterically modulated by adenosine deaminase

artículo científico publicado en 2011

Adenosine/dopamine receptor-receptor interactions in the central nervous system

scholarly article by Rafael Franco et al published January 2001 in Drug Development Research

Basic concepts in G-protein-coupled receptor homo- and heterodimerization.

artículo científico publicado en 2007

Cannabinoid receptors CB1 and CB2 form functional heteromers in brain

artículo científico publicado en 2012

Circadian-related heteromerization of adrenergic and dopamine D₄ receptors modulates melatonin synthesis and release in the pineal gland

artículo científico publicado en 2012

Coaggregation, cointernalization, and codesensitization of adenosine A2A receptors and dopamine D2 receptors

artículo científico publicado en 2002

Cocaine inhibits dopamine D2 receptor signaling via sigma-1-D2 receptor heteromers

artículo científico publicado en 2013

Detection of heteromerization of more than two proteins by sequential BRET-FRET.

artículo científico publicado en 2008

Detection of heteromers formed by cannabinoid CB1, dopamine D2, and adenosine A2A G-protein-coupled receptors by combining bimolecular fluorescence complementation and bioluminescence energy transfer.

artículo científico publicado en 2008

Detection of receptor heteromers involving dopamine receptors by the sequential BRET-FRET technology

artículo científico publicado en 2013

Dimer-based model for heptaspanning membrane receptors

scientific article published on 01 July 2005

Direct involvement of sigma-1 receptors in the dopamine D1 receptor-mediated effects of cocaine

artículo científico publicado en 2010

Dopamine D1-histamine H3 receptor heteromers provide a selective link to MAPK signaling in GABAergic neurons of the direct striatal pathway

artículo científico publicado en 2010

Functional μ-Opioid-Galanin Receptor Heteromers in the Ventral Tegmental Area.

artículo científico publicado en 2016

GPCR homomers and heteromers: a better choice as targets for drug development than GPCR monomers?

artículo científico publicado en 2009

Gi protein coupling to adenosine A1-A2A receptor heteromers in human brain caudate nucleus.

artículo científico publicado en 2010

Heptaspanning membrane receptors and cytoskeletal/scaffolding proteins: focus on adenosine, dopamine, and metabotropic glutamate receptor function

artículo científico publicado en 2005

Homodimerization of adenosine A2A receptors: qualitative and quantitative assessment by fluorescence and bioluminescence energy transfer

artículo científico publicado en 2004

Human adenosine deaminase as an allosteric modulator of human A(1) adenosine receptor: abolishment of negative cooperativity for [H](R)-pia binding to the caudate nucleus

artículo científico publicado en 2008

Interactions between calmodulin, adenosine A2A, and dopamine D2 receptors

artículo científico publicado en 2009

Interactions between intracellular domains as key determinants of the quaternary structure and function of receptor heteromers

artículo científico publicado en 2010

Involvement of caveolin in ligand-induced recruitment and internalization of A(1) adenosine receptor and adenosine deaminase in an epithelial cell line

artículo científico publicado en 2001

L-DOPA disrupts adenosine A(2A)-cannabinoid CB(1)-dopamine D(2) receptor heteromer cross-talk in the striatum of hemiparkinsonian rats: biochemical and behavioral studies

artículo científico publicado en 2014

L-DOPA-treatment in primates disrupts the expression of A(2A) adenosine-CB(1) cannabinoid-D(2) dopamine receptor heteromers in the caudate nucleus

artículo científico publicado en 2013

Ligand-induced caveolae-mediated internalization of A1 adenosine receptors: morphological evidence of endosomal sorting and receptor recycling

artículo científico publicado en 2003

Marked changes in signal transduction upon heteromerization of dopamine D1 and histamine H3 receptors

artículo científico publicado en 2009

Metabotropic glutamate type 1alpha receptor localizes in low-density caveolin-rich plasma membrane fractions

artículo científico publicado en 2003

Molecular mechanisms involved in the adenosine A and A receptor-induced neuronal differentiation in neuroblastoma cells and striatal primary cultures

artículo científico publicado en 2005

Mutual regulation between metabotropic glutamate type 1alpha receptor and caveolin proteins: from traffick to constitutive activity

artículo científico publicado en 2004

Novel pharmacological targets based on receptor heteromers

artículo científico publicado en 2008

Old and new ways to calculate the affinity of agonists and antagonists interacting with G-protein-coupled monomeric and dimeric receptors: the receptor-dimer cooperativity index.

artículo científico publicado en 2007

Orexin-corticotropin-releasing factor receptor heteromers in the ventral tegmental area as targets for cocaine

artículo científico publicado en 2015

Partners for adenosine A1 receptors

artículo científico publicado en 2005

Presynaptic control of striatal glutamatergic neurotransmission by adenosine A1-A2A receptor heteromers

artículo científico publicado en 2006

Regulation of epithelial and lymphocyte cell adhesion by adenosine deaminase-CD26 interaction

artículo científico publicado en 2002

Regulation of heptaspanning-membrane-receptor function by dimerization and clustering

artículo científico publicado en 2003

The adenosine A2A receptor interacts with the actin-binding protein alpha-actinin

scientific journal article

The catalytic site structural gate of adenosine deaminase allosterically modulates ligand binding to adenosine receptors

artículo científico publicado en 2012

The neuronal Ca(2+) -binding protein 2 (NECAB2) interacts with the adenosine A(2A) receptor and modulates the cell surface expression and function of the receptor

artículo científico publicado en 2007

The two-state dimer receptor model: a general model for receptor dimers

artículo científico publicado en 2006

Up-regulation of the Kv3.4 potassium channel subunit in early stages of Alzheimer's disease.

artículo científico publicado en 2004

Useful pharmacological parameters for G-protein-coupled receptor homodimers obtained from competition experiments. Agonist-antagonist binding modulation.

artículo científico publicado en 2009