Lista de obras -

(18)F- and (68)Ga-Labeled Neurotensin Peptides for PET Imaging of Neurotensin Receptor 1.

artículo científico publicado en 2016

(18)F-glyco-RGD peptides for PET imaging of integrin expression: efficient radiosynthesis by click chemistry and modulation of biodistribution by glycosylation

artículo científico publicado en 2013

18F-Labeled FAUC 346 and BP 897 derivatives as subtype-selective potential PET radioligands for the dopamine D3 receptor.

artículo científico publicado en 2008

18F-labelled triazolyl-linked argininamides targeting the neuropeptide Y Y1R for PET imaging of mammary carcinoma

artículo científico publicado en 2019

3,4,6-Tri-O-acetyl-2-deoxy-2-[18F]fluoroglucopyranosyl Phenylthiosulfonate: A Thiol-Reactive Agent for the Chemoselective18F-Glycosylation of Peptides

scientific article published on 01 January 2007

99mTc-MIP-1404 SPECT/CT for Assessment of Whole-Body Tumor Burden and Treatment Response in Patients With Biochemical Recurrence of Prostate Cancer

scientific article published on 17 June 2020

99mTc-MIP-1404 SPECT/CT for Patients With Metastatic Prostate Cancer: Interobserver and Intraobserver Variability in Treatment-Related Longitudinal Tracer Uptake Assessments of Prostate-Specific Membrane Antigen-Positive Lesions

artículo científico publicado en 2020

A dopaminergic mechanism of antipsychotic drug efficacy, failure, and failure reversal: the role of the dopamine transporter

artículo científico publicado en 2018

A series of 18F-labelled pyridinylphenyl amides as subtype-selective radioligands for the dopamine D3 receptor

artículo científico publicado en 2010

A series of 2-O-trifluoromethylsulfonyl-D-mannopyranosides as precursors for concomitant 18F-labeling and glycosylation by click chemistry

artículo científico publicado en 2009

Assessment of Treatment Response by 99mTc-MIP-1404 SPECT/CT: A Pilot Study in Patients With Metastatic Prostate Cancer

artículo científico publicado en 2018

Biodistribution studies of two 18F-labeled pyridinylphenyl amides as subtype selective radioligands for the dopamine D3 receptor

artículo científico publicado en 2013

Characterization of 18F-FDG uptake in human endothelial cells in vitro

artículo científico publicado en 2004

Characterization of uptake of 3-[(131)I]iodo-alpha-methyl-L-tyrosine in human monocyte-macrophages

artículo científico publicado en 2004

Click chemistry based synthesis of dopamine D4 selective receptor ligands for the selection of potential PET tracers

artículo científico publicado en 2013

Detection of monoamine oxidase a in brain of living rats with [18F]fluoroethyl-harmol PET.

artículo científico publicado en 2014

Development of 18F-Fluoroglycosylated PSMA-Ligands with Improved Renal Clearance Behavior

artículo científico publicado en 2020

Development of molecular tools based on the dopamine D3 receptor ligand FAUC 329 showing inhibiting effects on drug and food maintained behavior

artículo científico publicado en 2017

Discovery of a dopamine D4 selective PET ligand candidate taking advantage of a click chemistry based REM linker

artículo científico publicado en 2008

Disentangling inflammatory from fibrotic disease activity by fibroblast activation protein imaging

artículo científico publicado en 2020

Effects of Recombinant Human Thyroid-Stimulating Hormone Superagonists on Thyroidal Uptake of18F-Fluorodeoxyglucose and Radioiodide ⬇️

artículo científico publicado el 13 de mayo de 2011

Estimation of [177Lu]PSMA-617 tumor uptake based on voxel-wise 3D Monte Carlo tumor dosimetry in patients with metastasized castration resistant prostate cancer

artículo científico publicado en 2020

Evaluation of18F-Labeled Benzodioxine Piperazine-Based Dopamine D4Receptor Ligands: Lipophilicity as a Determinate of Nonspecific Binding

scientific article published on 23 November 2011

Fast and efficient (18) F-labeling by [(18) f]fluorophenylazocarboxylic esters

artículo científico publicado en 2013

First Experience With SPECT/CT Using a 99mTc-Labeled Inhibitor for Prostate-Specific Membrane Antigen in Patients With Biochemical Recurrence of Prostate Cancer

artículo científico publicado en 2017

H-CRRETAWAC-OH, a lead structure for the development of radiotracer targeting integrin α5β1?

artículo científico publicado en 2014

Identification of Boronic Acid Derivatives as an Active Form of N-Alkylaminoferrocene-Based Anticancer Prodrugs and Their Radiolabeling with 18F

artículo científico publicado en 2019

Improved radiosynthesis and preliminary in vivo evaluation of a (18)F-labeled glycopeptide-peptoid hybrid for PET imaging of neurotensin receptor 2.

artículo científico publicado en 2015

In Vitro and In Vivo Characterization of Selected Fluorine-18 Labeled Radioligands for PET Imaging of the Dopamine D3 Receptor.

artículo científico publicado en 2016

In vitro and initial in vivo evaluation of (68)Ga-labeled transferrin receptor (TfR) binding peptides as potential carriers for enhanced drug transport into TfR expressing cells

artículo científico publicado en 2011

In vitro characterization of the thyroidal uptake of O-(2-[(18)F]fluoroethyl)-L-tyrosine

artículo científico publicado en 2007

In vitro studies on the signal transduction of thyroidal uptake of 18F-FDG and 131I-Iodide.

artículo científico publicado en 2006

In vivo monitoring of the antiangiogenic effect of neurotensin receptor-mediated radiotherapy by small-animal positron emission tomography: a pilot study

artículo científico publicado en 2014

Induction and repair of DNA double-strand breaks in blood lymphocytes of patients undergoing 18F-FDG PET/CT examinations ⬇️

artículo científico publicado el 2 de agosto de 2012

Labeling and glycosylation of peptides using click chemistry: a general approach to (18)F-glycopeptides as effective imaging probes for positron emission tomography

artículo científico publicado en 2010

Microwave-Assisted Rapid One-Pot Synthesis of Fused and Non-Fused Indoles and 5-[18 F]Fluoroindoles from Phenylazocarboxylates

artículo científico publicado en 2017

Multimerization of cRGD Peptides by Click Chemistry: Synthetic Strategies, Chemical Limitations, and Influence on Biological Properties ⬇️

artículo científico publicado el 18 de octubre de 2010

Multimodal Bone Metastasis-associated Epidermal Growth Factor Receptor Imaging in an Orthotopic Rat Model

artículo científico publicado en 2021

Non-Invasive Characterization of Experimental Bone Metastasis in Obesity Using Multiparametric MRI and PET/CT

artículo científico publicado en 2022

Optimization and synthesis of an18F-labeled dopamine D3receptor ligand using [18F]fluorophenylazocarboxylictert-butylester

artículo científico publicado en 2015

PET radiopharmaceuticals for imaging integrin expression: tracers in clinical studies and recent developments.

artículo científico

Perturbed Development of Striatal Dopamine Transporters in Fatty Versus Lean Zucker Rats: a Follow-up Small Animal PET Study

artículo científico publicado en 2014

Pharmacological characterization of low-to-moderate affinity opioid receptor agonists and brain imaging with 18F-labeled derivatives in rats

artículo científico publicado en 2020

Prediction of early metastatic disease in experimental breast cancer bone metastasis by combining PET/CT and MRI parameters to a Model-Averaged Neural Network

scientific article published on 13 November 2018

Prototypic 18F-Labeled Argininamide-Type Neuropeptide Y Y1R Antagonists as Tracers for PET Imaging of Mammary Carcinoma.

artículo científico publicado en 2017

Radioligands for the dopamine receptor subtypes

artículo científico

Radiopharmaceuticals for imaging and endoradiotherapy of neurotensin receptor-positive tumors.

artículo científico publicado en 2017

Radiosynthesis and Preclinical Evaluation of 18F-Fluoroglycosylated Octreotate for Somatostatin Receptor Imaging.

artículo científico publicado en 2016

Radiosynthesis and evaluation of 18F-labeled dopamine D4-receptor ligands

scientific article published on 16 July 2020

Radiosynthesis and validation of ¹⁸F-FP-CMT, a phenyltropane with superior properties for imaging the dopamine transporter in living brain.

artículo científico publicado en 2014

Radiosynthesis of an F-fluoroglycosylated aminoferrocene for in-vivo imaging of reactive oxygen species activity by PET

article

Recent trends in pharmaceutical radiochemistry for molecular PET imaging

artículo científico publicado en 2014

Regulation of uptake of 18F-FDG by a follicular human thyroid cancer cell line with mutation-activated K-ras

artículo científico publicado en 2009

Specific binding of [(18)F]fluoroethyl-harmol to monoamine oxidase A in rat brain cryostat sections, and compartmental analysis of binding in living brain

artículo científico publicado en 2015

Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands

artículo científico publicado en 2007

Sweetening pharmaceutical radiochemistry by (18)f-fluoroglycosylation: a short review.

artículo científico

Syntheses and radiofluorination of two derivatives of 5-cyano-indole as selective ligands for the dopamine subtype-4 receptor

Syntheses, receptor bindings, in vitro and in vivo stabilities and biodistributions of DOTA-neurotensin(8-13) derivatives containing β-amino acid residues - a lesson about the importance of animal experiments

artículo científico publicado en 2013

Synthesis and evaluation of 18F-labeled dopamine D3 receptor ligands as potential PET imaging agents

artículo científico publicado en 2005

Synthesis and evaluation of a (18)F-labeled diarylpyrazole glycoconjugate for the imaging of NTS1-positive tumors

artículo científico publicado en 2013

Synthesis and evaluation of fluoro substituted pyridinylcarboxamides and their phenylazo analogues for potential dopamine D3 receptor PET imaging

artículo científico publicado en 2014

Synthesis and in vitro and in vivo evaluation of an (18)F-labeled neuropeptide Y analogue for imaging of breast cancer by PET.

artículo científico publicado en 2015

Synthesis and in vivo evaluation of an (18)F-labeled glycoconjugate of PD156707 for imaging ETA receptor expression in thyroid carcinoma by positron emission tomography

artículo científico publicado en 2013

Synthesis and radioiodination of selective ligands for the dopamine D3 receptor subtype

artículo científico publicado en 2004

Synthesis of a (68)ga-labeled peptoid-Peptide hybrid for imaging of neurotensin receptor expression in vivo

artículo científico publicado en 2010

Synthesis, biological evaluation and radiosynthesis of buprenorphine-derived phenylazocarboxamides as novel μ-opioid receptor ligands

scientific article published on 06 May 2020

Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET.

artículo científico publicado en 2008

Targeting Fibroblast Activation Protein: Radiosynthesis and Preclinical Evaluation of an 18F-labeled FAP Inhibitor

scientific article published on 24 April 2020

Theranostic Value of Multimers: Lessons Learned from Trimerization of Neurotensin Receptor Ligands and Other Targeting Vectors

artículo científico publicado en 2017

[(68)Ga]Ga-DO(2)A-(OBu-l-tyr)(2): synthesis, (68)Ga-radiolabeling and in vitro studies of a novel (68)Ga-DO(2)A-tyrosine conjugate as potential tumor tracer for PET.

artículo científico publicado en 2009

[18F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor

artículo científico publicado en 2017

Lista de obras de

(18)F- and (68)Ga-Labeled Neurotensin Peptides for PET Imaging of Neurotensin Receptor 1.

(18)F-glyco-RGD peptides for PET imaging of integrin expression: efficient radiosynthesis by click chemistry and modulation of biodistribution by glycosylation

18F-Labeled FAUC 346 and BP 897 derivatives as subtype-selective potential PET radioligands for the dopamine D3 receptor.

18F-labelled triazolyl-linked argininamides targeting the neuropeptide Y Y1R for PET imaging of mammary carcinoma

3,4,6-Tri-O-acetyl-2-deoxy-2-[18F]fluoroglucopyranosyl Phenylthiosulfonate: A Thiol-Reactive Agent for the Chemoselective18F-Glycosylation of Peptides

99mTc-MIP-1404 SPECT/CT for Assessment of Whole-Body Tumor Burden and Treatment Response in Patients With Biochemical Recurrence of Prostate Cancer

99mTc-MIP-1404 SPECT/CT for Patients With Metastatic Prostate Cancer: Interobserver and Intraobserver Variability in Treatment-Related Longitudinal Tracer Uptake Assessments of Prostate-Specific Membrane Antigen-Positive Lesions

A dopaminergic mechanism of antipsychotic drug efficacy, failure, and failure reversal: the role of the dopamine transporter

A series of 18F-labelled pyridinylphenyl amides as subtype-selective radioligands for the dopamine D3 receptor

A series of 2-O-trifluoromethylsulfonyl-D-mannopyranosides as precursors for concomitant 18F-labeling and glycosylation by click chemistry

Assessment of Treatment Response by 99mTc-MIP-1404 SPECT/CT: A Pilot Study in Patients With Metastatic Prostate Cancer

Biodistribution studies of two 18F-labeled pyridinylphenyl amides as subtype selective radioligands for the dopamine D3 receptor

Characterization of 18F-FDG uptake in human endothelial cells in vitro

Characterization of uptake of 3-[(131)I]iodo-alpha-methyl-L-tyrosine in human monocyte-macrophages

Click chemistry based synthesis of dopamine D4 selective receptor ligands for the selection of potential PET tracers

Detection of monoamine oxidase a in brain of living rats with [18F]fluoroethyl-harmol PET.

Development of 18F-Fluoroglycosylated PSMA-Ligands with Improved Renal Clearance Behavior

Development of molecular tools based on the dopamine D3 receptor ligand FAUC 329 showing inhibiting effects on drug and food maintained behavior

Discovery of a dopamine D4 selective PET ligand candidate taking advantage of a click chemistry based REM linker

Disentangling inflammatory from fibrotic disease activity by fibroblast activation protein imaging

Effects of Recombinant Human Thyroid-Stimulating Hormone Superagonists on Thyroidal Uptake of18F-Fluorodeoxyglucose and Radioiodide ⬇️

Estimation of [177Lu]PSMA-617 tumor uptake based on voxel-wise 3D Monte Carlo tumor dosimetry in patients with metastasized castration resistant prostate cancer

Evaluation of18F-Labeled Benzodioxine Piperazine-Based Dopamine D4Receptor Ligands: Lipophilicity as a Determinate of Nonspecific Binding

Fast and efficient (18) F-labeling by [(18) f]fluorophenylazocarboxylic esters

First Experience With SPECT/CT Using a 99mTc-Labeled Inhibitor for Prostate-Specific Membrane Antigen in Patients With Biochemical Recurrence of Prostate Cancer

H-CRRETAWAC-OH, a lead structure for the development of radiotracer targeting integrin α5β1?

Identification of Boronic Acid Derivatives as an Active Form of N-Alkylaminoferrocene-Based Anticancer Prodrugs and Their Radiolabeling with 18F

Improved radiosynthesis and preliminary in vivo evaluation of a (18)F-labeled glycopeptide-peptoid hybrid for PET imaging of neurotensin receptor 2.

In Vitro and In Vivo Characterization of Selected Fluorine-18 Labeled Radioligands for PET Imaging of the Dopamine D3 Receptor.

In vitro and initial in vivo evaluation of (68)Ga-labeled transferrin receptor (TfR) binding peptides as potential carriers for enhanced drug transport into TfR expressing cells

In vitro characterization of the thyroidal uptake of O-(2-[(18)F]fluoroethyl)-L-tyrosine

In vitro studies on the signal transduction of thyroidal uptake of 18F-FDG and 131I-Iodide.

In vivo monitoring of the antiangiogenic effect of neurotensin receptor-mediated radiotherapy by small-animal positron emission tomography: a pilot study

Induction and repair of DNA double-strand breaks in blood lymphocytes of patients undergoing 18F-FDG PET/CT examinations ⬇️

Labeling and glycosylation of peptides using click chemistry: a general approach to (18)F-glycopeptides as effective imaging probes for positron emission tomography

Microwave-Assisted Rapid One-Pot Synthesis of Fused and Non-Fused Indoles and 5-[18 F]Fluoroindoles from Phenylazocarboxylates

Multimerization of cRGD Peptides by Click Chemistry: Synthetic Strategies, Chemical Limitations, and Influence on Biological Properties ⬇️

Multimodal Bone Metastasis-associated Epidermal Growth Factor Receptor Imaging in an Orthotopic Rat Model

Non-Invasive Characterization of Experimental Bone Metastasis in Obesity Using Multiparametric MRI and PET/CT

Optimization and synthesis of an18F-labeled dopamine D3receptor ligand using [18F]fluorophenylazocarboxylictert-butylester

PET radiopharmaceuticals for imaging integrin expression: tracers in clinical studies and recent developments.

Perturbed Development of Striatal Dopamine Transporters in Fatty Versus Lean Zucker Rats: a Follow-up Small Animal PET Study

Pharmacological characterization of low-to-moderate affinity opioid receptor agonists and brain imaging with 18F-labeled derivatives in rats

Prediction of early metastatic disease in experimental breast cancer bone metastasis by combining PET/CT and MRI parameters to a Model-Averaged Neural Network

Prototypic 18F-Labeled Argininamide-Type Neuropeptide Y Y1R Antagonists as Tracers for PET Imaging of Mammary Carcinoma.

Radioligands for the dopamine receptor subtypes

Radiopharmaceuticals for imaging and endoradiotherapy of neurotensin receptor-positive tumors.

Radiosynthesis and Preclinical Evaluation of 18F-Fluoroglycosylated Octreotate for Somatostatin Receptor Imaging.

Radiosynthesis and evaluation of 18F-labeled dopamine D4-receptor ligands

Radiosynthesis and validation of ¹⁸F-FP-CMT, a phenyltropane with superior properties for imaging the dopamine transporter in living brain.

Radiosynthesis of an F-fluoroglycosylated aminoferrocene for in-vivo imaging of reactive oxygen species activity by PET

Recent trends in pharmaceutical radiochemistry for molecular PET imaging

Regulation of uptake of 18F-FDG by a follicular human thyroid cancer cell line with mutation-activated K-ras

Specific binding of [(18)F]fluoroethyl-harmol to monoamine oxidase A in rat brain cryostat sections, and compartmental analysis of binding in living brain

Structure-selectivity investigations of D2-like receptor ligands by CoMFA and CoMSIA guiding the discovery of D3 selective PET radioligands

Sweetening pharmaceutical radiochemistry by (18)f-fluoroglycosylation: a short review.

Syntheses and radiofluorination of two derivatives of 5-cyano-indole as selective ligands for the dopamine subtype-4 receptor

Syntheses, receptor bindings, in vitro and in vivo stabilities and biodistributions of DOTA-neurotensin(8-13) derivatives containing β-amino acid residues - a lesson about the importance of animal experiments

Synthesis and evaluation of 18F-labeled dopamine D3 receptor ligands as potential PET imaging agents

Synthesis and evaluation of a (18)F-labeled diarylpyrazole glycoconjugate for the imaging of NTS1-positive tumors

Synthesis and evaluation of fluoro substituted pyridinylcarboxamides and their phenylazo analogues for potential dopamine D3 receptor PET imaging

Synthesis and in vitro and in vivo evaluation of an (18)F-labeled neuropeptide Y analogue for imaging of breast cancer by PET.

Synthesis and in vivo evaluation of an (18)F-labeled glycoconjugate of PD156707 for imaging ETA receptor expression in thyroid carcinoma by positron emission tomography

Synthesis and radioiodination of selective ligands for the dopamine D3 receptor subtype

Synthesis of a (68)ga-labeled peptoid-Peptide hybrid for imaging of neurotensin receptor expression in vivo

Synthesis, biological evaluation and radiosynthesis of buprenorphine-derived phenylazocarboxamides as novel μ-opioid receptor ligands

Synthesis, radiofluorination, and in vitro evaluation of pyrazolo[1,5-a]pyridine-based dopamine D4 receptor ligands: discovery of an inverse agonist radioligand for PET.

Targeting Fibroblast Activation Protein: Radiosynthesis and Preclinical Evaluation of an 18F-labeled FAP Inhibitor

Theranostic Value of Multimers: Lessons Learned from Trimerization of Neurotensin Receptor Ligands and Other Targeting Vectors

[(68)Ga]Ga-DO(2)A-(OBu-l-tyr)(2): synthesis, (68)Ga-radiolabeling and in vitro studies of a novel (68)Ga-DO(2)A-tyrosine conjugate as potential tumor tracer for PET.

[18F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor