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A Vancomycin Derivative with a Pyrophosphate-Binding Group: A Strategy to Combat Vancomycin-Resistant Bacteria

artículo científico publicado en 2016

Amide side chain amphiphilic polymers disrupt surface established bacterial bio-films and protect mice from chronic Acinetobacter baumannii infection.

artículo científico publicado en 2015

Antibacterial and Antibiofilm Activity of Cationic Small Molecules with Spatial Positioning of Hydrophobicity: An in Vitro and in Vivo Evaluation.

artículo científico publicado en 2016

Autophosphorylation of gatekeeper tyrosine by symbiosis receptor kinase.

artículo científico publicado en 2013

Battle Against Vancomycin-Resistant Bacteria: Recent Developments in Chemical Strategies

artículo científico publicado en 2018

Chitosan Derivatives Active against Multidrug-Resistant Bacteria and Pathogenic Fungi: In Vivo Evaluation as Topical Antimicrobials

artículo científico publicado en 2016

Cyclization and unsaturation rather than isomerisation of side chains govern the selective antibacterial activity of cationic-amphiphilic polymers.

artículo científico publicado en 2016

Designing Simple Lipidated Lysines: Bifurcation Imparts Selective Antibacterial Activity.

artículo científico publicado en 2016

Gatekeeper Tyrosine Phosphorylation of SYMRK Is Essential for Synchronizing the Epidermal and Cortical Responses in Root Nodule Symbiosis

artículo científico publicado en 2016

Gatekeeper tyrosine phosphorylation is autoinhibitory for Symbiosis Receptor Kinase.

artículo científico publicado en 2014

Intracellular activity of a membrane-active glycopeptide antibiotic against meticillin-resistant Staphylococcus aureus infection

artículo científico publicado en 2016

Isosteric substitution in cationic-amphiphilic polymers reveals an important role for hydrogen bonding in bacterial membrane interactions.

artículo científico publicado en 2016

Membrane Active Small Molecules Show Selective Broad Spectrum Antibacterial Activity with No Detectable Resistance and Eradicate Biofilms

artículo científico publicado en 2015

Membrane Disruption and Enhanced Inhibition of Cell-Wall Biosynthesis: A Synergistic Approach to Tackle Vancomycin-Resistant Bacteria.

artículo científico publicado en 2015

Membrane active phenylalanine conjugated lipophilic norspermidine derivatives with selective antibacterial activity.

artículo científico publicado en 2014

Membrane-active macromolecules kill antibiotic-tolerant bacteria and potentiate antibiotics towards Gram-negative bacteria.

artículo científico publicado en 2017

Selective and broad spectrum amphiphilic small molecules to combat bacterial resistance and eradicate biofilms.

artículo científico publicado en 2015

Side Chain Degradable Cationic-Amphiphilic Polymers with Tunable Hydrophobicity Show in Vivo Activity.

artículo científico publicado en 2016

Structure-Activity Relationship of Amino Acid Tunable Lipidated Norspermidine Conjugates: Disrupting Biofilms with Potent Activity against Bacterial Persisters.

artículo científico publicado en 2015

Vancomycin Analogue Restores Meropenem Activity against NDM-1 Gram-Negative Pathogens

artículo científico publicado en 2018

l-Lysine based lipidated biphenyls as agents with anti-biofilm and anti-inflammatory properties that also inhibit intracellular bacteria.

artículo científico publicado en 2017