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1,2,3-Triazolyl-tetrahydropyrimidine Conjugates as Potential Sterol Carrier Protein-2 Inhibitors: Larvicidal Activity against the Malaria Vector and In Silico Molecular Docking Study

artículo científico publicado en 2022

1,2,3-Triazolyl-tetrahydropyrimidine Conjugates as Potential Sterol Carrier Protein-2 Inhibitors: Larvicidal Activity against the Malaria Vector and In Silico Molecular Docking Study

artículo científico publicado en 2022

7-Amino-2-aryl/hetero-aryl-5-oxo-5,8-dihydro[1,2,4]triazolo[1,5-a]pyridine-6-carbonitriles: Synthesis and adenosine receptor binding studies

scientific article published on 15 May 2019

<i>In vitro</i> anti-TB properties, <i>in silico</i> target validation, molecular docking and dynamics studies of substituted 1,2,4-oxadiazole analogues against <i>Mycobacterium tuberculosis</i>

artículo científico publicado en 2021

Anti-Tubercular Properties of 4-Amino-5-(4-Fluoro-3- Phenoxyphenyl)-4H-1,2,4-Triazole-3-Thiol and Its Schiff Bases: Computational Input and Molecular Dynamics

scientific article published on 31 August 2020

Antitubercular, Cytotoxicity, and Computational Target Validation of Dihydroquinazolinone Derivatives

artículo científico publicado en 2022

Crystallography, in Silico Studies, and In Vitro Antifungal Studies of 2,4,5 Trisubstituted 1,2,3-Triazole Analogues

artículo científico publicado en 2020

Cytotoxicity and Antimycobacterial Properties of Pyrrolo[1,2-a]quinoline Derivatives: Molecular Target Identification and Molecular Docking Studies

scientific article published on 07 May 2020

Evolving nanoformulation strategies for diagnosis and clinical interventions for Parkinson's disease

artículo científico publicado en 2019

Functionalized carbon nanotubes as emerging delivery system for the treatment of cancer

scientific article published on 08 July 2018

Imidazo[1,2-a]pyridine Scaffold as Prospective Therapeutic Agents

artículo científico publicado en 2016

In silico and saturation transfer difference NMR approaches to unravel the binding mode of an andrographolide derivative to K-Ras oncoprotein

artículo científico publicado en 2020

Larvicidal Activities of 2-Aryl-2,3-Dihydroquinazolin -4-ones against Malaria Vector Anopheles arabiensis, In Silico ADMET Prediction and Molecular Target Investigation

scientific article published on 13 March 2020

Medicinal Chemistry and Therapeutic Potential of Agonists, Antagonists and Allosteric Modulators of A1 Adenosine Receptor: Current Status and Perspectives

artículo científico publicado en 2019

Molecular docking and receptor-specific 3D-QSAR studies of acetylcholinesterase inhibitors.

artículo científico publicado en 2012

Molecular dynamics simulation strategies for designing carbon-nanotube-based targeted drug delivery

artículo científico publicado en 2017

Molecular modeling approaches for the discovery of adenosine A2B receptor antagonists: current status and future perspectives

artículo científico publicado en 2019

Molecular signaling of G-protein-coupled receptor in chronic heart failure and associated complications

scientific article published on 30 November 2019

Novel Therapies for the Treatment of Neuropathic Pain: Potential and Pitfalls

artículo científico publicado en 2022

P1 Receptor Agonists/Antagonists in Clinical Trials - Potential Drug Candidates of the Future

artículo científico publicado en 2019

Progress in the Development of Agonists, Antagonists and Allosteric Modulators of Adenosine Receptors

artículo científico publicado en 2019

Recent Updates in the Computer Aided Drug Design Strategies for the Discovery of Agonists and Antagonists of Adenosine Receptors

artículo científico publicado en 2019

Synthesis and evaluation of 2,4,5-trisubstitutedthiazoles as carbonic anhydrase-III inhibitors

artículo científico publicado en 2020

Synthesis, adenosine receptor binding and molecular modelling studies of novel thieno[2,3-d]pyrimidine derivatives.

artículo científico publicado en 2017

Synthesis, biological evaluation, and computational investigation of ethyl 2,4,6-trisubstituted-1,4-dihydropyrimidine-5-carboxylates as potential larvicidal agents against Anopheles arabiensis

artículo científico publicado en 2023

Synthesis, evaluation and docking studies on 3-alkoxy-4-methanesulfonamido acetophenone derivatives as non ulcerogenic anti-inflammatory agents

scientific article published on 18 January 2012

The Beneficial Effect of Boswellic Acid on Bone Metabolism and Possible Mechanisms of Action in Experimental Osteoporosis

artículo científico publicado en 2020

Therapeutic Potentials of Adenosine Receptors: The State of The Art

scientific article published on 01 January 2019