Lista de obras -

(2-Arylethenyl)-1,3,5-triazin-2-amines as a novel histamine H4 receptor ligands

artículo científico publicado en 2015

4-tert-Pentylphenoxyalkyl derivatives - Histamine H receptor ligands and monoamine oxidase B inhibitors

artículo científico publicado en 2018

8-Benzylaminoxanthine scaffold variations for selective ligands acting on adenosine A2A receptors. Design, synthesis and biological evaluation

artículo científico publicado en 2020

A Taxicab geometry quantification system to evaluate the performance of in silico methods: a case study on adenosine receptors ligands

artículo científico publicado en 2020

Alkyl derivatives of 1,3,5-triazine as histamine H4 receptor ligands

scientific article published on 12 February 2019

Anticonvulsive effect of nonimidazole histamine H3 receptor antagonists.

artículo científico publicado en 2014

Aryl-1,3,5-triazine derivatives as histamine H4 receptor ligands.

artículo científico publicado en 2014

Chlorophenoxy aminoalkyl derivatives as histamine H(3)R ligands and antiseizure agents.

artículo científico publicado en 2015

Cholinesterase inhibitory activity of chlorophenoxy derivatives-Histamine H3 receptor ligands.

artículo científico publicado en 2016

Corrigendum to "Search for new multi-target compounds against Alzheimer's disease among histamine H3 receptor ligands" [Eur. J. Med. Chem. 185 (2020) 111785]

artículo científico publicado en 2020

Diether (substituted) piperidine derivatives as novel, histamine H3 receptor ligands.

artículo científico publicado en 2009

Diether derivatives of homo- or substituted piperidines as non-imidazole histamine H3 receptor ligands

artículo científico publicado en 2009

Discovery of Potential, Dual-Active Histamine H Receptor Ligands with Combined Antioxidant Properties

artículo científico publicado en 2021

Discovery of novel lead in the group of N-substituted piperazine ether derivatives with potential histamine H3 receptor activity.

artículo científico publicado en 2014

Dual-acting diether derivatives of piperidine and homopiperidine with histamine H(3) receptor antagonistic and anticholinesterase activity

artículo científico publicado en 2012

Dual-targeting approach on histamine H3 and sigma-1 receptor ligands as promising pharmacological tools in the treatment of CNS-linked disorders

artículo científico publicado en 2020

Fluorescent GPCR ligands as new tools in pharmacology-update, years 2008-early 2014.

artículo científico

Fluorescent GPCR ligands as new tools in pharmacology.

artículo científico publicado en 2008

H3 histamine receptor antagonist pitolisant reverses some subchronic disturbances induced by olanzapine in mice.

artículo científico publicado en 2016

Histamine H Receptor Ligands-KSK-59 and KSK-73-Reduce Body Weight Gain in a Rat Model of Excessive Eating

artículo científico publicado en 2021

Histamine H3 receptor ligands in the group of (homo)piperazine derivatives

artículo científico publicado en 2017

KSK19 - Novel histamine H3 receptor ligand reduces body weight in diet induced obese mice

scientific article published on 08 July 2019

Monocyclic and Fused Azines and Azoles as Histamine H₄ Receptor Ligands

artículo científico publicado en 2016

N-substituted piperazine derivatives as potential multitarget agents acting on histamine H3 receptor and cancer resistance proteins

artículo científico publicado en 2020

Non-imidazole-based histamine H3 receptor antagonists with anticonvulsant activity in different seizure models in male adult rats.

artículo científico publicado en 2016

Novel multi-target directed ligands based on annelated xanthine scaffold with aromatic substituents acting on adenosine receptor and monoamine oxidase B. Synthesis, in vitro and in silico studies

scientific article published on 02 February 2019

Novel, Dual Target-Directed Annelated Xanthine Derivatives Acting on Adenosine Receptors and Monoamine Oxidase B

scientific article published on 12 March 2020

Optimization and preclinical evaluation of novel histamine H3receptor ligands: Acetyl and propionyl phenoxyalkyl piperazine derivatives

scientific article published on 10 November 2018

Piperidine variations in search for non-imidazole histamine H(3) receptor ligands.

artículo científico publicado en 2008

Probing an artificial polypeptide receptor library using a series of novel histamine H3 receptor ligands

artículo científico publicado en 2014

Rational design of new multitarget histamine H3 receptor ligands as potential candidates for treatment of Alzheimer's disease

artículo científico publicado en 2020

Search for new multi-target compounds against Alzheimer's disease among histamine H3 receptor ligands

scientific article published on 17 October 2019

Search for novel, high affinity histamine H3 receptor ligands with fluorescent properties

artículo científico publicado en 2010

Structural modifications and in vitro pharmacological evaluation of 4-pyridyl-piperazine derivatives as an active and selective histamine H3 receptor ligands

artículo científico publicado en 2019

Structural modifications in the distal, regulatory region of histamine H<sub>3</sub> receptor antagonists leading to the identification of a potent anti-obesity agent

artículo científico publicado en 2020

Synthesis and biological activity of novel tert-amylphenoxyalkyl (homo)piperidine derivatives as histamine H3R ligands.

artículo científico publicado en 2017

Synthesis and biological activity of novel tert-butyl and tert-pentylphenoxyalkyl piperazine derivatives as histamine H3R ligands

Synthesis and biological activity of tricyclic cycloalkylimidazo-, pyrimido- and diazepinopurinediones.

artículo científico publicado en 2011

The histamine H3 receptor inverse agonist pitolisant reduces body weight in obese mice

artículo científico publicado en 2018

Lista de obras de

(2-Arylethenyl)-1,3,5-triazin-2-amines as a novel histamine H4 receptor ligands

4-tert-Pentylphenoxyalkyl derivatives - Histamine H receptor ligands and monoamine oxidase B inhibitors

8-Benzylaminoxanthine scaffold variations for selective ligands acting on adenosine A2A receptors. Design, synthesis and biological evaluation

A Taxicab geometry quantification system to evaluate the performance of in silico methods: a case study on adenosine receptors ligands

Alkyl derivatives of 1,3,5-triazine as histamine H4 receptor ligands

Anticonvulsive effect of nonimidazole histamine H3 receptor antagonists.

Aryl-1,3,5-triazine derivatives as histamine H4 receptor ligands.

Chlorophenoxy aminoalkyl derivatives as histamine H(3)R ligands and antiseizure agents.

Cholinesterase inhibitory activity of chlorophenoxy derivatives-Histamine H3 receptor ligands.

Corrigendum to "Search for new multi-target compounds against Alzheimer's disease among histamine H3 receptor ligands" [Eur. J. Med. Chem. 185 (2020) 111785]

Diether (substituted) piperidine derivatives as novel, histamine H3 receptor ligands.

Diether derivatives of homo- or substituted piperidines as non-imidazole histamine H3 receptor ligands

Discovery of Potential, Dual-Active Histamine H Receptor Ligands with Combined Antioxidant Properties

Discovery of novel lead in the group of N-substituted piperazine ether derivatives with potential histamine H3 receptor activity.

Dual-acting diether derivatives of piperidine and homopiperidine with histamine H(3) receptor antagonistic and anticholinesterase activity

Dual-targeting approach on histamine H3 and sigma-1 receptor ligands as promising pharmacological tools in the treatment of CNS-linked disorders

Fluorescent GPCR ligands as new tools in pharmacology-update, years 2008-early 2014.

Fluorescent GPCR ligands as new tools in pharmacology.

H3 histamine receptor antagonist pitolisant reverses some subchronic disturbances induced by olanzapine in mice.

Histamine H Receptor Ligands-KSK-59 and KSK-73-Reduce Body Weight Gain in a Rat Model of Excessive Eating

Histamine H3 receptor ligands in the group of (homo)piperazine derivatives

KSK19 - Novel histamine H3 receptor ligand reduces body weight in diet induced obese mice

Monocyclic and Fused Azines and Azoles as Histamine H₄ Receptor Ligands

N-substituted piperazine derivatives as potential multitarget agents acting on histamine H3 receptor and cancer resistance proteins

Non-imidazole-based histamine H3 receptor antagonists with anticonvulsant activity in different seizure models in male adult rats.

Novel multi-target directed ligands based on annelated xanthine scaffold with aromatic substituents acting on adenosine receptor and monoamine oxidase B. Synthesis, in vitro and in silico studies

Novel, Dual Target-Directed Annelated Xanthine Derivatives Acting on Adenosine Receptors and Monoamine Oxidase B

Optimization and preclinical evaluation of novel histamine H3receptor ligands: Acetyl and propionyl phenoxyalkyl piperazine derivatives

Piperidine variations in search for non-imidazole histamine H(3) receptor ligands.

Probing an artificial polypeptide receptor library using a series of novel histamine H3 receptor ligands

Rational design of new multitarget histamine H3 receptor ligands as potential candidates for treatment of Alzheimer's disease

Search for new multi-target compounds against Alzheimer's disease among histamine H3 receptor ligands

Search for novel, high affinity histamine H3 receptor ligands with fluorescent properties

Structural modifications and in vitro pharmacological evaluation of 4-pyridyl-piperazine derivatives as an active and selective histamine H3 receptor ligands

Structural modifications in the distal, regulatory region of histamine H<sub>3</sub> receptor antagonists leading to the identification of a potent anti-obesity agent

Synthesis and biological activity of novel tert-amylphenoxyalkyl (homo)piperidine derivatives as histamine H3R ligands.

Synthesis and biological activity of novel tert-butyl and tert-pentylphenoxyalkyl piperazine derivatives as histamine H3R ligands

Synthesis and biological activity of tricyclic cycloalkylimidazo-, pyrimido- and diazepinopurinediones.

The histamine H3 receptor inverse agonist pitolisant reduces body weight in obese mice