Lista de obras -

A Multicomponent Route to Functionalized Amides and Oxazolidinones

artículo científico publicado en 2017

A flow platform for degradation-free CuAAC bioconjugation

artículo científico publicado en 2018

A modular synthesis of functionalised phenols enabled by controlled boron speciation

scientific article published on 01 March 2015

A one-pot tandem chemoselective allylation/cross-coupling via temperature control of a multi-nucleophile/electrophile system

artículo científico publicado en 2017

Amidation of esters with amino alcohols using organobase catalysis

artículo científico publicado en 2014

Amidation of unactivated ester derivatives mediated by trifluoroethanol

artículo científico publicado en 2017

Biocatalytic Synthesis of Chiral N-Functionalized Amino Acids

artículo científico publicado en 2018

Bismesitylmagnesium: a thermally stable and non-nucleophilic carbon-centred base reagent for the efficient preparation of silyl enol ethers

artículo científico publicado en 2007

Catalytic Enantioselective Synthesis of α-Chiral Azaheteroaryl Ethylamines by Asymmetric Protonation

scientific article published on 01 August 2018

Chan-Evans-Lam Amination of Boronic Acid Pinacol (BPin) Esters: Overcoming the Aryl Amine Problem

scientific article published on 18 April 2016

Chemoselective One-Pot Synthesis of Functionalized Amino-azaheterocycles Enabled by COware

artículo científico publicado en 2017

Chemoselective Suzuki-Miyaura Cross-Coupling via Kinetic Transmetallation.

artículo científico publicado en 2016

Chemoselective boronic ester synthesis by controlled speciation.

artículo científico publicado en 2014

Chemoselective oxidation of aryl organoboron systems enabled by boronic acid-selective phase transfer

artículo científico publicado en 2016

Contra-Thermodynamic, Photocatalytic E→Z Isomerization of Styrenyl Boron Species: Vectors to Facilitate Exploration of 2D Chemical Space.

artículo científico publicado en 2018

Correction to "Modular, Step-Efficient Palladium-Catalyzed Cross-Coupling Strategy To Access C6-Heteroaryl 2-Aminopurine Ribonucleosides".

artículo científico publicado en 2017

Cyrene as a bio-based solvent for HATU mediated amide coupling

artículo científico publicado en 2018

Deoxyfluorination with CuF2 : Enabled by Using a Lewis Base Activating Group

artículo científico publicado en 2020

Determining the Origin of Rate-Independent Chemoselectivity in CuAAC Reactions: An Alkyne-Specific Shift in Rate-Determining Step.

artículo científico publicado en 2017

Discovery of Tetrahydroquinoxalines as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the Second Bromodomain.

artículo científico publicado en 2018

Emergence of Small-Molecule Non-RGD-Mimetic Inhibitors for RGD Integrins.

artículo científico publicado en 2017

First experimental evidence for a bis-ethene chromium(I) complex forming from an activated ethene oligomerization catalyst

artículo científico publicado en 2020

In situ generation of Mes2Mg as a non-nucleophilic carbon-centred base reagent for the efficient one-pot conversion of ketones to silyl enol ethers.

artículo científico publicado en 2008

Interrogating Pd(II) Anion Metathesis Using a Bifunctional Chemical Probe: A Transmetalation Switch.

artículo científico publicado en 2017

Mechanism of Cu-Catalyzed Aryl Boronic Acid Halodeboronation Using Electrophilic Halogen: Development of a Base-Catalyzed Iododeboronation for Radiolabeling Applications

scientific article published on 25 March 2019

Mechanistic Development and Recent Applications of the Chan-Lam Amination

scientific article published on 22 November 2019

Modular, Step-Efficient Palladium-Catalyzed Cross-Coupling Strategy To Access C6-Heteroaryl 2-Aminopurine Ribonucleosides.

artículo científico publicado en 2017

N-Alkyl-α-amino acids in Nature and their biocatalytic preparation

scientific article published on 26 January 2019

Ni vs. Pd in Suzuki-Miyaura sp2-sp2 cross-coupling: a head-to-head study in a comparable precatalyst/ligand system

scientific article published on 03 May 2019

One-Pot Homologation of Boronic Acids: A Platform for Diversity-Oriented Synthesis

artículo científico publicado en 2015

Practical synthesis of pharmaceutically relevant molecules enriched in sp3 character.

artículo científico publicado en 2017

Rational Design of Autotaxin Inhibitors by Structural Evolution of Endogenous Modulators

artículo científico publicado en 2017

Scalable total synthesis and comprehensive structure-activity relationship studies of the phytotoxin coronatine.

artículo científico publicado en 2018

Scope and limitations of a DMF bio-alternative within Sonogashira cross-coupling and Cacchi-type annulation

artículo científico publicado en 2016

Soft scorpionate anions as platforms for novel heterocycles.

artículo científico publicado en 2013

Speciation control during Suzuki-Miyaura cross-coupling of haloaryl and haloalkenyl MIDA boronic esters

artículo científico publicado en 2015

Spectroscopic Studies of the Chan-Lam Amination: A Mechanism-Inspired Solution to Boronic Ester Reactivity.

artículo científico publicado en 2017

Strategy for Conditional Orthogonal Sequential CuAAC Reactions Using a Protected Aromatic Ynamine.

artículo científico publicado en 2017

Structure-Activity Relationships of Small Molecule Autotaxin Inhibitors with a Discrete Binding Mode

artículo científico publicado en 2016

Synthesis of 2-BMIDA 6,5-bicyclic heterocycles by Cu(i)/Pd(0)/Cu(ii) cascade catalysis of 2-iodoaniline/phenols

artículo científico publicado en 2016

Synthesis of functionalised 4H-quinolizin-4-ones via tandem Horner-Wadsworth-Emmons olefination/cyclisation.

artículo científico publicado en 2013

Tandem Chemoselective Suzuki-Miyaura Cross-Coupling Enabled by Nucleophile Speciation Control

artículo científico publicado en 2015

Towards energetically viable asymmetric deprotonations: selectivity at more elevated temperatures with C2-symmetric magnesium bisamides

artículo científico publicado en 2011

Lista de obras de

A Multicomponent Route to Functionalized Amides and Oxazolidinones

A flow platform for degradation-free CuAAC bioconjugation

A modular synthesis of functionalised phenols enabled by controlled boron speciation

A one-pot tandem chemoselective allylation/cross-coupling via temperature control of a multi-nucleophile/electrophile system

Amidation of esters with amino alcohols using organobase catalysis

Amidation of unactivated ester derivatives mediated by trifluoroethanol

Biocatalytic Synthesis of Chiral N-Functionalized Amino Acids

Bismesitylmagnesium: a thermally stable and non-nucleophilic carbon-centred base reagent for the efficient preparation of silyl enol ethers

Catalytic Enantioselective Synthesis of α-Chiral Azaheteroaryl Ethylamines by Asymmetric Protonation

Chan-Evans-Lam Amination of Boronic Acid Pinacol (BPin) Esters: Overcoming the Aryl Amine Problem

Chemoselective One-Pot Synthesis of Functionalized Amino-azaheterocycles Enabled by COware

Chemoselective Suzuki-Miyaura Cross-Coupling via Kinetic Transmetallation.

Chemoselective boronic ester synthesis by controlled speciation.

Chemoselective oxidation of aryl organoboron systems enabled by boronic acid-selective phase transfer

Contra-Thermodynamic, Photocatalytic E→Z Isomerization of Styrenyl Boron Species: Vectors to Facilitate Exploration of 2D Chemical Space.

Correction to "Modular, Step-Efficient Palladium-Catalyzed Cross-Coupling Strategy To Access C6-Heteroaryl 2-Aminopurine Ribonucleosides".

Cyrene as a bio-based solvent for HATU mediated amide coupling

Deoxyfluorination with CuF2 : Enabled by Using a Lewis Base Activating Group

Determining the Origin of Rate-Independent Chemoselectivity in CuAAC Reactions: An Alkyne-Specific Shift in Rate-Determining Step.

Discovery of Tetrahydroquinoxalines as Bromodomain and Extra-Terminal Domain (BET) Inhibitors with Selectivity for the Second Bromodomain.

Emergence of Small-Molecule Non-RGD-Mimetic Inhibitors for RGD Integrins.

First experimental evidence for a bis-ethene chromium(I) complex forming from an activated ethene oligomerization catalyst

In situ generation of Mes2Mg as a non-nucleophilic carbon-centred base reagent for the efficient one-pot conversion of ketones to silyl enol ethers.

Interrogating Pd(II) Anion Metathesis Using a Bifunctional Chemical Probe: A Transmetalation Switch.

Mechanism of Cu-Catalyzed Aryl Boronic Acid Halodeboronation Using Electrophilic Halogen: Development of a Base-Catalyzed Iododeboronation for Radiolabeling Applications

Mechanistic Development and Recent Applications of the Chan-Lam Amination

Modular, Step-Efficient Palladium-Catalyzed Cross-Coupling Strategy To Access C6-Heteroaryl 2-Aminopurine Ribonucleosides.

N-Alkyl-α-amino acids in Nature and their biocatalytic preparation

Ni vs. Pd in Suzuki-Miyaura sp2-sp2 cross-coupling: a head-to-head study in a comparable precatalyst/ligand system

One-Pot Homologation of Boronic Acids: A Platform for Diversity-Oriented Synthesis

Practical synthesis of pharmaceutically relevant molecules enriched in sp3 character.

Rational Design of Autotaxin Inhibitors by Structural Evolution of Endogenous Modulators

Scalable total synthesis and comprehensive structure-activity relationship studies of the phytotoxin coronatine.

Scope and limitations of a DMF bio-alternative within Sonogashira cross-coupling and Cacchi-type annulation

Soft scorpionate anions as platforms for novel heterocycles.

Speciation control during Suzuki-Miyaura cross-coupling of haloaryl and haloalkenyl MIDA boronic esters

Spectroscopic Studies of the Chan-Lam Amination: A Mechanism-Inspired Solution to Boronic Ester Reactivity.

Strategy for Conditional Orthogonal Sequential CuAAC Reactions Using a Protected Aromatic Ynamine.

Structure-Activity Relationships of Small Molecule Autotaxin Inhibitors with a Discrete Binding Mode

Synthesis of 2-BMIDA 6,5-bicyclic heterocycles by Cu(i)/Pd(0)/Cu(ii) cascade catalysis of 2-iodoaniline/phenols

Synthesis of functionalised 4H-quinolizin-4-ones via tandem Horner-Wadsworth-Emmons olefination/cyclisation.

Tandem Chemoselective Suzuki-Miyaura Cross-Coupling Enabled by Nucleophile Speciation Control

Towards energetically viable asymmetric deprotonations: selectivity at more elevated temperatures with C2-symmetric magnesium bisamides