Lista de obras -

A phosphonamidate containing aromatic N-terminal amino group as inhibitor of leucine aminopeptidase-design, synthesis and stability.

artículo científico publicado en 2006

A structural insight into the P1S1 binding mode of diaminoethylphosphonic and phosphinic acids, selective inhibitors of alanine aminopeptidases

artículo científico publicado en 2016

A synthetic method for diversification of the P1' substituent in phosphinic dipeptides as a tool for exploration of the specificity of the S1' binding pockets of leucine aminopeptidases

artículo científico publicado en 2007

Addition of thiols to the double bond of dipeptide C-terminal dehydroalanine as a source of new inhibitors of cathepsin C

artículo científico publicado en 2017

Individual stereoisomers of phosphinic dipeptide inhibitor of leucine aminopeptidase.

artículo científico publicado en 2008

N-Benzyl Residues as the P1' Substituents in Phosphorus-Containing Extended Transition State Analog Inhibitors of Metalloaminopeptidases

artículo científico publicado en 2020

Phosphonic Acid Analogues of Phenylglycine as Inhibitors of Aminopeptidases: Comparison of Porcine Aminopeptidase N, Bovine Leucine Aminopeptidase, Tomato Acidic Leucine Aminopeptidase and Aminopeptidase from Barley Seeds

artículo científico publicado en 2019

Purification and partial characterization of aminopeptidase from barley (Hordeum vulgare L.) seeds ⬇️

artículo científico publicado el 8 de febrero de 2013

Stereoselective synthesis of 1-aminoalkanephosphonic acids with two chiral centers and their activity towards leucine aminopeptidase.

artículo científico publicado en 2003

Structure-guided, single-point modifications in the phosphinic dipeptide structure yield highly potent and selective inhibitors of neutral aminopeptidases.

artículo científico publicado en 2014

Substituted phosphonic analogues of phenylglycine as inhibitors of phenylalanine ammonia lyase from potatoes

artículo científico publicado en 2018

Substrate specificity screening of oat (Avena sativa) seeds aminopeptidase demonstrate unusually broad tolerance in S1 pocket ⬇️

artículo científico publicado el 8 de febrero de 2012

Synthesis of Hybrid Tripeptide Peptidomimetics Containing Dehydroamino Acid and Aminophosphonic Acid in the Chain and Evaluation of Their Activity toward Cathepsin C

artículo científico publicado en 2022

Synthesis of dehydrodipeptide esters and their evaluation as inhibitors of cathepsin C.

artículo científico publicado en 2015

Toward very potent, non-covalent organophosphonate inhibitors of cathepsin C and related enzymes by 2-amino-1-hydroxy-alkanephosphonates dipeptides

artículo científico publicado en 2013

Unusual activity pattern of leucine aminopeptidase inhibitors based on phosphorus containing derivatives of methionine and norleucine

artículo científico publicado en 2010

Lista de obras de