Lista de obras -

3D QSAR analyses-guided rational design of novel ligands for the (alpha4)2(beta2)3 nicotinic acetylcholine receptor

artículo científico publicado en 2003

6H,13H-Pyrazino[1,2-a;4,5-a']diindole analogs: probing the pharmacophore for allosteric ligands of muscarinic M2 receptors

artículo científico publicado en 2006

A hydrazide linker strategy for heterobivalent compounds as ortho- and allosteric ligands of acetylcholine-binding proteins

artículo científico publicado en 2011

Bispidine as a Privileged Scaffold

artículo científico publicado en 2015

Carbazole Scaffold in Medicinal Chemistry and Natural Products: A Review from 2010-2015.

artículo científico publicado en 2015

Cytisine-based nicotinic partial agonists as novel antidepressant compounds

artículo científico publicado en 2009

Development of a 5-Hydroxytryptamine2A Receptor Binding Assay for High Throughput Screening Using 96-Well Microfilter Plates

scholarly article by Antje Harms et al published 1 August 2000 in Journal of Biomolecular Screening

Effects of Abeta1-42 fibrils and of the tetrapeptide Pr-IIGL on the phosphorylation state of the tau-protein and on the alpha7 nicotinic acetylcholine receptor in vitro

artículo científico publicado en 2005

Feasibility of 2-deoxy-2-[18F]fluoro-D-glucose- A85380-PET for imaging of human cardiac nicotinic acetylcholine receptors in vivo.

artículo científico publicado en 2006

Feasibility of [18F]-2-Fluoro-A85380-PET imaging of human vascular nicotinic acetylcholine receptors in vivo

artículo científico publicado en 2012

Halogenated and isosteric cytisine derivatives with increased affinity and functional activity at nicotinic acetylcholine receptors

artículo científico publicado en 2005

Heliotropiumides A and B, new phenolamides with N-carbamoyl putrescine moiety from Heliotropium foertherianum collected in Hawaii and their biological activities

artículo científico publicado en 2017

In vitro characterization of 6-[18F]fluoro-A-85380, a high-affinity ligand for alpha4beta2* nicotinic acetylcholine receptors

artículo científico publicado en 2005

In vitro evaluation of nicotinic acetylcholine receptors with 2-[18F]F-A85380 in Parkinson's disease

artículo científico publicado en 2006

Nicotine decreases food intake through activation of POMC neurons

artículo científico publicado en 2011

Nicotinic acetylcholine receptor ligands, a patent review (2006 – 2011) ⬇️

artículo científico publicado el 1 de diciembre de 2011

Prenylated indole alkaloids from Flustra foliacea with subtype specific binding on NAChRs

artículo científico publicado en 2004

Semisynthetic analogues of toxiferine I and their pharmacological properties at α7 nAChRs, muscle-type nAChRs, and the allosteric binding site of muscarinic M2 receptors

artículo científico publicado en 2014

Smoking upregulates alpha4beta2* nicotinic acetylcholine receptors in the human brain

artículo científico publicado en 2007

Syntheses and evaluation of pyridazine and pyrimidine containing bioisosteres of (+/-)-pyrido[3.4-b]homotropane and pyrido-[3.4-b]tropane as novel nAChR ligands

artículo científico publicado en 2002

Synthesis and evaluation of phenylcarbamate derivatives as ligands for nicotinic acetylcholine receptors

artículo científico publicado en 2004

Synthesis and nicotinic binding studies on enantiopure diazine analogues of the novel (2-chloro-5-pyridyl)-9-azabicyclo[4.2.1]non-2-ene UB-165.

artículo científico publicado en 2002

Synthetic approaches and bio-distribution studies of [11C]methyl-phenidate.

artículo científico publicado en 2007

The 3,7-diazabicyclo[3.3.1]nonane scaffold for subtype selective nicotinic acetylcholine receptor (nAChR) ligands. Part 1: the influence of different hydrogen bond acceptor systems on alkyl and (hetero)aryl substituents

artículo científico publicado en 2013

The 3,7-diazabicyclo[3.3.1]nonane scaffold for subtype selective nicotinic acetylcholine receptor ligands. Part 2: carboxamide derivatives with different spacer motifs

artículo científico publicado en 2013

The twin drug approach for novel nicotinic acetylcholine receptor ligands

artículo científico publicado en 2015

[Nuclides and tracers--mechanisms and application. Radiodiagnosis for peripheral organ diseases].

artículo científico publicado en 2005

Lista de obras de

3D QSAR analyses-guided rational design of novel ligands for the (alpha4)2(beta2)3 nicotinic acetylcholine receptor

6H,13H-Pyrazino[1,2-a;4,5-a']diindole analogs: probing the pharmacophore for allosteric ligands of muscarinic M2 receptors

A hydrazide linker strategy for heterobivalent compounds as ortho- and allosteric ligands of acetylcholine-binding proteins

Bispidine as a Privileged Scaffold

Carbazole Scaffold in Medicinal Chemistry and Natural Products: A Review from 2010-2015.

Cytisine-based nicotinic partial agonists as novel antidepressant compounds

Development of a 5-Hydroxytryptamine2A Receptor Binding Assay for High Throughput Screening Using 96-Well Microfilter Plates

Effects of Abeta1-42 fibrils and of the tetrapeptide Pr-IIGL on the phosphorylation state of the tau-protein and on the alpha7 nicotinic acetylcholine receptor in vitro

Feasibility of 2-deoxy-2-[18F]fluoro-D-glucose- A85380-PET for imaging of human cardiac nicotinic acetylcholine receptors in vivo.

Feasibility of [18F]-2-Fluoro-A85380-PET imaging of human vascular nicotinic acetylcholine receptors in vivo

Halogenated and isosteric cytisine derivatives with increased affinity and functional activity at nicotinic acetylcholine receptors

Heliotropiumides A and B, new phenolamides with N-carbamoyl putrescine moiety from Heliotropium foertherianum collected in Hawaii and their biological activities

In vitro characterization of 6-[18F]fluoro-A-85380, a high-affinity ligand for alpha4beta2* nicotinic acetylcholine receptors

In vitro evaluation of nicotinic acetylcholine receptors with 2-[18F]F-A85380 in Parkinson's disease

Nicotine decreases food intake through activation of POMC neurons

Nicotinic acetylcholine receptor ligands, a patent review (2006 – 2011) ⬇️

Prenylated indole alkaloids from Flustra foliacea with subtype specific binding on NAChRs

Semisynthetic analogues of toxiferine I and their pharmacological properties at α7 nAChRs, muscle-type nAChRs, and the allosteric binding site of muscarinic M2 receptors

Smoking upregulates alpha4beta2* nicotinic acetylcholine receptors in the human brain

Syntheses and evaluation of pyridazine and pyrimidine containing bioisosteres of (+/-)-pyrido[3.4-b]homotropane and pyrido-[3.4-b]tropane as novel nAChR ligands

Synthesis and evaluation of phenylcarbamate derivatives as ligands for nicotinic acetylcholine receptors

Synthesis and nicotinic binding studies on enantiopure diazine analogues of the novel (2-chloro-5-pyridyl)-9-azabicyclo[4.2.1]non-2-ene UB-165.

Synthetic approaches and bio-distribution studies of [11C]methyl-phenidate.

The 3,7-diazabicyclo[3.3.1]nonane scaffold for subtype selective nicotinic acetylcholine receptor (nAChR) ligands. Part 1: the influence of different hydrogen bond acceptor systems on alkyl and (hetero)aryl substituents

The 3,7-diazabicyclo[3.3.1]nonane scaffold for subtype selective nicotinic acetylcholine receptor ligands. Part 2: carboxamide derivatives with different spacer motifs

The twin drug approach for novel nicotinic acetylcholine receptor ligands

[Nuclides and tracers--mechanisms and application. Radiodiagnosis for peripheral organ diseases].