Lista de obras - D G Vander Velde - Dominio Público Uruguay

18Oxygen incorporation into inorganic phosphate in the reaction catalyzed by N5,10-methenyltetrahydrofolate synthetase

artículo científico publicado en 1995

A 19F NMR study of lomefloxacin in human erythrocytes and its interaction with hemoglobin

artículo científico publicado en 1995

A one-step synthesis of a deuterated paclitaxel analogue: 10-deacetoxy-(10alpha-2H)paclitaxel

artículo científico publicado en 1999

A tandem Prins/Schmidt reaction approach to marine alkaloids: formal and total syntheses of lepadiformines A and C

artículo científico publicado en 2010

Alternate substrates of human glutaryl-CoA dehydrogenase: structure and reactivity of substrates, and identification of a novel 2-enoyl-CoA product.

artículo científico publicado en 2002

An Initial Event in the Insect Innate Immune Response: Structural and Biological Studies of Interactions between β-1,3-Glucan and the N-Terminal Domain of β-1,3-Glucan Recognition Protein

artículo científico publicado en 2013

Biofilm-specific extracellular matrix proteins of nontypeable Haemophilus influenzae

artículo científico publicado en 2014

CO Coupling Chemistry of a Terminal Mo Carbide: Sequential Addition of Proton, Hydride, and CO Releases Ethenone

scientific article published on 19 September 2019

Characterization and dynamics of substituted ruthenacyclobutanes relevant to the olefin cross-metathesis reaction

artículo científico publicado en 2011

Characterization of the complexation of fluoroquinolone antimicrobials with metal ions by nuclear magnetic resonance spectroscopy

scientific article published on 01 January 1993

Comparative effects of (SBE)7m-beta-CD and HP-beta-CD on the stability of two anti-neoplastic agents, melphalan and carmustine

artículo científico publicado en 2000

Comprehensive study of sansalvamide A derivatives and their structure-activity relationships against drug-resistant colon cancer cell lines.

artículo científico publicado en 2008

Conformation of ATP and ADP bound to N10-formyltetrahydrofolate synthetase determined by TRNOE NMR spectroscopy.

artículo científico publicado en 1994

Conformational analysis of the beta-amyloid peptide fragment, beta(12-28)

artículo científico publicado en 1995

Conformational studies on resiniferatoxin (RTX), an ultrapotent vanilloid agonist

artículo científico publicado en 1998

Conformationally restricted paclitaxel analogues: macrocyclic mimics of the "hydrophobic collapse" conformation

artículo científico publicado en 1999

Cyclodextrin-catalyzed deacetylation of spironolactone is pH and cyclodextrin dependent

scientific article published on 01 February 2000

Deamidation of model beta-turn cyclic peptides in the solid state

artículo científico publicado en 2005

Diastereomeric phosphonate ester adducts of chymotrypsin: 31P-NMR measurements

scientific article published on 01 January 1993

Effect of buffer species on the thermally induced aggregation of interferon-tau

artículo científico publicado en 2006

Effect of conformation on the rate of deamidation of vancomycin in aqueous solutions

scientific article published on 01 June 2000

Effect of progressive benzyl substitution on the conformations of aminocaproic acid-cyclized dipeptides.

artículo científico publicado en 2001

Effect of restricted conformational flexibility on the permeation of model hexapeptides across Caco-2 cell monolayers

artículo científico publicado en 1997

Effect of stereochemistry on the transport of Aca-linked β-turn peptidomimetics across a human intestinal cell line ⬇️

artículo científico publicado el 1 de septiembre de 1997

Effect of zinc binding on the structure and stability of fibrolase, a fibrinolytic protein from snake venom

artículo científico publicado en 1992

Effects of amino acid chirality and the chemical linker on the cell permeation characteristics of cyclic prodrugs of opioid peptides.

artículo científico publicado en 2006

Evaluation of NMR diffusion measurements for the conformational analysis of flexible peptides.

artículo científico publicado en 2001

Experimental and theoretical investigations into the unusual regioselectivity of 4,5-, 5,6-, and 6,7-indole aryne cycloadditions

artículo científico publicado en 2010

Fibrolase. A fibrinolytic protein from snake venom.

artículo científico publicado en 1993

Fluoride-facilitated deuterium exchange from DMSO-d6 to polyamide-based cryptands.

artículo científico publicado en 2004

Get5 Carboxyl-terminal Domain Is a Novel Dimerization Motif That Tethers an Extended Get4/Get5 Complex

artículo científico publicado en 2012

Highly regioirregular polypropylene from asymmetric group 4 anilide(pyridine)phenoxide complexes.

artículo científico publicado en 2012

Hydrocotylosides I-VII, new oleanane saponins from hydrocotylesibthorpioides.

artículo científico publicado en 2004

Hydrolysis of the prodrug, 2',3',5'-triacetyl-6-azauridine.

artículo científico publicado en 1995

Improved preparation and structural conformation of the fluorescence labelling reagents 1,2-diamino-4,5-dimethoxybenzene and 3,4-dihydro-6,7-dimethoxy-4-methyl-3-oxo-quinoxaline-2-carbonyl chloride

scientific article published on 01 January 1990

Indole-derived arynes and their Diels-Alder reactivity with furans

artículo científico publicado en 2007

Isolation and characterization by NMR spectroscopy of three monosubstituted 4-sulfobutyl ether derivatives of cyclomaltoheptaose (beta-cyclodextrin)

scientific article published on 01 April 1997

Isolation of endogenous modulators for the GABAA and taurine receptors

scientific article published on 01 November 1993

Kinetics and products of the acid-catalyzed ring-opening of atmospherically relevant butyl epoxy alcohols.

artículo científico publicado en 2010

Lewis Acid Enhancement of Proton Induced CO2 Cleavage: Bond Weakening and Ligand Residence Time Effects

artículo científico publicado en 2018

Lewis acid promoted titanium alkylidene formation: off-cycle intermediates relevant to olefin trimerization catalysis

artículo científico publicado en 2014

Modulating the Folding Landscape of Superoxide Dismutase 1 with Targeted Molecular Binders.

artículo científico publicado en 2018

New polyamide cryptand for anion binding.

artículo científico publicado en 2003

Nitrogen Insertion into a Corrole Ring: Iridium Monoazaporphyrins ⬇️

artículo científico publicado el 30 de agosto de 2011

Novel d-seco paclitaxel analogues: synthesis, biological evaluation, and model testing.

artículo científico publicado en 2001

Nucleoside triphosphate specificity of tubulin

artículo científico publicado en 2000

Optimum doses of deuterium oxide and sodium bromide for the determination of total body water and extracellular fluid ⬇️

artículo científico publicado el 1 de enero de 1991

Paclitaxel Analogues fromTaxus×mediacv. Hicksii

scientific article published on 01 February 1999

Poly(L-lysine) as a model drug macromolecule with which to investigate secondary structure and microporous membrane transport, part 2: diffusion studies

artículo científico publicado en 2002

Preparation and physicochemical characterization of a novel water-soluble prodrug of carbamazepine.

artículo científico publicado en 2010

Protonation of crotonyl-CoA dienolate by human glutaryl-CoA dehydrogenase occurs by solvent-derived protons.

artículo científico publicado en 2005

Reactivity of Metabolic Intermediates and Cofactor Stability under Model Early Earth Conditions

artículo científico publicado en 2020

Reactivity toward deamidation of asparagine residues in beta-turn structures.

artículo científico publicado en 2000

Redox and pH gradients drive amino acid synthesis in iron oxyhydroxide mineral systems

scientific article published on 25 February 2019

Regioselective Diels-Alder cycloadditions and other reactions of 4,5-, 5,6-, and 6,7-indole arynes.

artículo científico publicado en 2009

Secondary structure of a dynamic type I'beta-hairpin peptide.

artículo científico publicado en 2004

Site-specifically traced drug release and biodistribution of a paclitaxel-antibody conjugate toward improvement of the linker structure.

artículo científico publicado en 2004

Solution behavior of a novel type 1 interferon, interferon-tau.

artículo científico publicado en 2005

Stability of the thrombolytic protein fibrolase: effect of temperature and pH on activity and conformation

artículo científico publicado en 1991

Structure-activity studies of antitumor taxanes: synthesis of novel C-13 side chain homologated taxol and taxotere analogs

scientific article published on 01 September 1994

Synthesis and conformation of Gly-Gly dipeptides constrained with phenylalanine-like aminocaproic acid linkers

artículo científico publicado en 2000

Synthesis and conformational analysis of a coumarinic acid-based cyclic prodrug of an opioid peptide with modified sensitivity to esterase-catalyzed bioconversion.

artículo científico publicado en 2002

The dormancy-specific regulator, SutA, is intrinsically disordered and modulates transcription initiation in Pseudomonas aeruginosa

scientific article published on 10 July 2019

The effect of beta-turn structure on the passive diffusion of peptides across Caco-2 cell monolayers

scientific article published on 01 October 1997

The effect of conformation on membrane permeability of an acyloxyalkoxy-linked cyclic prodrug of a model hexapeptide

scientific article published on 01 November 1996

The effect of conformation on the membrane permeation of coumarinic acid- and phenylpropionic acid-based cyclic prodrugs of opioid peptides.

artículo científico publicado en 1999

The effect of the aromatic rings of taxol on biological activity and solution conformation: synthesis and evaluation of saturated taxol and taxotere analogues

scientific article published on 01 September 1994

The oxetane conformational lock of paclitaxel: structural analysis of D-secopaclitaxel.

artículo científico publicado en 1999

Total Synthesis and Characterization of 7-Hypoquinuclidonium Tetrafluoroborate and 7-Hypoquinuclidone BF3 Complex

artículo científico publicado en 2016

Total synthesis and evaluation of C25-benzyloxyepothilone C for tubulin assembly and cytotoxicity against MCF-7 breast cancer cells.

artículo científico publicado en 2008

Total synthesis and evaluation of C26-hydroxyepothilone D derivatives for photoaffinity labeling of beta-tubulin.

artículo científico publicado en 2010

Transport characteristics of peptides and peptidomimetics: II. Hydroxyethylamine bioisostere-containing peptidomimetics as substrates for the oligopeptide transporter and P-glycoprotein in the intestinal mucosa.

artículo científico publicado en 2001

Two-, three-, and four-dimensional nuclear magnetic resonance spectroscopy of protein pharmaceuticals.

artículo científico publicado en 1995

Lista de obras de D G Vander Velde

18Oxygen incorporation into inorganic phosphate in the reaction catalyzed by N5,10-methenyltetrahydrofolate synthetase

A 19F NMR study of lomefloxacin in human erythrocytes and its interaction with hemoglobin

A one-step synthesis of a deuterated paclitaxel analogue: 10-deacetoxy-(10alpha-2H)paclitaxel

A tandem Prins/Schmidt reaction approach to marine alkaloids: formal and total syntheses of lepadiformines A and C

Alternate substrates of human glutaryl-CoA dehydrogenase: structure and reactivity of substrates, and identification of a novel 2-enoyl-CoA product.

An Initial Event in the Insect Innate Immune Response: Structural and Biological Studies of Interactions between β-1,3-Glucan and the N-Terminal Domain of β-1,3-Glucan Recognition Protein

Biofilm-specific extracellular matrix proteins of nontypeable Haemophilus influenzae

CO Coupling Chemistry of a Terminal Mo Carbide: Sequential Addition of Proton, Hydride, and CO Releases Ethenone

Characterization and dynamics of substituted ruthenacyclobutanes relevant to the olefin cross-metathesis reaction

Characterization of the complexation of fluoroquinolone antimicrobials with metal ions by nuclear magnetic resonance spectroscopy

Comparative effects of (SBE)7m-beta-CD and HP-beta-CD on the stability of two anti-neoplastic agents, melphalan and carmustine

Comprehensive study of sansalvamide A derivatives and their structure-activity relationships against drug-resistant colon cancer cell lines.

Conformation of ATP and ADP bound to N10-formyltetrahydrofolate synthetase determined by TRNOE NMR spectroscopy.

Conformational analysis of the beta-amyloid peptide fragment, beta(12-28)

Conformational studies on resiniferatoxin (RTX), an ultrapotent vanilloid agonist

Conformationally restricted paclitaxel analogues: macrocyclic mimics of the "hydrophobic collapse" conformation

Cyclodextrin-catalyzed deacetylation of spironolactone is pH and cyclodextrin dependent

Deamidation of model beta-turn cyclic peptides in the solid state

Diastereomeric phosphonate ester adducts of chymotrypsin: 31P-NMR measurements

Effect of buffer species on the thermally induced aggregation of interferon-tau

Effect of conformation on the rate of deamidation of vancomycin in aqueous solutions

Effect of progressive benzyl substitution on the conformations of aminocaproic acid-cyclized dipeptides.

Effect of restricted conformational flexibility on the permeation of model hexapeptides across Caco-2 cell monolayers

Effect of stereochemistry on the transport of Aca-linked β-turn peptidomimetics across a human intestinal cell line ⬇️

Effect of zinc binding on the structure and stability of fibrolase, a fibrinolytic protein from snake venom

Effects of amino acid chirality and the chemical linker on the cell permeation characteristics of cyclic prodrugs of opioid peptides.

Evaluation of NMR diffusion measurements for the conformational analysis of flexible peptides.

Experimental and theoretical investigations into the unusual regioselectivity of 4,5-, 5,6-, and 6,7-indole aryne cycloadditions

Fibrolase. A fibrinolytic protein from snake venom.

Fluoride-facilitated deuterium exchange from DMSO-d6 to polyamide-based cryptands.

Get5 Carboxyl-terminal Domain Is a Novel Dimerization Motif That Tethers an Extended Get4/Get5 Complex

Highly regioirregular polypropylene from asymmetric group 4 anilide(pyridine)phenoxide complexes.

Hydrocotylosides I-VII, new oleanane saponins from hydrocotylesibthorpioides.

Hydrolysis of the prodrug, 2',3',5'-triacetyl-6-azauridine.

Improved preparation and structural conformation of the fluorescence labelling reagents 1,2-diamino-4,5-dimethoxybenzene and 3,4-dihydro-6,7-dimethoxy-4-methyl-3-oxo-quinoxaline-2-carbonyl chloride

Indole-derived arynes and their Diels-Alder reactivity with furans

Isolation and characterization by NMR spectroscopy of three monosubstituted 4-sulfobutyl ether derivatives of cyclomaltoheptaose (beta-cyclodextrin)

Isolation of endogenous modulators for the GABAA and taurine receptors

Kinetics and products of the acid-catalyzed ring-opening of atmospherically relevant butyl epoxy alcohols.

Lewis Acid Enhancement of Proton Induced CO2 Cleavage: Bond Weakening and Ligand Residence Time Effects

Lewis acid promoted titanium alkylidene formation: off-cycle intermediates relevant to olefin trimerization catalysis

Modulating the Folding Landscape of Superoxide Dismutase 1 with Targeted Molecular Binders.

New polyamide cryptand for anion binding.

Nitrogen Insertion into a Corrole Ring: Iridium Monoazaporphyrins ⬇️

Novel d-seco paclitaxel analogues: synthesis, biological evaluation, and model testing.

Nucleoside triphosphate specificity of tubulin

Optimum doses of deuterium oxide and sodium bromide for the determination of total body water and extracellular fluid ⬇️

Paclitaxel Analogues fromTaxus×mediacv. Hicksii

Poly(L-lysine) as a model drug macromolecule with which to investigate secondary structure and microporous membrane transport, part 2: diffusion studies

Preparation and physicochemical characterization of a novel water-soluble prodrug of carbamazepine.

Protonation of crotonyl-CoA dienolate by human glutaryl-CoA dehydrogenase occurs by solvent-derived protons.

Reactivity of Metabolic Intermediates and Cofactor Stability under Model Early Earth Conditions

Reactivity toward deamidation of asparagine residues in beta-turn structures.

Redox and pH gradients drive amino acid synthesis in iron oxyhydroxide mineral systems

Regioselective Diels-Alder cycloadditions and other reactions of 4,5-, 5,6-, and 6,7-indole arynes.

Secondary structure of a dynamic type I'beta-hairpin peptide.

Site-specifically traced drug release and biodistribution of a paclitaxel-antibody conjugate toward improvement of the linker structure.

Solution behavior of a novel type 1 interferon, interferon-tau.

Stability of the thrombolytic protein fibrolase: effect of temperature and pH on activity and conformation

Structure-activity studies of antitumor taxanes: synthesis of novel C-13 side chain homologated taxol and taxotere analogs

Synthesis and conformation of Gly-Gly dipeptides constrained with phenylalanine-like aminocaproic acid linkers

Synthesis and conformational analysis of a coumarinic acid-based cyclic prodrug of an opioid peptide with modified sensitivity to esterase-catalyzed bioconversion.

The dormancy-specific regulator, SutA, is intrinsically disordered and modulates transcription initiation in Pseudomonas aeruginosa

The effect of beta-turn structure on the passive diffusion of peptides across Caco-2 cell monolayers

The effect of conformation on membrane permeability of an acyloxyalkoxy-linked cyclic prodrug of a model hexapeptide

The effect of conformation on the membrane permeation of coumarinic acid- and phenylpropionic acid-based cyclic prodrugs of opioid peptides.

The effect of the aromatic rings of taxol on biological activity and solution conformation: synthesis and evaluation of saturated taxol and taxotere analogues

The oxetane conformational lock of paclitaxel: structural analysis of D-secopaclitaxel.

Total Synthesis and Characterization of 7-Hypoquinuclidonium Tetrafluoroborate and 7-Hypoquinuclidone BF3 Complex

Total synthesis and evaluation of C25-benzyloxyepothilone C for tubulin assembly and cytotoxicity against MCF-7 breast cancer cells.

Total synthesis and evaluation of C26-hydroxyepothilone D derivatives for photoaffinity labeling of beta-tubulin.

Transport characteristics of peptides and peptidomimetics: II. Hydroxyethylamine bioisostere-containing peptidomimetics as substrates for the oligopeptide transporter and P-glycoprotein in the intestinal mucosa.

Two-, three-, and four-dimensional nuclear magnetic resonance spectroscopy of protein pharmaceuticals.