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Lista de obras de Ryo Yazaki

Amino Acid Schiff Base Bearing Benzophenone Imine As a Platform for Highly Congested Unnatural α-Amino Acid Synthesis

artículo científico publicado en 2020

An Expeditious Route to trans-Configured Tetrahydrothiophenes Enabled by Fe(OTf)3 -Catalyzed [3+2] Cycloaddition of Donor-Acceptor Cyclopropanes with Thionoesters

artículo científico publicado en 2018

Asymmetric synthesis of isothiazoles through Cu catalysis: direct catalytic asymmetric conjugate addition of allyl cyanide to α,β-unsaturated thioamides

artículo científico publicado en 2011

Catalytic Aerobic Chemoselective α-Oxidation of Acylpyrazoles en Route to α-Hydroxy Acid Derivatives.

artículo científico publicado en 2017

Catalytic Aerobic Cross-Dehydrogenative Coupling of Azlactones en Route to α,α-Disubstituted α-Amino Acids

artículo científico publicado en 2020

Catalytic Chemoselective Conjugate Addition of Amino Alcohols to α,β-Unsaturated Ester: Hydroxy Group over Amino Group and Conjugate Addition over Transesterification

artículo científico publicado en 2017

Chemo- and Regioselective Direct Functional Group Installation through Catalytic Hydroxy Group Selective Conjugate Addition of Amino Alcohols to α,β-Unsaturated Sulfonyl Compounds

artículo científico publicado en 2016

Chemoselective Catalytic α-Oxidation of Carboxylic Acids: Iron/Alkali Metal Cooperative Redox Active Catalysis

artículo científico publicado en 2020

Chemoselective catalytic conjugate addition of alcohols over amines

artículo científico publicado en 2014

Concise enantioselective synthesis of duloxetine via direct catalytic asymmetric aldol reaction of thioamide.

artículo científico publicado en 2012

Cooperative activation of alkyne and thioamide functionalities; direct catalytic asymmetric conjugate addition of terminal alkynes to α,β-unsaturated thioamides.

artículo científico publicado en 2011

Direct Catalytic Chemoselective α-Amination of Acylpyrazoles: A Concise Route to Unnatural α-Amino Acid Derivatives

artículo científico publicado en 2016

Direct catalytic asymmetric Mannich-type reaction of thioamides.

artículo científico publicado en 2009

Direct catalytic asymmetric addition of allyl cyanide to ketones.

artículo científico publicado en 2009

Direct catalytic asymmetric addition of allylic cyanides to ketoimines.

artículo científico publicado en 2008

Direct catalytic asymmetric aldol reactions of thioamides: toward a stereocontrolled synthesis of 1,3-polyols.

artículo científico publicado en 2009

Direct catalytic asymmetric alkynylation of ketoimines

scientific article published on 18 January 2013

Direct catalytic asymmetric conjugate addition of terminal alkynes to alpha,beta-unsaturated thioamides.

artículo científico publicado en 2010

Direct catalytic asymmetric intramolecular conjugate addition of thioamide to α,β-unsaturated esters

artículo científico publicado en 2011

Direct catalytic enantio- and diastereoselective aldol reaction of thioamides

artículo científico publicado en 2011

Enantioselective synthesis of a GPR40 agonist AMG 837 via catalytic asymmetric conjugate addition of terminal alkyne to α,β-unsaturated thioamide

scientific article published on 03 February 2011

Growth Suppression of Human Colorectal Cancer Cells with Mutated KRAS by 3-Deaza-cytarabine in 3D Floating Culture

artículo científico publicado en 2018

Intermediate as catalyst: catalytic asymmetric conjugate addition of nitroalkanes to α,β-unsaturated thioamides

artículo científico publicado en 2011

Oxetanyl peptides: novel peptidomimetic modules for medicinal chemistry

artículo científico publicado en 2014

Strategy for Catalytic Chemoselective Cross-Enolate Coupling Reaction via a Transient Homocoupling Dimer

scientific article published on 31 May 2018

Toward the total synthesis of onchidin, a cytotoxic cyclic depsipeptide from a mollusc

scientific article published on 01 January 2007

μ-Oxo-Dinuclear-Iron(III)-Catalyzed O-Selective Acylation of Aliphatic and Aromatic Amino Alcohols and Transesterification of Tertiary Alcohols.

artículo científico publicado en 2016