Lista de obras - Steven Verhelst - Dominio Público Uruguay

4-Bromophenacyl bromide specifically inhibits rhoptry secretion during Toxoplasma invasion

artículo científico publicado en 2009

A General Solid Phase Method for the Preparation of Diverse Azapeptide Probes Directed Against Cysteine Proteases

artículo científico publicado en 2005

A Mild Chemically Cleavable Linker System for Functional Proteomic Applications

scientific article published on 01 January 2007

A Substrate-Inspired Probe Monitors Translocation, Activation, and Subcellular Targeting of Bacterial Type III Effector Protease AvrPphB

artículo científico publicado en 2013

A selective activity-based probe for the papain family cysteine protease dipeptidyl peptidase I/cathepsin C.

artículo científico publicado en 2006

A simple and effective cleavable linker for chemical proteomics applications

artículo científico publicado en 2012

A stereoselective route towards highly functionalized 4,6-diaminocyclohexene derivatives

ATP13A3 is a major component of the enigmatic mammalian polyamine transport system

artículo científico publicado en 2020

Activity-Based Protein Profiling of Rhomboid Proteases in Liposomes

artículo científico publicado en 2015

Activity-Based Protein Profiling of Serine Proteases in Immune Cells

artículo científico publicado en 2020

Activity-based probes for rhomboid proteases discovered in a mass spectrometry-based assay

artículo científico publicado en 2013

Activity-based probes for the study of proteases: recent advances and developments.

artículo científico publicado en 2012

Alkyne derivatives of isocoumarins as clickable activity-based probes for serine proteases.

artículo científico publicado en 2011

Bioorthogonal Reactions in Activity-Based Protein Profiling

artículo científico publicado en 2020

Chemical Tools for the Study of Intramembrane Proteases

artículo científico

Cleavable trifunctional biotin reagents for protein labelling, capture and release.

artículo científico publicado en 2013

Clickable polyamine derivatives as chemical probes for the polyamine transport system

artículo científico publicado en 2018

Comparative analysis of click chemistry mediated activity-based protein profiling in cell lysates.

artículo científico publicado en 2013

Design and synthesis of a protein:Farnesyltransferase inhibitor based on sugar amino acids

article by Herman S Overkleeft et al published May 1999 in Tetrahedron Letters

Detection of protease activity in cells and animals.

artículo científico

Development of calpain-specific inactivators by screening of positional scanning epoxide libraries

artículo científico publicado en 2007

Discovery of Cellular Roles of Intramembrane Proteases

artículo científico publicado en 2019

Inhibitor Fingerprinting of Rhomboid Proteases by Activity-Based Protein Profiling Reveals Inhibitor Selectivity and Rhomboid Autoprocessing

artículo científico publicado en 2015

Inhibitors of rhomboid proteases

artículo científico

Kinase Photoaffinity Labeling Reveals Low Selectivity Profile of the IRE1 Targeting Imidazopyrazine-Based KIRA6 Inhibitor

scientific article published on 08 December 2020

Minitags for small molecules: detecting targets of reactive small molecules in living plant tissues using 'click chemistry'.

artículo científico publicado en 2008

Mixed alkyl aryl phosphonate esters as quenched fluorescent activity-based probes for serine proteases

artículo científico publicado en 2015

Probing Functional Tyrosines ⬇️

artículo científico publicado el 18 de abril de 2013

Protease Specificity Profiling in a Pipet Tip Using "Charge-Synchronized" Proteome-Derived Peptide Libraries.

artículo científico publicado en 2018

Role for cathepsin F in invariant chain processing and major histocompatibility complex class II peptide loading by macrophages

artículo científico publicado en 2000

Short Peptides with Uncleavable Peptide Bond Mimetics as Photoactivatable Caspase-3 Inhibitors

artículo científico publicado en 2019

Solid-phase methods for the preparation of epoxysuccinate-based inhibitors of cysteine proteases.

artículo científico publicado en 2006

Solid-phase synthesis of double-headed epoxysuccinyl activity-based probes for selective targeting of papain family cysteine proteases.

artículo científico publicado en 2005

Specificity of aza-peptide electrophile activity-based probes of caspases

artículo científico publicado en 2006

Stress-induced inflammation evoked by immunogenic cell death is blunted by the IRE1α kinase inhibitor KIRA6 through HSP60 targeting

artículo científico publicado en 2021

Surface plasmon resonance evaluation of various aminoglycoside-RNA hairpin interactions reveals low degree of selectivity.

artículo científico publicado en 2004

Synthesis of orthogonally protected 2-deoxystreptamine stereoisomers

Tagging and detection strategies for activity-based proteomics.

artículo científico publicado en 2006

Target profiling of 4-hydroxyderricin in S. aureus reveals seryl-tRNA synthetase binding and inhibition by covalent modification.

artículo científico publicado en 2013

The structural basis for catalysis and substrate specificity of a rhomboid protease

artículo científico publicado en 2010

Tuning activity-based probe selectivity for serine proteases by on-resin 'click' construction of peptide diphenyl phosphonates.

artículo científico publicado en 2013

Tuning probe selectivity for chemical proteomics applications ⬇️

artículo científico publicado el 28 de diciembre de 2012

Lista de obras de Steven Verhelst

4-Bromophenacyl bromide specifically inhibits rhoptry secretion during Toxoplasma invasion

A General Solid Phase Method for the Preparation of Diverse Azapeptide Probes Directed Against Cysteine Proteases

A Mild Chemically Cleavable Linker System for Functional Proteomic Applications

A Substrate-Inspired Probe Monitors Translocation, Activation, and Subcellular Targeting of Bacterial Type III Effector Protease AvrPphB

A selective activity-based probe for the papain family cysteine protease dipeptidyl peptidase I/cathepsin C.

A simple and effective cleavable linker for chemical proteomics applications

A stereoselective route towards highly functionalized 4,6-diaminocyclohexene derivatives

ATP13A3 is a major component of the enigmatic mammalian polyamine transport system

Activity-Based Protein Profiling of Rhomboid Proteases in Liposomes

Activity-Based Protein Profiling of Serine Proteases in Immune Cells

Activity-based probes for rhomboid proteases discovered in a mass spectrometry-based assay

Activity-based probes for the study of proteases: recent advances and developments.

Alkyne derivatives of isocoumarins as clickable activity-based probes for serine proteases.

Bioorthogonal Reactions in Activity-Based Protein Profiling

Chemical Tools for the Study of Intramembrane Proteases

Cleavable trifunctional biotin reagents for protein labelling, capture and release.

Clickable polyamine derivatives as chemical probes for the polyamine transport system

Comparative analysis of click chemistry mediated activity-based protein profiling in cell lysates.

Design and synthesis of a protein:Farnesyltransferase inhibitor based on sugar amino acids

Detection of protease activity in cells and animals.

Development of calpain-specific inactivators by screening of positional scanning epoxide libraries

Discovery of Cellular Roles of Intramembrane Proteases

Inhibitor Fingerprinting of Rhomboid Proteases by Activity-Based Protein Profiling Reveals Inhibitor Selectivity and Rhomboid Autoprocessing

Inhibitors of rhomboid proteases

Kinase Photoaffinity Labeling Reveals Low Selectivity Profile of the IRE1 Targeting Imidazopyrazine-Based KIRA6 Inhibitor

Minitags for small molecules: detecting targets of reactive small molecules in living plant tissues using 'click chemistry'.

Mixed alkyl aryl phosphonate esters as quenched fluorescent activity-based probes for serine proteases

Probing Functional Tyrosines ⬇️

Protease Specificity Profiling in a Pipet Tip Using "Charge-Synchronized" Proteome-Derived Peptide Libraries.

Role for cathepsin F in invariant chain processing and major histocompatibility complex class II peptide loading by macrophages

Short Peptides with Uncleavable Peptide Bond Mimetics as Photoactivatable Caspase-3 Inhibitors

Solid-phase methods for the preparation of epoxysuccinate-based inhibitors of cysteine proteases.

Solid-phase synthesis of double-headed epoxysuccinyl activity-based probes for selective targeting of papain family cysteine proteases.

Specificity of aza-peptide electrophile activity-based probes of caspases

Stress-induced inflammation evoked by immunogenic cell death is blunted by the IRE1α kinase inhibitor KIRA6 through HSP60 targeting

Surface plasmon resonance evaluation of various aminoglycoside-RNA hairpin interactions reveals low degree of selectivity.

Synthesis of orthogonally protected 2-deoxystreptamine stereoisomers

Tagging and detection strategies for activity-based proteomics.

Target profiling of 4-hydroxyderricin in S. aureus reveals seryl-tRNA synthetase binding and inhibition by covalent modification.

The structural basis for catalysis and substrate specificity of a rhomboid protease

Tuning activity-based probe selectivity for serine proteases by on-resin 'click' construction of peptide diphenyl phosphonates.

Tuning probe selectivity for chemical proteomics applications ⬇️