Lista de obras - Valentina Onnis - Dominio Público Uruguay

2-(Arylamino)-6-(trifluoromethyl)nicotinic Acid Derivatives: New HIV-1 RT Dual Inhibitors Active on Viral Replication

scientific article published on 15 March 2020

A new convenient synthetic method and preliminary pharmacological characterization of triazinediones as prokineticin receptor antagonists

artículo científico publicado en 2014

Benzofuran hydrazones as potential scaffold in the development of multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity

artículo científico publicado en 2018

Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors

artículo científico publicado en 2019

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment

scientific article published on 14 October 2020

Design, Synthesis and Evaluation of Antiproliferative Activity of New Benzimidazolehydrazones.

artículo científico publicado en 2016

Design, synthesis and <i>in vitro</i> and <i>in vivo</i> biological evaluation of flurbiprofen amides as new fatty acid amide hydrolase/cyclooxygenase-2 dual inhibitory potential analgesic agents

artículo científico publicado en 2021

Discovery of thiazolin-4-one-based aromatic sulfamates as a new class of carbonic anhydrase isoforms I, II, IV, and IX inhibitors.

artículo científico publicado en 2018

Effect of lysine at C-terminus of the Dmt-Tic opioid pharmacophore.

artículo científico publicado en 2006

Effect of the T-type channel blocker KYS-05090S in mouse models of acute and neuropathic pain

artículo científico publicado en 2015

Exploring the fatty acid amide hydrolase and cyclooxygenase inhibitory properties of novel amide derivatives of ibuprofen

artículo científico publicado en 2020

Flavones and structurally related 4-chromenones inhibit carbonic anhydrases by a different mechanism of action compared to coumarins

scientific article published on 27 March 2012

Further studies on the effect of lysine at the C-terminus of the Dmt-Tic opioid pharmacophore.

artículo científico publicado en 2007

In vitro antimycobacterial activity of newly synthesised S-alkylisothiosemicarbazone derivatives and synergistic interactions in combination with rifamycins against Mycobacterium avium.

artículo científico publicado en 2005

Indole derivatives as multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity of indole hydrazones

scientific article published on 10 February 2019

Inhibition of fatty acid amide hydrolase and cyclooxygenase by the N-(3-methylpyridin-2-yl)amide derivatives of flurbiprofen and naproxen

artículo científico publicado en 2013

Inhibitory effect of positively charged triazine antagonists of prokineticin receptors on the transient receptor vanilloid type-1 (TRPV1) channel.

artículo científico publicado en 2015

Inhibitory properties of ibuprofen and its amide analogues towards the hydrolysis and cyclooxygenation of the endocannabinoid anandamide.

artículo científico publicado en 2012

Interaction of the N-(3-Methylpyridin-2-yl)amide Derivatives of Flurbiprofen and Ibuprofen with FAAH: Enantiomeric Selectivity and Binding Mode

artículo científico publicado en 2015

Nematicidal activity of acetophenones and chalcones against Meloidogyne incognita and structure-activity considerations

artículo científico publicado en 2015

Novel propanamides as fatty acid amide hydrolase inhibitors.

artículo científico publicado en 2017

PPARγ controls pregnancy outcome through activation of EG-VEGF: new insights into the mechanism of placental development

artículo científico publicado en 2015

Synthesis and Biological Evaluation of 2-Substituted Benzyl-/Phenylethylamino-4-amino-5-aroylthiazoles as Apoptosis-Inducing Anticancer Agents

scientific article published on 06 May 2020

Synthesis and antimycobacterial activity of new S-alkylisothiosemicarbazone derivatives.

artículo científico publicado en 2002

Synthesis and antiproliferative activity of 2,6-dibenzylamino-3,5-dicyanopyridines on human cancer cell lines.

artículo científico publicado en 2005

Synthesis and antitumor evaluation of 6-thioxo-, 6-oxo- and 2,4-dioxopyrimidine derivatives.

artículo científico publicado en 2001

Synthesis and biological evaluation of novel acylhydrazone derivatives as potential antitumor agents

artículo científico publicado en 2013

Synthesis and biological evaluation of novel pyrazoline-based aromatic sulfamates with potent carbonic anhydrase isoforms II, IV and IX inhibitory efficacy.

artículo científico publicado en 2018

Synthesis and carbonic anhydrase I, II, IX and XII inhibition studies of 4-N,N-disubstituted sulfanilamides incorporating 4,4,4-trifluoro-3-oxo-but-1-enyl, phenacylthiourea and imidazol-2(3H)-one/thione moieties

artículo científico publicado en 2014

Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties

artículo científico publicado en 2015

Synthesis and evaluation of anticancer activity of 2-arylamino-6-trifluoromethyl-3-(hydrazonocarbonyl)pyridines.

artículo científico publicado en 2009

Synthesis and evaluation of antitumoral activity of ester and amide derivatives of 2-arylamino-6-trifluoromethyl-3-pyridinecarboxylic acids.

artículo científico publicado en 2007

Synthesis and evaluation of paracetamol esters as novel fatty acid amide hydrolase inhibitors.

artículo científico publicado en 2010

Synthesis and in vitro antitumor activity of new 4,5-dihydropyrazole derivatives.

artículo científico publicado en 2010

Synthesis and in vitro antitumoral activity of new 3,5-dicyanopyridine derivatives.

artículo científico publicado en 2006

Synthesis and in vitro antitumoral activity of new N-phenyl-3-pyrrolecarbothioamides.

artículo científico publicado en 2003

Synthesis of new 2-arylamino-6-trifluoromethylpyridine-3-carboxylic acid derivatives and investigation of their analgesic activity

artículo científico publicado en 2004

Synthesis of new N-(2-(trifluoromethyl)pyridin-4-yl)anthranilic acid derivatives and their evaluation as anticancer agents.

artículo científico publicado en 2004

Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity

artículo científico publicado en 2015

Synthesis, characterisation and insulin-mimetic activity of oxovanadium(IV) complexes with amidrazone derivatives

scientific article published on 05 August 2006

Synthetic Flavonoids, Aminoisoflavones: Interaction and Reactivity with Metal-Free and Metal-Associated Amyloid-β Species

artículo científico publicado en 2014

TRPV1 modulators: Synthesis and in vitro evaluation of 1-heteroaryl piperidinecarboxamide and piperazinylurea derivatives

artículo científico publicado en 2015

Lista de obras de Valentina Onnis

2-(Arylamino)-6-(trifluoromethyl)nicotinic Acid Derivatives: New HIV-1 RT Dual Inhibitors Active on Viral Replication

A new convenient synthetic method and preliminary pharmacological characterization of triazinediones as prokineticin receptor antagonists

Benzofuran hydrazones as potential scaffold in the development of multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity

Benzylamides and piperazinoarylamides of ibuprofen as fatty acid amide hydrolase inhibitors

Carbonic Anhydrase Inhibitors Targeting Metabolism and Tumor Microenvironment

Design, Synthesis and Evaluation of Antiproliferative Activity of New Benzimidazolehydrazones.

Design, synthesis and <i>in vitro</i> and <i>in vivo</i> biological evaluation of flurbiprofen amides as new fatty acid amide hydrolase/cyclooxygenase-2 dual inhibitory potential analgesic agents

Discovery of thiazolin-4-one-based aromatic sulfamates as a new class of carbonic anhydrase isoforms I, II, IV, and IX inhibitors.

Effect of lysine at C-terminus of the Dmt-Tic opioid pharmacophore.

Effect of the T-type channel blocker KYS-05090S in mouse models of acute and neuropathic pain

Exploring the fatty acid amide hydrolase and cyclooxygenase inhibitory properties of novel amide derivatives of ibuprofen

Flavones and structurally related 4-chromenones inhibit carbonic anhydrases by a different mechanism of action compared to coumarins

Further studies on the effect of lysine at the C-terminus of the Dmt-Tic opioid pharmacophore.

In vitro antimycobacterial activity of newly synthesised S-alkylisothiosemicarbazone derivatives and synergistic interactions in combination with rifamycins against Mycobacterium avium.

Indole derivatives as multifunctional drugs: Synthesis and evaluation of antioxidant, photoprotective and antiproliferative activity of indole hydrazones

Inhibition of fatty acid amide hydrolase and cyclooxygenase by the N-(3-methylpyridin-2-yl)amide derivatives of flurbiprofen and naproxen

Inhibitory effect of positively charged triazine antagonists of prokineticin receptors on the transient receptor vanilloid type-1 (TRPV1) channel.

Inhibitory properties of ibuprofen and its amide analogues towards the hydrolysis and cyclooxygenation of the endocannabinoid anandamide.

Interaction of the N-(3-Methylpyridin-2-yl)amide Derivatives of Flurbiprofen and Ibuprofen with FAAH: Enantiomeric Selectivity and Binding Mode

Nematicidal activity of acetophenones and chalcones against Meloidogyne incognita and structure-activity considerations

Novel propanamides as fatty acid amide hydrolase inhibitors.

PPARγ controls pregnancy outcome through activation of EG-VEGF: new insights into the mechanism of placental development

Synthesis and Biological Evaluation of 2-Substituted Benzyl-/Phenylethylamino-4-amino-5-aroylthiazoles as Apoptosis-Inducing Anticancer Agents

Synthesis and antimycobacterial activity of new S-alkylisothiosemicarbazone derivatives.

Synthesis and antiproliferative activity of 2,6-dibenzylamino-3,5-dicyanopyridines on human cancer cell lines.

Synthesis and antitumor evaluation of 6-thioxo-, 6-oxo- and 2,4-dioxopyrimidine derivatives.

Synthesis and biological evaluation of novel acylhydrazone derivatives as potential antitumor agents

Synthesis and biological evaluation of novel pyrazoline-based aromatic sulfamates with potent carbonic anhydrase isoforms II, IV and IX inhibitory efficacy.

Synthesis and carbonic anhydrase I, II, IX and XII inhibition studies of 4-N,N-disubstituted sulfanilamides incorporating 4,4,4-trifluoro-3-oxo-but-1-enyl, phenacylthiourea and imidazol-2(3H)-one/thione moieties

Synthesis and carbonic anhydrase I, II, IX and XII inhibitory activity of sulfamates incorporating piperazinyl-ureido moieties

Synthesis and evaluation of anticancer activity of 2-arylamino-6-trifluoromethyl-3-(hydrazonocarbonyl)pyridines.

Synthesis and evaluation of antitumoral activity of ester and amide derivatives of 2-arylamino-6-trifluoromethyl-3-pyridinecarboxylic acids.

Synthesis and evaluation of paracetamol esters as novel fatty acid amide hydrolase inhibitors.

Synthesis and in vitro antitumor activity of new 4,5-dihydropyrazole derivatives.

Synthesis and in vitro antitumoral activity of new 3,5-dicyanopyridine derivatives.

Synthesis and in vitro antitumoral activity of new N-phenyl-3-pyrrolecarbothioamides.

Synthesis of new 2-arylamino-6-trifluoromethylpyridine-3-carboxylic acid derivatives and investigation of their analgesic activity

Synthesis of new N-(2-(trifluoromethyl)pyridin-4-yl)anthranilic acid derivatives and their evaluation as anticancer agents.

Synthesis of sulfonamides incorporating piperazinyl-ureido moieties and their carbonic anhydrase I, II, IX and XII inhibitory activity

Synthesis, characterisation and insulin-mimetic activity of oxovanadium(IV) complexes with amidrazone derivatives

Synthetic Flavonoids, Aminoisoflavones: Interaction and Reactivity with Metal-Free and Metal-Associated Amyloid-β Species

TRPV1 modulators: Synthesis and in vitro evaluation of 1-heteroaryl piperidinecarboxamide and piperazinylurea derivatives