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Lista de obras de Christer Halldin

(18)F-MCL-524, an (18)F-Labeled Dopamine D2 and D3 Receptor Agonist Sensitive to Dopamine: A Preliminary PET Study

artículo científico publicado en 2014

(S)- and (R)-[11C]nicotine and the metabolite (R/S)-[11C]cotinine. Preparation, metabolite studies and in vivo distribution in the human brain using PET

artículo científico publicado el 1 de noviembre de 1992

11C- and 76Br-labelled NNC 22-0010, selective dopamine D1 receptor radioligands for PET.

artículo científico publicado en 1996

11C-Methionine Kinetics in Pregnant Rhesus Monkeys Studied by Positron Emission Tomography: A New Approach to Feto-Maternal Metabolism ⬇️

artículo científico publicado el 1 de enero de 1984

11C-SCH 39166, a selective ligand for visualization of dopamine-D1 receptor binding in the monkey brain using PET ⬇️

artículo científico publicado el 1 de enero de 1991

11C-labelling of Ro 15-1788 in two different positions, and also 11C-labelling of its main metabolite Ro 15-3890, for PET studies of benzodiazepine receptors

artículo científico publicado en 1988

11C-labelling of dimethylphenethylamine in two different positions and biodistribution studies

artículo científico publicado en 1989

11CRo 15-4513, a ligand for visualization of benzodiazepine receptor binding. Preparation, autoradiography and positron emission tomography

artículo científico publicado el 1 de enero de 1992

125Iβ-CIT-FE and 125Iβ-CIT-FP are superior to 125Iβ-CIT for dopamine transporter visualization: Autoradiographic evaluation in the human brain ⬇️

artículo científico publicado el 1 de octubre de 1997

18Fβ-CIT-FP is superior to 11Cβ-CIT-FP for quantitation of the dopamine transporter ⬇️

artículo científico publicado el 1 de octubre de 1997

5-HT(1A) receptor and 5-HTT binding during the menstrual cycle in healthy women examined with [(11)C] WAY100635 and [(11)C] MADAM PET.

artículo científico publicado en 2009

5-HT1B receptor imaging and cognition: a positron emission tomography study in control subjects and Parkinson's disease patients

artículo científico

5-HT2 and D2 dopamine receptor occupancy in the living human brain. A PET study with risperidone

artículo científico publicado en 1993

5-HTT and 5-HT(1A) receptor occupancy of the novel substance vortioxetine (Lu AA21004). A PET study in control subjects

artículo científico publicado en 2013

76Br-beta-CBT, a PET tracer for investigating dopamine neuronal uptake

artículo científico publicado en 1995

A Comparative PET-study of five carbon-11 or fluorine-18 labelled salicylamides. Preparation and in vitro dopamine D-2 receptor binding ⬇️

artículo científico publicado el 1 de enero de 1991

A Nonhuman Primate PET Study: Measurement of Brain PDE4 Occupancy by Roflumilast Using (R)-[11C]Rolipram

artículo científico publicado en 2018

A PET study comparing receptor occupancy by five selective cannabinoid 1 receptor antagonists in non-human primates

artículo científico publicado en 2015

A PET study of

artículo científico publicado en 2000

A PET study of 5-HT1A receptors at different phases of the menstrual cycle in women with premenstrual dysphoria

artículo científico publicado en 2006

A PET study of 5-HT2 and D2 dopamine receptor occupancy induced by olanzapine in healthy subjects

scientific article published on 01 January 1997

A PET study of D(1)-like dopamine receptor ligand binding during altered endogenous dopamine levels in the primate brain

artículo científico publicado en 1999

A PET study of D2 and 5-HT2 receptor occupancy induced by risperidone in poor metabolizers of debrisoquin and risperidone

artículo científico publicado en 1995

A PET study of D2 dopamine receptor density at different phases of the menstrual cycle

artículo científico publicado en 1998

A PET study on regional coexpression of 5-HT1A receptors and 5-HTT in the human brain

artículo científico publicado en 2007

A PET study with [11C]AZ10419369 to determine brain 5-HT1B receptor occupancy of zolmitriptan in healthy male volunteers

artículo científico publicado en 2013

A PET-study of [ 11 C]FLB 457 binding to extrastriatal D 2 -dopamine receptors in healthy subjects and antipsychotic drug-treated patients ⬇️

artículo científico publicado el 1 de octubre de 1997

A comparative autoradiography study in post mortem whole hemisphere human brain slices taken from Alzheimer patients and age-matched controls using two radiolabelled DAA1106 analogues with high affinity to the peripheral benzodiazepine receptor (PBR

artículo científico publicado en 2008

A comparison of recent parametric neuroreceptor mapping approaches based on measurements with the high affinity PET radioligands [11C]FLB 457 and [11C]WAY 100635.

artículo científico publicado en 2006

A cross-validation study on the relationship between central D2 receptor occupancy and serum perphenazine concentration

artículo científico publicado en 2004

A direct comparison of the brain uptake and plasma clearance of N-[11C]methylspiroperidol and [18F]N-methylspiroperidol in baboon using PET.

artículo científico publicado en 1986

A fully automated one-pot synthesis of [carbonyl-11C]WAY-100635 for clinical PET applications

artículo científico publicado en 2008

A human [(11)C]T-773 PET study of PDE10A binding after oral administration of TAK-063, a PDE10A inhibitor

artículo científico publicado en 2016

A novel electrophilic synthesis and evaluation of medium specific radioactivity (1R,2S)-4-[18F]fluorometaraminol, a tracer for the assessment of cardiac sympathetic nerve integrity with PET.

artículo científico publicado en 2004

A positron emission tomography study in healthy volunteers to estimate mGluR5 receptor occupancy of AZD2066 - estimating occupancy in the absence of a reference region

artículo científico publicado en 2013

A preliminary PET evaluation of the new dopamine D2 receptor agonist [11C]MNPA in cynomolgus monkey

artículo científico publicado en 2005

A radiometabolite study of the serotonin transporter PET radioligand [(11)C]MADAM.

artículo científico publicado en 2014

A simplified radiometabolite analysis procedure for PET radioligands using a solid phase extraction with micellar medium

artículo científico publicado en 2013

ABC transporter-dependent brain uptake of the 5-HT1B receptor radioligand [ (11)C]AZ10419369: a comparative PET study in mouse, rat, and guinea pig

artículo científico publicado en 2014

AZD5213: a novel histamine H3 receptor antagonist permitting high daytime and low nocturnal H3 receptor occupancy, a PET study in human subjects

artículo científico publicado en 2012

Activation of glucocorticoid receptors increases 5-HT2A receptor levels

artículo científico publicado en 2009

Advancement in PET quantification using 3D-OP-OSEM point spread function reconstruction with the HRRT.

artículo científico publicado en 2009

Age and disease related changes in the translocator protein (TSPO) system in the human brain: positron emission tomography measurements with [11C]vinpocetine

artículo científico publicado en 2011

Age-related cognitive deficits mediated by changes in the striatal dopamine system.

artículo científico publicado en 2000

Age-related diurnal effect on D2 receptor binding: a preliminary PET study

artículo científico publicado en 2008

Age-related reduction in dopamine D1 receptors in the human brain: from late childhood to adulthood, a positron emission tomography study

artículo científico publicado en 2010

Amphetamine decreases α2C-adrenoceptor binding of [11C]ORM-13070: a PET study in the primate brain

artículo científico publicado en 2014

Amyloid binding properties of curcumin analogues in Alzheimer's disease postmortem brain tissue

artículo científico publicado en 2016

An HPLC-method for determination of ligand metabolism during PET studies with [11C]metaraminol and [11C]norepinephrine

artículo científico publicado en 1995

Application of cross-species PET imaging to assess neurotransmitter release in brain

artículo científico publicado en 2015

Approaches to quantify radioligands that wash out slowly from target organs

artículo científico publicado en 2010

Arrestin3 mediates D(2) dopamine receptor internalization

scientific article published on July 2009

Arterial input function derived from pairwise correlations between PET-image voxels

artículo científico publicado en 2013

Association between striatal and extrastriatal dopamine D2-receptor binding and social desirability

artículo científico publicado en 2009

Associations between cognition and serotonin receptor 1B binding in patients with major depressive disorder - A pilot study

artículo científico publicado en 2017

Associations between dopamine D2-receptor binding and cognitive performance indicate functional compartmentalization of the human striatum

artículo científico publicado en 2008

Atomoxetine occupies the norepinephrine transporter in a dose-dependent fashion: a PET study in nonhuman primate brain using (S,S)-[18F]FMeNER-D2.

artículo científico publicado en 2006

Attempts to visualize nicotinic receptors in the brain of monkey and man by positron emission tomography

artículo científico publicado en 1989

Autoradiographic Comparison of [125I]Epidepride and [125I]NCQ 298 Binding to Human Brain Extrastriated Dopamine Receptors ⬇️

artículo científico publicado el 1 de julio de 1997

Autoradiographic distribution of serotonin transporters and receptor subtypes in human brain

artículo científico publicado en 2004

Autoradiographic evaluation of [11C]vinpocetine binding in the human postmortem brain

artículo científico publicado en 2002

Autoradiographic localisation of D3-dopamine receptors in the human brain using the selective D3-dopamine receptor agonist (+)-[3H]PD 128907.

artículo científico publicado en 1996

Autoradiographic localization of 5-HT(2A) receptors in the human brain using [(3)H]M100907 and [(11)C]M100907.

artículo científico publicado en 2000

Autoradiographic localization of 5-HT1A receptors in the post-mortem human brain using [3H]WAY-100635 and [11C]way-100635

scientific article published on 01 January 1997

Autoradiographic localization of extrastriatal D2-dopamine receptors in the human brain using [125I]epidepride

scientific article published on 01 June 1996

Autoradiography and saturation experiments with 11C-RO 15-1788 binding to human brain

artículo científico publicado el 1 de enero de 1991

Autoradiography with saturation experiments of 11C-Ro 15-1788 binding to human brain sections

scientific article published on 01 January 1991

Binding of [3H]SCH 39166 to human post mortem brain tissue

artículo científico publicado en 1993

Biocompatible branched copolymer nanoparticles prepared by RAFT polymerization as MRI/PET bimodal tracers

artículo científico publicado en 2015

Biodistribution and dosimetry in humans of two inverse agonists to image cannabinoid CB1 receptors using positron emission tomography

artículo científico publicado en 2010

Biodistribution and radiation dosimetry of the norepinephrine transporter radioligand (S,S)-[18F]FMeNER-D2: a human whole-body PET study

artículo científico publicado en 2007

Brain PET measurement of PDE10A occupancy by TAK-063, a new PDE10A inhibitor, using [11 C]T-773 in nonhuman primates

artículo científico publicado en 2016

Brain radioligands--state of the art and new trends

artículo científico publicado en 2001

Brain uptake and distribution of the dopamine D3 /D2 receptor partial agonist [11 C]cariprazine: an in vivo positron emission tomography study in nonhuman primates

artículo científico publicado en 2013

Brain uptake and plasma metabolism of [11C]vinpocetine: a preliminary PET study in a cynomolgus monkey

artículo científico publicado en 1999

Bromine-76 and carbon-11 labelled NNC 13-8199, metabolically stable benzodiazepine receptor agonists as radioligands for positron emission tomography (PET) ⬇️

artículo científico publicado el 1 de octubre de 1997

Carbon-11 epidepride: a suitable radioligand for PET investigation of striatal and extrastriatal dopamine D2 receptors

artículo científico publicado en 1999

Carbon-11 labelling of eticlopride in two different positions--a selective high-affinity ligand for the study of dopamine D-2 receptors using PET

artículo científico publicado en 1990

Carbon-11 pb-12: an attempt to visualize the dopamine d(4) receptor in the primate brain with positron emission tomography

artículo científico publicado en 2000

Carbon-11-FLB 457: a radioligand for extrastriatal D2 dopamine receptors

artículo científico publicado en 1995

Carbon-11-NNC 112: a radioligand for PET examination of striatal and neocortical D1-dopamine receptors.

artículo científico publicado en 1998

Central 5-HT 2A and D 2 dopamine receptor occupancy after sublingual administration of ORG 5222 in healthy men ⬇️

artículo científico publicado el 1 de junio de 1997

Central D2 receptor occupancy and effects of zuclopenthixol acetate in humans.

artículo científico publicado en 1995

Central D2-dopamine receptor occupancy in relation to antipsychotic drug effects: a double-blind PET study of schizophrenic patients

artículo científico publicado en 1993

Central D2-dopamine receptor occupancy in schizophrenic patients treated with antipsychotic drugs

artículo científico publicado en 1988

Cerebral glucose utilization measured by positron emission tomography. [1-11C]-D-glucose compared with [2-18F]-2-fluoro-2-deoxy-D-glucose

artículo científico publicado el 1 de enero de 1991

Cerebral uptake of [ethyl-11C]vinpocetine and 1-[11C]ethanol in cynomolgous monkeys: a comparative preclinical PET study

artículo científico publicado en 2002

Changes in dopamine D2-receptor binding are associated to symptom reduction after psychotherapy in social anxiety disorder

artículo científico publicado en 2012

Changes in striatal D2-receptor density following chronic treatment with amphetamine as assessed with PET in nonhuman primates

artículo científico publicado en 1999

Characterisation of the appearance of radioactive metabolites in monkey and human plasma from the 5-HT1A receptor radioligand, [carbonyl-11C]WAY-100635--explanation of high signal contrast in PET and an aid to biomathematical modelling.

artículo científico publicado en 1998

Characterization of [(11)C]Cimbi-36 as an agonist PET radioligand for the 5-HT(2A) and 5-HT(2C) receptors in the nonhuman primate brain

artículo científico publicado en 2013

Characterization of bromine-76-labelled 5-bromo-6-nitroquipazine for PET studies of the serotonin transporter

artículo científico publicado en 1999

Characterization of the binding properties of T-773 as a PET radioligand for phosphodiesterase 10A.

artículo científico publicado en 2014

Characterization of the radioactive metabolites of the 5-HT1A receptor radioligand, [O-methyl-11C]WAY-100635, in monkey and human plasma by HPLC: comparison of the behaviour of an identified radioactive metabolite with parent radioligand in monkey u

artículo científico publicado en 1996

Clinical melperone treatment blocks D2-dopamine receptors in the human brain as determined by PET

scientific article published on 01 January 1989

Clinical validation of 18F-AZD4694, an amyloid-β-specific PET radioligand

artículo científico publicado en 2012

Clozapine binds preferentially to cortical D1-like dopamine receptors in the primate brain: a PET study

artículo científico publicado en 2006

Comparative double-tracer whole-body autoradiography: uptake of 11C-, 18F- and 3H-labeled compounds in rat tumors

artículo científico publicado en 1988

Comparison of D₂ dopamine receptor occupancy after oral administration of quetiapine fumarate immediate-release and extended-release formulations in healthy subjects

artículo científico publicado en 2011

Comparison of [11C]methyl triflate and [11C]methyl iodide in the synthesis of PET radioligands such as [11C]beta-CIT and [11C]beta-CFT.

artículo científico publicado en 1995

Comparison of the in vitro receptor binding properties of N-[3H]methylspiperone and [3H]raclopride to rat and human brain membranes

artículo científico publicado en 1990

Confirmation of fenfluramine effect on 5-HT(1B) receptor binding of [(11)C]AZ10419369 using an equilibrium approach

artículo científico publicado en 2011

Contribution of non-genetic factors to dopamine and serotonin receptor availability in the adult human brain

artículo científico publicado en 2015

Current state of agonist radioligands for imaging of brain dopamine D2/D3 receptors in vivo with positron emission tomography

scientific article published on January 2010

D(2)- and 5-HT(2) receptor occupancy in high-dose neuroleptic-treated patients

artículo científico publicado en 1998

D1, D2, and 5-HT2 receptor occupancy in relation to clozapine serum concentration: a PET study of schizophrenic patients

scientific article published on 01 October 1995

D1-, D2-, and 5-HT2-receptor occupancy in clozapine-treated patients

scientific article published on 01 September 1994

D2 dopamine receptor internalization prolongs the decrease of radioligand binding after amphetamine: a PET study in a receptor internalization-deficient mouse model

artículo científico publicado en 2010

D2 dopamine receptor occupancy during low-dose treatment with haloperidol decanoate

scientific article published on 01 February 1995

D2 dopamine receptors in neuroleptic-naive schizophrenic patients. A positron emission tomography study with [11C]raclopride

artículo científico publicado en 1990

D2 occupancy, extrapyramidal side effects and antipsychotic drug treatment: a pilot study with sertindole in healthy subjects

scientific article published on 01 February 1997

Decrease of mGluR5 receptor density goes parallel with changes in enkephalin and substance P immunoreactivity in Huntington's disease: a preliminary investigation in the postmortem human brain

artículo científico publicado en 2014

Decreased defluorination using the novel beta-cell imaging agent [18F]FE-DTBZ-d4 in pigs examined by PET

artículo científico publicado en 2011

Decreased dopamine D2 receptor binding in the anterior cingulate cortex in schizophrenia

artículo científico publicado en 2002

Decreased thalamic D2/D3 receptor binding in drug-naive patients with schizophrenia: a PET study with [11C]FLB 457.

artículo científico publicado en 2003

Delayed normalization of central D2 dopamine receptor availability after discontinuation of haloperidol decanoate. Preliminary findings

artículo científico publicado en 1997

Detection of amyloid in Alzheimer's disease with positron emission tomography using [11C]AZD2184.

artículo científico publicado en 2009

Determination of plasma protein binding of positron emission tomography radioligands by high-performance frontal analysis.

artículo científico publicado en 2014

Development of 123I-labelled NNC 13-8241 as a radioligand for SPECT visualization of benzodiazepine receptor binding

artículo científico publicado en 1996

Development of [11C]/[3H]THK-5351 - A potential novel carbon-11 tau imaging PET radioligand

artículo científico publicado en 2016

Development of a Novel Carbon-11 Labeled PET Radioligand for Melanin-Concentrating Hormone Receptor 1.

artículo científico publicado en 2016

Development of a PET radioligand for the central 5-HT1B receptor: radiosynthesis and characterization in cynomolgus monkeys of eight radiolabeled compounds

artículo científico publicado en 2010

Development of a series of novel carbon-11 labeled PDE10A inhibitors

artículo científico publicado en 2015

Development of a small D-enantiomeric Alzheimer's amyloid-β binding peptide ligand for future in vivo imaging applications

artículo científico publicado en 2012

Development of new brain imaging agents based upon nocaine-modafinil hybrid monoamine transporter inhibitors

artículo científico publicado en 2006

Development of radioligands for imaging of brain norepinephrine transporters in vivo with positron emission tomography

artículo científico publicado en 2007

Development of rapid multistep carbon-11 radiosynthesis of the myeloperoxidase inhibitor AZD3241 to assess brain exposure by PET microdosing

artículo científico publicado en 2015

Development of two fluorine-18 labeled PET radioligands targeting PDE10A and in vivo PET evaluation in nonhuman primates

artículo científico publicado en 2017

Different brain radioactivity curves in a PET study with [11C]beta-CIT labelled in two different positions

artículo científico publicado en 1999

Differentiation of extrastriatal dopamine D2 receptor density and affinity in the human brain using PET.

artículo científico publicado en 2004

Discovery and labeling of high-affinity 3,4-diarylpyrazolines as candidate radioligands for in vivo imaging of cannabinoid subtype-1 (CB1) receptors

artículo científico publicado en 2008

Discrepancies in brain tumor extent as shown by computed tomography and positron emission tomography using [68Ga]EDTA, [11C]glucose, and [11C]methionine

artículo científico publicado en 1983

Distribution and binding of 18F-labeled and 125I-labeled analogues of ACI-80, a prospective molecular imaging biomarker of disease: a whole hemisphere post mortem autoradiography study in human brains obtained from Alzheimer's disease patients

artículo científico publicado en 2011

Distribution of 5-HT4 receptors in the postmortem human brain--an autoradiographic study using [125I]SB 207710.

artículo científico publicado en 2003

Distribution of D1- and D2-dopamine receptors, and dopamine and its metabolites in the human brain

scientific article published on 01 December 1994

Distribution of messenger RNAs for D1 dopamine receptors and DARPP-32 in striatum and cerebral cortex of the cynomolgus monkey: relationship to D1 dopamine receptors

scientific article published on 01 July 1995

Dopamine D(2) receptor quantification in extrastriatal brain regions using [(123)I]epidepride with bolus/infusion

artículo científico publicado en 2000

Dopamine D(2/3) receptor occupancy of apomorphine in the nonhuman primate brain--a comparative PET study with [11C]raclopride and [11C]MNPA.

artículo científico publicado en 2009

Dopamine D1 receptor number--a sensitive PET marker for early brain degeneration in Huntington's disease

artículo científico publicado en 1994

Dopamine D1-receptor binding in the living human brain.

artículo científico publicado en 1986

Dopamine D2 receptor binding in drug-naïve patients with schizophrenia examined with raclopride-C11 and positron emission tomography

artículo científico publicado en 2006

Dopamine D2 receptors in the rat, monkey and the post-mortem human hippocampus. An autoradiographic study using the novel D2-selective ligand 125I-NCQ 298 ⬇️

artículo científico publicado el 15 de abril de 1991

Dopamine beta-hydroxylase-deficient mice have normal densities of D(2) dopamine receptors in the high-affinity state based on in vivo PET imaging and in vitro radioligand binding

artículo científico publicado en 2010

Dose-dependent binding of AZD3783 to brain 5-HT1B receptors in non-human primates and human subjects: a positron emission tomography study with [11C]AZ10419369.

artículo científico publicado en 2011

Drug distribution in man: a positron emission tomography study after oral administration of the labelled neuroprotective drug vinpocetine

artículo científico publicado en 2002

Dual tracer tau PET imaging reveals different molecular targets for C-THK5351 and C-PBB3 in the Alzheimer brain

Dynamic study of supratentorial gliomas with L-methyl-11C-methionine and positron emission tomography

artículo científico publicado en 1985

EANM procedure guidelines for brain tumour imaging using labelled amino acid analogues

artículo científico publicado en 2006

Effect of a single dose of escitalopram on serotonin concentration in the non-human and human primate brain

artículo científico publicado en 2013

Effect of amphetamine on dopamine D2 receptor binding in nonhuman primate brain: a comparison of the agonist radioligand [11C]MNPA and antagonist [11C]raclopride

artículo científico publicado en 2006

Effect of amphetamine on extrastriatal D2 dopamine receptor binding in the primate brain: a PET study

artículo científico publicado en 2000

Effect of clozapine and risperidone on 5-HT2 and D2-dopamine receptor binding in the post-mortem human brain. An autoradiographic study

artículo científico publicado en 1995

Effect of reserpine-induced depletion of synaptic dopamine on [11C]raclopride binding to D2-dopamine receptors in the monkey brain

artículo científico publicado en 1997

Effect of the myeloperoxidase inhibitor AZD3241 on microglia: a PET study in Parkinson's disease

artículo científico publicado en 2015

Effects of cocaine on [11C]norepinephrine and [11C] beta-CIT uptake in the primate peripheral organs measured by PET.

artículo científico publicado en 1996

Effects of estrogen and testosterone treatment on serotonin transporter binding in the brain of surgically postmenopausal women--a PET study

artículo científico publicado en 2014

Error analysis for quantification of [(11)C]FLB 457 binding to extrastriatal D(2) dopamine receptors in the human brain

artículo científico publicado en 2001

European Association of Nuclear Medicine procedure guidelines for brain perfusion SPET using (99m)Tc-labelled radiopharmaceuticals.

artículo científico publicado en 2002

Evaluation and metabolite studies of 125I- and 123I-labelled E-(R,R)-IQNP: potential radioligands for visualization of M1 muscarinic acetylcholine receptors in brain

artículo científico publicado en 1998

Evaluation of SCH 39166 as PET ligand for central D1 dopamine receptor binding and occupancy in man

artículo científico publicado en 1995

Evaluation of [11C]PipISB and [18F]PipISB in monkey as candidate radioligands for imaging brain cannabinoid type-1 receptors in vivo

artículo científico publicado en 2009

Evaluation of a novel PDE10A PET radioligand, [(11) C]T-773, in nonhuman primates: brain and whole body PET and brain autoradiography

artículo científico publicado en 2015

Evaluation of two automated methods for PET region of interest analysis

artículo científico publicado en 2014

Evidence of fatigue, disordered sleep and peripheral inflammation, but not increased brain TSPO expression, in seasonal allergy: A [11C]PBR28 PET study

artículo científico publicado en 2017

Evolution of microglial activation in ischaemic core and peri-infarct regions after stroke: a PET study with the TSPO molecular imaging biomarker [((11))C]vinpocetine

artículo científico publicado en 2012

Extrastriatal dopamine D(2) receptor binding in Huntington's disease

artículo científico publicado en 2010

Extrastriatal dopamine D2 and D3 receptors in early and advanced Parkinson's disease

scholarly article by V. Kaasinen et al published 11 April 2000 in Neurology

Extrastriatal dopamine D2 receptor density and affinity in the human brain measured by 3D PET.

artículo científico publicado en 1999

Fenfluramine Reduces [11C]Cimbi-36 Binding to the 5-HT2A Receptor in the Nonhuman Primate Brain

artículo científico publicado en 2017

Fenfluramine-induced serotonin release decreases [11C]AZ10419369 binding to 5-HT1B-receptors in the primate brain

artículo científico publicado en 2010

Fluorine-18 labeling of three novel D-peptides by conjugation with N-succinimidyl-4-[18F]fluorobenzoate and preliminary examination by postmortem whole-hemisphere human brain autoradiography.

artículo científico publicado en 2011

Fluorine-18-labelled NCQ 115, a selective dopamine D-2 receptor ligand. Preparation and positron emission tomography ⬇️

artículo científico publicado el 1 de mayo de 1994

Functional neuroimaging in multiple sclerosis with radiolabelled glia markers: preliminary comparative PET studies with [11C]vinpocetine and [11C]PK11195 in patients.

artículo científico publicado en 2007

GABAA receptor availability is not altered in adults with autism spectrum disorder or in mouse models

article

GABAA receptor occupancy by subtype selective GABAAα2,3 modulators: PET studies in humans

artículo científico

Gpp(NH)p stimulates [3H]raclopride binding to homogenates from human putamen and accumbens ⬇️

artículo científico publicado el 17 de febrero de 1992

Guideline to regulations for radiopharmaceuticals in early phase clinical trials in the EU.

artículo científico publicado en 2008

High 5-HT2 receptor occupancy in clozapine treated patients demonstrated by PET.

artículo científico publicado en 1993

High 5HT2A receptor occupancy in M100907-treated schizophrenic patients

artículo científico publicado en 2000

High specific radioactivity (1R,2S)-4-[(18)F]fluorometaraminol: a PET radiotracer for mapping sympathetic nerves of the heart

scientific article published on 01 April 2000

Identification and regional distribution in rat brain of radiometabolites of the dopamine transporter PET radioligand [11C]PE2I.

artículo científico publicado en 2006

Identification of PET radiometabolites by cytochrome P450, UHPLC/Q-ToF-MS and fast radio-LC: applied to the PET radioligands [11C]flumazenil, [18F]FE-PE2I, and [11C]PBR28.

artículo científico publicado en 2012

Imaging and quantitation of cannabinoid CB1 receptors in human and monkey brains using (18)F-labeled inverse agonist radioligands

artículo científico publicado en 2009

Imaging of dopamine receptors using PET and SPECT

artículo científico publicado el 1 de marzo de 1992

Imaging of the striatal and extrastriatal dopamine transporter with (18)F-LBT-999: quantification, biodistribution, and radiation dosimetry in nonhuman primates

artículo científico publicado en 2011

Imaging the norepinephrine transporter with positron emission tomography: initial human studies with (S,S)-[18F]FMeNER-D2.

artículo científico publicado en 2007

Immunohistoblot analysis on whole human hemispheres from normal and Alzheimer diseased brains

artículo científico publicado en 2008

Implications of brain imaging for the management of schizophrenia

artículo científico publicado en 1998

Improved mapping and quantification of serotonin transporter availability in the human brainstem with the HRRT.

artículo científico publicado en 2012

Improved synthesis of some commonly used PET radioligands by the use of [11C]methyl triflate

artículo científico publicado en 1995

In Vivo Visualization of Beta Cells by Targeting of GPR44.

artículo científico publicado en 2017

In Vivo and In Vitro Characterization of a Novel MAO-B Inhibitor Radioligand, 18F-Labeled Deuterated Fluorodeprenyl.

artículo científico publicado en 2015

In vitro and in vivo characterisation of nor-beta-CIT: a potential radioligand for visualisation of the serotonin transporter in the brain

artículo científico publicado en 1997

In vitro and in vivo evaluation of (11)C-SD5024, a novel PET radioligand for human brain imaging of cannabinoid CB1 receptors

artículo científico publicado en 2013

In vitro autoradiography and in vivo evaluation in cynomolgus monkey of [18F]FE-PE2I, a new dopamine transporter PET radioligand.

artículo científico publicado en 2009

In vivo TSPO imaging in patients with multiple sclerosis: a brain PET study with [18F]FEDAA1106.

artículo científico publicado en 2013

In vivo and in vitro characterization of [18F]-FE-(+)-DTBZ as a tracer for beta-cell mass

artículo científico publicado en 2010

In vivo evidence of a functional association between immune cells in blood and brain in healthy human subjects

artículo científico publicado en 2016

In vivo imaging of the 18-kDa translocator protein (TSPO) with [18F]FEDAA1106 and PET does not show increased binding in Alzheimer's disease patients

artículo científico publicado en 2013

In-target produced [11C]methane: Increased specific radioactivity

artículo científico publicado en 2008

Initial human studies with single-photon emission tomography using iodine-123 labelled 3-(5-cyclopropyl-1,2,4-oxadiazo-3-yl)- 7-iodo-5, 6-dihydro-5-methyl-6-oxo-4H-imidazo[1,5-a][1,4]-benzodiazepine (NNC 13-8241)

artículo científico publicado en 1996

Integrated Strategy for Use of Positron Emission Tomography in Nonhuman Primates to Confirm Multitarget Occupancy of Novel Psychotropic Drugs: An Example with AZD3676.

artículo científico publicado en 2016

Investigation of the metabolites of (S,S)-[(11)C]MeNER in humans, monkeys and rats

scientific article published on 18 September 2008

In vivo measurement of PDE10A enzyme occupancy by positron emission tomography (PET) following single oral dose administration of PF-02545920 in healthy male subjects

artículo científico publicado en 2017

Iodine-123 labeled nor-?-CIT as a potential tracer for serotonin transporter imaging in the human brain with single-photon emission tomography ⬇️

artículo científico publicado el 1 de enero de 1998

Iodine-123 labelled Z-(R,R)-IQNP: a potential radioligand for visualization of M(1 )and M(2) muscarinic acetylcholine receptors in Alzheimer's disease

scientific article published on 01 November 1999

Is dopamine D1 receptor availability related to social behavior? A positron emission tomography replication study.

artículo científico publicado en 2018

Joint explorative analysis of neuroreceptor subsystems in the human brain: application to receptor-transporter correlation using PET data

artículo científico publicado en 2004

Kinetic analysis and quantification of the dopamine transporter in the nonhuman primate brain with 11C-PE2I and 18F-FE-PE2I.

artículo científico publicado en 2011

Kinetic analysis and test-retest variability of the radioligand [11C](R)-PK11195 binding to TSPO in the human brain - a PET study in control subjects

artículo científico publicado en 2012

Kinetic brain analysis and whole-body imaging in monkey of [11C]MNPA: a dopamine agonist radioligand

artículo científico publicado en 2008

Lack of effect of reserpine-induced dopamine depletion on the binding of the dopamine-D3 selective radioligand, [11C]RGH-1756.

artículo científico publicado en 2005

Large Variation in Brain Exposure of Reference CNS Drugs: a PET Study in Nonhuman Primates

artículo científico publicado en 2015

Ligand selection for PET studies of D1 dopamine receptors. Relationship between distribution of binding sites and mRNA for DAARPP32 in the human brain

artículo científico publicado el 1 de enero de 1992

Limbic reductions of 5-HT1A receptor binding in human temporal lobe epilepsy

artículo científico publicado en 2004

Lipophilic metabolite of [123I]beta-CIT in human plasma may obstruct quantitation of the dopamine transporter

artículo científico publicado en 1995

Localization of monoamine oxidase B in human brain by autoradiographical use of 11C-labelled L-deprenyl

artículo científico publicado en 1989

Low background and high contrast PET imaging of amyloid-β with [11C]AZD2995 and [11C]AZD2184 in Alzheimer's disease patients

artículo científico publicado en 2013

Low brain CB1 receptor occupancy by a second generation CB1 receptor antagonist TM38837 in comparison with rimonabant in nonhuman primates: a PET study

artículo científico publicado en 2013

Low dopamine d(2) receptor binding in subregions of the thalamus in schizophrenia

artículo científico publicado en 2004

Low striatal and extra-striatal D2 receptor occupancy during treatment with the atypical antipsychotic sertindole

artículo científico publicado en 2002

Lower levels of the glial cell marker TSPO in drug-naive first-episode psychosis patients as measured using PET and [11C]PBR28.

artículo científico publicado en 2017

Lysosomal trapping of a radiolabeled substrate of P-glycoprotein as a mechanism for signal amplification in PET ⬇️

artículo científico publicado el 24 de enero de 2011

Mapping of central D2 dopamine receptors in man using [11C]raclopride: PET with anatomic standardization technique

artículo científico publicado en 1999

Mapping of the norepinephrine transporter in the human brain using PET with (S,S)-[18F]FMeNER-D2.

artículo científico publicado en 2008

Mapping the distribution of serotonin transporter in the human brainstem with high-resolution PET: Validation using postmortem autoradiography data

artículo científico publicado en 2016

Maps of receptor binding parameters in the human brain--a kinetic analysis of PET measurements.

artículo científico publicado en 1990

Measurement of serotonin transporter binding with PET and [11C]MADAM: a test-retest reproducibility study

artículo científico publicado en 2006

Measurement of striatal and extrastriatal dopamine D1 receptor binding potential with [11C]NNC 112 in humans: validation and reproducibility.

artículo científico publicado en 2000

Measurement of striatal and extrastriatal dopamine transporter binding with high-resolution PET and [11C]PE2I: quantitative modeling and test-retest reproducibility

artículo científico publicado en 2008

Metabolism of [123I]epidepride may affect brain dopamine D2 receptor imaging with single-photon emission tomography

artículo científico publicado en 2000

Modulation of striatal dopamine D1 binding by cognitive processing.

artículo científico publicado en 2009

Molecular Imaging of PDE10A Knockout Mice with a Novel PET Radiotracer: [(11)C]T-773.

artículo científico publicado en 2015

Molecular imaging of the dopamine transporter

artículo científico publicado en 2010

N-(4-Cyanotetrahydro-2H-pyran-4-yl) and N-(1-Cyanocyclohexyl) Derivatives of 1,5-Diarylpyrazole-3-carboxamides Showing High Affinity for 18 kDa Translocator Protein and/or Cannabinoid Receptors ⬇️

artículo científico publicado el 23 de marzo de 2011

N-(5-Fluoro-2-phenoxyphenyl)-N-(2-[(131)I]iodo-5-me thoxybenzyl)acetamide: a potent iodinated radioligand for the peripheral-type benzodiazepine receptor in brain

artículo científico publicado en 2007

N-desmethyl-loperamide is selective for P-glycoprotein among three ATP-binding cassette transporters at the blood-brain barrier

artículo científico publicado en 2010

N-oxide analogs of WAY-100635: new high affinity 5-HT(1A) receptor antagonists

artículo científico publicado en 2005

NCQ 298, a new selective iodinated salicylamide ligand for the labelling of dopamine D2 receptors ⬇️

artículo científico publicado el 1 de enero de 1991

NET occupancy by clomipramine and its active metabolite, desmethylclomipramine, in non-human primates in vivo.

artículo científico publicado en 2011

Neuroimaging and physiological evidence for involvement of glutamatergic transmission in regulation of the striatal dopaminergic system

artículo científico publicado en 2009

New alpha(1)-adrenoceptor antagonists derived from the antipsychotic sertindole - carbon-11 labelling and pet examination of brain uptake in the cynomolgus monkey

artículo científico publicado en 2004

New developments of dopaminergic imaging in Parkinson's disease.

artículo científico

New halogenated [11C]WAY analogues, [11C]6FPWAY and [11C]6BPWAY--radiosynthesis and assessment as radioligands for the study of brain 5-HT1A receptors in living monkey

artículo científico publicado en 2001

New methodologies for the preparation of carbon-11 labeled radiopharmaceuticals

artículo científico publicado en 2017

Nigrostriatal dopamine transporter availability in early Parkinson's disease

artículo científico publicado en 2018

No D2 receptor increase in PET study of schizophrenia

artículo científico publicado en 1987

No correlation between serotonin and its metabolite 5-HIAA in the cerebrospinal fluid and [(11) C]AZ10419369 binding measured with PET in healthy volunteers

artículo científico publicado en 2014

No elevated D2 dopamine receptors in neuroleptic-naive schizophrenic patients revealed by positron emission tomography and [11C]N-methylspiperone.

artículo científico publicado en 1995

No support for regional selectivity in clozapine-treated patients: a PET study with [(11)C]raclopride and [(11)C]FLB 457.

artículo científico publicado en 2001

Norepinephrine transporter occupancy by antidepressant in human brain using positron emission tomography with (S,S)-[18F]FMeNER-D2.

artículo científico publicado en 2010

Norepinephrine transporter occupancy in the human brain after oral administration of quetiapine XR.

artículo científico publicado en 2013

Occupancy of 5-HT1A receptors by clozapine in the primate brain: a PET study

artículo científico publicado en 2003

Occupancy of dopamine D2/3 receptors in rat brain by endogenous dopamine measured with the agonist positron emission tomography radioligand [11C]MNPA.

artículo científico publicado en 2008

Occupancy of dopamine D₂ and D₃ and serotonin 5-HT₁A receptors by the novel antipsychotic drug candidate, cariprazine (RGH-188), in monkey brain measured using positron emission tomography

artículo científico publicado en 2011

On-line synthesis of [11C]nitroalkanes

artículo científico publicado en 1989

Optimal Acquisition Time Window and Simplified Quantification of Dopamine Transporter Availability Using 18F-FE-PE2I in Healthy Controls and Parkinson Disease Patients.

artículo científico publicado en 2016

Oral administration of NNC 756 — a placebo controlled PET study of D1-dopamine receptor occupancy and pharmacodynamics in man ⬇️

artículo científico publicado el 1 de mayo de 1995

PET analysis of [11C]flumazenil binding to benzodiazepine receptors in chronic alcohol-dependent men and healthy controls

artículo científico publicado en 1993

PET analysis of alcohol interaction with the brain disposition of [11C]flumazenil ⬇️

artículo científico publicado el 1 de enero de 1992

PET analysis of human dopamine receptor subtypes using 11C-SCH 23390 and 11C-raclopride

artículo científico publicado en 1987

PET analysis of the 5-HT2A receptor inverse agonist ACP-103 in human brain

artículo científico publicado en 2007

PET and SPET tracers for mapping the cardiac nervous system

artículo científico publicado en 2002

PET evaluation of novel radiofluorinated reboxetine analogs as norepinephrine transporter probes in the monkey brain

artículo científico publicado en 2004

PET examination of [(11)C]5-methyl-6-nitroquipazine, a radioligand for visualization of the serotonin transporter

artículo científico publicado en 2002

PET examination of [11C]NNC 687 and [11C]NNC 756 as new radioligands for the D1-dopamine receptor

artículo científico publicado en 1993

PET examination of the monkey heart with high specific radioactivity [11C]norepinephrine and [11C]metaraminol

artículo científico publicado en 1995

PET examination of three potent cocaine derivatives as specific radioligands for the serotonin transporter

artículo científico publicado en 1999

PET for drug development.

artículo científico publicado en 2004

PET imaging of central 5-HT2A receptors with carbon-11-MDL 100,907.

artículo científico publicado en 1998

PET imaging of neuroreceptors in schizophrenia

artículo científico publicado en 1995

PET mapping of extrastriatal D2-like dopamine receptors in the human brain using an anatomic standardization technique and [11C]FLB 457

artículo científico publicado en 1999

PET measurement of serotonin transporter occupancy: a comparison of escitalopram and citalopram

artículo científico publicado en 2007

PET radioligands for dopamine receptors and re-uptake sites: chemistry and biochemistry

artículo científico publicado el 1 de mayo de 1992

PET radioligands targeting the brain GABAA /benzodiazepine receptor complex

artículo científico

PET studies of D2-receptor binding in striatal and extrastriatal brain regions: Biochemical support in vivo for separate dopaminergic systems in humans

artículo científico publicado en 2010

PET studies of binding competition between endogenous dopamine and the D1 radiotracer [11C]NNC 756.

artículo científico publicado en 1999

PET studies of dopamine receptors in relation to antipsychotic drug treatment

artículo científico publicado el 1 de enero de 1992

PET studies of the uptake of (S)- and (R)-[11C]nicotine in the human brain: difficulties in visualizing specific receptor binding in vivo

artículo científico publicado en 1994

PET studies on the brain uptake and regional distribution of [11C]vinpocetine in human subjects

artículo científico publicado en 2002

PET studies with carbon-11 radioligands in neuropsychopharmacological drug development

artículo científico publicado en 2001

PET study of D(1) dopamine receptor binding in neuroleptic-naive patients with schizophrenia

artículo científico publicado en 2002

PET study of [11C]beta-CIT binding to monoamine transporters in the monkey and human brain

artículo científico publicado en 1994

PET study of the M1-agonists [11C]xanomeline and [11C]butylthio-TZTP in monkey and man.

artículo científico publicado en 1996

PET study of the pre- and post-synaptic dopaminergic markers for the neurodegenerative process in Huntington's disease

artículo científico publicado en 1997

PET-Determination of robalzotan (NAD-299) induced 5-HT(1A) receptor occupancy in the monkey brain

scientific article published on 01 April 2000

PET-MR and SPECT-MR multimodality probes: Development and challenges

PET-characterization of [ carbonyl - 11 C]WAY-100635 binding to 5-HT 1A receptors in the primate brain ⬇️

artículo científico publicado el 1 de septiembre de 1997

PET-determination of benzodiazepine receptor binding in studies on alcoholism

artículo científico publicado en 1994

PET-examination and metabolite evaluation in monkey of [(11)C]NAD-299, a radioligand for visualisation of the 5-HT(1A) receptor

artículo científico publicado en 2002

Palladium mediated ¹¹C-cyanation and characterization in the non-human primate brain of the novel mGluR5 radioligand [¹¹C]AZD9272.

artículo científico publicado en 2013

Patterns of age related changes for phosphodiesterase type-10A in comparison with dopamine D2/3 receptors and sub-cortical volumes in the human basal ganglia: A PET study with 18F-MNI-659 and 11C-raclopride with correction for partial volume effect

artículo científico publicado en 2017

Peripheral benzodiazepine binding sites in human gliomas evaluated with positron emission tomography

artículo científico publicado en 1986

Pharmacokinetic analysis of plasma curves obtained after i.v. injection of the PET radioligand [11C] raclopride provides a likely explanation for rapid radioligand metabolism

artículo científico publicado en 2012

Pharmacokinetics and dosimetry of iodine-123 labelled PE2I in humans, a radioligand for dopamine transporter imaging

artículo científico publicado en 1998

Pharmacological characterization of (E)-N-(4-fluorobut-2-enyl)-2beta-carbomethoxy-3beta-(4'-tolyl)nortropane (LBT-999) as a highly promising fluorinated ligand for the dopamine transporter

artículo científico publicado en 2005

Pharmacological characterization of 2-methoxy-N-propylnorapomorphine's interactions with D2 and D3 dopamine receptors

scientific article published on June 2009

Pindolol binding to 5-HT1A receptors in the human brain confirmed with positron emission tomography

artículo científico publicado en 1999

Positron Emission Tomography studies with [11C]PBR28 in the Healthy Rodent Brain: Validating SUV as an Outcome Measure of Neuroinflammation

artículo científico publicado en 2015

Positron emission tomographic analysis of central D1 and D2 dopamine receptor occupancy in patients treated with classical neuroleptics and clozapine. Relation to extrapyramidal side effects

artículo científico publicado el 1 de julio de 1992

Positron emission tomographic analysis of dose-dependent MDL 100,907 binding to 5-hydroxytryptamine-2A receptors in the human brain

artículo científico publicado en 1998

Positron emission tomographic analysis of dose-dependent NAD-299 binding to 5-hydroxytryptamine-1A receptors in the human brain

artículo científico publicado en 2003

Positron emission tomographic evaluation of the putative dopamine-D3 receptor ligand, [11C]RGH-1756 in the monkey brain

artículo científico publicado en 2004

Positron emission tomographic measurements of cerebral glucose utilization using [1-11C]D-glucose

artículo científico publicado en 1990

Positron emission tomography imaging of 5-hydroxytryptamine1B receptors in Parkinson's disease

artículo científico publicado en 2013

Positron emission tomography imaging of the 18-kDa translocator protein (TSPO) with [18F]FEMPA in Alzheimer's disease patients and control subjects.

artículo científico publicado en 2014

Positron emission tomography imaging using an inverse agonist radioligand to assess cannabinoid CB1 receptors in rodents

artículo científico publicado en 2008

Positron emission tomography measurement of brain MAO-B inhibition in patients with Alzheimer's disease and elderly controls after oral administration of sembragiline

scientific article published on 16 September 2016

Positron emission tomography of in-vivo binding characteristics of atypical antipsychotic drugs. Review of D2 and 5-HT2 receptor occupancy studies and clinical response.

artículo científico publicado en 1996

Positron emission tomography shows high specific uptake of racemic carbon-11 labelled norepinephrine in the primate heart

scientific article published on 01 April 1994

Positron emission tomography studies on D2 and 5-HT2 receptor binding in risperidone-treated schizophrenic patients

artículo científico publicado en 1995

Positron emission tomography studies on D2 dopamine receptor occupancy and plasma antipsychotic drug levels in man

scientific article published on 01 September 1995

Post-mortem human brain autoradiography of the norepinephrine transporter using (S,S)-[18F]FMeNER-D2.

artículo científico publicado en 2005

Preclinical characterization of a novel class of 18F-labeled PET tracers for amyloid-β.

artículo científico publicado en 2012

Preparation of 11C-labelled SCH 23390 for the in vivo study of dopamine D-1 receptors using positron emission tomography

artículo científico publicado en 1986

Preparation of [1-11C]dopamine, [1-11C]p-tyramine and [1-11C]m-tyramine. Autoradiography and PET examination of [1-11C]dopamine in primates

artículo científico publicado en 1993

Preparation of [76Br]FLB 457 and [76Br]FLB 463 for examination of striatal and extrastriatal dopamine D-2 receptors with PET.

artículo científico publicado en 1996

Preparation of a potential positron emission tomographic radioligand for the dopamine transporter

artículo científico publicado en 1994

Preparation of highly specific radioactivity [18F]flumazenil and its evaluation in cynomolgus monkey by positron emission tomography

artículo científico publicado en 2005

Production method for [11C]-D-glucose labeled in carbon-1 for positron emission tomography of glucose metabolism

artículo científico publicado el 1 de enero de 1991

Quantification and wavelet-aided parametric imaging of cerebral amyloid using the HRRT PET-system and [18F]AZD4694

Quantification of 11C-MADAM binding to the serotonin transporter in the human brain.

artículo científico publicado en 2005

Quantification of [11C]FLB 457 binding to extrastriatal dopamine receptors in the human brain

scientific article published on 01 October 1999

Quantification of dopamine transporter in human brain using PET with 18F-FE-PE2I.

artículo científico publicado en 2012

Quantification of serotonin transporter availability with [11C]MADAM--a comparison between the ECAT HRRT and HR systems

artículo científico publicado en 2011

Quantitation of cannabinoid CB1 receptors in healthy human brain using positron emission tomography and an inverse agonist radioligand

artículo científico publicado en 2009

Quantitative Analysis of ¹⁸F-(E)-N-(3-Iodoprop-2-Enyl)-2β-Carbofluoroethoxy-3β-(4'-Methyl-Phenyl) Nortropane Binding to the Dopamine Transporter in Parkinson Disease

artículo científico publicado en 2015

Quantitative PET analyses of regional [11C]PE2I binding to the dopamine transporter--application to juvenile myoclonic epilepsy

artículo científico publicado en 2011

Quantitative PET analysis of the dopamine D2 receptor agonist radioligand 11C-(R)-2-CH3O-N-n-propylnorapomorphine in the human brain

artículo científico publicado en 2009

Quantitative analyses of carbonyl-carbon-11-WAY-100635 binding to central 5-hydroxytryptamine-1A receptors in man.

artículo científico publicado en 1998

Quantitative analyses of regional [11C]PE2I binding to the dopamine transporter in the human brain: a PET study

artículo científico publicado en 2006

Quantitative analysis of [11C]AZ10419369 binding to 5-HT1B receptors in human brain

artículo científico publicado en 2010

Quantitative analysis of norepinephrine transporter in the human brain using PET with (S,S)-18F-FMeNER-D2.

artículo científico publicado en 2008

Quantitative localization of human brain monoamine oxidase B by large section autoradiography using L-[3H]deprenyl

artículo científico publicado en 1991

Radioiodinated SB 207710 as a radioligand in vivo: imaging of brain 5-HT4 receptors with SPET.

artículo científico publicado en 2003

Radiolabeling of the cannabinoid receptor agonist AZD1940 with carbon-11 and PET microdosing in non-human primate

artículo científico publicado en 2013

Radioligands for PET studies of central benzodiazepine receptors and PK (peripheral benzodiazepine) binding sites--current status

artículo científico publicado en 1993

Radioligands for the study of brain 5-HT(1A) receptors in vivo--development of some new analogues of way.

artículo científico publicado en 2000

Radiopharmaceuticals for positron emission tomography investigations of Alzheimer's disease

artículo científico publicado en 2009

Radiosynthesis and autoradiographic evaluation of [11C]NAD-299, a radioligand for visualization of the 5-HT1A receptor

artículo científico publicado en 1999

Radiosynthesis and evaluation of new α1-adrenoceptor antagonists as PET radioligands for brain imaging.

artículo científico publicado en 2013

Radiosynthesis of the candidate beta-amyloid radioligand [(11)C]AZD2184: Positron emission tomography examination and metabolite analysis in cynomolgus monkeys

artículo científico publicado en 2010

Radiotoxicity of 11C-methionine measured by the accumulation of DNA strand breaks in mammalian cells

artículo científico publicado en 1985

Receptor binding of N-(methyl-11C) clozapine in the brain of rhesus monkey studied by positron emission tomography (PET).

artículo científico publicado en 1986

Reduced 5-HT(1B) receptor binding in the dorsal brain stem after cognitive behavioural therapy of major depressive disorder

artículo científico publicado en 2014

Reduced midbrain dopamine transporter binding in male adolescents with attention-deficit/hyperactivity disorder: association between striatal dopamine markers and motor hyperactivity

artículo científico publicado en 2005

Reduction of [11 C]CO2 to [11 C]CO using solid supported zinc

artículo científico publicado en 2017

Regional cerebral oxidative and total glucose consumption during rest and activation studied with positron emission tomography

artículo científico publicado en 1994

Regional increases in [11C]flumazenil binding after epilepsy surgery

artículo científico publicado en 1998

Regional reductions in serotonin 1A receptor binding in juvenile myoclonic epilepsy

artículo científico publicado en 2005

Reliability of volumetric and surface-based normalisation and smoothing techniques for PET analysis of the cortex: A test-retest analysis using [11C]SCH-23390.

artículo científico publicado en 2017

Reproducibility of PET measurement for presynaptic dopaminergic functions using L-[β-(11)C]DOPA and [(18)F]FE-PE2I in humans.

artículo científico publicado en 2014

Reproducibility of [11 C]FLB 457 binding in extrastriatal regions

artículo científico publicado en 2001

Revisiting the Logan plot to account for non-negligible blood volume in brain tissue

artículo científico publicado en 2017

SERT and NET occupancy by venlafaxine and milnacipran in nonhuman primates: a PET study

artículo científico publicado en 2012

SPET imaging of central muscarinic acetylcholine receptors with iodine-123 labelled E-IQNP and Z-IQNP.

artículo científico publicado en 2001

Safety and tolerability of intracerebroventricular PDGF-BB in Parkinson's disease patients

artículo científico publicado en 2015

Saturated norepinephrine transporter occupancy by atomoxetine relevant to clinical doses: a rhesus monkey study with (S,S)-[(18)F]FMeNER-D (2).

artículo científico publicado en 2009

Saturation of striatal D(2) dopamine receptors by clozapine.

artículo científico publicado en 2002

Search for correlations between serotonin 5-HT1A receptor expression and cognitive functions--a strategy in translational psychopharmacology

artículo científico publicado en 2006

Selective synthesis of racemic 1-11C-labelled norepinephrine, octopamine, norphenylephrine and phenylethanolamine using [11C]nitromethane

artículo científico publicado en 1994

Selective, irreversible in vivo binding of [11C]clorgyline and [11C]-L-deprenyl in mice: potential for measurement of functional monoamine oxidase activity in brain using positron emission tomography

artículo científico publicado en 1985

Serotonin and norepinephrine transporter occupancy of tramadol in non-human primate using positron emission tomography

artículo científico publicado en 2019

Serotonin concentration enhancers at clinically relevant doses reduce [11C]AZ10419369 binding to the 5-HT1B receptors in the nonhuman primate brain.

artículo científico publicado en 2018

Serotonin transporter genotype is associated with cognitive performance but not regional 5-HT1A receptor binding in humans

artículo científico publicado en 2009

Serotonin transporter occupancy by escitalopram and citalopram in the non-human primate brain: a [(11)C]MADAM PET study

artículo científico publicado en 2015

Sex differences in the serotonin 1A receptor and serotonin transporter binding in the human brain measured by PET.

artículo científico publicado en 2007

Short and efficient syntheses of analogues of WAY-100635: new and potent 5-HT1A receptor antagonists

artículo científico publicado en 2001

Signal transduction pathway activity compensates dopamine D₂/D₃ receptor density changes in Parkinson's disease: a preliminary comparative human brain receptor autoradiography study with [³H]raclopride and [³⁵S]GTPγS.

artículo científico publicado en 2012

Simplified estimation of binding parameters based on image-derived reference tissue models for dopamine transporter bindings in non-human primates using [18F]FE-PE2I and PET.

artículo científico publicado en 2017

Simplified quantification and whole-body distribution of [18F]FE-PE2I in nonhuman primates: prediction for human studies.

artículo científico publicado en 2011

Simultaneous determination of protein-free and total positron emission tomography radioligand concentrations in plasma using high-performance frontal analysis followed by mixed micellar liquid chromatography: application to [11C]PBR28 in human plasm

artículo científico publicado en 2013

Some new methods for the synthesis of cardiac neurotransmission PET radiotracers.

artículo científico publicado en 1995

Specific in vitro binding of (S,S)-[3H]MeNER to norepinephrine transporters

artículo científico publicado en 2005

Specific in vivo binding to the norepinephrine transporter demonstrated with the PET radioligand, (S,S)-[11C]MeNER.

artículo científico publicado en 2003

Stereoselective binding of 11C-raclopride in living human brain--a search for extrastriatal central D2-dopamine receptors by PET.

artículo científico publicado en 1988

Striatal and extrastriatal imaging of dopamine D2 receptors in the living human brain with [123I]epidepride single-photon emission tomography

artículo científico publicado en 1997

Suggested minimal effective dose of risperidone based on PET-measured D2 and 5-HT2A receptor occupancy in schizophrenic patients

artículo científico publicado en 1999

Support for dopaminergic hypoactivity in restless legs syndrome: a PET study on D2-receptor binding

artículo científico publicado en 2006

Syntheses of [123I]-, [125I]- and unlabelled (S)-3-iodo-5,6-dimethoxy-N-[(1-ethyl-2-pyrrolidinyl)methyl]salicylamide (NCQ 298), selective ligands for the study of dopamine D-2 receptors.

artículo científico publicado en 1990

Synthesis and binding properties of [3H]NNC 12-0781, a new radioligand for the dopamine reuptake system

artículo científico publicado en 1995

Synthesis and binding properties of the fluorinated substituted benzamide [3H]NCQ 115, a new selective dopamine D2 receptor ligand ⬇️

artículo científico publicado el 16 de agosto de 1991

Synthesis and biological evaluation of [¹¹C]AZ12504948; a novel tracer for imaging of glucokinase in pancreas and liver.

artículo científico publicado en 2014

Synthesis and biological evaluation of technetium(III) mixed-ligand complexes with high affinity for the cerebral 5-HT(1A) receptor and the alpha1-adrenergic receptor

artículo científico publicado en 2002

Synthesis and evaluation of 2-chloro N-[(S)-{(S)-1-[11 C]methylpiperidin-2-yl} (phenyl)methyl]3-trifluoromethyl-benzamide ([11 C]N-methyl-SSR504734) as a PET radioligand for glycine transporter 1.

artículo científico publicado en 2012

Synthesis and evaluation of N-(5-fluoro-2-phenoxyphenyl)-N-(2-[(18)F]fluoromethoxy-d(2)-5-methoxybenzyl)acetamide: a deuterium-substituted radioligand for peripheral benzodiazepine receptor

artículo científico publicado en 2005

Synthesis and in vitro autoradiographic evaluation of a novel high-affinity radioiodinated ligand for imaging brain cannabinoid subtype-1 receptors

artículo científico publicado en 2009

Synthesis and initial evaluation of [11C](R)-RWAY in monkey-a new, simply labeled antagonist radioligand for imaging brain 5-HT1A receptors with PET.

artículo científico publicado en 2007

Synthesis and positron emission tomography evaluation of three norepinephrine transporter radioligands: [C-11]desipramine, [C-11]talopram and [C-11]talsupram

artículo científico publicado en 2006

Synthesis and preclinical evaluation of [18F]FSL25.1188, a reversible PET radioligand for monoamine oxidase-B

scientific article published on 27 April 2019

Synthesis and structure-activity relationships (SARs) of 1,5-diarylpyrazole cannabinoid type-1 (CB(1)) receptor ligands for potential use in molecular imaging

artículo científico publicado en 2006

Synthesis of ([(11)C]carbonyl)raclopride and a comparison with ([(11)C]methyl)raclopride in a monkey PET study

artículo científico publicado en 2015

Synthesis of 11C-labelled (R)-OHDMI and CFMME and their evaluation as candidate radioligands for imaging central norepinephrine transporters with PET.

artículo científico publicado en 2006

Synthesis of 3H-labeled N-(3-iodoprop-2E-enyl)-2beta-carbomethoxy-3beta-(4-methylphenyl)nortropane (PE2I) and its interaction with mice striatal membrane fragments

artículo científico publicado en 2006

Synthesis of L- and D-[methyl-11C]methionine

artículo científico publicado en 1987

Synthesis of [1-11C]-beta-hydroxybutyric acid

artículo científico publicado en 1991

Synthesis of [1-11C]D-glucose and [1-11C]D-mannose from on-line produced [11C]nitromethane

artículo científico publicado en 1991

Synthesis of [11C]sodium thiocyanate for in vivo studies of anion kinetics using positron emission tomography (PET)

artículo científico publicado en 1989

Synthesis of [18F]NNC 12-0817 and [18F]NNC 12-0818; two potential radioligands for the dopamine transporter ⬇️

artículo científico publicado el 1 de mayo de 1995

Synthesis of [isopropyl-11C]nimodipine for in vivo studies of dihydropyridine binding in man using positron emission tomography ⬇️

artículo científico publicado el 1 de enero de 1991

Synthesis of a [6-pyridinyl-18F]-labelled fluoro derivative of WAY-100635 as a candidate radioligand for brain 5-HT1A receptor imaging with PET.

artículo científico publicado en 2003

Synthesis of carbon-11 labelled SCH 39166, a new selective dopamine D-1 receptor ligand, and preliminary PET investigations ⬇️

artículo científico publicado el 1 de enero de 1991

Synthesis of five benzamide analogs. Comparison with positron emission tomography

artículo científico publicado el 1 de enero de 1991

Synthesis of high-specific-radioactivity 4- and 6-[18F]fluorometaraminol-PET tracers for the adrenergic nervous system of the heart

artículo científico publicado en 2001

Synthesis of nor-beta-CIT, beta-CIT and trimethylstannyl-beta-CT.

artículo científico publicado en 1995

Synthesis of three novel fluorine-18 labeled analogues of L-deprenyl for positron emission tomography (PET) studies of monoamine oxidase B (MAO-B).

artículo científico publicado en 2011

Synthesis, biological and autoradiographic evaluation of a novel Tc-99m radioligand derived from WAY 100635 with high affinity for the 5-HT(1A) receptor and the alpha1-adrenergic receptor

artículo científico publicado en 2002

Synthesis, ex vivo evaluation, and radiolabeling of potent 1,5-diphenylpyrrolidin-2-one cannabinoid subtype-1 receptor ligands as candidates for in vivo imaging

artículo científico publicado en 2008

Synthesis, radiolabeling and preliminary biological evaluation of radiolabeled 5-methyl-6-nitroquipazine, a potential radioligand for the serotonin transporter

artículo científico publicado en 2002

Synthesis, radiolabeling and preliminary in vivo evaluation of [18F]FE-PE2I, a new probe for the dopamine transporter.

artículo científico publicado en 2009

Synthesis, radiolabeling, and in vivo pharmacokinetic evaluation of the amyloid beta radioligand [11C]AZD4694 in nonhuman primates

artículo científico publicado en 2014

Test-retest reliability of [11C]AZ10419369 binding to 5-HT(1B) receptors in human brain

artículo científico publicado en 2013

Test-retest reliability of central [11C]raclopride binding at high D2 receptor occupancy. A PET study in haloperidol-treated patients

artículo científico publicado en 1996

Test-retest reproducibility of dopamine D2/3 receptor binding in human brain measured by PET with [11C]MNPA and [11C]raclopride.

artículo científico publicado en 2012

The "specific" P-glycoprotein inhibitor Tariquidar is also a substrate and an inhibitor for breast cancer resistance protein (BCRP/ABCG2).

artículo científico publicado en 2010

The Bücherer-Strecker synthesis of D- and L-(1-11C)tyrosine and the in vivo study of L-(1-11C)tyrosine in human brain using positron emission tomography

artículo científico publicado en 1987

The Culprit Is in the Cave: The Core Sites Explain the Binding Profiles of Amyloid-Specific Tracers

artículo científico publicado en 2016

The PET radioligand [11C]MePPEP binds reversibly and with high specific signal to cannabinoid CB1 receptors in nonhuman primate brain

artículo científico publicado en 2007

The PET radioligand [carbonyl-(11)C]desmethyl-WAY-100635 binds to 5-HT(1A) receptors and provides a higher radioactive signal than [carbonyl-(11)C]WAY-100635 in the human brain

artículo científico publicado en 2002

The decrease of dopamine D₂/D₃ receptor densities in the putamen and nucleus caudatus goes parallel with maintained levels of CB₁ cannabinoid receptors in Parkinson's disease: a preliminary autoradiographic study with the selective dopamine D₂/D₃ an

artículo científico publicado en 2012

The development of a GPR44 targeting radioligand [C]AZ12204657 for in vivo assessment of beta cell mass

article

The dopamine D₁ receptor agonist (S)-[¹¹C]N-methyl-NNC 01-0259 is not sensitive to changes in dopamine concentration--a positron emission tomography examination in the monkey brain

artículo científico publicado en 2013

The immune response of the human brain to abdominal surgery

artículo científico publicado en 2017

The metabolite pattern of [123I]beta-CIT determined with a gradient HPLC method

artículo científico publicado en 1995

The norepinephrine transporter (NET) radioligand (S,S)-[18F]FMeNER-D2 shows significant decreases in NET density in the human brain in Alzheimer's disease: a post-mortem autoradiographic study

artículo científico publicado en 2010

The pyridinyl-6 position of WAY-100635 as a site for radiofluorination--effect on 5-HT1A receptor radioligand behavior in vivo

artículo científico publicado en 2004

The role of the striatal dopamine transporter in cognitive aging

artículo científico publicado en 2005

The transport of tyrosine into the human brain as determined with L-[1-11C]tyrosine and PET.

artículo científico publicado en 1991

Theoretical study of the binding profile of an allosteric modulator NS-1738 with a chimera structure of the α7 nicotinic acetylcholine receptor

artículo científico publicado en 2016

Time course of D2-dopamine receptor occupancy examined by PET after single oral doses of haloperidol

artículo científico publicado en 1992

Toxicity, mutagenicity, and behavioral effects of beta-CIT, a ligand for dopamine transporter exploration by SPECT.

artículo científico publicado en 1998

Turnover of brain monoamine oxidase measured in vivo by positron emission tomography using L-[11C]deprenyl

artículo científico publicado en 1987

Two C-methyl derivatives of [11C]WAY-100635--effects of an amido alpha-methyl group on metabolism and brain 5-HT1A receptor radioligand behavior in monkey

artículo científico publicado en 2005

Use of PET and the radioligand [carbonyl-(11)C]WAY-100635 in psychotropic drug development

scientific article published on 01 July 2000

Utilization of radioligands in schizophrenia research

artículo científico publicado el 1 de enero de 1995

Validation of [(11) C]ORM-13070 as a PET tracer for alpha2c -adrenoceptors in the human brain

artículo científico publicado en 2015

Variability in D2-dopamine receptor density and affinity: a PET study with [11C]raclopride in man

artículo científico publicado en 1995

Venlafaxine ER Blocks the Norepinephrine Transporter in the Brain of Patients with Major Depressive Disorder: a PET Study Using [18F]FMeNER-D2

scholarly article by Ryosuke Arakawa et al published 1 April 2019 in The International Journal of Neuropsychopharmacology

Visualization of the dopamine transporter in the human brain postmortem with the new selective ligand [125I]PE2I.

artículo científico publicado en 1999

Whole hemisphere autoradiography of the postmortem human brain

artículo científico publicado en 1998

Whole-body biodistribution and dosimetry of the dopamine transporter radioligand 18F-FE-PE2I in human subjects

artículo científico publicado en 2018

Whole-body biodistribution, radiation dosimetry estimates for the PET norepinephrine transporter probe (S,S)-[18F]FMeNER-D2 in non-human primates

artículo científico publicado en 2005

Z-IQNP: a potential radioligand for SPECT imaging of muscarinic acetylcholine receptors in Alzheimer's disease

artículo científico publicado en 2000

[(11)C]MADAM, a new serotonin transporter radioligand characterized in the monkey brain by PET.

artículo científico publicado en 2005

[(11)C]PE2I: a highly selective radioligand for PET examination of the dopamine transporter in monkey and human brain

artículo científico publicado en 2003

[11C] beta-CIT, a cocaine analogue. Preparation, autoradiography and preliminary PET investigations

artículo científico publicado en 1993

[11C]AZ10419369: a selective 5-HT1B receptor radioligand suitable for positron emission tomography (PET). Characterization in the primate brain

artículo científico publicado en 2008

[11C]LBT-999: a suitable radioligand for investigation of extra-striatal dopamine transporter with PET.

artículo científico publicado en 2007

[11C]MADAM Used as a Model for Understanding the Radiometabolism of Diphenyl Sulfide Radioligands for Positron Emission Tomography (PET).

artículo científico publicado en 2015

[11C]MDL 100907, a radioligland for selective imaging of 5-HT(2A) receptors with positron emission tomography

artículo científico publicado en 1996

[11C]NNC 22-0215, a metabolically stable dopamine D1 radioligand for PET.

artículo científico publicado en 1998

[11C]NNC 687 and [11C]NNC 756, dopamine D-1 receptor ligands. Preparation, autoradiography and PET investigation in monkey

scientific article published on 01 November 1993

[11C]beta-CIT-FE, a radioligand for quantitation of the dopamine transporter in the living brain using positron emission tomography

artículo científico publicado en 1996

[11C]cyclopropyl-FLB 457: a PET radioligand for low densities of dopamine D2 receptors

artículo científico publicado en 2008

[11C]metaraminol, a false neurotransmitter: preparation, metabolite studies and positron emission tomography examination in monkey

artículo científico publicado en 1996

[11C]vinpocetine: a prospective peripheral benzodiazepine receptor ligand for primate PET studies

artículo científico publicado en 2004

[18F]flumazenil binding to central benzodiazepine receptor studies by PET--quantitative analysis and comparisons with [11C]flumazenil

artículo científico publicado en 2008

[Cerebral uptake and regional distribution of [11C]-vinpocetin after intravenous administration to healthy men: a PET study].

artículo científico publicado en 2002

[O-methyl-11C]beta-CIT-FP, a potential radioligand for quantitation of the dopamine transporter: preparation, autoradiography, metabolite studies, and positron emission tomography examinations

scientific article published on 01 October 1995

[carbonyl-11C]Desmethyl-WAY-100635 (DWAY) is a potent and selective radioligand for central 5-HT1A receptors in vitro and in vivo

artículo científico publicado en 1998

[¹²⁵I]SD-7015 reveals fine modalities of CB₁ cannabinoid receptor density in the prefrontal cortex during progression of Alzheimer's disease

artículo científico publicado en 2011

β-Amyloid binding in elderly subjects with declining or stable episodic memory function measured with PET and [¹¹C]AZD2184.

artículo científico publicado en 2015

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