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Lista de obras de F Zetterberg

3-Substituted 1-Naphthamidomethyl-C-galactosyls Interact with Two Unique Sub-sites for High-Affinity and High-Selectivity Inhibition of Galectin-3

scientific article published on 12 December 2019

5-alkyl-1,3-oxazole derivatives of 6-amino-nicotinic acids as alkyl ester bioisosteres are antagonists of the P2Y12 receptor

artículo científico publicado en 2013

A novel series of piperazinyl-pyridine ureas as antagonists of the purinergic P2Y12 receptor

artículo científico publicado en 2011

Aminopyrimidine-galactose hybrids are highly selective galectin-3 inhibitors

artículo científico publicado en 2019

An orally active galectin-3 antagonist inhibits lung adenocarcinoma growth and augments response to PD-L1 blockade

scientific article published on 23 January 2019

Defining the mechanism of galectin-3–mediated TGF-β1 activation and its role in lung fibrosis

artículo científico publicado en 2024

Evaluating the affinity and kinetics of small molecule glycomimetics for human and mouse galectin-3 using surface plasmon resonance

artículo científico publicado en 2023

Extracellular and intracellular small-molecule galectin-3 inhibitors

Human trophoblast requires galectin-3 for cell migration and invasion

artículo científico publicado en 2019

In Vivo Veritas: 18F-Radiolabeled Glycomimetics Allow Insights into the Pharmacological Fate of Galectin-3 Inhibitors

scientific article published on 03 January 2020

Lead optimization of ethyl 6-aminonicotinate acyl sulfonamides as antagonists of the P2Y12 receptor. separation of the antithrombotic effect and bleeding for candidate drug AZD1283.

artículo científico publicado en 2013

Monosaccharide Derivatives with Low-Nanomolar Lectin Affinity and High Selectivity Based on Combined Fluorine-Amide, Phenyl-Arginine, Sulfur-π, and Halogen Bond Interactions.

artículo científico publicado en 2017

Optimization of ketone-based P2Y(12) receptor antagonists as antithrombotic agents: pharmacodynamics and receptor kinetics considerations.

artículo científico publicado en 2014

State of affairs: Design and structure-activity relationships of reversible P2Y12 receptor antagonists.

artículo científico publicado en 2016

Synthesis, structure-property relationships and pharmacokinetic evaluation of ethyl 6-aminonicotinate sulfonylureas as antagonists of the P2Y₁₂ receptor.

artículo científico publicado en 2013

Systematic Tuning of Fluoro-galectin-3 Interactions Provides Thiodigalactoside Derivatives with Single-Digit nM Affinity and High Selectivity

artículo científico publicado en 2017