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A MedChem toolbox for cereblon-directed PROTACs

artículo científico publicado en 2019

A Short Peptide Inhibitor as an Activity-Based Probe for Matriptase-2.

artículo científico publicado en 2018

Andrographolide Derivatives Target the KEAP1/NRF2 Axis and Possess Potent Anti-SARS-CoV-2 Activity

artículo científico publicado en 2022

Antiangiogenic Activity and in Silico Cereblon Binding Analysis of Novel Thalidomide Analogs

scientific article published on 02 December 2020

Azanitrile Inhibitors of the SmCB1 Protease Target Are Lethal to <i>Schistosoma mansoni</i>: Structural and Mechanistic Insights into Chemotype Reactivity

scientific article published on 10 December 2020

BIM-46174 fragments as potential ligands of G proteins

artículo científico publicado en 2019

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-3

scientific article published on 30 June 2018

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-5

scientific article published on 30 June 2019

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-6

scientific article published on 28 December 2019

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes⁻4

scientific article published on 31 December 2018

Can Cysteine Protease Cross-Class Inhibitors Achieve Selectivity?

scientific article published on 15 August 2019

Cell-permeable high-affinity tracers for Gq proteins provide structural insights, reveal distinct binding kinetics and identify small molecule inhibitors

artículo científico publicado en 2020

Design of an Activity-Based Probe for Human Neutrophil Elastase: Implementation of the Lossen Rearrangement To Induce Förster Resonance Energy Transfers

artículo científico publicado en 2017

Discovery of Thanafactin A, a Linear, Proline-Containing Octalipopeptide from Pseudomonas sp. SH-C52, Motivated by Genome Mining ⬇️

scientific article published on 31 December 2020

Hit expansion through computational selectivity searching

artículo científico publicado en 2009

Homo-PROTACs for the Chemical Knockdown of Cereblon

artículo científico publicado en 2018

Identification of Interaction Hot Spots in Structures of Drug Targets on the Basis of Three-Dimensional Activity Cliff Information

artículo científico publicado en 2015

Inhibitors of cathepsins K and S identified using the DynaMAD virtual screening algorithm

artículo científico publicado en 2010

Mapping the S1 and S1' subsites of cysteine proteases with new dipeptidyl nitrile inhibitors as trypanocidal agents

artículo científico publicado en 2020

Solubility and Stability Enhanced Oral Formulations for the Anti-Infective Corallopyronin A

artículo científico publicado en 2020

Synthesis of Novel Potent Archazolids: Pharmacology of an Emerging Class of Anticancer Drugs

scientific article published on 13 February 2020

Synthesis, Structural Characterization, and Antiangiogenic Activity of Polyfluorinated Benzamides

artículo científico publicado en 2018

Systematic identification and classification of three-dimensional activity cliffs

artículo científico publicado en 2012

X-ray Structures of Target-Ligand Complexes Containing Compounds with Assay Interference Potential

artículo científico publicado en 2018

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