Lista de obras - P Scholze - Dominio Público Uruguay

A Human Polymorphism in CHRNA5 Is Linked to Relapse to Nicotine Seeking in Transgenic Rats

scientific article published on 04 October 2018

A benzodiazepine ligand with improved GABA<sub>A</sub>-receptor α5-subunit-selectivity driven by interactions with loop C

scientific article published on 02 December 2020

A novel de novo variant of GABRA1 causes increased sensitivity for GABA in vitro

artículo científico publicado en 2020

A photoswitchable GABA receptor channel blocker

scientific article published on 26 June 2019

Amphetamines take two to tango: an oligomer-based counter-transport model of neurotransmitter transport explores the amphetamine action

Attaining in vivo selectivity of positive modulation of α3βγ2 GABAA receptors in rats: A hard task!

artículo científico publicado en 2018

Bi-directional transport of GABA in human embryonic kidney (HEK-293) cells stably expressing the rat GABA transporter GAT-1

artículo científico publicado en 2002

Biochemical and functional properties of distinct nicotinic acetylcholine receptors in the superior cervical ganglion of mice with targeted deletions of nAChR subunit genes.

artículo científico publicado en 2010

Catecholamine outflow from mouse and rat brain slice preparations evoked by nicotinic acetylcholine receptor activation and electrical field stimulation

artículo científico publicado en 2007

Characterization of carrier-mediated efflux in human embryonic kidney 293 cells stably expressing the rat serotonin transporter: a superfusion study.

artículo científico publicado en 2000

Chronic exposure to manganese decreases striatal dopamine turnover in human alpha-synuclein transgenic mice

artículo científico publicado en 2011

Coronaridine congeners potentiate GABAA receptors and induce sedative activity in mice in a benzodiazepine-insensitive manner

artículo científico publicado en 2020

Detection Methods for Autoantibodies in Suspected Autoimmune Encephalitis

artículo científico publicado en 2018

Different Benzodiazepines Bind with Distinct Binding Modes to GABAA Receptors

scientific article published on 23 July 2018

Disturbed neurotransmitter homeostasis in ether lipid deficiency.

artículo científico publicado en 2019

Dual mode of stimulation by the beta-carboline ZK 91085 of recombinant GABA(A) receptor currents: molecular determinants affecting its action

artículo científico publicado en 1999

Engineered Flumazenil Recognition Site Provides Mechanistic Insight Governing Benzodiazepine Modulation in GABA Receptors

artículo científico publicado en 2018

Ester to amide substitution improves selectivity, efficacy and kinetic behavior of a benzodiazepine positive modulator of GABAA receptors containing the α5 subunit

artículo científico publicado en 2016

Exploring the polyamine regulatory site of the NMDA receptor: a parallel synthesis approach.

artículo científico publicado en 2012

Extensive heterogeneity of recombinant gamma-aminobutyric acidA receptors expressed in alpha 4 beta 3 gamma 2-transfected human embryonic kidney 293 cells.

artículo científico publicado en 1996

GABAA Receptor Ligands Often Interact with Binding Sites in the Transmembrane Domain and in the Extracellular Domain-Can the Promiscuity Code Be Cracked?

scientific article published on 03 January 2020

Investigation of neurotrophic factor concentrations with a novel in vitro concept for peripheral nerve regeneration.

artículo científico publicado en 2015

Molecular tools for GABAA receptors: High affinity ligands for β1-containing subtypes.

artículo científico publicado en 2017

Nicotinic acetylcholine receptor-subunit mRNAs in the mouse superior cervical ganglion are regulated by development but not by deletion of distinct subunit genes.

artículo científico publicado en 2008

Nicotinic acetylcholine receptors control acetylcholine and noradrenaline release in the rodent habenulo-interpeduncular complex

artículo científico publicado en 2014

Nicotinic acetylcholine receptors modulate osteoclastogenesis

artículo científico publicado en 2016

Novel Benzodiazepine-Like Ligands with Various Anxiolytic, Antidepressant, or Pro-Cognitive Profiles

scientific article published on 23 January 2019

Oligomerization of the human serotonin transporter and of the rat GABA transporter 1 visualized by fluorescence resonance energy transfer microscopy in living cells.

artículo científico publicado en 2000

Role of α5-containing nicotinic receptors in neuropathic pain and response to nicotine

artículo científico publicado en 2015

SAR-Guided Scoring Function and Mutational Validation Reveal the Binding Mode of CGS-8216 at the α1+/γ2– Benzodiazepine Site

artículo científico publicado en 2018

Serotonin-transporter mediated efflux: a pharmacological analysis of amphetamines and non-amphetamines

artículo científico publicado en 2005

Single-channel properties of α3β4, α3β4α5 and α3β4β2 nicotinic acetylcholine receptors in mice lacking specific nicotinic acetylcholine receptor subunits.

artículo científico publicado en 2013

Substantial loss of substrate by diffusion during uptake in HEK-293 cells expressing neurotransmitter transporters.

artículo científico publicado en 2001

The role of the nAChR subunits α5, β2, and β4 on synaptic transmission in the mouse superior cervical ganglion

article

The role of zinc ions in reverse transport mediated by monoamine transporters.

artículo científico publicado en 2002

Towards functional selectivity for α6β3γ2 GABAA receptors: a series of novel pyrazoloquinolinones.

artículo científico publicado en 2017

Trigeminal neuropathic pain development and maintenance in rats are suppressed by a positive modulator of α6 GABAA receptors

scientific article published on 04 February 2019

Two discontinuous segments in the carboxyl terminus are required for membrane targeting of the rat gamma-aminobutyric acid transporter-1 (GAT1)

scientific journal article

Unexpected Properties of δ-Containing GABAA Receptors in Response to Ligands Interacting with the α+ β- Site.

artículo científico publicado en 2013

Lista de obras de P Scholze

A Human Polymorphism in CHRNA5 Is Linked to Relapse to Nicotine Seeking in Transgenic Rats

A benzodiazepine ligand with improved GABA<sub>A</sub>-receptor α5-subunit-selectivity driven by interactions with loop C

A novel de novo variant of GABRA1 causes increased sensitivity for GABA in vitro

A photoswitchable GABA receptor channel blocker

Amphetamines take two to tango: an oligomer-based counter-transport model of neurotransmitter transport explores the amphetamine action

Attaining in vivo selectivity of positive modulation of α3βγ2 GABAA receptors in rats: A hard task!

Bi-directional transport of GABA in human embryonic kidney (HEK-293) cells stably expressing the rat GABA transporter GAT-1

Biochemical and functional properties of distinct nicotinic acetylcholine receptors in the superior cervical ganglion of mice with targeted deletions of nAChR subunit genes.

Catecholamine outflow from mouse and rat brain slice preparations evoked by nicotinic acetylcholine receptor activation and electrical field stimulation

Characterization of carrier-mediated efflux in human embryonic kidney 293 cells stably expressing the rat serotonin transporter: a superfusion study.

Chronic exposure to manganese decreases striatal dopamine turnover in human alpha-synuclein transgenic mice

Coronaridine congeners potentiate GABAA receptors and induce sedative activity in mice in a benzodiazepine-insensitive manner

Detection Methods for Autoantibodies in Suspected Autoimmune Encephalitis

Different Benzodiazepines Bind with Distinct Binding Modes to GABAA Receptors

Disturbed neurotransmitter homeostasis in ether lipid deficiency.

Dual mode of stimulation by the beta-carboline ZK 91085 of recombinant GABA(A) receptor currents: molecular determinants affecting its action

Engineered Flumazenil Recognition Site Provides Mechanistic Insight Governing Benzodiazepine Modulation in GABA Receptors

Ester to amide substitution improves selectivity, efficacy and kinetic behavior of a benzodiazepine positive modulator of GABAA receptors containing the α5 subunit

Exploring the polyamine regulatory site of the NMDA receptor: a parallel synthesis approach.

Extensive heterogeneity of recombinant gamma-aminobutyric acidA receptors expressed in alpha 4 beta 3 gamma 2-transfected human embryonic kidney 293 cells.

GABAA Receptor Ligands Often Interact with Binding Sites in the Transmembrane Domain and in the Extracellular Domain-Can the Promiscuity Code Be Cracked?

Investigation of neurotrophic factor concentrations with a novel in vitro concept for peripheral nerve regeneration.

Molecular tools for GABAA receptors: High affinity ligands for β1-containing subtypes.

Nicotinic acetylcholine receptor-subunit mRNAs in the mouse superior cervical ganglion are regulated by development but not by deletion of distinct subunit genes.

Nicotinic acetylcholine receptors control acetylcholine and noradrenaline release in the rodent habenulo-interpeduncular complex

Nicotinic acetylcholine receptors modulate osteoclastogenesis

Novel Benzodiazepine-Like Ligands with Various Anxiolytic, Antidepressant, or Pro-Cognitive Profiles

Oligomerization of the human serotonin transporter and of the rat GABA transporter 1 visualized by fluorescence resonance energy transfer microscopy in living cells.

Role of α5-containing nicotinic receptors in neuropathic pain and response to nicotine

SAR-Guided Scoring Function and Mutational Validation Reveal the Binding Mode of CGS-8216 at the α1+/γ2– Benzodiazepine Site

Serotonin-transporter mediated efflux: a pharmacological analysis of amphetamines and non-amphetamines

Single-channel properties of α3β4, α3β4α5 and α3β4β2 nicotinic acetylcholine receptors in mice lacking specific nicotinic acetylcholine receptor subunits.

Substantial loss of substrate by diffusion during uptake in HEK-293 cells expressing neurotransmitter transporters.

The role of the nAChR subunits α5, β2, and β4 on synaptic transmission in the mouse superior cervical ganglion

The role of zinc ions in reverse transport mediated by monoamine transporters.

Towards functional selectivity for α6β3γ2 GABAA receptors: a series of novel pyrazoloquinolinones.

Trigeminal neuropathic pain development and maintenance in rats are suppressed by a positive modulator of α6 GABAA receptors

Two discontinuous segments in the carboxyl terminus are required for membrane targeting of the rat gamma-aminobutyric acid transporter-1 (GAT1)

Unexpected Properties of δ-Containing GABAA Receptors in Response to Ligands Interacting with the α+ β- Site.