Lista de obras - Richard M van Rijn - Dominio Público Uruguay

A FLIPR assay for evaluating agonists and antagonists of GPCR heterodimers.

artículo científico publicado en 2013

A Review of the Therapeutic Potential of Recently Developed G Protein-Biased Kappa Agonists

article

A critical evaluation of TRPA1-mediated locomotor behavior in zebrafish as a screening tool for novel anti-nociceptive drug discovery

scientific article published on 20 February 2019

A non-convulsant delta-opioid receptor agonist, KNT-127, reduces cortical spreading depression and nitroglycerin-induced allodynia

scientific article published on 16 December 2020

Adolescent intake of caffeinated energy drinks does not affect adult alcohol consumption in C57BL/6 and BALB/c mice

artículo científico publicado en 2016

An integrated perspective on diabetic, alcoholic, and drug-induced neuropathy, etiology, and treatment in the US.

artículo científico publicado en 2017

Anti-analgesic effect of the mu/delta opioid receptor heteromer revealed by ligand-biased antagonism

artículo científico publicado en 2013

Arrestin recruitment and signaling by G protein-coupled receptor heteromers

scientific article published on 09 November 2018

Behavioral Characterization of β-Arrestin 1 Knockout Mice in Anxiety-Like and Alcohol Behaviors.

artículo científico publicado en 2018

Commonly Used Anesthesia/Euthanasia Methods for Brain Collection Differentially Impact MAPK Activity in Male and Female C57BL/6 Mice

artículo científico publicado en 2019

Critical Role for Gi/o-Protein Activity in the Dorsal Striatum in the Reduction of Voluntary Alcohol Intake in C57Bl/6 Mice.

artículo científico publicado en 2018

Delta Opioid Pharmacology in Relation to Alcohol Behaviors.

artículo científico publicado en 2016

Discovery of naturally occurring splice variants of the rat histamine H3 receptor that act as dominant-negative isoforms

artículo científico publicado en 2006

Distinctive modulation of ethanol place preference by delta opioid receptor-selective agonists ⬇️

artículo científico publicado el 21 de octubre de 2011

Drug screening with zebrafish visual behavior identifies carvedilol as a potential treatment for an autosomal dominant form of retinitis pigmentosa

artículo científico publicado en 2021

Emergence of functional spinal delta opioid receptors after chronic ethanol exposure

artículo científico publicado en 2011

Functional histamine H3 and adenosine A2A receptor heteromers in recombinant cells and rat striatum.

artículo científico publicado en 2017

G protein-biased kratom-alkaloids and synthetic carfentanil-amide opioids as potential treatments for alcohol use disorder

artículo científico publicado en 2020

Identification of a selective small-molecule inhibitor of type 1 adenylyl cyclase activity with analgesic properties.

artículo científico publicado en 2017

Involvement of delta opioid receptors in alcohol withdrawal-induced mechanical allodynia in male C57BL/6 mice.

artículo científico publicado en 2016

Isolation and Pharmacological Characterization of Six Opioidergic Picralima nitida Alkaloids

artículo científico publicado en 2020

Isolation of acetylcholinesterase inhibitory alkaloids from Nerine bowdenii.

artículo científico publicado en 2010

Methadone antinociception is dependent on peripheral opioid receptors

artículo científico publicado en 2009

Oligomerization of recombinant and endogenously expressed human histamine H(4) receptors

artículo científico publicado en 2006

Optimization of a 1,3,4-oxadiazole series for inhibition of Ca2+/calmodulin-stimulated activity of adenylyl cyclases 1 and 8 for the treatment of chronic pain

artículo científico publicado en 2018

Pharmacological traits of delta opioid receptors: pitfalls or opportunities?

artículo científico publicado en 2013

Repeated Use of the Psychoactive Substance Ethylphenidate Impacts Neurochemistry and Reward Learning in Adolescent Male and Female Mice

artículo científico publicado en 2019

Rubiscolins are naturally occurring G protein-biased delta opioid receptor peptides

artículo científico publicado en 2018

Selection of DNA-Encoded Libraries to Protein Targets within and on Living Cells

scientific article published on 22 October 2019

Synthesis and structure-activity relationships of indole and benzimidazole piperazines as histamine H(4) receptor antagonists.

artículo científico publicado en 2004

The Meta-Position of Phe4 in Leu-Enkephalin Regulates Potency, Selectivity, Functional Activity, and Signaling Bias at the Delta and Mu Opioid Receptors

artículo científico publicado en 2019

The delta(1) opioid receptor is a heterodimer that opposes the actions of the delta(2) receptor on alcohol intake

artículo científico publicado en 2009

The only way is up: preventing opioid tolerance by promoting cell surface expression of MOR-DOR heterodimers?

artículo científico publicado en 2008

Unique Behavioral and Neurochemical Effects Induced by Repeated Adolescent Consumption of Caffeine-Mixed Alcohol in C57BL/6 Mice

artículo científico publicado en 2016

β-Arrestin 2 dependence of δ opioid receptor agonists is correlated with alcohol intake

artículo científico publicado en 2016

β-Arrestin-Dependent Dopaminergic Regulation of Calcium Channel Activity in the Axon Initial Segment.

artículo científico publicado en 2016

Lista de obras de Richard M van Rijn

A FLIPR assay for evaluating agonists and antagonists of GPCR heterodimers.

A Review of the Therapeutic Potential of Recently Developed G Protein-Biased Kappa Agonists

A critical evaluation of TRPA1-mediated locomotor behavior in zebrafish as a screening tool for novel anti-nociceptive drug discovery

A non-convulsant delta-opioid receptor agonist, KNT-127, reduces cortical spreading depression and nitroglycerin-induced allodynia

Adolescent intake of caffeinated energy drinks does not affect adult alcohol consumption in C57BL/6 and BALB/c mice

An integrated perspective on diabetic, alcoholic, and drug-induced neuropathy, etiology, and treatment in the US.

Anti-analgesic effect of the mu/delta opioid receptor heteromer revealed by ligand-biased antagonism

Arrestin recruitment and signaling by G protein-coupled receptor heteromers

Behavioral Characterization of β-Arrestin 1 Knockout Mice in Anxiety-Like and Alcohol Behaviors.

Commonly Used Anesthesia/Euthanasia Methods for Brain Collection Differentially Impact MAPK Activity in Male and Female C57BL/6 Mice

Critical Role for Gi/o-Protein Activity in the Dorsal Striatum in the Reduction of Voluntary Alcohol Intake in C57Bl/6 Mice.

Delta Opioid Pharmacology in Relation to Alcohol Behaviors.

Discovery of naturally occurring splice variants of the rat histamine H3 receptor that act as dominant-negative isoforms

Distinctive modulation of ethanol place preference by delta opioid receptor-selective agonists ⬇️

Drug screening with zebrafish visual behavior identifies carvedilol as a potential treatment for an autosomal dominant form of retinitis pigmentosa

Emergence of functional spinal delta opioid receptors after chronic ethanol exposure

Functional histamine H3 and adenosine A2A receptor heteromers in recombinant cells and rat striatum.

G protein-biased kratom-alkaloids and synthetic carfentanil-amide opioids as potential treatments for alcohol use disorder

Identification of a selective small-molecule inhibitor of type 1 adenylyl cyclase activity with analgesic properties.

Involvement of delta opioid receptors in alcohol withdrawal-induced mechanical allodynia in male C57BL/6 mice.

Isolation and Pharmacological Characterization of Six Opioidergic Picralima nitida Alkaloids

Isolation of acetylcholinesterase inhibitory alkaloids from Nerine bowdenii.

Methadone antinociception is dependent on peripheral opioid receptors

Oligomerization of recombinant and endogenously expressed human histamine H(4) receptors

Optimization of a 1,3,4-oxadiazole series for inhibition of Ca2+/calmodulin-stimulated activity of adenylyl cyclases 1 and 8 for the treatment of chronic pain

Pharmacological traits of delta opioid receptors: pitfalls or opportunities?

Repeated Use of the Psychoactive Substance Ethylphenidate Impacts Neurochemistry and Reward Learning in Adolescent Male and Female Mice

Rubiscolins are naturally occurring G protein-biased delta opioid receptor peptides

Selection of DNA-Encoded Libraries to Protein Targets within and on Living Cells

Synthesis and structure-activity relationships of indole and benzimidazole piperazines as histamine H(4) receptor antagonists.

The Meta-Position of Phe4 in Leu-Enkephalin Regulates Potency, Selectivity, Functional Activity, and Signaling Bias at the Delta and Mu Opioid Receptors

The delta(1) opioid receptor is a heterodimer that opposes the actions of the delta(2) receptor on alcohol intake

The only way is up: preventing opioid tolerance by promoting cell surface expression of MOR-DOR heterodimers?

Unique Behavioral and Neurochemical Effects Induced by Repeated Adolescent Consumption of Caffeine-Mixed Alcohol in C57BL/6 Mice

β-Arrestin 2 dependence of δ opioid receptor agonists is correlated with alcohol intake

β-Arrestin-Dependent Dopaminergic Regulation of Calcium Channel Activity in the Axon Initial Segment.