Lista de obras - Anna Lesniak - Dominio Público Uruguay

5-HT1A and 5-HT2A receptors affinity, docking studies and pharmacological evaluation of a series of 8-acetyl-7-hydroxy-4-methylcoumarin derivatives

artículo científico publicado en 2017

An imidazole based H-Phe-Phe-NH2 peptidomimetic with anti-allodynic effect in spared nerve injury mice

artículo científico publicado en 2018

Analogues of deltorphin I containing conformationally restricted amino acids in position 2: structure and opioid activity.

artículo científico publicado en 2014

Antinociceptive effect induced by a combination of opioid and neurotensin moieties vs. their hybrid peptide [Ile(9)]PK20 in an acute pain treatment in rodents.

artículo científico publicado en 2016

Antinociceptive effect of co-administered NMDA and histamine H4 receptor antagonists in a rat model of acute pain.

artículo científico publicado en 2016

Bidirectional selection for high and low stress-induced analgesia affects G-protein activity

article

Biological evaluation and molecular docking studies of AA3052, a compound containing a μ-selective opioid peptide agonist DALDA and d-Phe-Phe-d-Phe-Leu-Leu-NH2, a substance P analogue.

artículo científico publicado en 2016

Biphalin analogs containing β(3)-homo-amino acids at the 4,4' positions: Synthesis and opioid activity profiles

artículo científico publicado en 2015

Biphalin preferentially recruits peripheral opioid receptors to facilitate analgesia in a mouse model of cancer pain - A comparison with morphine.

artículo científico publicado en 2016

Biphalin protects against cognitive deficits in a mouse model of mild traumatic brain injury (mTBI).

artículo científico publicado en 2015

Canine olfactory receptor gene polymorphism and its relation to odor detection performance by sniffer dogs.

artículo científico publicado en 2008

Central antinociceptive effect of tapentadol is increased by nitric oxide synthase inhibitors

artículo científico publicado en 2016

Delta-opioid receptor antagonism leads to excessive ethanol consumption in mice with enhanced activity of the endogenous opioid system

artículo científico publicado en 2017

Distinct susceptibility to inoculated melanoma and sensitivity to cancer pain in mouse lines with high and low sensitivity to stress.

artículo científico publicado en 2012

Divergent Response to Cannabinoid Receptor Stimulation in High and Low Stress-Induced Analgesia Mouse Lines Is Associated with Differential G-Protein Activation

scientific article published on 20 February 2019

Effects of the presence or absence of a protein corona on silica nanoparticle uptake and impact on cells

artículo científico publicado en 2012

Ethanol consumption following mild traumatic brain injury is related to blood-brain barrier permeability

artículo científico publicado en 2018

Fate and effects of CeO2 nanoparticles in aquatic ecotoxicity tests.

artículo científico publicado en 2009

Hydrazone Linker as a Useful Tool for Preparing Chimeric Peptide/Nonpeptide Bifunctional Compounds.

artículo científico publicado en 2016

Identification of Dmt-D-Lys-Phe-Phe-OH as a highly antinociceptive tetrapeptide metabolite of the opioid-neurotensin hybrid peptide PK20.

artículo científico publicado en 2013

Impact of N-methylation of the substance P 1-7 amide on anti-allodynic effect in mice after peripheral administration.

artículo científico publicado en 2017

Importance of N- and C-terminal residues of substance P 1-7 for alleviating allodynia in mice after peripheral administration.

artículo científico publicado en 2017

In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt(1)-DALDA Analogues

artículo científico publicado en 2014

In vitro developmental toxicity test detects inhibition of stem cell differentiation by silica nanoparticles.

artículo científico publicado en 2009

Inhibitory effect of Ligustrum vulgare leaf extract on the development of neuropathic pain in a streptozotocin-induced rat model of diabetes

scientific article published on 11 June 2018

N-terminal guanidinylation of the cyclic 1,4-ureido-deltorphin analogues: the synthesis, receptor binding studies, and resistance to proteolytic digestion

artículo científico publicado en 2015

Naloxone exacerbates memory impairments and depressive-like behavior after mild traumatic brain injury (mTBI) in mice with upregulated opioid system activity.

artículo científico publicado en 2017

Nanoparticle adhesion to the cell membrane and its effect on nanoparticle uptake efficiency

artículo científico publicado en 2013

Opioid agonist--tachykinin antagonist as a new analgesic with adjuvant anticancer properties.

artículo científico publicado en 2013

Opioid peptides in peripheral pain control ⬇️

artículo científico publicado el 1 de enero de 2011

Role of the blood-brain barrier in differential response to opioid peptides and morphine in mouse lines divergently bred for high and low swim stress-induced analgesia

artículo científico publicado en 2014

Serum heat inactivation affects protein corona composition and nanoparticle uptake

artículo científico publicado en 2010

Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist - neurokinin-1 antagonist peptidomimetics

artículo científico publicado en 2014

The Discovery and Development of Drug Combinations for the Treatment of Various Diseases from Patent Literature (1980-Present).

artículo científico publicado en 2016

The biological consequences of replacing D-Ala in biphalin with amphiphilic α-alkylserines

artículo científico publicado en 2014

Lista de obras de Anna Lesniak

5-HT1A and 5-HT2A receptors affinity, docking studies and pharmacological evaluation of a series of 8-acetyl-7-hydroxy-4-methylcoumarin derivatives

An imidazole based H-Phe-Phe-NH2 peptidomimetic with anti-allodynic effect in spared nerve injury mice

Analogues of deltorphin I containing conformationally restricted amino acids in position 2: structure and opioid activity.

Antinociceptive effect induced by a combination of opioid and neurotensin moieties vs. their hybrid peptide [Ile(9)]PK20 in an acute pain treatment in rodents.

Antinociceptive effect of co-administered NMDA and histamine H4 receptor antagonists in a rat model of acute pain.

Bidirectional selection for high and low stress-induced analgesia affects G-protein activity

Biological evaluation and molecular docking studies of AA3052, a compound containing a μ-selective opioid peptide agonist DALDA and d-Phe-Phe-d-Phe-Leu-Leu-NH2, a substance P analogue.

Biphalin analogs containing β(3)-homo-amino acids at the 4,4' positions: Synthesis and opioid activity profiles

Biphalin preferentially recruits peripheral opioid receptors to facilitate analgesia in a mouse model of cancer pain - A comparison with morphine.

Biphalin protects against cognitive deficits in a mouse model of mild traumatic brain injury (mTBI).

Canine olfactory receptor gene polymorphism and its relation to odor detection performance by sniffer dogs.

Central antinociceptive effect of tapentadol is increased by nitric oxide synthase inhibitors

Delta-opioid receptor antagonism leads to excessive ethanol consumption in mice with enhanced activity of the endogenous opioid system

Distinct susceptibility to inoculated melanoma and sensitivity to cancer pain in mouse lines with high and low sensitivity to stress.

Divergent Response to Cannabinoid Receptor Stimulation in High and Low Stress-Induced Analgesia Mouse Lines Is Associated with Differential G-Protein Activation

Effects of the presence or absence of a protein corona on silica nanoparticle uptake and impact on cells

Ethanol consumption following mild traumatic brain injury is related to blood-brain barrier permeability

Fate and effects of CeO2 nanoparticles in aquatic ecotoxicity tests.

Hydrazone Linker as a Useful Tool for Preparing Chimeric Peptide/Nonpeptide Bifunctional Compounds.

Identification of Dmt-D-Lys-Phe-Phe-OH as a highly antinociceptive tetrapeptide metabolite of the opioid-neurotensin hybrid peptide PK20.

Impact of N-methylation of the substance P 1-7 amide on anti-allodynic effect in mice after peripheral administration.

Importance of N- and C-terminal residues of substance P 1-7 for alleviating allodynia in mice after peripheral administration.

In Vitro Membrane Permeation Studies and in Vivo Antinociception of Glycosylated Dmt(1)-DALDA Analogues

In vitro developmental toxicity test detects inhibition of stem cell differentiation by silica nanoparticles.

Inhibitory effect of Ligustrum vulgare leaf extract on the development of neuropathic pain in a streptozotocin-induced rat model of diabetes

N-terminal guanidinylation of the cyclic 1,4-ureido-deltorphin analogues: the synthesis, receptor binding studies, and resistance to proteolytic digestion

Naloxone exacerbates memory impairments and depressive-like behavior after mild traumatic brain injury (mTBI) in mice with upregulated opioid system activity.

Nanoparticle adhesion to the cell membrane and its effect on nanoparticle uptake efficiency

Opioid agonist--tachykinin antagonist as a new analgesic with adjuvant anticancer properties.

Opioid peptides in peripheral pain control ⬇️

Role of the blood-brain barrier in differential response to opioid peptides and morphine in mouse lines divergently bred for high and low swim stress-induced analgesia

Serum heat inactivation affects protein corona composition and nanoparticle uptake

Synthesis and biological evaluation of compact, conformationally constrained bifunctional opioid agonist - neurokinin-1 antagonist peptidomimetics

The Discovery and Development of Drug Combinations for the Treatment of Various Diseases from Patent Literature (1980-Present).

The biological consequences of replacing D-Ala in biphalin with amphiphilic α-alkylserines