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Lista de obras de Franciszek Sączewski

1-[(Imidazolidin-2-yl)imino]-1H-indoles as new hypotensive agents: synthesis and in vitro and in vivo biological studies

artículo científico publicado en 2016

1-[(Imidazolidin-2-yl)imino]indazole. Highly alpha 2/I1 selective agonist: synthesis, X-ray structure, and biological activity

artículo científico publicado en 2008

1H-Benzimidazole-2-carboxylic acid monohydrate

2-(4,5-Dihydro-1H-imidazol-2-yl)indazole (indazim) derivatives as selective I2 imidazoline receptor ligands ⬇️

artículo científico publicado el 1 de octubre de 2003

2-Amino-4,5-dihydro-1H-imidazol-3-ium 7,8-dihydroimidazo[1,2-c][1,3,5]thiadiazine-2,4(6H)-dithione(1−) dimethylformamide disolvate

2-Amino-6-(1-imidazolylmethyl)-4-(3,5,5-trimethyl-2-pyrazolin-1-yl)-1,3,5-triazine and 2-amino-6-(1-benzimidazolylmethyl)-4-(3,5,5-trimethyl-2-pyrazolin-1-yl)-1,3,5-triazine hemihydrate

artículo científico publicado en 2003

2-Chloro-4,5-dihydroimidazole. Part VII. Reactions with carbon disulfide and potassium O-alkyl dithiocarbonates. Synthesis and transformations of 2,3,7,8-tetrahydro-5H-diimidazo[2,1-b : 1′,2′-e][1,3,5]thiadiazine-5-thione

3-[(Imidazolidin-2-yl)imino]indazole ligands with selectivity for the α2-adrenoceptor compared to the imidazoline I1 receptor

scientific article published on 11 November 2010

5-Methyl-3,6,7,8a-tetra-hydro-2H-diimidazo[1,2-c:1',2'-e]pyrido[1,2-a][1,3,5]triazin-5-ium iodide

artículo científico publicado en 2010

A new imidazoline-containing Bunte salt: synthesis, molecular and electronic structure

A new type of mixed anhydride and its applications to the synthesis of 7-substituted 8-chloro-5,5-dioxoimidazo[1,2-b][1,4,2]benzodithiazines with in vitro antitumor activity

artículo científico publicado en 2002

A search for new antihypertensive agents. II. Circulatory activity and selection of structures among 2-methylbenzimidazole derivatives

scientific article published on 01 July 1987

Anion-pi interactions in cyanuric acids: a combined crystallographic and computational study

artículo científico publicado en 2005

Application of CoMFA and CoMSIA 3D-QSAR and docking studies in optimization of mercaptobenzenesulfonamides as HIV-1 integrase inhibitors

artículo científico publicado en 2004

Are Alpha-2D Adrenoceptor Subtypes Involved in Rat Mydriasis Evoked by New Imidazoline Derivatives: Marsanidine and 7-Methylmarsanidine?

artículo científico publicado en 2017

Biological activities of guanidine compounds

scientific article published on October 2009

Biological activities of guanidine compounds, 2008 - 2012 update

artículo científico publicado en 2013

COMPARISON OF THE EFFECTS OF MARSANIDINE DERIVATIVES ON RAT CARDIOVASCULAR SYSTEM

Carbon disulfide promoted reactions of 2-chloro-4,5-dihydro-imidazole with some N-nucleophiles

artículo científico publicado en 2001

Carbonic anhydrase inhibitors. Inhibition of the cytosolic human isozymes I and II, and the transmembrane, tumor-associated isozymes IX and XII with substituted aromatic sulfonamides activatable in hypoxic tumors

scientific article published on 30 June 2006

Carbonic anhydrase inhibitors. Selective inhibition of human tumor-associated isozymes IX and XII and cytosolic isozymes I and II with some substituted-2-mercapto-benzenesulfonamides

Carbonic anhydrase inhibitors: inhibition of human cytosolic isozymes I and II and tumor-associated isozymes IX and XII with S-substituted 4-chloro-2-mercapto-5-methyl-benzenesulfonamides.

artículo científico publicado en 2008

Carbonic anhydrase inhibitors: synthesis and inhibition of the human cytosolic isozymes I and II and transmembrane isozymes IX, XII (cancer-associated) and XIV with 4-substituted 3-pyridinesulfonamides

artículo científico publicado en 2010

Circulatory effect of TCS-80, a new imidazoline compound, in rats.

artículo científico publicado en 2016

Comparative pharmacodynamic analysis of imidazoline compounds using rat model of ocular mydriasis with a test of quantitative structure-activity relationships.

artículo científico publicado en 2017

Copper(II)-assisted hydrolysis of cyclic ureas: Transformation of 1-(pyridin-2-yl)-2,3,7,8-tetrahydro-1 H -imidazo[2,1- b ][1,3,5]triazepin-5(6 H )-ones into N 1 -[1-(pyridin-2-yl)imidazolidin-2-ylidene]-ethane-1,2-diamine ligands

Crystal and molecular structure of 3-(4-chlorobenzoylimino)-5,6-dihydro-3H-imidazo[2,1-c]-1,2,4-dithiazole

Experimental and theoretical studies on the tautomerism and reactivity of isoxazolo[3,4-b]quinolin-3(1H)-ones

First StableO-Amidinylhydroxylamines and Their Transformations into Sulfenamides by Intramolecular 1,5-O→S Amine Migration

Fluorinated analogues of marsanidine, a highly α2-AR/imidazoline I1 binding site-selective hypotensive agent. Synthesis and biological activities

artículo científico publicado en 2014

Hybrid Molecules Composed of 2,4-Diamino-1,3,5-triazines and 2-Imino-Coumarins and Coumarins. Synthesis and Cytotoxic Properties

artículo científico publicado en 2018

Imidazoline scaffold in medicinal chemistry: a patent review (2012-2015).

artículo científico publicado en 2016

Marsanidine and 7-Me-marsanidine, the new hypotensive imidazolines augment sodium and urine excretion in rats.

artículo científico publicado en 2013

N-Amidinio-3,5,5-trimethyl-2-pyrazoline-1-carboxamidine chloride (BPC-151), an oral hypoglycaemic agent

Polymeric (anion-π)n interactions in crystals of 2-(2,4,6-trioxo-[1,3,5]triazinan-1-yl)ethylammonium iodide

Preparation, structure and affinity for imidazoline I2 receptors and alpha2-adrenoceptors of 1-[(4,5-dihydroimidazolidin-2-yl)imino]indan-2-ols

artículo científico publicado en 2005

Radiosynthesis and Preclinical Evaluation of an α2A-Adrenoceptor Tracer Candidate, 6-[18F]Fluoro-marsanidine

scientific article published on 01 October 2019

Structural diversity of copper(II) complexes with N-(2-pyridyl)imidazolidin-2-ones(thiones) and their in vitro antitumor activity.

artículo científico publicado en 2014

Structure of New Imidazoline Derivatives and Their Cardiovascular Effect in Ratsa

artículo científico publicado en 1999

Structure-activity relationships of novel heteroaryl-acrylonitriles as cytotoxic and antibacterial agents.

artículo científico publicado en 2007

Studies of benzimidazole derivatives. XIII. Synthesis of various 2-alpha-hydroxy- and 2-beta-hydroxyalkyl-benzimidazoles

artículo científico publicado en 1986

Syntheses and biological activities of 2-(adamantylmethyl)benzimidazoles and -imidazolines

scientific article published on 01 September 1986

Synthesis and Fluorescent Properties of Novel Isoquinoline Derivatives

scientific article published on 10 November 2019

Synthesis and Preliminary Cytotoxicity Studies of 1-[1-(4,5-Dihydrooxazol-2-yl)-1H-indazol-3-yl]-3-phenylurea and 3-phenylthiourea Derivatives

artículo científico publicado en 2017

Synthesis and anti-HIV-1 activity of a novel series of 1,4,2-benzodithiazine-dioxides

artículo científico publicado en 2006

Synthesis and anti-HIV-1 integrase activities of 3-aroyl-2,3-dihydro-1,1-dioxo-1,4,2-benzodithiazines

artículo científico publicado en 2008

Synthesis and antitumor activity of novel 2-amino-4-(3,5,5-trimethyl-2-pyrazolino)-1,3,5-triazine derivatives

artículo científico publicado en 2002

Synthesis and biological activities of 2-[(heteroaryl)methyl]imidazolines

scientific article published on 25 November 2011

Synthesis and biological activities of some 7,8-dihydroimidazo[1,2-a]-1,3,5-triazine derivatives

scientific article published on 01 May 1995

Synthesis and cytotoxic activity of imidazo[1,2-a]-1,3,5-triazine analogues of 6-mercaptopurine

artículo científico publicado en 2008

Synthesis and in vitro anti-tumor activity of N-{1-[(3-thioxo-5,6-dihydroimidazo[2,1-c][1,2,4]thiadiazol-7-ylthio)thiocarbonyl]-2-imidazolidene}arylsulfonamides

artículo científico publicado en 2006

Synthesis and structure of novel 2,3, 5,6-tetrahydro-1H-imidazo[2,1-b][1,3,5]benzotriazepines with vasocontractile activity in rabbit aortic rings

artículo científico publicado en 2003

Synthesis of 2,3,5,6-tetrahydro-3H-imidazo[2,1-b] [1,3,5]benzotriazepines and their oxidative ring contraction into 1-(4,5-dihydro-1H-imidazol-2-yl)-1H-benzimidazoles

artículo científico publicado en 2004

Synthesis of HBB analogs with potential antiviral activity

scientific article published on 01 January 1978

Synthesis of N-(2-pyridyl)imidazolidin-2-ones and 1-(2-pyridyl)-2,3,7,8-tetrahydro-1H-imidazo[2,1-b][1,3,5]triazepin-5(6H)-ones with potential biological activities

Synthesis of novel 3-amino-2-(4-chloro-2-mercaptobenzenesulfonyl)-guanidine derivatives as potential antitumor agents

artículo científico publicado en 2007

Synthesis of novel aryl(heteroaryl)sulfonyl ureas of possible biological interest

artículo científico publicado en 2010

Synthesis, Structure and Cytotoxicity Testing of Novel 7-(4,5-dihydro-1<i>H</i>-imidazol-2-yl)-2-aryl-6,7-dihydro-2<i>H</i>-imidazo[2,1-<i>c</i>][1,2,4]triazol-3(5<i>H</i>)-Imine Derivatives

artículo científico publicado en 2020

Synthesis, Structure and Transformations of 2-Iminoimidazolidines into Novel Fused Heterocyclic Ring Systems

Synthesis, Structure, Chemical Stability, and In Vitro Cytotoxic Properties of Novel Quinoline-3-Carbaldehyde Hydrazones Bearing a 1,2,4-Triazole or Benzotriazole Moiety

artículo científico publicado en 2018

Synthesis, X-ray crystal structures, stabilities, and in vitro cytotoxic activities of new heteroarylacrylonitriles

artículo científico publicado en 2004

Synthesis, X-ray structure analysis and computational studies of novel bis(thiocarbamoyl) disulfides with non-covalent S⋯N and S⋯S interactions

Synthesis, anti-HIV-1 integrase, and cytotoxic activities of 4-chloro-N-(4-oxopyrimidin-2-yl)-2-mercaptobenzenesulfonamide derivatives

artículo científico publicado en 2007

Synthesis, antitumor and anti-HIV activities of benzodithiazine-dioxides

artículo científico publicado en 2006

Synthesis, antiviral, and anti-HIV-1 integrase activities of 3-aroyl-1,1-dioxo-1,4,2-benzodithiazines

artículo científico publicado en 2004

Synthesis, crystal structure and biological activities of copper(II) complexes with chelating bidentate 2-substituted benzimidazole ligands

artículo científico publicado en 2006

Synthesis, crystal structure, cytotoxic and superoxide dismutase activities of copper(II) complexes of N-(4,5-dihydroimidazol-2-yl)azoles

artículo científico publicado en 2007

Synthesis, molecular structure and anticancer activity of 1-allyl-3-amino-2-(4-chloro-2-mercaptobenzenesulphonyl)guanidine derivatives

artículo científico publicado en 2002

Synthesis, molecular structure and reactivity of 5-methylidene-1,2,3,5-tetrahydroimidazo[2,1-b]quinazolines

artículo científico publicado en 2004

Synthesis, molecular structure, and applications of 2-hydroxylamino-4,5-dihydroimidazolium-O-sulfonate to the synthesis of novel heterocyclic ring systems

artículo científico publicado en 2003

Synthesis, structural characterization and antitumor activity of novel 2,4-diamino-1,3,5-triazine derivatives

artículo científico publicado en 2000

Synthesis, structural characterization and in vitro antitumor activity of 4-dimethylaminopyridinium (6-chloro-1,1-dioxo-1,4,2-benzodithiazin-3-yl)methanides

artículo científico publicado en 2003

Synthesis, structural characterization and in vitro antitumor activity of novel 6-chloro-1,1-dioxo-1,4,2-benzodithiazie derivatives

artículo científico publicado en 2003

Synthesis, structural characterization, and in vitro antitumor activity of novel N-(6-chloro-1,1-dioxo-1,4,2-benzodithiazin-3-yl)arylsulfonamides

artículo científico publicado en 2007

Synthesis, structure and antiaggregatory effects of some N-(4,5-dihydro-1H-imidazol-2-yl)indoles

artículo científico publicado en 2000

Synthesis, structure and antiaggregatory effects of some α-hydroxy analogues of 2-aryliminoimidazolines in human platelets

Synthesis, structure and anticancer activity of novel 2,4-diamino-1,3,5-triazine derivatives.

artículo científico publicado en 2005

Synthesis, structure and anticancer activity of novel alkenyl-1,3,5-triazine derivatives

artículo científico publicado en 2006

Synthesis, structure, and binding of some 2-imidazolines to rat brain alfa-1 and alfa-2-adrenergic receptors

artículo científico publicado en 2000

Synthesis, structure, and biological activities of some N-(4,5-dihydro-1H-imidazol-2-yl)-1,3-dihydrobenzimidazole derivatives

artículo científico publicado en 1998

Synthesis, transformations and tuberculostatic activity of 1-(N-aroylthiocarbamoyl)imidiazolidine-2-thiones

artículo científico publicado en 1993

The effect of 7-fluoro-marsanidine, a novel α2-adrenoceptor agonist, on extracellular noradrenaline in rat frontal cortex: a microdialysis study

artículo científico publicado en 2015

Transfer of SAR information from hypotensive indazole to indole derivatives acting at α-adrenergic receptors: In vitro and in vivo studies

artículo científico publicado en 2016

Vagotomy reveals the importance of the imidazoline receptors in the cardiovascular effects of marsanidine and 7-ME-marsanidine in rats

artículo científico publicado en 2014

α-Iminohydroxylamine-α-aminonitrone tautomerism: a 1∶1 mixture of two tautomeric forms in crystals of N-(4,5-dihydro-1H-imidazol-2-yl)-N-phenyl-hydroxylamine

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