Lista de obras -

A new and useful method for the macrocyclization of linear peptides

artículo científico publicado en 2012

An asymmetric synthesis of (2S,5S)-5-substituted azepane-2-carboxylate derivatives.

artículo científico publicado en 2011

Comparative pharmacokinetic profile of cyclosporine (CsA) with a decapeptide and a linear analogue

artículo científico publicado en 2017

Cyclic Peptide Design Guided by Residual Dipolar Couplings, J-Couplings, and Intramolecular Hydrogen Bond Analysis

artículo científico publicado en 2019

Delineating the role of cooperativity in the design of potent PROTACs for BTK.

artículo científico publicado en 2018

Design and evaluation of a 2-(2,3,6-trifluorophenyl)acetamide derivative as an agonist of the GPR119 receptor ⬇️

artículo científico publicado el 25 de enero de 2011

Discovery of azetidinyl ketolides for the treatment of susceptible and multidrug resistant community-acquired respiratory tract infections.

artículo científico publicado en 2009

Discovery of cytotoxic dolastatin 10 analogues with N-terminal modifications

artículo científico publicado en 2014

Efficient use of the iron ortho-nitrophenylporphyrin chloride to mimic biological oxidations of dimethylaminoantipyrine

artículo científico publicado en 2007

Integrating Intramolecular Hydrogen Bonding (IMHB) Considerations in Drug Discovery Using ΔlogP As a Tool

artículo científico publicado en 2013

Macrocyclizations for medicinal chemistry: synthesis of druglike macrocycles by high-concentration Ullmann coupling.

artículo científico publicado en 2012

Optimizing PK properties of cyclic peptides: the effect of side chain substitutions on permeability and clearance().

artículo científico publicado en 2012

Revisiting N-to-O acyl shift for synthesis of natural product-like cyclic depsipeptides

artículo científico publicado en 2014

Screening of compound libraries for protein binding using flow-injection nuclear magnetic resonance spectroscopy.

artículo científico publicado en 2001

Structural analysis of bovine somatotropin using monoclonal antibodies and the conformation-sensitive immunoassay

artículo científico publicado en 1996

Utilizing on- and off-line monitoring tools to follow a kinetic resolution step during flow synthesis

artículo científico publicado en 2016

Lista de obras de

A new and useful method for the macrocyclization of linear peptides

An asymmetric synthesis of (2S,5S)-5-substituted azepane-2-carboxylate derivatives.

Comparative pharmacokinetic profile of cyclosporine (CsA) with a decapeptide and a linear analogue

Cyclic Peptide Design Guided by Residual Dipolar Couplings, J-Couplings, and Intramolecular Hydrogen Bond Analysis

Delineating the role of cooperativity in the design of potent PROTACs for BTK.

Design and evaluation of a 2-(2,3,6-trifluorophenyl)acetamide derivative as an agonist of the GPR119 receptor ⬇️

Discovery of azetidinyl ketolides for the treatment of susceptible and multidrug resistant community-acquired respiratory tract infections.

Discovery of cytotoxic dolastatin 10 analogues with N-terminal modifications

Efficient use of the iron ortho-nitrophenylporphyrin chloride to mimic biological oxidations of dimethylaminoantipyrine

Integrating Intramolecular Hydrogen Bonding (IMHB) Considerations in Drug Discovery Using ΔlogP As a Tool

Macrocyclizations for medicinal chemistry: synthesis of druglike macrocycles by high-concentration Ullmann coupling.

Optimizing PK properties of cyclic peptides: the effect of side chain substitutions on permeability and clearance().

Revisiting N-to-O acyl shift for synthesis of natural product-like cyclic depsipeptides

Screening of compound libraries for protein binding using flow-injection nuclear magnetic resonance spectroscopy.

Structural analysis of bovine somatotropin using monoclonal antibodies and the conformation-sensitive immunoassay

Utilizing on- and off-line monitoring tools to follow a kinetic resolution step during flow synthesis