Filtros de búsqueda

Lista de obras de Alberto Dal Corso

A non-internalizing antibody-drug conjugate based on an anthracycline payload displays potent therapeutic activity in vivo.

artículo científico publicado en 2017

Acetazolamide Serves as Selective Delivery Vehicle for Dipeptide-Linked Drugs to Renal Cell Carcinoma

scientific article published on 08 September 2016

Affinity enhancement of protein ligands by reversible covalent modification of neighboring lysine residues

artículo científico publicado en 2018

Chemically Defined Antibody- and Small Molecule-Drug Conjugates for in Vivo Tumor Targeting Applications: A Comparative Analysis.

artículo científico publicado en 2018

Cyclic isoDGR and RGD peptidomimetics containing bifunctional diketopiperazine scaffolds are integrin antagonists.

artículo científico publicado en 2015

Cyclic isoDGR peptidomimetics as low-nanomolar αvβ3 integrin ligands.

artículo científico publicado en 2013

Fast Cyclization of a Proline-Derived Self-Immolative Spacer Improves the Efficacy of Carbamate Prodrugs

artículo científico publicado en 2020

Impact of a Central Scaffold on the Binding Affinity of Fragment Pairs Isolated from DNA-Encoded Self-Assembling Chemical Libraries.

artículo científico publicado en 2017

Innovative Linker Strategies for Tumor-Targeted Drug Conjugates

scientific article published on 20 September 2019

Linker stability influences the anti-tumor activity of acetazolamide-drug conjugates for the therapy of renal cell carcinoma

artículo científico publicado en 2016

Multivalency Increases the Binding Strength of RGD Peptidomimetic-Paclitaxel Conjugates to Integrin αV β3.

artículo científico publicado en 2017

Neutrophil Elastase Promotes Linker Cleavage and Paclitaxel Release from an Integrin-Targeted Conjugate

scientific article published on 27 December 2018

Protease-Cleavable Linkers Modulate the Anticancer Activity of Noninternalizing Antibody-Drug Conjugates.

artículo científico publicado en 2017

Synthesis and Biological Evaluation of RGD and isoDGR-Monomethyl Auristatin Conjugates Targeting Integrin αV β3

artículo científico publicado en 2019

Synthesis and biological evaluation of RGD peptidomimetic-paclitaxel conjugates bearing lysosomally cleavable linkers

artículo científico publicado en 2015

Synthesis and biological evaluation of dual action cyclo-RGD/SMAC mimetic conjugates targeting α(v)β(3)/α(v)β(5) integrins and IAP proteins.

artículo científico publicado en 2014

Synthesis, Characterization, and Biological Evaluation of a Dual-Action Ligand Targeting αvβ3 Integrin and VEGF Receptors

artículo científico publicado en 2015

Targeted Delivery of Cytotoxic Drugs: Challenges, Opportunities and New Developments

artículo científico publicado en 2017

Targeted Small-Molecule Conjugates: the Future is Now

artículo científico publicado en 2020

αvβ3 Integrin-Targeted Peptide/Peptidomimetic-Drug Conjugates: In-Depth Analysis of the Linker Technology

artículo científico

Dominio Público Uruguay está sostenido por:

Acerca de Dominio Público Uruguay

Ayuda