Lista de obras - Alberto Minassi - Dominio Público Uruguay

8-Prenylnaringenin, inhibits estrogen receptor-alpha mediated cell growth and induces apoptosis in MCF-7 breast cancer cells

artículo científico publicado en 2007

A Multicomponent Carba-Betti Strategy to Alkylidene Heterodimers - Total Synthesis and Structure-Activity Relationships of Arzanol

A Regiodivergent Synthesis of Ring A C-Prenylflavones

artículo científico publicado en 2008

A multicomponent synthesis of gem-(β-dicarbonyl)arylmethanes

A structure-activity relationship study on N-arachidonoyl-amino acids as possible endogenous inhibitors of fatty acid amide hydrolase

artículo científico publicado en 2004

Amines Bearing Tertiary Substituents by Tandem Enantioselective Carbolithiation–Rearrangement of Vinylureas

artículo científico publicado en 2013

Amines Bearing Tertiary Substituents by Tandem Enantioselective Carbolithiation–Rearrangement of Vinylureas

artículo científico publicado en 2012

An NMR spectroscopic method to identify and classify thiol-trapping agents: revival of Michael acceptors for drug discovery?

artículo científico publicado en 2011

An expeditious hydroxyamidation of carboxylic acids

Anti-inflammatory and vascularprotective properties of 8-prenylapigenin

artículo científico publicado en 2009

Antimicrobial phenolics and unusual glycerides from Helichrysum italicum subsp. microphyllum

artículo científico publicado en 2012

Carbolithiation of N-alkenyl ureas and N-alkenyl carbamates

artículo científico publicado en 2013

Cerium(III) chloride-promoted chemoselective esterification of phenolic alcohols

Chemoproteomic fishing identifies arzanol as a positive modulator of brain glycogen phosphorylase

artículo científico publicado en 2018

Chemoselective Esterification of Phenolic Acids and Alcohols

scientific article published on 01 October 2002

Cloning of the first sn1-DAG lipases points to the spatial and temporal regulation of endocannabinoid signaling in the brain

artículo científico publicado en 2003

Conformationally constrained fatty acid ethanolamides as cannabinoid and vanilloid receptor probes

artículo científico publicado en 2009

Development of the first potent and specific inhibitors of endocannabinoid biosynthesis

artículo científico publicado en 2006

Development of the first ultra-potent "capsaicinoid" agonist at transient receptor potential vanilloid type 1 (TRPV1) channels and its therapeutic potential

artículo científico publicado en 2004

Differential effects of phorbol-13-monoesters on human immunodeficiency virus reactivation.

artículo científico publicado en 2007

Discovery of non-electrophilic capsaicinoid-type TRPA1 ligands

artículo científico publicado en 2015

Dissecting the pharmacophore of curcumin. Which structural element is critical for which action?

artículo científico publicado en 2013

Exploring the Universe of Natural Products: Recent Advances in Synthesis, Isolation and Structural Elucidation

artículo científico publicado en 2021

First "hybrid" ligands of vanilloid TRPV1 and cannabinoid CB2 receptors and non-polyunsaturated fatty acid-derived CB2-selective ligands

artículo científico publicado en 2005

Flavonoid-induced autophagy in hormone sensitive breast cancer cells

artículo científico publicado en 2009

Functionalization of β-Caryophyllene Generates Novel Polypharmacology in the Endocannabinoid System

artículo científico publicado en 2014

Geometry-Selective Synthesis ofEorZN-Vinyl Ureas (N-Carbamoyl Enamines)

artículo científico publicado en 2010

Homologues and isomers of noladin ether, a putative novel endocannabinoid: interaction with rat cannabinoid CB(1) receptors

artículo científico publicado en 2003

Identification of a Strigoterpenoid with Dual Nrf2 and Nf-κB Modulatory Activity

scientific article published on 08 January 2019

Immunosuppressive activity of capsaicinoids: capsiate derived from sweet peppers inhibits NF-kappaB activation and is a potent antiinflammatory compound in vivo

artículo científico publicado en 2002

In vivo estrogenic comparisons of Trifolium pratense (red clover) Humulus lupulus (hops), and the pure compounds isoxanthohumol and 8-prenylnaringenin

artículo científico publicado en 2008

Involvement of reactive oxygen species in capsaicinoid-induced apoptosis in transformed cells

artículo científico publicado en 2003

Iodinated N-acylvanillamines: potential "multiple-target" anti-inflammatory agents acting via the inhibition of t-cell activation and antagonism at vanilloid TRPV1 channels.

artículo científico publicado en 2006

Iodine-mediated cyclization of cannabigerol (CBG) expands the cannabinoid biological and chemical space

scientific article published on 27 July 2018

Ischemic neuroprotection by TRPV1 receptor-induced hypothermia

artículo científico publicado en 2012

Modulation of the transient receptor potential vanilloid channel TRPV4 by 4alpha-phorbol esters: a structure-activity study

artículo científico publicado en 2009

N-Acylvanillamides: development of an expeditious synthesis and discovery of new acyl templates for powerful activation of the vanilloid receptor

artículo científico publicado en 2002

Noladin ether, a putative novel endocannabinoid: inactivation mechanisms and a sensitive method for its quantification in rat tissues

artículo científico publicado en 2002

Non-pungent capsaicinoids from sweet pepper synthesis and evaluation of the chemopreventive and anticancer potential

artículo científico publicado en 2003

Oligomeric acylphloroglucinols from myrtle (Myrtus communis).

artículo científico publicado en 2002

One-Pot Total Synthesis of Cannabinol via Iodine-Mediated Deconstructive Annulation

scientific article published on 24 July 2019

Oxyhomologation of the amide bond potentiates neuroprotective effects of the endolipid N-palmitoylethanolamine

artículo científico publicado en 2006

Oxyhomologues of anandamide and related endolipids: chemoselective synthesis and biological activity

artículo científico publicado en 2006

Prenylation preserves antioxidant properties and effect on cell viability of the natural dietary phenol curcumin

Protective activation of the endocannabinoid system during ischemia in dopamine neurons

artículo científico publicado en 2006

Protective effect and relation structure-activity of nonivamide and iododerivatives in several models of lipid oxidation

artículo científico publicado en 2009

Recreational drug discovery: natural products as lead structures for the synthesis of smart drugs

artículo científico publicado en 2014

Roasting impact on the contents of clovamide (N-caffeoyl-L-DOPA) and the antioxidant activity of cocoa beans (Theobroma cacao L.)

SAR Studies on Curcumin’s Pro-inflammatory Targets: Discovery of Prenylated Pyrazolocurcuminoids as Potent and Selective Novel Inhibitors of 5-Lipoxygenase

scientific article published on 24 June 2014

Sesquiterpenoids from Common Ragweed (Ambrosia artemisiifolia L.), an Invasive Biological Polluter

Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The side chain benzylic methylene

artículo científico publicado en 2009

Structure–activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The homovanillyl moiety

artículo científico publicado en 2006

Synthesis and Biological Evaluation of Phorbol-Resiniferatoxin (RTX) Hybrids

Synthesis and tubulin-binding properties of non-symmetrical click C5-curcuminoids ⬇️

artículo científico publicado el 13 de junio de 2013

Tandem beta-alkylation-alpha-arylation of amines by carbolithiation and rearrangement of N-carbamoyl enamines (vinyl ureas).

artículo científico publicado en 2010

Targeting oncogenic serine/threonine-protein kinase BRAF in cancer cells inhibits angiogenesis and abrogates hypoxia

artículo científico publicado en 2011

The 1,2,3-triazole ring as a peptido- and olefinomimetic element: discovery of click vanilloids and cannabinoids

artículo científico publicado en 2007

The Thia-Michael Reactivity of Zerumbone and Related Cross-Conjugated Dienones: Disentangling Stoichiometry, Regiochemistry, and Addition Mode with an NMR-Spectroscopy-Based Cysteamine Assay

The biosynthesis of N-arachidonoyl dopamine (NADA), a putative endocannabinoid and endovanilloid, via conjugation of arachidonic acid with dopamine

scientific article published on 30 June 2009

The role of natural products in the ligand deorphanization of TRP channels.

artículo científico publicado en 2008

The taming of capsaicin. Reversal of the vanilloid activity of N-acylvanillamines by aromatic iodination

artículo científico publicado en 2005

Triazole-curcuminoids: A new class of derivatives for 'tuning' curcumin bioactivities?

artículo científico publicado en 2015

Triterpenoid Hydroxamates as HIF Prolyl Hydrolase Inhibitors

artículo científico publicado en 2018

Umbellulone modulates TRP channels

artículo científico publicado en 2011

Lista de obras de Alberto Minassi

8-Prenylnaringenin, inhibits estrogen receptor-alpha mediated cell growth and induces apoptosis in MCF-7 breast cancer cells

A Multicomponent Carba-Betti Strategy to Alkylidene Heterodimers - Total Synthesis and Structure-Activity Relationships of Arzanol

A Regiodivergent Synthesis of Ring A C-Prenylflavones

A multicomponent synthesis of gem-(β-dicarbonyl)arylmethanes

A structure-activity relationship study on N-arachidonoyl-amino acids as possible endogenous inhibitors of fatty acid amide hydrolase

Amines Bearing Tertiary Substituents by Tandem Enantioselective Carbolithiation–Rearrangement of Vinylureas

Amines Bearing Tertiary Substituents by Tandem Enantioselective Carbolithiation–Rearrangement of Vinylureas

An NMR spectroscopic method to identify and classify thiol-trapping agents: revival of Michael acceptors for drug discovery?

An expeditious hydroxyamidation of carboxylic acids

Anti-inflammatory and vascularprotective properties of 8-prenylapigenin

Antimicrobial phenolics and unusual glycerides from Helichrysum italicum subsp. microphyllum

Carbolithiation of N-alkenyl ureas and N-alkenyl carbamates

Cerium(III) chloride-promoted chemoselective esterification of phenolic alcohols

Chemoproteomic fishing identifies arzanol as a positive modulator of brain glycogen phosphorylase

Chemoselective Esterification of Phenolic Acids and Alcohols

Cloning of the first sn1-DAG lipases points to the spatial and temporal regulation of endocannabinoid signaling in the brain

Conformationally constrained fatty acid ethanolamides as cannabinoid and vanilloid receptor probes

Development of the first potent and specific inhibitors of endocannabinoid biosynthesis

Development of the first ultra-potent "capsaicinoid" agonist at transient receptor potential vanilloid type 1 (TRPV1) channels and its therapeutic potential

Differential effects of phorbol-13-monoesters on human immunodeficiency virus reactivation.

Discovery of non-electrophilic capsaicinoid-type TRPA1 ligands

Dissecting the pharmacophore of curcumin. Which structural element is critical for which action?

Exploring the Universe of Natural Products: Recent Advances in Synthesis, Isolation and Structural Elucidation

First "hybrid" ligands of vanilloid TRPV1 and cannabinoid CB2 receptors and non-polyunsaturated fatty acid-derived CB2-selective ligands

Flavonoid-induced autophagy in hormone sensitive breast cancer cells

Functionalization of β-Caryophyllene Generates Novel Polypharmacology in the Endocannabinoid System

Geometry-Selective Synthesis ofEorZN-Vinyl Ureas (N-Carbamoyl Enamines)

Homologues and isomers of noladin ether, a putative novel endocannabinoid: interaction with rat cannabinoid CB(1) receptors

Identification of a Strigoterpenoid with Dual Nrf2 and Nf-κB Modulatory Activity

Immunosuppressive activity of capsaicinoids: capsiate derived from sweet peppers inhibits NF-kappaB activation and is a potent antiinflammatory compound in vivo

In vivo estrogenic comparisons of Trifolium pratense (red clover) Humulus lupulus (hops), and the pure compounds isoxanthohumol and 8-prenylnaringenin

Involvement of reactive oxygen species in capsaicinoid-induced apoptosis in transformed cells

Iodinated N-acylvanillamines: potential "multiple-target" anti-inflammatory agents acting via the inhibition of t-cell activation and antagonism at vanilloid TRPV1 channels.

Iodine-mediated cyclization of cannabigerol (CBG) expands the cannabinoid biological and chemical space

Ischemic neuroprotection by TRPV1 receptor-induced hypothermia

Modulation of the transient receptor potential vanilloid channel TRPV4 by 4alpha-phorbol esters: a structure-activity study

N-Acylvanillamides: development of an expeditious synthesis and discovery of new acyl templates for powerful activation of the vanilloid receptor

Noladin ether, a putative novel endocannabinoid: inactivation mechanisms and a sensitive method for its quantification in rat tissues

Non-pungent capsaicinoids from sweet pepper synthesis and evaluation of the chemopreventive and anticancer potential

Oligomeric acylphloroglucinols from myrtle (Myrtus communis).

One-Pot Total Synthesis of Cannabinol via Iodine-Mediated Deconstructive Annulation

Oxyhomologation of the amide bond potentiates neuroprotective effects of the endolipid N-palmitoylethanolamine

Oxyhomologues of anandamide and related endolipids: chemoselective synthesis and biological activity

Prenylation preserves antioxidant properties and effect on cell viability of the natural dietary phenol curcumin

Protective activation of the endocannabinoid system during ischemia in dopamine neurons

Protective effect and relation structure-activity of nonivamide and iododerivatives in several models of lipid oxidation

Recreational drug discovery: natural products as lead structures for the synthesis of smart drugs

Roasting impact on the contents of clovamide (N-caffeoyl-L-DOPA) and the antioxidant activity of cocoa beans (Theobroma cacao L.)

SAR Studies on Curcumin’s Pro-inflammatory Targets: Discovery of Prenylated Pyrazolocurcuminoids as Potent and Selective Novel Inhibitors of 5-Lipoxygenase

Sesquiterpenoids from Common Ragweed (Ambrosia artemisiifolia L.), an Invasive Biological Polluter

Structure-activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The side chain benzylic methylene

Structure–activity relationships of the ultrapotent vanilloid resiniferatoxin (RTX): The homovanillyl moiety

Synthesis and Biological Evaluation of Phorbol-Resiniferatoxin (RTX) Hybrids

Synthesis and tubulin-binding properties of non-symmetrical click C5-curcuminoids ⬇️

Tandem beta-alkylation-alpha-arylation of amines by carbolithiation and rearrangement of N-carbamoyl enamines (vinyl ureas).

Targeting oncogenic serine/threonine-protein kinase BRAF in cancer cells inhibits angiogenesis and abrogates hypoxia

The 1,2,3-triazole ring as a peptido- and olefinomimetic element: discovery of click vanilloids and cannabinoids

The Thia-Michael Reactivity of Zerumbone and Related Cross-Conjugated Dienones: Disentangling Stoichiometry, Regiochemistry, and Addition Mode with an NMR-Spectroscopy-Based Cysteamine Assay

The biosynthesis of N-arachidonoyl dopamine (NADA), a putative endocannabinoid and endovanilloid, via conjugation of arachidonic acid with dopamine

The role of natural products in the ligand deorphanization of TRP channels.

The taming of capsaicin. Reversal of the vanilloid activity of N-acylvanillamines by aromatic iodination

Triazole-curcuminoids: A new class of derivatives for 'tuning' curcumin bioactivities?

Triterpenoid Hydroxamates as HIF Prolyl Hydrolase Inhibitors

Umbellulone modulates TRP channels