Lista de obras - Samuel Estrada-Soto - Dominio Público Uruguay

1,5-Diarylpyrazole and vanillin hybrids: Synthesis, biological activity and DFT studies

artículo científico publicado en 2015

2-(2-Benzyl-oxyphen-yl)-1H-benzimid-azole.

artículo científico publicado en 2008

4-Meth-oxy-N-[6-methyl-2,3-dihydro-1,3-benzothia-zol-2-yl-idene]benzene-sulfonamide.

artículo científico publicado en 2007

A comparative study of flavonoid analogues on streptozotocin-nicotinamide induced diabetic rats: quercetin as a potential antidiabetic agent acting via 11beta-hydroxysteroid dehydrogenase type 1 inhibition.

artículo científico publicado en 2010

Acute and sub-acute toxicity methanolic extract from Brickellia cavanillesii in mice

Acute and subacute antidiabetic studies of ENP-9, a new 1,5-diarylpyrazole derivative

scientific article published on 17 May 2018

Analysis of Flavonoids Bioactivity for Cholestatic Liver Disease: Systematic Literature Search and Experimental Approaches

artículo científico publicado en 2019

Anti-diabetic effect on alloxanized and normoglycemic rats and some pharmacological evaluations of Tournefortia hartwegiana.

artículo científico publicado en 2005

Antidiabetic activity of N-(6-substituted-1,3-benzothiazol-2-yl)benzenesulfonamides.

artículo científico publicado en 2008

Antidiabetic activity of some pentacyclic acid triterpenoids, role of PTP-1B: in vitro, in silico, and in vivo approaches

artículo científico publicado en 2011

Antidiabetic and toxicological evaluations of naringenin in normoglycaemic and NIDDM rat models and its implications on extra-pancreatic glucose regulation.

artículo científico publicado en 2008

Antidiabetic, antidyslipidemic and toxicity profile of ENV-2: A potent pyrazole derivative against diabetes and related diseases.

artículo científico publicado en 2017

Antidiabetic, antihyperlipidemic and anti-inflammatory effects of tilianin in streptozotocin-nicotinamide diabetic rats.

artículo científico publicado en 2016

Antihypertensive and vasorelaxant activities of Laelia autumnalis are mainly through calcium channel blockade.

artículo científico publicado en 2008

Antihypertensive and vasorelaxant effects of dihydrospinochalcone-A isolated from Lonchocarpus xuul Lundell by NO production: computational and ex vivo approaches.

artículo científico publicado en 2013

Antihypertensive and vasorelaxant effects of tilianin isolated from Agastache mexicana are mediated by NO/cGMP pathway and potassium channel opening.

artículo científico publicado en 2009

Anxiolytic-like effects and toxicological studies of Brickellia cavanillesii (Cass.) A. Gray in experimental mice models

artículo científico publicado en 2016

Anxiolytic-like effects of Brickellia cavanillesii and their bioactive compounds nicotiflorin and acacetin in experimental models in mice

Biopharmaceutical Characterization and Bioavailability Study of a Tetrazole Analog of Clofibric Acid in Rat.

artículo científico publicado en 2017

Chemical constituents of the hemiparasitic plant Phoradendron brachystachyum DC Nutt (Viscaceae)

artículo científico publicado en 2012

Chrysin Induces Antidiabetic, Antidyslipidemic and Anti-Inflammatory Effects in Athymic Nude Diabetic Mice.

artículo científico publicado en 2017

Cochlospermum vitifolium induces vasorelaxant and antihypertensive effects mainly by activation of NO/cGMP signaling pathway.

artículo científico publicado en 2010

Crystal structure of 4-methyl-7-prop-oxy-2H-chromen-2-one

artículo científico publicado en 2014

Depressant effects of Agastache mexicana methanol extract and one of major metabolites tilianin

scientific article published on 01 March 2015

Design, Synthesis and in Combo Antidiabetic Bioevaluation of Multitarget Phenylpropanoic Acids.

artículo científico publicado en 2018

Design, microwave-assisted synthesis, and spasmolytic activity of 2-(alkyloxyaryl)-1H-benzimidazole derivatives as constrained stilbene bioisosteres

artículo científico publicado en 2006

Design, synthesis, and in vitro antiprotozoal, antimycobacterial activities of N-{2-[(7-chloroquinolin-4-yl)amino]ethyl}ureas.

artículo científico publicado en 2010

Differential role of cyclooxygenase-1 and -2 on renal vasoconstriction to α₁-adrenoceptor stimulation in normotensive and hypertensive rats

artículo científico publicado en 2013

Discovery of 2-(3,4-dichlorophenoxy)-N-(2-morpholin-4-ylethyl)acetamide: A selective σ1 receptor ligand with antinociceptive effect

scientific article published on 14 March 2016

Discovery of new dual PPARγ-GPR40 agonists with robust antidiabetic activity: Design, synthesis and in combo drug evaluation

artículo científico publicado en 2017

Discovery of thiazolidine-2,4-dione/biphenylcarbonitrile hybrid as dual PPAR α/γ modulator with antidiabetic effect: in vitro, in silico and in vivo approaches.

artículo científico publicado en 2013

Discovery, synthesis and in combo studies of a tetrazole analogue of clofibric acid as a potent hypoglycemic agent

scientific article published on 05 April 2013

Dose-dependent antihypertensive determination and toxicological studies of tilianin isolated from Agastache mexicana.

artículo científico publicado en 2012

Endothelium-independent relaxation of aorta rings by two stilbenoids from the orchids Scaphyglottis livida.

artículo científico publicado en 2006

Evaluation of the neuroprotective activity of stansin 6, a resin glycoside from Ipomoea stans.

artículo científico publicado en 2014

Ex Vivo Study of the Vasorelaxant Activity Induced by Phenanthrene Derivatives Isolated from Maxillaria densa

artículo científico publicado en 2012

Functional mechanism of tracheal relaxation, antiasthmatic, and toxicological studies of 6-hydroxyflavone

artículo científico publicado en 2018

Glycolipid ester-type heterodimers from Ipomoea tyrianthina and their pharmacological activity.

artículo científico publicado en 2009

Hypoglycemic, vasorelaxant and hepatoprotective effects of Cochlospermum vitifolium (Willd.) Sprengel: a potential agent for the treatment of metabolic syndrome.

artículo científico publicado en 2006

Identification of fatty acid esters and hydrocarbon derivatives from Cyrtocarpa procera Kunth by GC-MS.

artículo científico publicado en 2006

In vitro and in silico PTP-1B inhibition and in vivo antidiabetic activity of semisynthetic moronic acid derivatives

artículo científico publicado en 2016

Insights on the vasorelaxant mode of action of malbrancheamide

artículo científico publicado en 2015

Metronidazole and Secnidazole Carbamates: Synthesis, Antiprotozoal Activity, and Molecular Dynamics Studies

scientific article published on 12 February 2020

Micropropagation and vasorelaxant activity of Laelia autumnalis (Orchidaceae).

artículo científico publicado en 2010

New phenanthrene derivatives from maxillaria densa(1)

scientific article published on 01 August 1999

New triterpenoids from the orchids Scaphyglottis livida and Nidema boothii.

artículo científico publicado en 2002

Postprandial glycaemia and inhibition of α-glucosidase activity by aqueous extract from Coriandrum sativum

artículo científico publicado en 2014

QSAR study on the relaxant agents from some Mexican medicinal plants and synthetic related organic compounds.

artículo científico publicado en 2007

Relaxant activity of 2-(substituted phenyl)-1H-benzimidazoles on isolated rat aortic rings: design and synthesis of 5-nitro derivatives.

artículo científico publicado en 2006

Relaxant effects of Artemisia ludoviciana on isolated rat smooth muscle tissues

article

Resin glycosides from Ipomoea tyrianthina and their sedative and vasorelaxant effects

artículo científico publicado en 2014

Resin glycosides from the roots of Ipomoea tyrianthina and their biological activity

artículo científico publicado en 2007

Sedative, vasorelaxant, and cytotoxic effects of convolvulin from Ipomoea tyrianthina.

artículo científico publicado en 2011

Semisynthesis, ex vivo evaluation, and SAR studies of coumarin derivatives as potential antiasthmatic drugs.

artículo científico publicado en 2014

Smooth muscle relaxing flavonoids and terpenoids from Conyza filaginoides

scientific article published on 01 February 1997

Spasmolytic action of Lepechinia caulescens is through calcium channel blockade and NO release.

artículo científico publicado en 2007

Spasmolytic activity of several extracts obtained from some Mexican medicinal plants.

artículo científico publicado en 2003

Spasmolytic effect of Mentha pulegium L. involves ionic flux regulation in rat ileum strips.

artículo científico publicado en 2010

Spasmolytic stilbenoids from Maxillaria densa

artículo científico publicado en 2004

Synthesis and antimycobacterial activity of 4-(5-substituted-1,3,4-oxadiazol-2-yl)pyridines

scientific article published on 25 May 2007

Synthesis and molecular docking of N'-arylidene-5-(4-chlorophenyl)-1-(3,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carbohydrazides as novel hypoglycemic and antioxidant dual agents.

artículo científico publicado en 2016

Synthesis of 2-{2-[(α/β-naphthalen-1-ylsulfonyl)amino]-1,3-thiazol-4-yl} acetamides with 11β-hydroxysteroid dehydrogenase inhibition and in combo antidiabetic activities

artículo científico publicado en 2014

Synthesis of nitro(benzo)thiazole acetamides and in vitro antiprotozoal effect against amitochondriate parasites Giardia intestinalis and Trichomonas vaginalis

artículo científico publicado en 2015

Synthesis of oleanolic acid derivatives: In vitro, in vivo and in silico studies for PTP-1B inhibition

artículo científico publicado en 2014

Synthesis, ex vivo and in silico studies of 3-cyano-2-pyridone derivatives with vasorelaxant activity.

artículo científico publicado en 2013

Synthesis, hypoglycemic activity and molecular modeling studies of pyrazole-3-carbohydrazides designed by a CoMFA model.

artículo científico publicado en 2013

Synthesis, in vitro and computational studies of protein tyrosine phosphatase 1B inhibition of a small library of 2-arylsulfonylaminobenzothiazoles with antihyperglycemic activity.

artículo científico publicado en 2009

Synthesis, in vitro and in silico screening of ethyl 2-(6-substituted benzo[d]thiazol-2-ylamino)-2-oxoacetates as protein-tyrosine phosphatase 1B inhibitors

artículo científico publicado en 2012

Synthesis, in vitro and in silico studies of a PPARγ and GLUT-4 modulator with hypoglycemic effect

artículo científico publicado en 2014

Tracheal relaxation of five medicinal plants used in Mexico for the treatment of several diseases.

artículo científico publicado en 2014

Ursolic acid derivatives as potential antidiabetic agents: In vitro, in vivo, and in silico studies.

artículo científico publicado en 2018

Ursolic acid mediates the vasorelaxant activity of Lepechinia caulescens via NO release in isolated rat thoracic aorta

artículo científico publicado en 2006

Vasorelaxant activity of some structurally related triterpenic acids from Phoradendron reichenbachianum (Viscaceae) mainly by NO production: ex vivo and in silico studies

artículo científico publicado en 2012

Vasorelaxant and antihypertensive effects of methanolic extract from roots of Laelia anceps are mediated by calcium-channel antagonism.

artículo científico publicado en 2009

Vasorelaxant effect of Valeriana edulis ssp. procera (Valerianaceae) and its mode of action as calcium channel blocker.

artículo científico publicado en 2010

Vasorelaxant effect of flavonoids through calmodulin inhibition: Ex vivo, in vitro, and in silico approaches

artículo científico publicado en 2010

Vasorelaxant mode of action of dichloromethane-soluble extract from Agastache mexicana and its main bioactive compounds.

artículo científico publicado en 2016

alpha-Glucosidase inhibitory activity of the methanolic extract from Tournefortia hartwegiana: an anti-hyperglycemic agent

scientific article published on 08 July 2006

Lista de obras de Samuel Estrada-Soto

1,5-Diarylpyrazole and vanillin hybrids: Synthesis, biological activity and DFT studies

2-(2-Benzyl-oxyphen-yl)-1H-benzimid-azole.

4-Meth-oxy-N-[6-methyl-2,3-dihydro-1,3-benzothia-zol-2-yl-idene]benzene-sulfonamide.

A comparative study of flavonoid analogues on streptozotocin-nicotinamide induced diabetic rats: quercetin as a potential antidiabetic agent acting via 11beta-hydroxysteroid dehydrogenase type 1 inhibition.

Acute and sub-acute toxicity methanolic extract from Brickellia cavanillesii in mice

Acute and subacute antidiabetic studies of ENP-9, a new 1,5-diarylpyrazole derivative

Analysis of Flavonoids Bioactivity for Cholestatic Liver Disease: Systematic Literature Search and Experimental Approaches

Anti-diabetic effect on alloxanized and normoglycemic rats and some pharmacological evaluations of Tournefortia hartwegiana.

Antidiabetic activity of N-(6-substituted-1,3-benzothiazol-2-yl)benzenesulfonamides.

Antidiabetic activity of some pentacyclic acid triterpenoids, role of PTP-1B: in vitro, in silico, and in vivo approaches

Antidiabetic and toxicological evaluations of naringenin in normoglycaemic and NIDDM rat models and its implications on extra-pancreatic glucose regulation.

Antidiabetic, antidyslipidemic and toxicity profile of ENV-2: A potent pyrazole derivative against diabetes and related diseases.

Antidiabetic, antihyperlipidemic and anti-inflammatory effects of tilianin in streptozotocin-nicotinamide diabetic rats.

Antihypertensive and vasorelaxant activities of Laelia autumnalis are mainly through calcium channel blockade.

Antihypertensive and vasorelaxant effects of dihydrospinochalcone-A isolated from Lonchocarpus xuul Lundell by NO production: computational and ex vivo approaches.

Antihypertensive and vasorelaxant effects of tilianin isolated from Agastache mexicana are mediated by NO/cGMP pathway and potassium channel opening.

Anxiolytic-like effects and toxicological studies of Brickellia cavanillesii (Cass.) A. Gray in experimental mice models

Anxiolytic-like effects of Brickellia cavanillesii and their bioactive compounds nicotiflorin and acacetin in experimental models in mice

Biopharmaceutical Characterization and Bioavailability Study of a Tetrazole Analog of Clofibric Acid in Rat.

Chemical constituents of the hemiparasitic plant Phoradendron brachystachyum DC Nutt (Viscaceae)

Chrysin Induces Antidiabetic, Antidyslipidemic and Anti-Inflammatory Effects in Athymic Nude Diabetic Mice.

Cochlospermum vitifolium induces vasorelaxant and antihypertensive effects mainly by activation of NO/cGMP signaling pathway.

Crystal structure of 4-methyl-7-prop-oxy-2H-chromen-2-one

Depressant effects of Agastache mexicana methanol extract and one of major metabolites tilianin

Design, Synthesis and in Combo Antidiabetic Bioevaluation of Multitarget Phenylpropanoic Acids.

Design, microwave-assisted synthesis, and spasmolytic activity of 2-(alkyloxyaryl)-1H-benzimidazole derivatives as constrained stilbene bioisosteres

Design, synthesis, and in vitro antiprotozoal, antimycobacterial activities of N-{2-[(7-chloroquinolin-4-yl)amino]ethyl}ureas.

Differential role of cyclooxygenase-1 and -2 on renal vasoconstriction to α₁-adrenoceptor stimulation in normotensive and hypertensive rats

Discovery of 2-(3,4-dichlorophenoxy)-N-(2-morpholin-4-ylethyl)acetamide: A selective σ1 receptor ligand with antinociceptive effect

Discovery of new dual PPARγ-GPR40 agonists with robust antidiabetic activity: Design, synthesis and in combo drug evaluation

Discovery of thiazolidine-2,4-dione/biphenylcarbonitrile hybrid as dual PPAR α/γ modulator with antidiabetic effect: in vitro, in silico and in vivo approaches.

Discovery, synthesis and in combo studies of a tetrazole analogue of clofibric acid as a potent hypoglycemic agent

Dose-dependent antihypertensive determination and toxicological studies of tilianin isolated from Agastache mexicana.

Endothelium-independent relaxation of aorta rings by two stilbenoids from the orchids Scaphyglottis livida.

Evaluation of the neuroprotective activity of stansin 6, a resin glycoside from Ipomoea stans.

Ex Vivo Study of the Vasorelaxant Activity Induced by Phenanthrene Derivatives Isolated from Maxillaria densa

Functional mechanism of tracheal relaxation, antiasthmatic, and toxicological studies of 6-hydroxyflavone

Glycolipid ester-type heterodimers from Ipomoea tyrianthina and their pharmacological activity.

Hypoglycemic, vasorelaxant and hepatoprotective effects of Cochlospermum vitifolium (Willd.) Sprengel: a potential agent for the treatment of metabolic syndrome.

Identification of fatty acid esters and hydrocarbon derivatives from Cyrtocarpa procera Kunth by GC-MS.

In vitro and in silico PTP-1B inhibition and in vivo antidiabetic activity of semisynthetic moronic acid derivatives

Insights on the vasorelaxant mode of action of malbrancheamide

Metronidazole and Secnidazole Carbamates: Synthesis, Antiprotozoal Activity, and Molecular Dynamics Studies

Micropropagation and vasorelaxant activity of Laelia autumnalis (Orchidaceae).

New phenanthrene derivatives from maxillaria densa(1)

New triterpenoids from the orchids Scaphyglottis livida and Nidema boothii.

Postprandial glycaemia and inhibition of α-glucosidase activity by aqueous extract from Coriandrum sativum

QSAR study on the relaxant agents from some Mexican medicinal plants and synthetic related organic compounds.

Relaxant activity of 2-(substituted phenyl)-1H-benzimidazoles on isolated rat aortic rings: design and synthesis of 5-nitro derivatives.

Relaxant effects of Artemisia ludoviciana on isolated rat smooth muscle tissues

Resin glycosides from Ipomoea tyrianthina and their sedative and vasorelaxant effects

Resin glycosides from the roots of Ipomoea tyrianthina and their biological activity

Sedative, vasorelaxant, and cytotoxic effects of convolvulin from Ipomoea tyrianthina.

Semisynthesis, ex vivo evaluation, and SAR studies of coumarin derivatives as potential antiasthmatic drugs.

Smooth muscle relaxing flavonoids and terpenoids from Conyza filaginoides

Spasmolytic action of Lepechinia caulescens is through calcium channel blockade and NO release.

Spasmolytic activity of several extracts obtained from some Mexican medicinal plants.

Spasmolytic effect of Mentha pulegium L. involves ionic flux regulation in rat ileum strips.

Spasmolytic stilbenoids from Maxillaria densa

Synthesis and antimycobacterial activity of 4-(5-substituted-1,3,4-oxadiazol-2-yl)pyridines

Synthesis and molecular docking of N'-arylidene-5-(4-chlorophenyl)-1-(3,4-dichlorophenyl)-4-methyl-1H-pyrazole-3-carbohydrazides as novel hypoglycemic and antioxidant dual agents.

Synthesis of 2-{2-[(α/β-naphthalen-1-ylsulfonyl)amino]-1,3-thiazol-4-yl} acetamides with 11β-hydroxysteroid dehydrogenase inhibition and in combo antidiabetic activities

Synthesis of nitro(benzo)thiazole acetamides and in vitro antiprotozoal effect against amitochondriate parasites Giardia intestinalis and Trichomonas vaginalis

Synthesis of oleanolic acid derivatives: In vitro, in vivo and in silico studies for PTP-1B inhibition

Synthesis, ex vivo and in silico studies of 3-cyano-2-pyridone derivatives with vasorelaxant activity.

Synthesis, hypoglycemic activity and molecular modeling studies of pyrazole-3-carbohydrazides designed by a CoMFA model.

Synthesis, in vitro and computational studies of protein tyrosine phosphatase 1B inhibition of a small library of 2-arylsulfonylaminobenzothiazoles with antihyperglycemic activity.

Synthesis, in vitro and in silico screening of ethyl 2-(6-substituted benzo[d]thiazol-2-ylamino)-2-oxoacetates as protein-tyrosine phosphatase 1B inhibitors

Synthesis, in vitro and in silico studies of a PPARγ and GLUT-4 modulator with hypoglycemic effect

Tracheal relaxation of five medicinal plants used in Mexico for the treatment of several diseases.

Ursolic acid derivatives as potential antidiabetic agents: In vitro, in vivo, and in silico studies.

Ursolic acid mediates the vasorelaxant activity of Lepechinia caulescens via NO release in isolated rat thoracic aorta

Vasorelaxant activity of some structurally related triterpenic acids from Phoradendron reichenbachianum (Viscaceae) mainly by NO production: ex vivo and in silico studies

Vasorelaxant and antihypertensive effects of methanolic extract from roots of Laelia anceps are mediated by calcium-channel antagonism.

Vasorelaxant effect of Valeriana edulis ssp. procera (Valerianaceae) and its mode of action as calcium channel blocker.

Vasorelaxant effect of flavonoids through calmodulin inhibition: Ex vivo, in vitro, and in silico approaches

Vasorelaxant mode of action of dichloromethane-soluble extract from Agastache mexicana and its main bioactive compounds.

alpha-Glucosidase inhibitory activity of the methanolic extract from Tournefortia hartwegiana: an anti-hyperglycemic agent

α-Glucosidase inhibitory activity of extracts from Cordia morelosana