Lista de obras - Luigi André Agrofoglio - Dominio Público Uruguay

3'-(1,2,3-Triazol-1-yl)-3'-deoxythymidine analogs as substrates for human and Ureaplasma parvum thymidine kinase for structure-activity investigations.

artículo científico publicado en 2010

Active site labeling of cysteine cathepsins by a straightforward diazomethylketone probe derived from the N-terminus of human cystatin C.

artículo científico publicado en 2015

Alkyne-Azide Click Chemistry Mediated Carbanucleosides Synthesis

article

Analysis and validation of the phosphorylated metabolites of two anti-human immunodeficiency virus nucleotides (stavudine and didanosine) by pressure-assisted CE-ESI-MS/MS in cell extracts: sensitivity enhancement by the use of perfluorinated acids

artículo científico publicado en 2006

Artificial receptors for the extraction of nucleoside metabolite 7-methylguanosine from aqueous media made by molecular imprinting.

artículo científico publicado en 2014

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-2.

artículo científico publicado en 2017

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-3

scientific article published on 30 June 2018

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-5

scientific article published on 30 June 2019

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-6

scientific article published on 28 December 2019

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes⁻4

scientific article published on 31 December 2018

Combination of computational methods, adsorption isotherms and selectivity tests for the conception of a mixed non-covalent-semi-covalent molecularly imprinted polymer of vanillin.

artículo científico publicado en 2013

Cross-Metathesis Mediated Synthesis of New Acyclic Nucleoside Phosphonates

scientific article published on 01 January 2007

Design and Synthesis of Various 5'-Deoxy-5'-(4-Substituted-1,2,3-Triazol-1-yl)-Uridine Analogues as Inhibitors of Mycobacterium tuberculosis Mur Ligases

artículo científico publicado en 2020

Determination at ppb level of an anti-human immunodeficiency virus nucleoside drug by capillary electrophoresis-electrospray ionization tandem mass spectrometry.

artículo científico publicado en 2000

Efficient synthesis of D-[1'-13C]-ribonucleosides for incorporation into oligo-RNA

scientific article published on 01 April 2001

Efficient synthesis of unprotected C-5-aryl/heteroaryl-2'-deoxyuridine via a Suzuki-Miyaura reaction in aqueous media.

artículo científico publicado en 2012

Evaluation of molecularly imprinted polymers using 2',3',5'-tri-O-acyluridines as templates for pyrimidine nucleoside recognition

artículo científico publicado en 2014

HPLC and mass spectrometry analysis of the enzymatic hydrolysis of anti-HIV pronucleotide diastereomers.

artículo científico publicado en 2003

Highly convergent synthesis and antiviral activity of (E)-but-2-enyl nucleoside phosphonoamidates

artículo científico publicado en 2018

Human and viral nucleoside/nucleotide kinases involved in antiviral drug activation: structural and catalytic properties.

artículo científico publicado en 2010

Inhibition of human immunodeficiency virus type 1 reverse transcriptase by the 5'-triphosphate beta enantiomers of cytidine analogs

artículo científico publicado en 1994

Liquid chromatographic separation of phosphoramidate diastereomers on a polysaccharide-type chiral stationary phase.

artículo científico publicado en 2003

Looking for new pyrimidine acyclic nucleotide analogues designed for phosphorylation by human UMP-CMP kinase.

artículo científico publicado en 2007

Love Acoustic Wave-Based Devices and Molecularly-Imprinted Polymers as Versatile Sensors for Electronic Nose or Tongue for Cancer Monitoring.

artículo científico publicado en 2016

Mass spectrometry based methods for analysis of nucleosides as antiviral drugs and potential tumor biomarkers

artículo científico publicado en 2007

Microwave-Assisted Silylation-Amination of Uracil Acyclonucleosides to 4-Alkylamino-2(1H)-Pyrimidinone Analogues

Microwave-assisted syntheses of nucleosides and their precursors.

artículo científico publicado en 2010

Molecularly imprinted polymer of 5-methyluridine for solid-phase extraction of pyrimidine nucleoside cancer markers in urine.

artículo científico publicado en 2008

Novel antiviral C5-substituted pyrimidine acyclic nucleoside phosphonates selected as human thymidylate kinase substrates

artículo científico publicado en 2011

Nucleotide binding to human UMP-CMP kinase using fluorescent derivatives -- a screening based on affinity for the UMP-CMP binding site

artículo científico publicado en 2007

Olefin metathesis route to antiviral nucleosides

artículo científico publicado en 2005

Palladium-assisted routes to nucleosides.

artículo científico publicado en 2003

Phosphorylation of dGMP analogs by vaccinia virus TMP kinase and human GMP kinase

artículo científico publicado en 2009

Potential and perspectives of cyclonucleosides.

artículo científico publicado en 2010

Preparation of acyclo nucleoside phosphonate analogues based on cross-metathesis

article

Recent progress for the synthesis of selected carbocyclic nucleosides

artículo científico

Selective inhibition of human cathepsin S by 2,4,6-trisubstituted 1,3,5-triazine analogs

scientific article published on 19 July 2018

Simultaneous analysis of several antiretroviral nucleosides in rat-plasma by high-performance liquid chromatography with UV using acetic acid/hydroxylamine buffer Test of this new volatile medium-pH for HPLC-ESI-MS/MS.

artículo científico publicado en 2005

Simultaneous quantitation of nucleoside HIV-1 reverse transcriptase inhibitors by short-end injection capillary electrochromatography on a beta-cyclodextrin-bonded silica stationary phase.

artículo científico publicado en 2001

Sonication-Assisted Synthesis of(E)-2-Methyl-but-2-enyl Nucleoside Phosphonate Prodrugs

Specificity enhancement with LC-positive ESI-MS/MS for the measurement of nucleotides: application to the quantitative determination of carbovir triphosphate, lamivudine triphosphate and tenofovir diphosphate in human peripheral blood mononuclear ce

artículo científico publicado en 2008

Straightforward synthesis of 2,4,6-trisubstituted 1,3,5-triazine compounds targeting cysteine cathepsins K and S.

artículo científico publicado en 2016

Study of Copper(I) Catalysts for the Synthesis of Carbanucleosides via Azide-Alkyne 1,3-Dipolar Cycloaddition

Study of Different Copper (I) Catalysts for the “Click Chemistry” Approach to Carbanucleosides

artículo científico publicado en 2007

Synthesis and Anti-HIV Evaluation of 3′-Triazolo Nucleosides ⬇️

artículo científico publicado el 1 de abril de 2011

Synthesis and antiviral activity of novel acyclic nucleosides in the 5-alkynyl- and 6-alkylfuro[2,3-d]pyrimidine series.

artículo científico publicado en 2005

Synthesis and antiviral evaluation of C5-substituted-(1,3-diyne)-2'-deoxyuridines.

artículo científico publicado en 2012

Synthesis and antiviral evaluation of bis(POM) prodrugs of (E)-[4′-phosphono-but-2′-en-1′-yl]purine nucleosides

article

Synthesis and broad spectrum antiviral evaluation of bis(POM) prodrugs of novel acyclic nucleosides

artículo científico publicado en 2013

Synthesis and characterization of various 5'-dye-labeled ribonucleosides

artículo científico publicado en 2018

Synthesis of 1,2,3-triazolo-carbanucleoside analogues of ribavirin targeting an HCV in replicon.

artículo científico publicado en 2003

Synthesis of 5'-thioalkyl, sulfoxide and sulfone pyrimidine nucleosides

artículo científico publicado en 1999

Synthesis of 5-haloethynyl- and 5-(1,2-dihalo)vinyluracil nucleosides: antiviral activity and cellular toxicity.

artículo científico publicado en 2005

Synthesis of a molecularly imprinted polymer to isolate glucosamine from plant extracts by an ionic-non-covalent dual approach

artículo científico publicado en 2015

Synthesis of a novel heterocyclic ring system: 2-thia-3,5,6,7,9-pentaazabenz[cd]azulenes

artículo científico publicado en 2002

Synthesis of dihydropyrimidine α,γ-diketobutanoic acid derivatives targeting HIV integrase

artículo científico publicado en 2015

Synthesis of isotopically labeled D-[1'-13C]ribonucleoside phosphoramidites

scientific article published on 01 March 2001

Synthesis of new C5-(1-substituted-1,2,3-triazol-4 or 5-yl)-2'-deoxyuridines and their antiviral evaluation

artículo científico publicado en 2010

Synthesis of water-compatible imprinted polymers of in situ produced fructosazine and 2,5-deoxyfructosazine ⬇️

artículo científico publicado el 22 de julio de 2012

The Preparation of Trisubstituted Alkenyl Nucleoside Phosphonates under Ultrasound-Assisted Olefin Cross-Metathesis

artículo científico publicado en 2013

Thiopurine Derivative-Induced Fpg/Nei DNA Glycosylase Inhibition: Structural, Dynamic and Functional Insights

scientific article published on 17 March 2020

Lista de obras de Luigi André Agrofoglio

3'-(1,2,3-Triazol-1-yl)-3'-deoxythymidine analogs as substrates for human and Ureaplasma parvum thymidine kinase for structure-activity investigations.

Active site labeling of cysteine cathepsins by a straightforward diazomethylketone probe derived from the N-terminus of human cystatin C.

Alkyne-Azide Click Chemistry Mediated Carbanucleosides Synthesis

Analysis and validation of the phosphorylated metabolites of two anti-human immunodeficiency virus nucleotides (stavudine and didanosine) by pressure-assisted CE-ESI-MS/MS in cell extracts: sensitivity enhancement by the use of perfluorinated acids

Artificial receptors for the extraction of nucleoside metabolite 7-methylguanosine from aqueous media made by molecular imprinting.

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-2.

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-3

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-5

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-6

Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes⁻4

Combination of computational methods, adsorption isotherms and selectivity tests for the conception of a mixed non-covalent-semi-covalent molecularly imprinted polymer of vanillin.

Cross-Metathesis Mediated Synthesis of New Acyclic Nucleoside Phosphonates

Design and Synthesis of Various 5'-Deoxy-5'-(4-Substituted-1,2,3-Triazol-1-yl)-Uridine Analogues as Inhibitors of Mycobacterium tuberculosis Mur Ligases

Determination at ppb level of an anti-human immunodeficiency virus nucleoside drug by capillary electrophoresis-electrospray ionization tandem mass spectrometry.

Efficient synthesis of D-[1'-13C]-ribonucleosides for incorporation into oligo-RNA

Efficient synthesis of unprotected C-5-aryl/heteroaryl-2'-deoxyuridine via a Suzuki-Miyaura reaction in aqueous media.

Evaluation of molecularly imprinted polymers using 2',3',5'-tri-O-acyluridines as templates for pyrimidine nucleoside recognition

HPLC and mass spectrometry analysis of the enzymatic hydrolysis of anti-HIV pronucleotide diastereomers.

Highly convergent synthesis and antiviral activity of (E)-but-2-enyl nucleoside phosphonoamidates

Human and viral nucleoside/nucleotide kinases involved in antiviral drug activation: structural and catalytic properties.

Inhibition of human immunodeficiency virus type 1 reverse transcriptase by the 5'-triphosphate beta enantiomers of cytidine analogs

Liquid chromatographic separation of phosphoramidate diastereomers on a polysaccharide-type chiral stationary phase.

Looking for new pyrimidine acyclic nucleotide analogues designed for phosphorylation by human UMP-CMP kinase.

Love Acoustic Wave-Based Devices and Molecularly-Imprinted Polymers as Versatile Sensors for Electronic Nose or Tongue for Cancer Monitoring.

Mass spectrometry based methods for analysis of nucleosides as antiviral drugs and potential tumor biomarkers

Microwave-Assisted Silylation-Amination of Uracil Acyclonucleosides to 4-Alkylamino-2(1H)-Pyrimidinone Analogues

Microwave-assisted syntheses of nucleosides and their precursors.

Molecularly imprinted polymer of 5-methyluridine for solid-phase extraction of pyrimidine nucleoside cancer markers in urine.

Novel antiviral C5-substituted pyrimidine acyclic nucleoside phosphonates selected as human thymidylate kinase substrates

Nucleotide binding to human UMP-CMP kinase using fluorescent derivatives -- a screening based on affinity for the UMP-CMP binding site

Olefin metathesis route to antiviral nucleosides

Palladium-assisted routes to nucleosides.

Phosphorylation of dGMP analogs by vaccinia virus TMP kinase and human GMP kinase

Potential and perspectives of cyclonucleosides.

Preparation of acyclo nucleoside phosphonate analogues based on cross-metathesis

Recent progress for the synthesis of selected carbocyclic nucleosides

Selective inhibition of human cathepsin S by 2,4,6-trisubstituted 1,3,5-triazine analogs

Simultaneous analysis of several antiretroviral nucleosides in rat-plasma by high-performance liquid chromatography with UV using acetic acid/hydroxylamine buffer Test of this new volatile medium-pH for HPLC-ESI-MS/MS.

Simultaneous quantitation of nucleoside HIV-1 reverse transcriptase inhibitors by short-end injection capillary electrochromatography on a beta-cyclodextrin-bonded silica stationary phase.

Sonication-Assisted Synthesis of(E)-2-Methyl-but-2-enyl Nucleoside Phosphonate Prodrugs

Specificity enhancement with LC-positive ESI-MS/MS for the measurement of nucleotides: application to the quantitative determination of carbovir triphosphate, lamivudine triphosphate and tenofovir diphosphate in human peripheral blood mononuclear ce

Straightforward synthesis of 2,4,6-trisubstituted 1,3,5-triazine compounds targeting cysteine cathepsins K and S.

Study of Copper(I) Catalysts for the Synthesis of Carbanucleosides via Azide-Alkyne 1,3-Dipolar Cycloaddition

Study of Different Copper (I) Catalysts for the “Click Chemistry” Approach to Carbanucleosides

Synthesis and Anti-HIV Evaluation of 3′-Triazolo Nucleosides ⬇️

Synthesis and antiviral activity of novel acyclic nucleosides in the 5-alkynyl- and 6-alkylfuro[2,3-d]pyrimidine series.

Synthesis and antiviral evaluation of C5-substituted-(1,3-diyne)-2'-deoxyuridines.

Synthesis and antiviral evaluation of bis(POM) prodrugs of (E)-[4′-phosphono-but-2′-en-1′-yl]purine nucleosides

Synthesis and broad spectrum antiviral evaluation of bis(POM) prodrugs of novel acyclic nucleosides

Synthesis and characterization of various 5'-dye-labeled ribonucleosides

Synthesis of 1,2,3-triazolo-carbanucleoside analogues of ribavirin targeting an HCV in replicon.

Synthesis of 5'-thioalkyl, sulfoxide and sulfone pyrimidine nucleosides

Synthesis of 5-haloethynyl- and 5-(1,2-dihalo)vinyluracil nucleosides: antiviral activity and cellular toxicity.

Synthesis of a molecularly imprinted polymer to isolate glucosamine from plant extracts by an ionic-non-covalent dual approach

Synthesis of a novel heterocyclic ring system: 2-thia-3,5,6,7,9-pentaazabenz[cd]azulenes

Synthesis of dihydropyrimidine α,γ-diketobutanoic acid derivatives targeting HIV integrase

Synthesis of isotopically labeled D-[1'-13C]ribonucleoside phosphoramidites

Synthesis of new C5-(1-substituted-1,2,3-triazol-4 or 5-yl)-2'-deoxyuridines and their antiviral evaluation

Synthesis of water-compatible imprinted polymers of in situ produced fructosazine and 2,5-deoxyfructosazine ⬇️

The Preparation of Trisubstituted Alkenyl Nucleoside Phosphonates under Ultrasound-Assisted Olefin Cross-Metathesis

Thiopurine Derivative-Induced Fpg/Nei DNA Glycosylase Inhibition: Structural, Dynamic and Functional Insights