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A dual read-out assay to evaluate the potency of compounds active against Mycobacterium tuberculosis

artículo científico publicado en 2013

Advancement of Imidazo[1,2-a]pyridines with Improved Pharmacokinetics and Nanomolar Activity Against Mycobacterium tuberculosis

artículo científico publicado en 2013

Advent of Imidazo[1,2-a]pyridine-3-carboxamides with Potent Multi- and Extended Drug Resistant Antituberculosis Activity

artículo científico publicado en 2011

Allylic thiocyanates as a new class of antitubercular agents

artículo científico publicado en 2012

Bactericidal activity of an imidazo[1, 2-a]pyridine using a mouse M. tuberculosis infection model

artículo científico publicado en 2014

ChemInform Abstract: One-Step Syntheses of Nitrofuranyl Benzimidazoles that Are Active Against Multidrug-Resistant Bacteria

ChemInform Abstract: Utilization of the Suzuki Coupling to Enhance the Antituberculosis Activity of Aryloxazoles

Design, synthesis, and study of a mycobactin-artemisinin conjugate that has selective and potent activity against tuberculosis and malaria

artículo científico publicado en 2011

Generation and exploration of new classes of antitubercular agents: The optimization of oxazolines, oxazoles, thiazolines, thiazoles to imidazo[1,2-a]pyridines and isomeric 5,6-fused scaffolds

artículo científico publicado en 2012

Imidazo[1,2-a]Pyridine-3-Carboxamides Are Active Antimicrobial Agents against Mycobacterium avium Infection In Vivo

artículo científico publicado en 2016

N-((1-benzyl-1H-1,2,3-triazol-4-yl)methyl)arylamide as a new scaffold that provides rapid access to antimicrotubule agents: synthesis and evaluation of antiproliferative activity against select cancer cell lines

artículo científico publicado en 2010

One-step syntheses of nitrofuranyl benzimidazoles that are active against multidrug-resistant bacteria

artículo científico publicado en 2011

Preparation and Evaluation of Potent Pentafluorosulfanyl-Substituted Anti-Tuberculosis Compounds.

artículo científico publicado en 2017

Scaffold-switching: an exploration of 5,6-fused bicyclic heteroaromatics systems to afford antituberculosis activity akin to the imidazo[1,2-a]pyridine-3-carboxylates

artículo científico publicado en 2014

Streamlined Processes for the Synthesis of a Farnesyl Transferase Inhibitor Drug Candidate

Structure-Based Mechanism for Oxidative Decarboxylation Reactions Mediated by Amino Acids and Heme Propionates in Coproheme Decarboxylase (HemQ).

scientific article published on 12 December 2016

Structure-activity relationship of new anti-tuberculosis agents derived from oxazoline and oxazole benzyl esters

artículo científico publicado en 2010

Syntheses and biological studies of novel spiropiperazinyl oxazolidinone antibacterial agents using a spirocyclic diene derived acylnitroso Diels-Alder reaction

artículo científico publicado en 2012

Thiolates chemically induce redox activation of BTZ043 and related potent nitroaromatic anti-tuberculosis agents

artículo científico publicado en 2013

UTILIZTION OF THE SUZUKI COUPLING TO ENHANCE THE ANTITUBERCULOSIS ACTIVITY OF ARYL OXAZOLES.

artículo científico publicado en 2010

Unusual Peroxide-Dependent, Heme-Transforming Reaction Catalyzed by HemQ.

artículo científico publicado en 2015

Utilization of microbial iron assimilation processes for the development of new antibiotics and inspiration for the design of new anticancer agents

artículo científico publicado en 2009