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Lista de obras de Marta Artola

1,6-Cyclophellitol Cyclosulfates: A New Class of Irreversible Glycosidase Inhibitor

artículo científico publicado en 2017

A Divergent Synthesis ofl-arabino- andd-xylo-Configured Cyclophellitol Epoxides and Aziridines

Activity-Based Probes for Glycosidases: Profiling and Other Applications

artículo científico publicado en 2017

Activity-based probes for functional interrogation of retaining β-glucuronidases

artículo científico publicado en 2017

An overview of activity-based probes for glycosidases

artículo científico publicado en 2019

Carba-cyclophellitols Are Neutral Retaining-Glucosidase Inhibitors.

artículo científico publicado en 2017

Chemical Proteomics Identifies SLC25A20 as a Functional Target of the Ingenol Class of Actinic Keratosis Drugs

artículo científico publicado en 2017

Competitive and Covalent Inhibitors of Human Lysosomal Retaining Exoglucosidases

Direct Stereoselective Aziridination of Cyclohexenols with 3-Amino-2-(trifluoromethyl)quinazolin-4(3H )-one in the Synthesis of Cyclitol Aziridine Glycosidase Inhibitors

scientific article published on 11 January 2019

Discovering the Microbial Enzymes Driving Drug Toxicity with Activity-Based Protein Profiling

scientific article published on 12 December 2019

Distinguishing the differences in beta-glycosylceramidase folds, dynamics, and actions informs therapeutic uses

article

Effective GTP-Replacing FtsZ Inhibitors and Antibacterial Mechanism of Action

scientific article published on 30 December 2014

Functionalized Cyclophellitols Are Selective Glucocerebrosidase Inhibitors and Induce a Bona Fide Neuropathic Gaucher Model in Zebrafish

artículo científico publicado en 2019

Gluco-1 H-imidazole: A New Class of Azole-Type β-Glucosidase Inhibitor.

artículo científico publicado en 2018

Glycosphingolipids and lysosomal storage disorders as illustrated by gaucher disease

scientific article published on 26 November 2019

Human glucocerebrosidase mediates formation of xylosyl-cholesterol by β-xylosidase and transxylosidase reactions

scientific article published on 23 December 2020

Identification of a Novel Orally Bioavailable Phosphodiesterase 10A (PDE10A) Inhibitor with Efficacy in Animal Models of Schizophrenia

artículo científico publicado en 2015

In vivo inactivation of glycosidases by conduritol B epoxide and cyclophellitol as revealed by activity-based protein profiling

scientific article published on 02 February 2019

New irreversible α-L-iduronidase inhibitors and activity-based probes

artículo científico publicado en 2018

New synthetic inhibitors of fatty acid synthase with anticancer activity

artículo científico publicado en 2012

Novel activity-based probes for N-acylethanolamine acid amidase

artículo científico publicado en 2017

Plant Glycosides and Glycosidases: A Treasure-Trove for Therapeutics

artículo científico publicado en 2020

Rational Design of Mechanism-Based Inhibitors and Activity-Based Probes for the Identification of Retaining α-l-Arabinofuranosidases

artículo científico publicado en 2020

Role of cannabinoid receptor CB2 in HER2 pro-oncogenic signaling in breast cancer

artículo científico publicado en 2015

Role of β-glucosidase 2 in aberrant glycosphingolipid metabolism: model of glucocerebrosidase deficiency in zebrafish

artículo científico publicado en 2019

Structure of a GH51 α-L-arabinofuranosidase from Meripilus giganteus: conserved substrate recognition from bacteria to fungi

scientific article published on 16 October 2020

Synthetic inhibitors of bacterial cell division targeting the GTP-binding site of FtsZ.

artículo científico publicado en 2013

The Synthesis of Cyclophellitol-Aziridine and Its Configurational and Functional Isomers

The structural assembly switch of cell division protein FtsZ probed with fluorescent allosteric inhibitors.

artículo científico publicado en 2016

Towards broad spectrum activity-based glycosidase probes: synthesis and evaluation of deoxygenated cyclophellitol aziridines.

artículo científico publicado en 2017

Xylose-Configured Cyclophellitols as Selective Inhibitors for Glucocerebrosidase

artículo científico publicado en 2021

α-galactosidase A1.1 can functionally complement human α-galactosidase A deficiency associated with Fabry disease

artículo científico publicado en 2018