Lista de obras - Mikhail Reibarkh - Dominio Público Uruguay

13C NMR-Based Approaches for Solving Challenging Stereochemical Problems.

artículo científico publicado en 2019

1J(CC)-edited HSQC-1,n-ADEQUATE: a new paradigm for simultaneous direct and long-range carbon-carbon correlation

scientific article published on 19 September 2012

A multifunctional catalyst that stereoselectively assembles prodrugs.

artículo científico publicado en 2017

A new class of prolylcarboxypeptidase inhibitors, part 2: the aminocyclopentanes.

artículo científico publicado en 2012

Asymmetric synthesis of cyclic indole aminals via 1,3-stereoinduction

artículo científico publicado en 2014

Band-Selective 2D HSQMBC: A Universal Technique for Detection and Measurement of 35,37Cl Isotope Effects for 13C Nuclei

artículo científico publicado en 2016

Benzimidazole-based DGAT1 inhibitors with a [3.1.0] bicyclohexane carboxylic acid moiety

artículo científico publicado en 2019

Broadband inversion of 1J(CC) responses in 1,n-ADEQUATE spectra

artículo científico publicado en 2013

Complex macrocycle exploration: parallel, heuristic, and constraint-based conformer generation using ForceGen.

artículo científico publicado en 2019

Coniothyrione: anatomy of a structure revision

artículo científico publicado en 2013

Discovery of N-[Bis(4-methoxyphenyl)methyl]-4-hydroxy-2-(pyridazin-3-yl)pyrimidine-5-carboxamide (MK-8617), an Orally Active Pan-Inhibitor of Hypoxia-Inducible Factor Prolyl Hydroxylase 1-3 (HIF PHD1-3) for the Treatment of Anemia

artículo científico publicado en 2016

Discovery of Novel Indoline Cholesterol Ester Transfer Protein Inhibitors (CETP) through a Structure-Guided Approach

artículo científico publicado en 2016

Discovery of a Photoinduced Dark Catalytic Cycle Using in Situ LED-NMR Spectroscopy

artículo científico publicado en 2018

Discovery of highly potent and efficacious MC4R agonists with spiroindane N-Me-1,2,4-triazole privileged structures for the treatment of obesity

scientific article published on 19 September 2010

Eukaryotic initiation factor (eIF) 1 carries two distinct eIF5-binding faces important for multifactor assembly and AUG selection

artículo científico publicado en 2008

Facile Quantum Yield Determination via NMR Actinometry.

artículo científico publicado en 2018

Identification of individual protein-ligand NOEs in the limit of intermediate exchange

artículo científico publicado en 2006

Interatomic potentials and solvation parameters from protein engineering data for buried residues

artículo científico publicado en 2002

Investigation of Cardiovascular Effects of Tetrahydro-β-carboline sstr3 antagonists.

artículo científico publicado en 2014

NMR study of monomer-dimer equilibrium of barstar in solution.

artículo científico publicado en 2001

Oxyfunctionalization of the Remote C-H Bonds of Aliphatic Amines by Decatungstate Photocatalysis

artículo científico publicado en 2017

PBLG as a versatile liquid crystalline medium for anisotropic NMR data acquisition

scientific article published on 01 April 2019

Promotion of a Ti-Mediated Mannich Reaction by a Proton Source

artículo científico publicado en 2015

SAR exploration at the C-3 position of tetrahydro-β-carboline sstr3 antagonists

artículo científico publicado en 2016

Secondary amine selective Petasis (SASP) bioconjugation

artículo científico publicado en 2019

Selective pharmacological targeting of a DEAD box RNA helicase.

artículo científico publicado en 2008

Small molecule inhibition of phosphatidylinositol-3,4,5-triphosphate (PIP3) binding to pleckstrin homology domains ⬇️

artículo científico publicado el 16 de noviembre de 2010

Small-molecule inhibition of the interaction between the translation initiation factors eIF4E and eIF4G

artículo científico publicado en 2007

Structure elucidation of uniformly (13)C labeled small molecule natural products

artículo científico publicado en 2015

Structure elucidation of uniformly 13C labeled small molecule natural products ⬇️

artículo científico publicado en 2015

Substituted fused bicyclic pyrrolizinones as potent, orally bioavailable hNK1 antagonists.

artículo científico publicado en 2010

The C-terminal domain of eukaryotic initiation factor 5 promotes start codon recognition by its dynamic interplay with eIF1 and eIF2β

artículo científico publicado en 2012

The Discovery of MK-4256, a Potent SSTR3 Antagonist as a Potential Treatment of Type 2 Diabetes.

artículo científico publicado en 2012

The protecting-group free selective 3'-functionalization of nucleosides

artículo científico publicado en 2017

Three-dimensional structure of toxin OSK1 from Orthochirus scrobiculosus scorpion venom

artículo científico publicado en 1997

Three‐dimensional structure of binase in solution ⬇️

artículo científico publicado el 17 de julio de 1998

Trapping‐Enrichment Multi‐dimensional Liquid Chromatography with On‐Line Deuterated Solvent Exchange for Streamlined Structure Elucidation at the Microgram Scale

Use of hydrostatic pressure for modulation of protein chemical modification and enzymatic selectivity

artículo científico publicado en 2016

Using Electron Paramagnetic Resonance Spectroscopy To Facilitate Problem Solving in Pharmaceutical Research and Development.

artículo científico publicado en 2016

Visualizing small differences using subtractive chromatographic analysis.

artículo científico publicado en 2016

[I87E mutation prevents barstar dimerization]

artículo científico publicado en 2004

pK measurements for the SAMPL6 prediction challenge for a set of kinase inhibitor-like fragments

scientific article published on 01 October 2018

Lista de obras de Mikhail Reibarkh

13C NMR-Based Approaches for Solving Challenging Stereochemical Problems.

1J(CC)-edited HSQC-1,n-ADEQUATE: a new paradigm for simultaneous direct and long-range carbon-carbon correlation

A multifunctional catalyst that stereoselectively assembles prodrugs.

A new class of prolylcarboxypeptidase inhibitors, part 2: the aminocyclopentanes.

Asymmetric synthesis of cyclic indole aminals via 1,3-stereoinduction

Band-Selective 2D HSQMBC: A Universal Technique for Detection and Measurement of 35,37Cl Isotope Effects for 13C Nuclei

Benzimidazole-based DGAT1 inhibitors with a [3.1.0] bicyclohexane carboxylic acid moiety

Broadband inversion of 1J(CC) responses in 1,n-ADEQUATE spectra

Complex macrocycle exploration: parallel, heuristic, and constraint-based conformer generation using ForceGen.

Coniothyrione: anatomy of a structure revision

Discovery of N-[Bis(4-methoxyphenyl)methyl]-4-hydroxy-2-(pyridazin-3-yl)pyrimidine-5-carboxamide (MK-8617), an Orally Active Pan-Inhibitor of Hypoxia-Inducible Factor Prolyl Hydroxylase 1-3 (HIF PHD1-3) for the Treatment of Anemia

Discovery of Novel Indoline Cholesterol Ester Transfer Protein Inhibitors (CETP) through a Structure-Guided Approach

Discovery of a Photoinduced Dark Catalytic Cycle Using in Situ LED-NMR Spectroscopy

Discovery of highly potent and efficacious MC4R agonists with spiroindane N-Me-1,2,4-triazole privileged structures for the treatment of obesity

Eukaryotic initiation factor (eIF) 1 carries two distinct eIF5-binding faces important for multifactor assembly and AUG selection

Facile Quantum Yield Determination via NMR Actinometry.

Identification of individual protein-ligand NOEs in the limit of intermediate exchange

Interatomic potentials and solvation parameters from protein engineering data for buried residues

Investigation of Cardiovascular Effects of Tetrahydro-β-carboline sstr3 antagonists.

NMR study of monomer-dimer equilibrium of barstar in solution.

Oxyfunctionalization of the Remote C-H Bonds of Aliphatic Amines by Decatungstate Photocatalysis

PBLG as a versatile liquid crystalline medium for anisotropic NMR data acquisition

Promotion of a Ti-Mediated Mannich Reaction by a Proton Source

SAR exploration at the C-3 position of tetrahydro-β-carboline sstr3 antagonists

Secondary amine selective Petasis (SASP) bioconjugation

Selective pharmacological targeting of a DEAD box RNA helicase.

Small molecule inhibition of phosphatidylinositol-3,4,5-triphosphate (PIP3) binding to pleckstrin homology domains ⬇️

Small-molecule inhibition of the interaction between the translation initiation factors eIF4E and eIF4G

Structure elucidation of uniformly (13)C labeled small molecule natural products

Structure elucidation of uniformly 13C labeled small molecule natural products ⬇️

Substituted fused bicyclic pyrrolizinones as potent, orally bioavailable hNK1 antagonists.

The C-terminal domain of eukaryotic initiation factor 5 promotes start codon recognition by its dynamic interplay with eIF1 and eIF2β

The Discovery of MK-4256, a Potent SSTR3 Antagonist as a Potential Treatment of Type 2 Diabetes.

The protecting-group free selective 3'-functionalization of nucleosides

Three-dimensional structure of toxin OSK1 from Orthochirus scrobiculosus scorpion venom

Three‐dimensional structure of binase in solution ⬇️

Trapping‐Enrichment Multi‐dimensional Liquid Chromatography with On‐Line Deuterated Solvent Exchange for Streamlined Structure Elucidation at the Microgram Scale

Use of hydrostatic pressure for modulation of protein chemical modification and enzymatic selectivity

Using Electron Paramagnetic Resonance Spectroscopy To Facilitate Problem Solving in Pharmaceutical Research and Development.

Visualizing small differences using subtractive chromatographic analysis.

[I87E mutation prevents barstar dimerization]

pK measurements for the SAMPL6 prediction challenge for a set of kinase inhibitor-like fragments

pKa measurements for the SAMPL6 prediction challenge for a set of kinase inhibitor-like fragments