Lista de obras - Ernesto G. Occhiato - Dominio Público Uruguay

19-Nor-10-azasteroids, a New Class of Steroid 5α-Reductase Inhibitors. 2.1X-ray Structure, Molecular Modeling, Conformational Analysis of 19-Nor-10-azasteroids and Comparison with 4-Azasteroids and 6-Azasteroids

artículo científico publicado en 1997

19-Nor-10-azasteroids. 5.(1) A Synthetic Strategy for the Preparation of (+)-17-(3-Pyridyl)-(5beta)-10-azaestra-1,16- dien-3-one, a Novel Potential Inhibitor for Human Cytochrome P450(17)(alpha) (17alpha-Hydroxylase/C(17,20)-lyase)

artículo científico publicado en 1999

19-nor-10-azasteroids: a novel class of inhibitors for human steroid 5alpha-reductases 1 and 2

scientific article published on 01 March 1997

5 alpha-reductase inhibitors, chemical and clinical models.

artículo científico publicado en 1998

A Short and Efficient Route to Enantiopure 3,5-Diarylpyrrolizidines

artículo científico publicado en 1999

A new class of conjugated strigolactone analogues with fluorescent properties: synthesis and biological activity

artículo científico publicado en 2009

A novel allergen-adjuvant conjugate suitable for specific immunotherapy of respiratory allergy

artículo científico publicado en 2013

Benzo[c]quinolizin-3-ones: a novel class of potent and selective nonsteroidal inhibitors of human steroid 5alpha-reductase 1

artículo científico publicado en 2000

Cyclopropane pipecolic acids as templates for linear and cyclic peptidomimetics: application in the synthesis of an Arg-Gly-Asp (RGD)-containing peptide as an αvβ3 integrin ligand

artículo científico publicado en 2014

Density functional studies on the Nazarov reaction involving cyclic systems

artículo científico publicado en 2006

Effect of C-ring modifications in benzo[c]quinolizin-3-ones, new selective inhibitors of human 5 alpha-reductase 1.

artículo científico publicado en 2001

High-performance liquid chromatographic determination of 3,5-dimethylhippuric acid in the occupational exposure to trimethylbenzenes

artículo científico publicado el 20 de mayo de 1992

Introduction of the new dipeptide isostere 7-endo-BtA as reverse turn inducer in a Bowman-Birk proteinase inhibitor: synthesis and conformational analysis.

artículo científico publicado en 2001

Lactam-derived Vinyl Triflates and Phosphates in the Synthesis of N-heterocycles

Low molecular weight, non-peptidic agonists of TrkA receptor with NGF-mimetic activity

artículo científico publicado en 2012

Modification of the aza-robinson annulation for the synthesis of 4-methyl-benzo[c]quinolizin-3-ones, potent inhibitors of steroid 5alpha-reductase 1.

artículo científico publicado en 2000

New Potent Fluorescent Analogues of Strigolactones: Synthesis and Biological Activity in Parasitic Weed Germination and Fungal Branching

New synthetic approach to cyclopenta-fused heterocycles based upon a mild Nazarov reaction.

artículo científico publicado en 2003

New synthetic approach to cyclopenta-fused heterocycles based upon a mild nazarov reaction. 2. Further studies on the torquoselectivity

scientific article published on 01 October 2004

One-Pot Access to 1,7a-Dihydro-1,3a-ethano-indene and 1,8a-Dihydro-1,3a-ethano-azulene Skeletons by a Sequential Gold(I)-Catalyzed Propargyl Claisen Rearrangement/Nazarov Cyclization/[4+2] Cycloaddition Reaction

scientific article published on 26 March 2020

Pentannulation Reaction by Tandem Gold(I)-Catalyzed Propargyl Claisen Rearrangement/Nazarov Cyclization of Enynyl Vinyl Ethers

scientific article published on 23 July 2018

Pentannulation of N-heterocycles by a tandem gold-catalyzed [3,3]-rearrangement/Nazarov reaction of propargyl ester derivatives: a computational study on the crucial role of the nitrogen atom

artículo científico publicado en 2020

Pharmacokinetics of 4-hydroxyandrostenedione in man after intramuscular injection of different formulations and the effect of this drug on plasma aromatizable androgens and 17β-estradiol concentrations

artículo científico publicado en 1993

Predicting reactivity and stereoselectivity in the Nazarov reaction: a combined computational and experimental study

artículo científico publicado en 2008

Preparation and cycloaddition reactions of enantiopure 2-(N-acylamino)-1,3-dienes for the synthesis of octahydroquinoline derivatives

artículo científico publicado en 2003

Remote stereocontrol in the Nazarov reaction: a new approach to the core of roseophilin.

artículo científico publicado en 2005

Selective non-steroidal inhibitors of 5 alpha-reductase type 1.

artículo científico publicado en 2004

Stereodivergent synthesis of 5-aminopipecolic acids and application in the preparation of a cyclic RGD peptidomimetic as a nanomolar αVβ3 integrin ligand

artículo científico publicado en 2018

Stereoselective Synthesis of Spirocyclic Ketones by Nazarov Reaction

artículo científico publicado en 2005

Strigolactone analogs as molecular probes in chasing the (SLs) receptor/s: design and synthesis of fluorescent labeled molecules.

artículo científico publicado en 2012

Structure–Function Relations of Strigolactone Analogs: Activity as Plant Hormones and Plant Interactions ⬇️

artículo científico publicado el 8 de diciembre de 2012

Suzuki reaction of vinyl triflates from six- and seven-membered N-alkoxycarbonyl lactams with boronic acids and esters.

artículo científico publicado en 2001

Synthesis and activity of 8-substituted benzo[c]quinolizin-3-ones as dual inhibitors of human 5alpha-reductases 1 and 2.

artículo científico publicado en 2005

Synthesis and conformational analysis of peptides embodying 2,3-methanopipecolic acids.

artículo científico publicado en 2017

Synthesis of 8-chloro-benzo[c]quinolizin-3-ones as potent and selective inhibitors of human steroid 5alpha-reductase 1

artículo científico publicado en 2000

Synthesis of Indenes by Tandem Gold(I)-Catalyzed Claisen Rearrangement/Hydroarylation Reaction of Propargyl Vinyl Ethers

scientific article published on 06 May 2019

Synthesis of Weinreb amides via Pd-catalyzed aminocarbonylation of heterocyclic-derived triflates

artículo científico publicado en 2008

Synthesis of benzo[c]quinolizin-3-ones: selective non-steroidal inhibitors of steroid 5 alpha-reductase 1

artículo científico publicado en 1998

Synthesis of vinylogous amides by gold(I)-catalyzed cyclization of N-Boc-protected 6-alkynyl-3,4-dihydro-2H-pyridines.

artículo científico publicado en 2013

Synthesis of α-Acyl-Functionalized Azacycles by Pd-Catalyzed Cross-Coupling Reactions of α-Alkoxyboronates with Lactam-Derived Vinyl Triflates

artículo científico publicado en 2002

Synthesis, biological activity, and three-dimensional quantitative structure-activity relationship model for a series of benzo[c]quinolizin-3-ones, nonsteroidal inhibitors of human steroid 5alpha-reductase 1.

artículo científico publicado en 2004

Tailoring fluorescent strigolactones for in vivo investigations: a computational and experimental study

scientific article published on 01 May 2014

The Lewis acid-catalyzed nazarov reaction of 2-(n-methoxycarbonylamino)-1,4-pentadien-3-ones

artículo científico publicado en 2006

Total Synthesis of Bruceolline I.

artículo científico publicado en 2017

Treatment with 8-OH-modified adenine (TLR7 ligand)-allergen conjugates decreases T helper type 2-oriented murine airway inflammation

artículo científico publicado en 2015

Lista de obras de Ernesto G. Occhiato

19-Nor-10-azasteroids, a New Class of Steroid 5α-Reductase Inhibitors. 2.1X-ray Structure, Molecular Modeling, Conformational Analysis of 19-Nor-10-azasteroids and Comparison with 4-Azasteroids and 6-Azasteroids

19-Nor-10-azasteroids. 5.(1) A Synthetic Strategy for the Preparation of (+)-17-(3-Pyridyl)-(5beta)-10-azaestra-1,16- dien-3-one, a Novel Potential Inhibitor for Human Cytochrome P450(17)(alpha) (17alpha-Hydroxylase/C(17,20)-lyase)

19-nor-10-azasteroids: a novel class of inhibitors for human steroid 5alpha-reductases 1 and 2

5 alpha-reductase inhibitors, chemical and clinical models.

A Short and Efficient Route to Enantiopure 3,5-Diarylpyrrolizidines

A new class of conjugated strigolactone analogues with fluorescent properties: synthesis and biological activity

A novel allergen-adjuvant conjugate suitable for specific immunotherapy of respiratory allergy

Benzo[c]quinolizin-3-ones: a novel class of potent and selective nonsteroidal inhibitors of human steroid 5alpha-reductase 1

Cyclopropane pipecolic acids as templates for linear and cyclic peptidomimetics: application in the synthesis of an Arg-Gly-Asp (RGD)-containing peptide as an αvβ3 integrin ligand

Density functional studies on the Nazarov reaction involving cyclic systems

Effect of C-ring modifications in benzo[c]quinolizin-3-ones, new selective inhibitors of human 5 alpha-reductase 1.

High-performance liquid chromatographic determination of 3,5-dimethylhippuric acid in the occupational exposure to trimethylbenzenes

Introduction of the new dipeptide isostere 7-endo-BtA as reverse turn inducer in a Bowman-Birk proteinase inhibitor: synthesis and conformational analysis.

Lactam-derived Vinyl Triflates and Phosphates in the Synthesis of N-heterocycles

Low molecular weight, non-peptidic agonists of TrkA receptor with NGF-mimetic activity

Modification of the aza-robinson annulation for the synthesis of 4-methyl-benzo[c]quinolizin-3-ones, potent inhibitors of steroid 5alpha-reductase 1.

New Potent Fluorescent Analogues of Strigolactones: Synthesis and Biological Activity in Parasitic Weed Germination and Fungal Branching

New synthetic approach to cyclopenta-fused heterocycles based upon a mild Nazarov reaction.

New synthetic approach to cyclopenta-fused heterocycles based upon a mild nazarov reaction. 2. Further studies on the torquoselectivity

One-Pot Access to 1,7a-Dihydro-1,3a-ethano-indene and 1,8a-Dihydro-1,3a-ethano-azulene Skeletons by a Sequential Gold(I)-Catalyzed Propargyl Claisen Rearrangement/Nazarov Cyclization/[4+2] Cycloaddition Reaction

Pentannulation Reaction by Tandem Gold(I)-Catalyzed Propargyl Claisen Rearrangement/Nazarov Cyclization of Enynyl Vinyl Ethers

Pentannulation of N-heterocycles by a tandem gold-catalyzed [3,3]-rearrangement/Nazarov reaction of propargyl ester derivatives: a computational study on the crucial role of the nitrogen atom

Pharmacokinetics of 4-hydroxyandrostenedione in man after intramuscular injection of different formulations and the effect of this drug on plasma aromatizable androgens and 17β-estradiol concentrations

Predicting reactivity and stereoselectivity in the Nazarov reaction: a combined computational and experimental study

Preparation and cycloaddition reactions of enantiopure 2-(N-acylamino)-1,3-dienes for the synthesis of octahydroquinoline derivatives

Remote stereocontrol in the Nazarov reaction: a new approach to the core of roseophilin.

Selective non-steroidal inhibitors of 5 alpha-reductase type 1.

Stereodivergent synthesis of 5-aminopipecolic acids and application in the preparation of a cyclic RGD peptidomimetic as a nanomolar αVβ3 integrin ligand

Stereoselective Synthesis of Spirocyclic Ketones by Nazarov Reaction

Strigolactone analogs as molecular probes in chasing the (SLs) receptor/s: design and synthesis of fluorescent labeled molecules.

Structure–Function Relations of Strigolactone Analogs: Activity as Plant Hormones and Plant Interactions ⬇️

Suzuki reaction of vinyl triflates from six- and seven-membered N-alkoxycarbonyl lactams with boronic acids and esters.

Synthesis and activity of 8-substituted benzo[c]quinolizin-3-ones as dual inhibitors of human 5alpha-reductases 1 and 2.

Synthesis and conformational analysis of peptides embodying 2,3-methanopipecolic acids.

Synthesis of 8-chloro-benzo[c]quinolizin-3-ones as potent and selective inhibitors of human steroid 5alpha-reductase 1

Synthesis of Indenes by Tandem Gold(I)-Catalyzed Claisen Rearrangement/Hydroarylation Reaction of Propargyl Vinyl Ethers

Synthesis of Weinreb amides via Pd-catalyzed aminocarbonylation of heterocyclic-derived triflates

Synthesis of benzo[c]quinolizin-3-ones: selective non-steroidal inhibitors of steroid 5 alpha-reductase 1

Synthesis of vinylogous amides by gold(I)-catalyzed cyclization of N-Boc-protected 6-alkynyl-3,4-dihydro-2H-pyridines.

Synthesis of α-Acyl-Functionalized Azacycles by Pd-Catalyzed Cross-Coupling Reactions of α-Alkoxyboronates with Lactam-Derived Vinyl Triflates

Synthesis, biological activity, and three-dimensional quantitative structure-activity relationship model for a series of benzo[c]quinolizin-3-ones, nonsteroidal inhibitors of human steroid 5alpha-reductase 1.

Tailoring fluorescent strigolactones for in vivo investigations: a computational and experimental study

The Lewis acid-catalyzed nazarov reaction of 2-(n-methoxycarbonylamino)-1,4-pentadien-3-ones

Total Synthesis of Bruceolline I.

Treatment with 8-OH-modified adenine (TLR7 ligand)-allergen conjugates decreases T helper type 2-oriented murine airway inflammation