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Lista de obras de Sebastiano Intagliata

Benzimidazolone-based selective σ2 receptor ligands: Synthesis and pharmacological evaluation

scientific article published on 09 January 2019

Characterization of Sigma 1 Receptor Antagonist CM-304 and Its Analog, AZ-66: Novel Therapeutics Against Allodynia and Induced Pain.

artículo científico publicado en 2019

Design and synthesis of new homo and hetero bis-piperazinyl-1-propanone derivatives as 5-HT7R selective ligands over 5-HT1AR.

artículo científico publicado en 2016

Divergent Cytotoxic and Metabolically Stimulative Functions of Sigma-2 Receptors: Structure-Activity Relationships of 6-Acetyl-3-(4-(4-(4-fluorophenyl)piperazin-1-yl)butyl)benzo[d]oxazol-2(3H)-one (SN79) Derivatives

scientific article published on 07 December 2018

Ginseng and heme oxygenase-1: The link between an old herb and a new protective system

artículo científico publicado en 2019

Heme Oxygenase-2 (HO-2) as a therapeutic target: Activators and inhibitors

artículo científico publicado en 2019

In Vitro Antioxidant and Anti-Glycation Activity of Resveratrol and Its Novel Triester with Trolox

artículo científico publicado en 2020

New Arylethanolimidazole Derivatives as HO-1 Inhibitors with Cytotoxicity against MCF-7 Breast Cancer Cells

scientific article published on 11 March 2020

New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines derivatives as 5-HT7 and 5-HT1A receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies

artículo científico publicado en 2016

Novel Structural Insight into Inhibitors of Heme Oxygenase-1 (HO-1) by New Imidazole-Based Compounds: Biochemical and In Vitro Anticancer Activity Evaluation

artículo científico publicado en 2018

Protective Effects of Caffeic Acid Phenethyl Ester (CAPE) and Novel Cape Analogue as Inducers of Heme Oxygenase-1 in Streptozotocin-Induced Type 1 Diabetic Rats

scientific article published on 17 May 2019

Solid Lipid Nanoparticles Loading Idebenone Ester with Pyroglutamic Acid: In Vitro Antioxidant Activity and In Vivo Topical Efficacy

artículo científico publicado en 2018

Strategies to Improve Resveratrol Systemic and Topical Bioavailability: An Update

artículo científico publicado en 2019

Structure–Activity Relationships and Therapeutic Potentials of 5-HT7 Receptor Ligands: An Update

artículo científico publicado en 2018

Structure–activity relationships and molecular modeling studies of novel arylpiperazinylalkyl 2-benzoxazolones and 2-benzothiazolones as 5-HT7 and 5-HT1A receptor ligands

artículo científico publicado en 2014

Synthesis and Molecular Modelling Studies of New 1,3-Diaryl-5-Oxo-Proline Derivatives as Endothelin Receptor Ligands

scientific article published on 17 April 2020

Synthesis and binding properties of new long-chain 4-substituted piperazine derivatives as 5-HT₁A and 5-HT₇ receptor ligands

artículo científico publicado en 2015

Synthesis, in vitro and in silico studies of HO-1 inducers and lung antifibrotic agents

scientific article published on 01 July 2019

Synthesis, in vitro and in vivo characterization of new benzoxazole and benzothiazole-based sigma receptor ligands

scientific article published on 21 April 2019

Targeting heme Oxygenase-1 with hybrid compounds to overcome Imatinib resistance in chronic myeloid leukemia cell lines

scientific article published on 17 September 2018

[1]Benzothieno[3,2-d]pyrimidine derivatives as ligands for the serotonergic 5-HT7 receptor

artículo científico publicado en 2019