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Lista de obras de Anthony G Coyne

Asymmetric electrocyclic reactions

artículo científico publicado en 2011

Correction to Fragment-Based Design of Mycobacterium tuberculosis InhA Inhibitors

artículo científico publicado en 2020

Corrigendum: Substrate Fragmentation for the Design of M. tuberculosis CYP121 Inhibitors

artículo científico publicado en 2016

Covalent inactivation of Mycobacterium thermoresistibile inosine-5'-monophosphate dehydrogenase (IMPDH)

scientific article published on 09 November 2019

Development of Inhibitors against Mycobacterium abscessus tRNA (m1G37) Methyltransferase (TrmD) Using Fragment-Based Approaches

scientific article published on 19 July 2019

Drugging challenging targets using fragment-based approaches

artículo científico publicado en 2010

Effect of DMSO on Protein Structure and Interactions Assessed by Collision-Induced Dissociation and Unfolding

artículo científico publicado en 2017

Fragment Profiling Approach to Inhibitors of the Orphan M. tuberculosis P450 CYP144A1.

artículo científico publicado en 2017

Fragment Screening against the EthR-DNA Interaction by Native Mass Spectrometry.

artículo científico publicado en 2017

Fragment-Based Approach to Targeting Inosine-5'-monophosphate Dehydrogenase (IMPDH) from Mycobacterium tuberculosis

artículo científico publicado en 2018

Fragment-Based Approaches to the Development of Mycobacterium tuberculosis CYP121 Inhibitors

artículo científico publicado en 2016

Fragment-Based Design of Mycobacterium tuberculosis InhA Inhibitors

scientific article published on 02 April 2020

Fragment-based approaches in drug discovery and chemical biology

artículo científico publicado en 2012

Fragment-based approaches to TB drugs

artículo científico publicado en 2016

Inhibiting Mycobacterium tuberculosis CoaBC by targeting an allosteric site

artículo científico publicado en 2021

Organic synthesis reactions on-water at the organic-liquid water interface

artículo científico publicado en 2016

Overcoming the Limitations of Fragment Merging: Rescuing a Strained Merged Fragment Series TargetingMycobacterium tuberculosisCYP121

artículo científico publicado en 2013

Regioselective conversion of arenes to N-aryl-1,2,3-triazoles using C-H borylation

artículo científico publicado en 2014

Small-molecule inhibitors that target protein-protein interactions in the RAD51 family of recombinases

artículo científico publicado en 2014

Spirooxindoles as novel 3D-fragment scaffolds: Synthesis and screening against CYP121 from M. tuberculosis

artículo científico publicado en 2016

Structural insights into the EthR-DNA interaction using native mass spectrometry.

artículo científico publicado en 2017

Substrate Fragmentation for the Design of M. tuberculosis CYP121 Inhibitors.

artículo científico publicado en 2016

Targeting of Fumarate Hydratase from Mycobacterium tuberculosis Using Allosteric Inhibitors with a Dimeric-Binding Mode

artículo científico publicado en 2019

The Application of HETPHOX Ligands to the Intramolecular Asymmetric Heck Reaction

The influence of water on the rates of 1,3-dipolar cycloaddition reactions: trigger points for exponential rate increases in water-organic solvent mixtures. Water-super versus water-normal dipolarophiles

artículo científico publicado en 2004

Trapping of palindromic ligands within native transthyretin prevents amyloid formation

artículo científico publicado en 2010

Understanding "on-water" catalysis of organic reactions. Effects of H+ and Li+ ions in the aqueous phase and nonreacting competitor H-bond acceptors in the organic phase: on H2O versus on D2O for Huisgen cycloadditions

artículo científico publicado en 2015

Water and organic synthesis: a focus on the in-water and on-water border. Reversal of the in-water Breslow hydrophobic enhancement of the normal endo-effect on crossing to on-water conditions for Huisgen cycloadditions with increasingly insoluble or

artículo científico publicado en 2013

Water: nature's reaction enforcer--comparative effects for organic synthesis "in-water" and "on-water".

artículo científico publicado en 2010