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Lista de obras de Samuele Maramai

(S)-2-Amino-3-(5-methyl-3-hydroxyisoxazol-4-yl)propanoic Acid (AMPA) and Kainate Receptor Ligands: Further Exploration of Bioisosteric Replacements, Structural and Biological Investigation

artículo científico publicado en 2018

A stereoselective approach to peptidomimetic BACE1 inhibitors

artículo científico publicado en 2013

Activation of the Wnt Pathway by Small Peptides: Rational Design, Synthesis and Biological Evaluation.

artículo científico publicado en 2017

Development and Pharmacological Characterization of Selective Blockers of 2-Arachidonoyl Glycerol Degradation with Efficacy in Rodent Models of Multiple Sclerosis and Pain

artículo científico publicado en 2016

Development of Potent Inhibitors of Fatty Acid Amide Hydrolase Useful for the Treatment of Neuropathic Pain

scholarly article by Margherita Brindisi et al published 30 August 2018 in ChemMedChem

Development of a practical and scalable route for the preparation of the deacetoxytubuvaline (dTuv) fragment of pretubulysin and analogs

Development of novel cyclic peptides as pro-apoptotic agents

artículo científico publicado en 2016

Discovery of potent inhibitors of human and mouse fatty acid amide hydrolases

artículo científico publicado en 2012

Disease-modifying anti-Alzheimer's drugs: inhibitors of human cholinesterases interfering with β-amyloid aggregation.

artículo científico publicado en 2014

Dopamine D3 Receptor Antagonists as Potential Therapeutics for the Treatment of Neurological Diseases

artículo científico publicado en 2016

Harnessing the pyrroloquinoxaline scaffold for FAAH and MAGL interaction: definition of the structural determinants for enzyme inhibition

scholarly article in RSC Advances, vol. 6 no. 69, 2016

Identification of a novel arylpiperazine scaffold for fatty acid amide hydrolase inhibition with improved drug disposition properties

artículo científico publicado en 2012

Multifunctional cholinesterase and amyloid Beta fibrillization modulators. Synthesis and biological investigation

artículo científico publicado en 2013

Multitarget Therapeutic Strategies for Alzheimer's Disease: Review on Emerging Target Combinations

artículo científico publicado en 2020

Phenylpyrrole-based HDAC inhibitors: synthesis, molecular modeling and biological studies

artículo científico publicado en 2016

Selective kainate receptor (GluK1) ligands structurally based upon 1H-cyclopentapyrimidin-2,4(1H,3H)-dione: synthesis, molecular modeling, and pharmacological and biostructural characterization

artículo científico publicado en 2011

Subtype Selective γ-Aminobutyric Acid Type A Receptor (GABAAR) Modulators Acting at the Benzodiazepine Binding Site: An Update

scientific article published on 05 December 2019