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Lista de obras de Damien Bosc

A new quinoline-based chemical probe inhibits the autophagy-related cysteine protease ATG4B

scientific article published in Scientific Reports

Aggrecanase-2 inhibitors based on the acylthiosemicarbazide zinc-binding group

artículo científico publicado en 2013

Catalytic site inhibition of insulin-degrading enzyme by a small molecule induces glucose intolerance in mice

artículo científico publicado en 2015

Comparative Study of the Synthesis and Structural and Physicochemical Properties of Diketopiperazines vs Aza-diketopiperazines.

artículo científico publicado en 2017

Controlling Plasma Stability of Hydroxamic Acids: A MedChem Toolbox.

artículo científico publicado en 2017

Development of fluorescent peptide substrates and assays for the key autophagy-initiating cysteine protease enzyme, ATG4B.

artículo científico publicado en 2015

Discovery of a new class of protein farnesyltransferase inhibitors in the arylthiophene series

artículo científico publicado en 2009

Highly improved antiparasitic activity after introduction of an N-benzylimidazole moiety on protein farnesyltransferase inhibitors

artículo científico publicado en 2015

Identification of ebselen as a potent inhibitor of insulin degrading enzyme by a drug repurposing screening

artículo científico publicado en 2019

Kinetic Target-Guided Synthesis: Reaching the Age of Maturity

scientific article published on 24 December 2019

Kinetic target-guided synthesis in drug discovery and chemical biology: a comprehensive facts and figures survey

artículo científico publicado en 2016

New protein farnesyltransferase inhibitors in the 3-arylthiophene 2-carboxylic acid series: diversification of the aryl moiety by solid-phase synthesis.

artículo científico publicado en 2012

Precision autophagy: Will the next wave of selective autophagy markers and specific autophagy inhibitors feed clinical pipelines?

artículo científico publicado en 2015

Structure-activity relationships of imidazole-derived 2-[N-carbamoylmethyl-alkylamino]acetic acids, dual binders of human insulin-degrading enzyme.

artículo científico publicado en 2014