Lista de obras - Pascal Dumy - Dominio Público Uruguay

1-Ethoxyethylidene, a new group for the stepwise SPPS of aminooxyacetic acid containing peptides.

artículo científico publicado en 2008

3-nitro-3-deaza-2'-deoxyadenosine as a versatile photocleavable 2'-deoxyadenosine mimic.

artículo científico publicado en 2004

67Cu-Radiolabeling of a multimeric RGD peptide for αVβ3 integrin-targeted radionuclide therapy: stability, therapeutic efficacy, and safety studies in mice

artículo científico publicado en 2017

A cyclodecapeptide ligand to vitamin B12.

artículo científico publicado en 2008

A dynamic combinatorial approach for identifying side groups that stabilize DNA-templated supramolecular self-assemblies.

artículo científico publicado en 2015

A gadolinium-binding cyclodecapeptide with a large high-field relaxivity involving second-sphere water

artículo científico publicado en 2009

A highly convergent approach to O- and N-linked glycopeptide analogues

scientific article published on 01 August 1999

A multimeric quinacrine conjugate as a potential inhibitor of Alzheimer's beta-amyloid fibril formation.

artículo científico publicado en 2008

Access to Biomolecular Assemblies through One-Pot Triple Orthogonal Chemoselective Ligations

artículo científico publicado en 2011

Access to bifunctionalized biomolecular platforms using oxime ligation.

artículo científico publicado en 2014

Activatable fluorescent probes for tumour-targeting imaging in live mice

artículo científico publicado en 2006

Activatable probes for non-invasive small animal fluorescence imaging

Amino- and glycoconjugates of pyrido[4,3,2-kl]acridine. Synthesis, antitumor activity, and DNA binding

artículo científico publicado en 2006

Amphipol mediated surface immobilization of FhuA: a platform for label-free detection of the bacteriophage protein pb5.

artículo científico publicado en 2012

An oxime-based glycocluster microarray.

artículo científico publicado en 2017

Antitumor activity of a self-adjuvanting glyco-lipopeptide vaccine bearing B cell, CD4+ and CD8+ T cell epitopes.

artículo científico publicado en 2008

Application of click-click chemistry to the synthesis of new multivalent RGD conjugates.

artículo científico publicado en 2010

Benzoxaboroles as Efficient Inhibitors of the β-Carbonic Anhydrases from Pathogenic Fungi: Activity and Modeling Study

artículo científico publicado en 2017

Bioactive clusters promoting cell penetration and nucleic acid complexation for drug and gene delivery applications: from designed to self-assembled and responsive systems.

artículo científico publicado en 2016

Biomolecular assembly by iterative oxime ligations

scientific article published on 28 March 2009

Carbonic Anhydrase Glycoinhibitors belonging to the Aminoxysulfonamide Series.

artículo científico publicado en 2015

Cell adhesion through clustered ligand on fluid supported lipid bilayers

artículo científico publicado en 2010

Chemical and biological evaluations of an (111)in-labeled RGD-peptide targeting integrin alpha(V) beta(3) in a preclinical tumor model.

artículo científico publicado en 2008

Chemical synthesis, DNA incorporation and biological study of a new photocleavable 2'-deoxyadenosine mimic.

artículo científico publicado en 2009

Chemoselectively Template-Assembled Glycoconjugates as Mimics for Multivalent Presentation of Carbohydrates

artículo científico publicado en 2003

Chemoselectively addressable HCan building blocks in peptide synthesis:L-homocanaline derivatives

artículo científico publicado en 1998

Clicked tacrine conjugates as acetylcholinesterase and β-amyloid directed compounds

scientific article published on 10 December 2010

Control of Amyloid β-Peptide Protofibril Formation by a Designed Template Assembly

scholarly article by Gunnar T. Dolphin et al published 21 April 2006 in Angewandte Chemie International Edition

Cyclic peptides bearing a side-chain tail: a tool to model the structure and reactivity of protein zinc sites.

artículo científico publicado en 2008

Cyclodecapeptides to mimic the radical site of tyrosyl-containing proteins

scholarly article by Mohammed Akhter Hossain published in January 2006

Degradable hybrid materials based on cationic acylhydrazone dynamic covalent polymers promote DNA complexation through multivalent interactions.

artículo científico

Dendri-RAFTs: a second generation of cyclopeptide-based glycoclusters

artículo científico publicado en 2011

Deoxyribonolactone lesion in DNA: synthesis of fluorinated analogues.

artículo científico publicado en 2003

Designed amyloid beta peptide fibril - a tool for high-throughput screening of fibril inhibitors

artículo científico publicado en 2007

Double threading through DNA: NMR structural study of a bis-naphthalene macrocycle bound to a thymine-thymine mismatch

artículo científico publicado en 2012

Drug development in oncology assisted by noninvasive optical imaging.

artículo científico publicado en 2009

Dynamic Expression of DNA Complexation with Self-assembled Biomolecular Clusters

artículo científico publicado en 2015

Effective Access to Multivalent Inhibitors of Carbonic Anhydrases Promoted by Peptide Bioconjugation.

artículo científico publicado en 2017

Efficient conjugation and characterization of distamycin-based peptides with selected oligonucleotide stretches.

artículo científico publicado en 2004

Efficient conjugation of oligonucleotides through aromatic oxime formation.

artículo científico publicado en 2009

Efficient surface patterning of oligonucleotides inside a glass capillary through oxime bond formation.

artículo científico publicado en 2007

Electrochemical detection of Arachis hypogaea (peanut) agglutinin binding to monovalent and clustered lactosyl motifs immobilized on a polypyrrole film.

artículo científico publicado en 2005

Electrochemically controlled adsorption of Fc-functionalized polymers on beta-CD-modified self-assembled monolayers.

artículo científico publicado en 2010

Emerging trends in enzyme inhibition by multivalent nanoconstructs.

artículo científico

Enhancing the Proline Effect: Pseudo-Prolines for TailoringCis/TransIsomerization

scientific article published in 1998

Expanding the scope of oxime ligation: facile synthesis of large cyclopeptide-based glycodendrimers

artículo científico publicado en 2013

Fluorescent ADP sensing in physiological conditions based on cooperative inhibition of a miniature esterase

artículo científico publicado en 2007

Fluorescent Silica Nanoparticles with Multivalent Inhibitory Effects towards Carbonic Anhydrases

artículo científico publicado en 2015

Glycoside and peptide clustering around the octasilsesquioxane scaffold via photoinduced free-radical thiol–ene coupling. The observation of a striking glycoside cluster effect

Head-to-Tail Oxime Cyclization of Oligodeoxynucleotides for the Efficient Synthesis of Circular DNA Analogues ⬇️

artículo científico publicado el 31 de octubre de 2003

Hepatocyte Targeting and Intracellular Copper Chelation by a Thiol-Containing Glycocyclopeptide

artículo científico publicado en 2010

High affinity glycodendrimers for the lectin LecB from Pseudomonas aeruginosa

artículo científico publicado en 2013

Hydrazinolysis of Dde: Complete orthogonality with Aloc protecting groups

artículo científico publicado en 1998

Hydroxylamine-O-sulfonamide is a versatile lead compound for the development of carbonic anhydrase inhibitors.

artículo científico publicado en 2015

In Vivo Noninvasive Optical Imaging of Receptor-Mediated RGD Internalization Using Self-Quenched Cy5-Labeled RAFT-c(-RGDfK-) 4

scholarly article by Zhao-Hui Jin et al published January 2007 in Molecular imaging : official journal of the Society for Molecular Imaging

In vivo molecular imaging of myocardial angiogenesis using the αvβ3 integrin-targeted tracer 99mTc-RAFT-RGD

artículo científico publicado en 2010

In vivo optical imaging of integrin alphaV-beta3 in mice using multivalent or monovalent cRGD targeting vectors.

artículo científico publicado en 2007

Influence of Pre-organised Architecture on Cell Adhesion by Using Multivalent RGD Compounds

artículo científico publicado en 2016

Inhibition of β-carbonic anhydrases from Brucella suis with C-cinnamoyl glycosides incorporating the phenol moiety

artículo científico publicado en 2015

Linear and branched glyco-lipopeptide vaccines follow distinct cross-presentation pathways and generate different magnitudes of antitumor immunity

artículo científico publicado en 2010

Luminescent probes for optical in vivo imaging

Metal-free synthesis of imino-disaccharides and calix-iminosugars by photoinduced radical thiol-ene coupling (TEC)

scientific article published on 01 April 2020

Micro-positron emission tomography/contrast-enhanced computed tomography imaging of orthotopic pancreatic tumor-bearing mice using the αvβ₃ integrin tracer ⁶⁴Cu-labeled cyclam-RAFT-c(-RGDfK-)₄.

artículo científico publicado en 2013

Model peptides based on the binding loop of the copper metallochaperone Atx1: selectivity of the consensus sequence MxCxxC for metal ions Hg(II), Cu(I), Cd(II), Pb(II), and Zn(II)

artículo científico publicado en 2006

Multilayer assemblies of polyelectrolyte-gold nanoparticles for the electrocatalytic oxidation and detection of arsenic(III)

artículo científico publicado en 2012

Multivalent Carbonic Anhydrases Inhibitors

scientific article published on 28 October 2019

Multivalent DNA recognition by self-assembled clusters: deciphering structural effects by fragments screening and evaluation as siRNA vectors.

artículo científico

Multivalent RGD synthetic peptides as potent alphaVbeta3 integrin ligands.

artículo científico publicado en 2006

Multivalent glyco(cyclo)peptides ⬇️

artículo científico publicado el 21 de diciembre de 2012

N-glycosyl-N-hydroxysulfamides as potent inhibitors of Brucella suis carbonic anhydrases

artículo científico publicado en 2015

New acridone derivatives for the electrochemical DNA-hybridisation labelling.

artículo científico publicado en 2004

New method to prepare peptide-oligonucleotide conjugates through glyoxylic oxime formation.

artículo científico publicado en 2004

Nitrobenzylcarbamate prodrugs of cytotoxic acridines for potential use with nitroreductase gene-directed enzyme prodrug therapy.

artículo científico publicado en 2006

Noninvasive visualization and quantification of tumor αVβ3 integrin expression using a novel positron emission tomography probe, 64Cu-cyclam-RAFT-c(-RGDfK-)4.

artículo científico publicado en 2011

Novel model peptide for Atx1-like metallochaperones.

artículo científico publicado en 2004

Oligonucleotide sequential bis-conjugation via click-oxime and click-Huisgen procedures.

artículo científico publicado en 2010

On-bead synthesis and binding assay of chemoselectively template-assembled multivalent neoglycopeptides

artículo científico publicado en 2006

One-Pot Self-Assembly of Peptide-Based Cage-Type Nanostructures Using Orthogonal Ligations.

artículo científico publicado en 2017

One-pot approach to well-defined biomolecular assemblies by orthogonal chemoselective ligations.

artículo científico publicado en 2009

Oxime ligation: a chemoselective click-type reaction for accessing multifunctional biomolecular constructs.

artículo científico

PET imaging and biodistribution analysis of the effects of succinylated gelatin combined with L-lysine on renal uptake and retention of ⁶⁴Cu-cyclam-RAFT-c(-RGDfK-)₄ in vivo

artículo científico publicado en 2013

Photoadduct leading to crosslinking in Ru(II)-derivatized oligonucleotides.

artículo científico publicado en 2003

Photocrosslinking in ruthenium-labelled duplex oligonucleotides.

artículo científico publicado en 2003

Photomodulation of DNA-Templated Supramolecular Assemblies.

artículo científico publicado en 2017

Photoreactive threading agent that specifically binds to abasic sites in DNA.

artículo científico publicado en 2005

Phthalimide-Oxy Derivatives for 3′- or 5′-Conjugation of Oligonucleotides by Oxime Ligation and Circularization of DNA by “Bis- or Tris-Click” Oxime Ligation

Polyhedral Oligomeric Silsesquioxane (POSS) Bearing Glyoxylic Aldehyde as Clickable Platform Towards Multivalent Conjugates.

artículo científico publicado en 2017

Positron emission tomography of cerebral angiogenesis and TSPO expression in a mouse model of chronic hypoxia.

artículo científico publicado en 2017

Probing secondary interactions in biomolecular recognition by dynamic combinatorial chemistry

artículo científico

Probing the importance of π-stacking interactions in DNA-templated self-assembly of bisfunctionalized guanidinium compounds

Promotion of sugar-lectin recognition through the multiple sugar presentation offered by regioselectively addressable functionalized templates (RAFT): a QCM-D and SPR study

artículo científico publicado en 2008

Properties of Some Variants of Human β2-Microglobulin and Amyloidogenesis

artículo científico publicado en 2003

Protein design: On the threshold of functional properties ⬇️

artículo científico publicado el 1 de enero de 1998

RGD-cyclam conjugate: synthesis and potential application for positron emission tomography.

artículo científico publicado en 2010

Radiotheranostic Agent 64Cu-cyclam-RAFT-c(-RGDfK-)4 for Management of Peritoneal Metastasis in Ovarian Cancer

scientific article published on 15 September 2020

Randomized combinatorial library of heteroglycoclusters (hGC).

artículo científico publicado en 2008

Re-evaluation of binding properties of recombinant lymphocyte receptors NKR-P1A and CD69 to chemically synthesized glycans and peptides

artículo científico publicado en 2014

Reactivity of pyrido[4,3,2-kl]acridines: regioselective formation of 6-substituted derivatives.

artículo científico publicado en 2004

Redox strategy for reversible attachment of biomolecules using bifunctional linkers

artículo científico publicado en 2011

Redox-Active Biomolecular Architectures and Self-Assembled Monolayers Based on a Cyclodecapeptide Regioselectively Addressable Functional Template

artículo científico publicado en 2006

Redox-driven host-guest interactions allow the controlled release of captured cells on RGD-functionalized surfaces

artículo científico publicado en 2014

Retraction of “Synthesis of Multivalent Glycoconjugates Containing the Immunoactive LELTE Peptide: Effect of Glycosylation on Cellular Activation and Natural Killing by Human Peripheral Blood Mononuclear Cells”

artículo científico publicado en 2014

Self-assembly and chiroptical properties in supramolecular complexes of adenosine phosphates and guanidinium-bispyrene.

artículo científico publicado en 2018

Solution structure of regioselectively addressable functionalized templates: an NMR and restrained molecular dynamics investigation

scientific article published on 01 September 1996

Stabilization of the biologically active conformation of the principal neutralizing determinant of HIV-1(IIIB) containing a cis-proline surrogate: 1H NMR and molecular modeling study.

artículo científico publicado en 2006

Structural and dynamic properties of calixarene bimetallic complexes: solution versus solid-state structure of dinuclear complexes of EuIII and LuIII with substituted calix[8]arenes †

Structural and folding dynamic properties of the T70N variant of human lysozyme.

artículo científico publicado en 2003

Surface patterning of (bio)molecules onto the inner wall of fused-silica capillary tubes.

artículo científico publicado en 2008

Synthesis and activity of HIV protease inhibitors

article

Synthesis and biological characterisation of targeted pro-apoptotic peptide.

artículo científico publicado en 2008

Synthesis and biological evaluation of clicked curcumin and clicked KLVFFA conjugates as inhibitors of beta-amyloid fibril formation.

artículo científico publicado en 2009

Synthesis and evaluation of fused bispyrimidinoacridines as novel pentacyclic analogues of quadruplex-binder BRACO-19.

artículo científico publicado en 2009

Synthesis of N-acridinyl-N'-alkylguanidines: dramatic influence of amine to guanidine replacement on the physicochemical properties.

artículo científico publicado en 2008

Synthesis of heteroglycoclusters by using orthogonal chemoselective ligations

artículo científico publicado en 2012

Synthesis of multitopic neoglycopeptides displaying recognition and detection motifs

artículo científico publicado en 2005

Synthesis of multivalent glycoconjugates containing the immunoactive LELTE peptide: effect of glycosylation on cellular activation and natural killing by human peripheral blood mononuclear cells.

artículo científico publicado en 2010

Synthetic Peptide templates for molecular recognition: recent advances and applications.

artículo científico publicado en 2006

Systemic Delivery of Tumor-Targeted Bax-Derived Membrane-Active Peptides for the Treatment of Melanoma Tumors in a Humanized SCID Mouse Model.

artículo científico publicado en 2017

Targeted delivery of a proapoptotic peptide to tumors in vivo.

artículo científico publicado en 2010

Targeted delivery of activatable fluorescent pro-apoptotic peptide into live cells

scientific article published on 17 November 2008

Template-assembled synthetic G-quadruplex (TASQ): a useful system for investigating the interactions of ligands with constrained quadruplex topologies.

artículo científico

Template-directed combinatorial surface assembly for protein–protein interaction mimetics

Tethered bilayer lipid membranes on mixed self-assembled monolayers of a novel anchoring thiol: impact of the anchoring thiol density on bilayer formation

scientific article published on 28 October 2011

Tetravalent glycocyclopeptide with nanomolar affinity to wheat germ agglutinin

artículo científico publicado en 2013

The oxime bond formation as an efficient chemical tool for the preparation of 3',5'-bifunctionalised oligodeoxyribonucleotides.

artículo científico publicado en 2004

Thiol-ene and thiol-yne-based synthesis of glycodendrimers as nanomolar inhibitors of wheat germ agglutinin

Towards a self-adjuvanting multivalent B and T cell epitope containing synthetic glycolipopeptide cancer vaccine.

artículo científico publicado en 2008

Versatile Introduction of Azido Moiety into Oligonucleotides through Diazo Transfer Reaction ⬇️

artículo científico publicado el 29 de septiembre de 2011

α and βl-Fucopyranosyl oxyamines: key intermediates for the preparation of fucose-containing glycoconjugates by oxime ligation

artículo científico publicado en 2007

αVβ3 Integrin-Targeted Radionuclide Therapy with 64Cu-cyclam-RAFT-c(-RGDfK-)4.

artículo científico publicado en 2016

Lista de obras de Pascal Dumy

1-Ethoxyethylidene, a new group for the stepwise SPPS of aminooxyacetic acid containing peptides.

3-nitro-3-deaza-2'-deoxyadenosine as a versatile photocleavable 2'-deoxyadenosine mimic.

67Cu-Radiolabeling of a multimeric RGD peptide for αVβ3 integrin-targeted radionuclide therapy: stability, therapeutic efficacy, and safety studies in mice

A cyclodecapeptide ligand to vitamin B12.

A dynamic combinatorial approach for identifying side groups that stabilize DNA-templated supramolecular self-assemblies.

A gadolinium-binding cyclodecapeptide with a large high-field relaxivity involving second-sphere water

A highly convergent approach to O- and N-linked glycopeptide analogues

A multimeric quinacrine conjugate as a potential inhibitor of Alzheimer's beta-amyloid fibril formation.

Access to Biomolecular Assemblies through One-Pot Triple Orthogonal Chemoselective Ligations

Access to bifunctionalized biomolecular platforms using oxime ligation.

Activatable fluorescent probes for tumour-targeting imaging in live mice

Activatable probes for non-invasive small animal fluorescence imaging

Amino- and glycoconjugates of pyrido[4,3,2-kl]acridine. Synthesis, antitumor activity, and DNA binding

Amphipol mediated surface immobilization of FhuA: a platform for label-free detection of the bacteriophage protein pb5.

An oxime-based glycocluster microarray.

Antitumor activity of a self-adjuvanting glyco-lipopeptide vaccine bearing B cell, CD4+ and CD8+ T cell epitopes.

Application of click-click chemistry to the synthesis of new multivalent RGD conjugates.

Benzoxaboroles as Efficient Inhibitors of the β-Carbonic Anhydrases from Pathogenic Fungi: Activity and Modeling Study

Bioactive clusters promoting cell penetration and nucleic acid complexation for drug and gene delivery applications: from designed to self-assembled and responsive systems.

Biomolecular assembly by iterative oxime ligations

Carbonic Anhydrase Glycoinhibitors belonging to the Aminoxysulfonamide Series.

Cell adhesion through clustered ligand on fluid supported lipid bilayers

Chemical and biological evaluations of an (111)in-labeled RGD-peptide targeting integrin alpha(V) beta(3) in a preclinical tumor model.

Chemical synthesis, DNA incorporation and biological study of a new photocleavable 2'-deoxyadenosine mimic.

Chemoselectively Template-Assembled Glycoconjugates as Mimics for Multivalent Presentation of Carbohydrates

Chemoselectively addressable HCan building blocks in peptide synthesis:L-homocanaline derivatives

Clicked tacrine conjugates as acetylcholinesterase and β-amyloid directed compounds

Control of Amyloid β-Peptide Protofibril Formation by a Designed Template Assembly

Cyclic peptides bearing a side-chain tail: a tool to model the structure and reactivity of protein zinc sites.

Cyclodecapeptides to mimic the radical site of tyrosyl-containing proteins

Degradable hybrid materials based on cationic acylhydrazone dynamic covalent polymers promote DNA complexation through multivalent interactions.

Dendri-RAFTs: a second generation of cyclopeptide-based glycoclusters

Deoxyribonolactone lesion in DNA: synthesis of fluorinated analogues.

Designed amyloid beta peptide fibril - a tool for high-throughput screening of fibril inhibitors

Double threading through DNA: NMR structural study of a bis-naphthalene macrocycle bound to a thymine-thymine mismatch

Drug development in oncology assisted by noninvasive optical imaging.

Dynamic Expression of DNA Complexation with Self-assembled Biomolecular Clusters

Effective Access to Multivalent Inhibitors of Carbonic Anhydrases Promoted by Peptide Bioconjugation.

Efficient conjugation and characterization of distamycin-based peptides with selected oligonucleotide stretches.

Efficient conjugation of oligonucleotides through aromatic oxime formation.

Efficient surface patterning of oligonucleotides inside a glass capillary through oxime bond formation.

Electrochemical detection of Arachis hypogaea (peanut) agglutinin binding to monovalent and clustered lactosyl motifs immobilized on a polypyrrole film.

Electrochemically controlled adsorption of Fc-functionalized polymers on beta-CD-modified self-assembled monolayers.

Emerging trends in enzyme inhibition by multivalent nanoconstructs.

Enhancing the Proline Effect: Pseudo-Prolines for TailoringCis/TransIsomerization

Expanding the scope of oxime ligation: facile synthesis of large cyclopeptide-based glycodendrimers

Fluorescent ADP sensing in physiological conditions based on cooperative inhibition of a miniature esterase

Fluorescent Silica Nanoparticles with Multivalent Inhibitory Effects towards Carbonic Anhydrases

Glycoside and peptide clustering around the octasilsesquioxane scaffold via photoinduced free-radical thiol–ene coupling. The observation of a striking glycoside cluster effect

Head-to-Tail Oxime Cyclization of Oligodeoxynucleotides for the Efficient Synthesis of Circular DNA Analogues ⬇️

Hepatocyte Targeting and Intracellular Copper Chelation by a Thiol-Containing Glycocyclopeptide

High affinity glycodendrimers for the lectin LecB from Pseudomonas aeruginosa

Hydrazinolysis of Dde: Complete orthogonality with Aloc protecting groups

Hydroxylamine-O-sulfonamide is a versatile lead compound for the development of carbonic anhydrase inhibitors.

In Vivo Noninvasive Optical Imaging of Receptor-Mediated RGD Internalization Using Self-Quenched Cy5-Labeled RAFT-c(-RGDfK-) 4

In vivo molecular imaging of myocardial angiogenesis using the αvβ3 integrin-targeted tracer 99mTc-RAFT-RGD

In vivo optical imaging of integrin alphaV-beta3 in mice using multivalent or monovalent cRGD targeting vectors.

Influence of Pre-organised Architecture on Cell Adhesion by Using Multivalent RGD Compounds

Inhibition of β-carbonic anhydrases from Brucella suis with C-cinnamoyl glycosides incorporating the phenol moiety

Linear and branched glyco-lipopeptide vaccines follow distinct cross-presentation pathways and generate different magnitudes of antitumor immunity

Luminescent probes for optical in vivo imaging

Metal-free synthesis of imino-disaccharides and calix-iminosugars by photoinduced radical thiol-ene coupling (TEC)

Micro-positron emission tomography/contrast-enhanced computed tomography imaging of orthotopic pancreatic tumor-bearing mice using the αvβ₃ integrin tracer ⁶⁴Cu-labeled cyclam-RAFT-c(-RGDfK-)₄.

Model peptides based on the binding loop of the copper metallochaperone Atx1: selectivity of the consensus sequence MxCxxC for metal ions Hg(II), Cu(I), Cd(II), Pb(II), and Zn(II)

Multilayer assemblies of polyelectrolyte-gold nanoparticles for the electrocatalytic oxidation and detection of arsenic(III)

Multivalent Carbonic Anhydrases Inhibitors

Multivalent DNA recognition by self-assembled clusters: deciphering structural effects by fragments screening and evaluation as siRNA vectors.

Multivalent RGD synthetic peptides as potent alphaVbeta3 integrin ligands.

Multivalent glyco(cyclo)peptides ⬇️

N-glycosyl-N-hydroxysulfamides as potent inhibitors of Brucella suis carbonic anhydrases

New acridone derivatives for the electrochemical DNA-hybridisation labelling.

New method to prepare peptide-oligonucleotide conjugates through glyoxylic oxime formation.

Nitrobenzylcarbamate prodrugs of cytotoxic acridines for potential use with nitroreductase gene-directed enzyme prodrug therapy.

Noninvasive visualization and quantification of tumor αVβ3 integrin expression using a novel positron emission tomography probe, 64Cu-cyclam-RAFT-c(-RGDfK-)4.

Novel model peptide for Atx1-like metallochaperones.

Oligonucleotide sequential bis-conjugation via click-oxime and click-Huisgen procedures.

On-bead synthesis and binding assay of chemoselectively template-assembled multivalent neoglycopeptides

One-Pot Self-Assembly of Peptide-Based Cage-Type Nanostructures Using Orthogonal Ligations.

One-pot approach to well-defined biomolecular assemblies by orthogonal chemoselective ligations.