Lista de obras - Maria Digiacomo - Dominio Público Uruguay

2-[(3-Methoxyphenylethyl)phenoxy]-based ABCB1 inhibitors: effect of different basic side-chains on their biological properties

artículo científico publicado en 2008

A Proteomic Approach to Uncover Neuroprotective Mechanisms of Oleocanthal against Oxidative Stress

artículo científico publicado en 2018

Anti-ischemic properties of a new spiro-cyclic benzopyran activator of the cardiac mito-KATP channel

artículo científico publicado en 2009

Arylmethyloxyphenyl derivatives: small molecules displaying P-glycoprotein inhibition

artículo científico publicado en 2006

Design, Synthesis, and Evaluation of Thyronamine Analogues as Novel Potent Mouse Trace Amine Associated Receptor 1 (mTAAR1) Agonists

artículo científico publicado en 2015

Design, synthesis and preliminary evaluation of 18F-labelled 1,8-naphthyridin- and quinolin-2-one-3-carboxamide derivatives for PET imaging of CB2 cannabinoid receptor

scientific article published on 25 April 2015

Diclofenac-Derived Hybrids for Treatment of Actinic Keratosis and Squamous Cell Carcinoma.

artículo científico publicado en 2019

Enantioselectivity in Cardioprotection induced by (S)- (−)-2,2-Dimethyl-N-(4′-acetamido-benzyl)-4-spiromorpholone-chromane

artículo científico publicado en 2009

Evaluation of the NO-releasing properties of NO-donor linkers

artículo científico publicado en 2008

Identification of the First Synthetic Allosteric Modulator of the CB2 Receptors and Evidence of Its Efficacy for Neuropathic Pain Relief

artículo científico publicado en 2018

Metabolically labile cannabinoid esters: A ‘soft drug’ approach for the development of cannabinoid-based therapeutic drugs

artículo científico publicado en 2007

NO-glibenclamide derivatives: prototypes of a new class of nitric oxide-releasing anti-diabetic drugs.

artículo científico publicado en 2009

NO-sartans: a new class of pharmacodynamic hybrids as cardiovascular drugs

artículo científico publicado en 2004

New NO-Releasing Pharmacodynamic Hybrids of Losartan and Its Active Metabolite: Design, Synthesis, and Biopharmacological Properties

artículo científico publicado en 2006

P-gp transporter and its role in neurodegenerative diseases

scientific article published on January 2009

Predictive models, based on classification algorithms, for compounds potentially active as mitochondrial ATP-sensitive potassium channel openers

artículo científico publicado en 2009

SAR study on arylmethyloxyphenyl scaffold: looking for a P-gp nanomolar affinity

artículo científico publicado en 2014

SodiumN-(Methylsulfonyl)-N-(4-nitro-2-phenoxyphenyl)sulfamate: A Water-Soluble Nimesulide Prodrug for Parenteral Use

artículo científico publicado en 2010

Spirocyclic benzopyran-based derivatives as new anti-ischemic activators of mitochondrial ATP-sensitive potassium channel

artículo científico publicado en 2008

Synthesis and Affinity Evaluation for AT1 Receptor of Phenylsalicylaldoxime-Derivatives Structurally Related to Sartans

Synthesis and Biological Evaluation of 2′-Oxo-2,3-dihydro-3′H- spiro[chromene-4,5′-[1,3]oxazolidin]-3′yl]acetic Acid Derivatives as Aldose Reductase Inhibitors

artículo científico publicado en 2011

Synthesis and biological evaluation of (hetero)arylmethyloxy- and arylmethylamine-phenyl derivatives as potent P-glycoprotein modulating agents

artículo científico publicado en 2008

Synthesis and biological evaluation of 5-membered spiro heterocycle-benzopyran derivatives against myocardial ischemia

artículo científico publicado en 2011

Synthesis and evaluation of multi-functional NO-donor/insulin-secretagogue derivatives for the treatment of type II diabetes and its cardiovascular complications

artículo científico publicado en 2014

Synthesis and pharmacological evaluation of multifunctional tacrine derivatives against several disease pathways of AD.

artículo científico publicado en 2015

Therapeutic potential of sulindac hydroxamic acid against human pancreatic and colonic cancer cells

artículo científico publicado en 2010

Traditional Uses of Cannabinoids and New Perspectives in the Treatment of Multiple Sclerosis

alpha-Naphthylaminopropan-2-ol Derivatives as BACE1 Inhibitors

artículo científico publicado en 2008

Lista de obras de Maria Digiacomo

2-[(3-Methoxyphenylethyl)phenoxy]-based ABCB1 inhibitors: effect of different basic side-chains on their biological properties

A Proteomic Approach to Uncover Neuroprotective Mechanisms of Oleocanthal against Oxidative Stress

Anti-ischemic properties of a new spiro-cyclic benzopyran activator of the cardiac mito-KATP channel

Arylmethyloxyphenyl derivatives: small molecules displaying P-glycoprotein inhibition

Design, Synthesis, and Evaluation of Thyronamine Analogues as Novel Potent Mouse Trace Amine Associated Receptor 1 (mTAAR1) Agonists

Design, synthesis and preliminary evaluation of 18F-labelled 1,8-naphthyridin- and quinolin-2-one-3-carboxamide derivatives for PET imaging of CB2 cannabinoid receptor

Diclofenac-Derived Hybrids for Treatment of Actinic Keratosis and Squamous Cell Carcinoma.

Enantioselectivity in Cardioprotection induced by (S)- (−)-2,2-Dimethyl-N-(4′-acetamido-benzyl)-4-spiromorpholone-chromane

Evaluation of the NO-releasing properties of NO-donor linkers

Identification of the First Synthetic Allosteric Modulator of the CB2 Receptors and Evidence of Its Efficacy for Neuropathic Pain Relief

Metabolically labile cannabinoid esters: A ‘soft drug’ approach for the development of cannabinoid-based therapeutic drugs

NO-glibenclamide derivatives: prototypes of a new class of nitric oxide-releasing anti-diabetic drugs.

NO-sartans: a new class of pharmacodynamic hybrids as cardiovascular drugs

New NO-Releasing Pharmacodynamic Hybrids of Losartan and Its Active Metabolite: Design, Synthesis, and Biopharmacological Properties

P-gp transporter and its role in neurodegenerative diseases

Predictive models, based on classification algorithms, for compounds potentially active as mitochondrial ATP-sensitive potassium channel openers

SAR study on arylmethyloxyphenyl scaffold: looking for a P-gp nanomolar affinity

SodiumN-(Methylsulfonyl)-N-(4-nitro-2-phenoxyphenyl)sulfamate: A Water-Soluble Nimesulide Prodrug for Parenteral Use

Spirocyclic benzopyran-based derivatives as new anti-ischemic activators of mitochondrial ATP-sensitive potassium channel

Synthesis and Affinity Evaluation for AT1 Receptor of Phenylsalicylaldoxime-Derivatives Structurally Related to Sartans

Synthesis and Biological Evaluation of 2′-Oxo-2,3-dihydro-3′H- spiro[chromene-4,5′-[1,3]oxazolidin]-3′yl]acetic Acid Derivatives as Aldose Reductase Inhibitors

Synthesis and biological evaluation of (hetero)arylmethyloxy- and arylmethylamine-phenyl derivatives as potent P-glycoprotein modulating agents

Synthesis and biological evaluation of 5-membered spiro heterocycle-benzopyran derivatives against myocardial ischemia

Synthesis and evaluation of multi-functional NO-donor/insulin-secretagogue derivatives for the treatment of type II diabetes and its cardiovascular complications

Synthesis and pharmacological evaluation of multifunctional tacrine derivatives against several disease pathways of AD.

Therapeutic potential of sulindac hydroxamic acid against human pancreatic and colonic cancer cells

Traditional Uses of Cannabinoids and New Perspectives in the Treatment of Multiple Sclerosis

alpha-Naphthylaminopropan-2-ol Derivatives as BACE1 Inhibitors