Lista de obras - Frédéric Bihel - Dominio Público Uruguay

A Yeast/Drosophila Screen to Identify New Compounds Overcoming Frataxin Deficiency

artículo científico publicado en 2015

Access to 4-alkylaminopyridazine derivatives via nitrogen-assisted regioselective Pd-catalyzed reactions

artículo científico publicado en 2014

Aminoguanidine hydrazone derivatives as non-peptide NPFF1 receptor antagonists reverse opioid induced hyperalgesia.

artículo científico publicado en 2018

CMTX1 patients' cells present genomic instability corrected by CamKII inhibitors

artículo científico publicado en 2015

CamKII inhibitors reduce mitotic instability, connexon anomalies and progression of the in vivo behavioral phenotype in transgenic animals expressing a mutated Gjb1 gene

artículo científico publicado en 2014

Design and validation of a homogeneous time-resolved fluorescence cell-based assay targeting the ligand-gated ion channel 5-HT3A.

artículo científico publicado en 2015

Development of Dipeptidic hGPR54 Agonists.

artículo científico publicado en 2016

Development of a peptidomimetic antagonist of neuropeptide FF receptors for the prevention of opioid-induced hyperalgesia

artículo científico publicado en 2015

Development of sub-nanomolar dipeptidic ligands of neuropeptide FF receptors

artículo científico publicado en 2012

Diastereoselective Synthesis of Nonplanar 3-Amino-1,2,4-oxadiazine Scaffold: Structure Revision of Alchornedine

artículo científico publicado en 2020

Direct guanidinylation of aryl and heteroaryl halides via copper-catalyzed cross-coupling reaction

scientific article published on 13 December 2011

Discovery of a Subnanomolar helical D-tridecapeptide inhibitor of gamma-secretase

scientific article published on 01 July 2004

Effects of systematic N-terminus deletions and benzoylations of endogenous RF-amide peptides on NPFF1R, NPFF2R, GPR10, GPR54 and GPR103

artículo científico publicado en 2015

Erratum to: CMTX1 patients' cells present genomic instability corrected by CamKII inhibitors

artículo científico publicado en 2016

Fukuyama Cross-Coupling Approach to Isoprekinamycin: Discovery of the Highly Active and Bench-Stable Palladium Precatalyst POxAP

scientific article published on 18 January 2019

Heteroarylguanidines as Allosteric Modulators of ASIC1a and ASIC3 Channels.

artículo científico publicado en 2018

Induction of ATP Release, PPIX Transport, and Cholesterol Uptake by Human Red Blood Cells Using a New Family of TSPO Ligands

scholarly article by Irene Marginedas-Freixa published in October 2018

Involvement of neuropeptide FF receptors in neuroadaptive responses to acute and chronic opiate treatments.

artículo científico publicado en 2012

Microwave-assisted cyclic amidine synthesis using TiCl4

artículo científico publicado en 2006

Mitochondria modulatory effects of new TSPO ligands in a cellular model of tauopathies

scientific article published on 13 October 2019

Neuropeptide FF receptors as novel targets for limbic seizure attenuation

artículo científico publicado en 2015

New 3'-azido-3'-deoxythymidin-5'-yl O-(omega-hydroxyalkyl) carbonate prodrugs: synthesis and anti-HIV evaluation.

artículo científico publicado en 2001

New PDE4 inhibitors based on pharmacophoric similarity between papaverine and tofisopam

scientific article published on 12 August 2011

Nucleophilic substitution of azide acting as a pseudo leaving group: one-step synthesis of various aza heterocycles

artículo científico publicado en 2013

Opioid adjuvant strategy: improving opioid effectiveness

artículo científico publicado en 2016

Pharmacological characterization of the mouse NPFF2 receptor.

artículo científico publicado en 2009

Structure-activity relationship study around guanabenz identifies two derivatives retaining antiprion activity but having lost α2-adrenergic receptor agonistic activity

artículo científico publicado en 2014

Substituted thiazolamide coupled to a redox delivery system: a new gamma-secretase inhibitor with enhanced pharmacokinetic profile.

artículo científico publicado en 2005

Synthesis and antiproliferative effects of 5,6-disubstituted Pyridazin-3(2H)-ones designed as conformationally constrained combretastatin A-4 Analogues

artículo científico publicado en 2013

Synthesis of new 3-alkoxy-7-amino-4-chloro-isocoumarin derivatives as new beta-amyloid peptide production inhibitors and their activities on various classes of protease

artículo científico publicado en 2003

The effect of neuropeptide FF in the amygdala kindling model.

artículo científico publicado en 2015

The long-lasting love affair between the budding yeast Saccharomyces cerevisiae and the Epstein-Barr virus

artículo científico

χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds.

artículo científico publicado en 2017

Lista de obras de Frédéric Bihel

A Yeast/Drosophila Screen to Identify New Compounds Overcoming Frataxin Deficiency

Access to 4-alkylaminopyridazine derivatives via nitrogen-assisted regioselective Pd-catalyzed reactions

Aminoguanidine hydrazone derivatives as non-peptide NPFF1 receptor antagonists reverse opioid induced hyperalgesia.

CMTX1 patients' cells present genomic instability corrected by CamKII inhibitors

CamKII inhibitors reduce mitotic instability, connexon anomalies and progression of the in vivo behavioral phenotype in transgenic animals expressing a mutated Gjb1 gene

Design and validation of a homogeneous time-resolved fluorescence cell-based assay targeting the ligand-gated ion channel 5-HT3A.

Development of Dipeptidic hGPR54 Agonists.

Development of a peptidomimetic antagonist of neuropeptide FF receptors for the prevention of opioid-induced hyperalgesia

Development of sub-nanomolar dipeptidic ligands of neuropeptide FF receptors

Diastereoselective Synthesis of Nonplanar 3-Amino-1,2,4-oxadiazine Scaffold: Structure Revision of Alchornedine

Direct guanidinylation of aryl and heteroaryl halides via copper-catalyzed cross-coupling reaction

Discovery of a Subnanomolar helical D-tridecapeptide inhibitor of gamma-secretase

Effects of systematic N-terminus deletions and benzoylations of endogenous RF-amide peptides on NPFF1R, NPFF2R, GPR10, GPR54 and GPR103

Erratum to: CMTX1 patients' cells present genomic instability corrected by CamKII inhibitors

Fukuyama Cross-Coupling Approach to Isoprekinamycin: Discovery of the Highly Active and Bench-Stable Palladium Precatalyst POxAP

Heteroarylguanidines as Allosteric Modulators of ASIC1a and ASIC3 Channels.

Induction of ATP Release, PPIX Transport, and Cholesterol Uptake by Human Red Blood Cells Using a New Family of TSPO Ligands

Involvement of neuropeptide FF receptors in neuroadaptive responses to acute and chronic opiate treatments.

Microwave-assisted cyclic amidine synthesis using TiCl4

Mitochondria modulatory effects of new TSPO ligands in a cellular model of tauopathies

Neuropeptide FF receptors as novel targets for limbic seizure attenuation

New 3'-azido-3'-deoxythymidin-5'-yl O-(omega-hydroxyalkyl) carbonate prodrugs: synthesis and anti-HIV evaluation.

New PDE4 inhibitors based on pharmacophoric similarity between papaverine and tofisopam

Nucleophilic substitution of azide acting as a pseudo leaving group: one-step synthesis of various aza heterocycles

Opioid adjuvant strategy: improving opioid effectiveness

Pharmacological characterization of the mouse NPFF2 receptor.

Structure-activity relationship study around guanabenz identifies two derivatives retaining antiprion activity but having lost α2-adrenergic receptor agonistic activity

Substituted thiazolamide coupled to a redox delivery system: a new gamma-secretase inhibitor with enhanced pharmacokinetic profile.

Synthesis and antiproliferative effects of 5,6-disubstituted Pyridazin-3(2H)-ones designed as conformationally constrained combretastatin A-4 Analogues

Synthesis of new 3-alkoxy-7-amino-4-chloro-isocoumarin derivatives as new beta-amyloid peptide production inhibitors and their activities on various classes of protease

The effect of neuropeptide FF in the amygdala kindling model.

The long-lasting love affair between the budding yeast Saccharomyces cerevisiae and the Epstein-Barr virus

χ-Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds.