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Lista de obras de Stephen Brand

A Fluorous, Pummerer Cyclative-Capture Strategy for the Synthesis of N-Heterocycles

scientific article published on 01 January 2007

A Fluorous-Phase Pummerer Cyclative-Capture Strategy for the Synthesis of Nitrogen Heterocycles

artículo científico publicado en 2005

An Enantioselective Ring Expansion Route Leading to Furanose and Pyranose Nucleosides Featuring Spirodiketopiperazines at the Anomeric Position

artículo científico publicado en 1999

Development of Small-Molecule Trypanosoma brucei N-Myristoyltransferase Inhibitors: Discovery and Optimisation of a Novel Binding Mode.

artículo científico publicado en 2015

Development of a Fluorescence-based Trypanosoma cruzi CYP51 Inhibition Assay for Effective Compound Triaging in Drug Discovery Programmes for Chagas Disease

artículo científico publicado en 2015

Discovery of a Novel Class of Orally Active Trypanocidal N -Myristoyltransferase Inhibitors

artículo científico publicado en 2012

Efficient Synthesis of 3-Aminocyclobut-2-en-1-ones:  Squaramide Surrogates as Potent VLA-4 Antagonists

artículo científico publicado en 2003

Lead optimization of a pyrazole sulfonamide series of Trypanosoma brucei N-myristoyltransferase inhibitors: identification and evaluation of CNS penetrant compounds as potential treatments for stage 2 human African trypanosomiasis

artículo científico publicado en 2014

N-myristoyltransferase inhibitors as new leads to treat sleeping sickness

artículo científico publicado en 2010

Solid phase approaches to N-heterocycles using a sulfur linker cleaved by SmI2.

artículo científico publicado en 2006

The first Pummerer cyclisations on solid phase. Convenient construction of oxindoles enabled by a sulfur-link to resin

scientific article published on 01 September 2003

Validation of N-myristoyltransferase as Potential Chemotherapeutic Target in Mammal-Dwelling Stages of Trypanosoma cruzi

artículo científico publicado en 2016