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Lista de obras de Werner Sieghart

6,3'-Dinitroflavone is a low efficacy modulator of GABA(A) receptors.

artículo científico publicado en 2008

8-Substituted Triazolobenzodiazepines: <i>In Vitro</i> and <i>In Vivo</i> Pharmacology in Relation to Structural Docking at the α1 Subunit-Containing GABA<sub>A</sub> Receptor

scientific article published on 20 April 2021

A novel positive allosteric modulator of the GABA(A) receptor: the action of (+)-ROD188

artículo científico publicado en 2000

A novel serine kinase with specificity for beta3-subunits is tightly associated with GABA(A) receptors

scientific article published on 01 July 1999

A novel site on gamma 3 subunits important for assembly of GABA(A) receptors

artículo científico publicado en 2002

A polymorphism (5-HTTLPR) in the serotonin transporter promoter gene is associated with DSM-IV depression subtypes in seasonal affective disorder.

artículo científico publicado en 2003

A propofol binding site on mammalian GABAA receptors identified by photolabeling

artículo científico publicado en 2013

A rapid and simple method for efficient coating of microtiter plates using low amounts of antigen in the presence of detergent

scientific article published on 01 December 1986

AMPA and kainate receptors mediate mutually exclusive effects on GABA(A) receptor expression in cultured mouse cerebellar granule neurones

artículo científico publicado en 2007

Abolition of zolpidem sensitivity in mice with a point mutation in the GABAA receptor gamma2 subunit.

artículo científico publicado en 2004

Additional support for linkage of schizophrenia and bipolar disorder to chromosome 3q29

artículo científico publicado en 2007

Affinity of various ligands for benzodiazepine receptors in rat cerebellum and hippocampus.

artículo científico publicado en 1984

Allosteric modulation of GABAA receptors via multiple drug-binding sites.

artículo científico publicado en 2014

Alterations in GABAA Receptor Subunit Expression in the Amygdala and Entorhinal Cortex in Human Temporal Lobe Epilepsy

scientific article published on 01 November 2019

Alterations in the expression of GABAA receptor subunits in cerebellar granule cells after the disruption of the alpha6 subunit gene.

artículo científico publicado en 1999

Altered receptor subtypes in the forebrain of GABA(A) receptor delta subunit-deficient mice: recruitment of gamma 2 subunits.

artículo científico publicado en 2002

Alternate use of distinct intersubunit contacts controls GABAA receptor assembly and stoichiometry.

artículo científico publicado en 2001

An updated unified pharmacophore model of the benzodiazepine binding site on gamma-aminobutyric acid(a) receptors: correlation with comparative models

artículo científico publicado en 2007

Antiallergic drug cromolyn may inhibit histamine secretion by regulating phosphorylation of a mast cell protein

artículo científico publicado en 1980

Antibodies specific for GABAA receptor alpha subunits reveal that chronic alcohol treatment down-regulates alpha-subunit expression in rat brain regions

artículo científico publicado en 1993

Antiseizure activity of novel gamma-aminobutyric acid (A) receptor subtype-selective benzodiazepine analogues in mice and rat models

artículo científico publicado en 2009

Anxiolytic-like effects of 8-acetylene imidazobenzodiazepines in a rhesus monkey conflict procedure ⬇️

artículo científico publicado el 18 de agosto de 2010

Anxioselective anxiolytics: additional perspective.

artículo científico publicado en 2013

Apparent identity of alpha-subunit of pyruvate dehydrogenase and the protein phosphorylated in the presence of glutamate in P2-fractions of rat cerebral cortex

scientific article published on 01 January 1984

Are GABAA receptors containing alpha5 subunits contributing to the sedative properties of benzodiazepine site agonists?

artículo científico publicado en 2007

Assembly of GABA(A) receptors (Review).

artículo científico publicado en 2008

Association Studies of Candidate Genes in Bipolar Disorders

article

Association of proteins irreversibly labeled by 3H-flunitrazepam with different benzodiazepine

artículo científico publicado el 1 de enero de 1983

Association study of schizophrenia spectrum disorders and dopamine D3 receptor gene: is schizoaffective disorder special?

article

Attenuated sensitivity to neuroactive steroids in gamma-aminobutyrate type A receptor delta subunit knockout mice.

artículo científico publicado en 1999

Azemiopsin from Azemiops feae viper venom, a novel polypeptide ligand of nicotinic acetylcholine receptor.

artículo científico publicado en 2012

Behavioural correlates of an altered balance between synaptic and extrasynaptic GABAAergic inhibition in a mouse model.

artículo científico publicado en 2004

Benzodiazepine receptors: multiple receptors or multiple conformations?

artículo científico publicado en 1985

Benzodiazepine-induced spatial learning deficits in rats are regulated by the degree of modulation of α1 GABA(A) receptors

artículo científico publicado en 2012

Benzodiazepine-mediated regulation of alpha1, alpha2, beta1-3 and gamma2 GABA(A) receptor subunit proteins in the rat brain hippocampus and cortex.

artículo científico publicado en 1999

Benzodiazepines modulate GABAreceptors by reducing a gamma-subunit-mediated inhibition of GABA sensitivity

artículo científico publicado en 2009

Bidirectional alterations of GABA(A) receptor subunit peptide levels in rat cortex during chronic ethanol consumption and withdrawal.

artículo científico publicado en 1997

Binding of gamma-aminobutyric acidA receptors to tubulin

artículo científico publicado en 1994

Binge alcohol drinking is associated with GABAAα2-regulated Toll-like receptor 4 (TLR4) expression in the central amygdala ⬇️

artículo científico publicado el 28 de febrero de 2011

Biochemical, immunological, and pharmacological characterization of GABAA-benzodiazepine receptor subtypes

artículo científico publicado el 1 de enero de 1992

Biological evaluation of 2'-[18F]fluoroflumazenil ([18F]FFMZ), a potential GABA receptor ligand for PET.

artículo científico publicado en 2004

Biperiden and Haloperidol Plasma Levels and Extrapyramidal Side Effects in Schizophrenic Patients

artículo científico publicado en 1997

CYP2D6 genotype and phenotyping by determination of dextromethorphan and metabolites in serum of healthy controls and of patients under psychotropic medication.

artículo científico publicado en 1997

Ca2+ and cyclic AMP regulate phosphorylation of same two membrane-associated proteins specific to nerve tissue ⬇️

scientific article published on May 1, 1979

Calcium-dependent protein phosphorylation during secretion by exocytosis in the mast cell ⬇️

artículo científico publicado el 28 de septiembre de 1978

Cellular localization and differential distribution of GABAA receptor subunit proteins and messenger RNAs within hypothalamic magnocellular neurons

scientific article published on 01 February 1995

Cerebellar α6 subunit-containing GABAA receptors: A novel therapeutic target for disrupted prepulse inhibition in neuropsychiatric disorders.

artículo científico publicado en 2018

Clinical-pharmacological study with the two isomers (d-, l-) of fenfluramine and its comparison with chlorpromazine and d-amphetamine: blood levels, EEG mapping and safety evaluation.

artículo científico publicado en 1993

Clusters of GABAA receptors on cultured hippocampal cells correlate only partially with functional synapses.

artículo científico publicado en 1999

Colocalization of GABA, glycine, and their receptors at synapses in the rat spinal cord

artículo científico publicado en 1996

Comparative bioavailability studies with a new mixed-micelles solution of diazepam utilizing radioreceptor assay, psychometry and EEG brain mapping.

artículo científico publicado en 1988

Comparative modeling of GABA(A) receptors: limits, insights, future developments.

artículo científico publicado en 2003

Comparative models of GABAA receptor extracellular and transmembrane domains: important insights in pharmacology and function.

artículo científico publicado en 2005

Comparison of benzodiazepine receptor binding in membranes from human or rat brain.

artículo científico publicado en 1985

Comparison of benzodiazepine receptors in cerebellum and inferior colliculus.

artículo científico publicado en 1986

Comparison of tryptic peptides of benzodiazepine binding proteins photolabeled with [3H]flunitrazepam or [3H]Ro 15-4513

artículo científico publicado en 1987

Comparison of two different benzodiazepine binding proteins by peptide mapping after limited proteolysis

scientific article published on 01 May 1988

Composition of the GABA(A) receptors of retinal dopaminergic neurons

artículo científico publicado en 1999

Cultured Hippocampal Pyramidal Neurons Express Two Kinds of GABAA Receptors

artículo científico publicado en 2004

Deep amino acid sequencing of native brain GABAA receptors using high-resolution mass spectrometry

artículo científico publicado en 2012

Deficits in phosphorylation of GABA(A) receptors by intimately associated protein kinase C activity underlie compromised synaptic inhibition during status epilepticus

artículo científico publicado en 2008

Deficits in spatial memory correlate with modified {gamma}-aminobutyric acid type A receptor tyrosine phosphorylation in the hippocampus.

artículo científico publicado en 2009

Design and Synthesis of Novel Deuterated Ligands Functionally Selective for the γ-Aminobutyric Acid Type A Receptor (GABAAR) α6 Subtype with Improved Metabolic Stability and Enhanced Bioavailability.

artículo científico publicado en 2018

Detection and binding properties of GABA(A) receptor assembly intermediates.

artículo científico publicado en 2001

Development of gamma-aminobutyric acidergic synapses in cultured hippocampal neurons

artículo científico publicado en 2006

Diazepam-bound GABAA receptor models identify new benzodiazepine binding-site ligands

artículo científico publicado en 2012

Differential degradation of different benzodiazepine binding proteins by incubation of membranes from cerebellum or hippocampus with trypsin.

artículo científico publicado en 1985

Differential localization of GABA(A) receptor subunits in relation to rat striatopallidal and pallidopallidal synapses.

artículo científico publicado en 2011

Differential regulation of GABA(A) receptor gene expression by ethanol in the rat hippocampus versus cerebral cortex.

artículo científico publicado en 1998

Differential regulation of synaptic GABAA receptors by cAMP-dependent protein kinase in mouse cerebellar and olfactory bulb neurones.

artículo científico publicado en 1999

Distribution of GABAA receptor alpha 1 subunit-like immunoreactivity in comparison with that of enkephalin and substance P in the rat forebrain

scientific article published on 01 June 1995

Distribution of alpha1, alpha4, gamma2, and delta subunits of GABAA receptors in hippocampal granule cells

artículo científico publicado en 2004

Dopamine D3 receptor gene polymorphism and response to clozapine in schizophrenic Pakistani patients

article

Drug interactions with cyclic nucleotide and protein phosphorylation systems

artículo científico publicado el 1 de enero de 1979

Dual mode of stimulation by the beta-carboline ZK 91085 of recombinant GABA(A) receptor currents: molecular determinants affecting its action

artículo científico publicado en 1999

EDPC: a novel high affinity ligand for the benzodiazepine site on rat GABA(A) receptors.

artículo científico publicado en 1999

Early postnatal switch in GABAA receptor α-subunits in the reticular thalamic nucleus

artículo científico publicado en 2015

Engineered Flumazenil Recognition Site Provides Mechanistic Insight Governing Benzodiazepine Modulation in GABA Receptors

artículo científico publicado en 2018

Establishing a new mouse model for investigating the function of amygdala neurons in anxiety.

artículo científico publicado en 2008

European multicentre association study of schizophrenia: a study of the DRD2 Ser311Cys and DRD3 Ser9Gly polymorphisms

artículo científico publicado en 1998

European multicentre evaluation of the analytical performance of the Abbott AxSYM Abused Drugs Assays

artículo científico publicado en 1997

Evidence That Sedative Effects of Benzodiazepines Involve Unexpected GABAA Receptor Subtypes: Quantitative Observation Studies in Rhesus Monkeys

scientific article published on 02 May 2018

Evidence for association of a high affinity avermectin binding site with the benzodiazepine receptor.

artículo científico publicado en 1984

Evidence for the existence of differential O-glycosylated alpha 5-subunits of the gamma-aminobutyric acidA receptor in the rat brain.

artículo científico publicado en 1993

Evidence for the existence of several different alpha- and beta-subunits of the GABA/benzodiazepine receptor complex from rat brain.

artículo científico publicado en 1989

Extensive heterogeneity of recombinant gamma-aminobutyric acidA receptors expressed in alpha 4 beta 3 gamma 2-transfected human embryonic kidney 293 cells.

artículo científico publicado en 1996

Fear learning induces structural and functional plasticity at GABAergic synapses in the basolateral amygdala.

artículo científico publicado en 2011

Fear learning triggers structural changes at GABAergic synapses in the basal amygdala.

artículo científico publicado en 2010

First In Vivo Testing of Compounds Targeting Group 3 Medulloblastomas Using an Implantable Microdevice as a New Paradigm for Drug Development.

artículo científico publicado en 2016

Formation of GABAA receptor complexes containing α1 and α5 subunits is paralleling a multiple T-maze learning task in mice

artículo científico publicado en 2016

From synapse to behavior: rapid modulation of defined neuronal types with engineered GABAA receptors.

artículo científico publicado en 2007

Functional correlation of GABA(A) receptor alpha subunits expression with the properties of IPSCs in the developing thalamus.

artículo científico publicado en 2000

GABA A receptors: subtypes provide diversity of function and pharmacology

artículo científico publicado en 2009

GABA expression dominates neuronal lineage progression in the embryonic rat neocortex and facilitates neurite outgrowth via GABA(A) autoreceptor/Cl- channels.

artículo científico publicado en 2001

GABA influences the development of the ventromedial nucleus of the hypothalamus.

artículo científico publicado en 2001

GABA receptor associated drug receptors.

artículo científico publicado en 1981

GABA(A) Receptors: Post-Synaptic Co-Localization and Cross-Talk with Other Receptors.

artículo científico publicado en 2011

GABA(A) benzodiazepine receptors and epilepsy

artículo científico publicado en 1990

GABA(A) receptor assembly. Identification and structure of gamma(2) sequences forming the intersubunit contacts with alpha(1) and beta(3) subunits

scientific article published on 01 March 2000

GABA(A) receptor subtype-selectivity of novel bicuculline derivatives

artículo científico publicado en 2015

GABA(A) receptor subunits in the rat hippocampus I: immunocytochemical distribution of 13 subunits.

artículo científico publicado en 1997

GABA(A) receptor subunits in the rat hippocampus II: altered distribution in kainic acid-induced temporal lobe epilepsy.

artículo científico publicado en 1997

GABA(A) receptor subunits in the rat hippocampus III: altered messenger RNA expression in kainic acid-induced epilepsy.

artículo científico publicado en 1997

GABA(A) receptors: immunocytochemical distribution of 13 subunits in the adult rat brain.

artículo científico publicado en 2000

GABAA alpha6-containing receptors are selectively compromised in cerebellar granule cells of the ataxic mouse, stargazer.

artículo científico publicado en 2007

GABAA receptor phosphorylation and functional modulation in cortical neurons by a protein kinase C-dependent pathway.

artículo científico publicado en 2000

GABAA receptor subunit composition and functional properties of Cl- channels with differential sensitivity to zolpidem in embryonic rat hippocampal cells.

artículo científico publicado en 1999

GABAA receptor subunits in the human amygdala and hippocampus: Immunohistochemical distribution of 7 subunits.

artículo científico publicado en 2017

GABAA, Receptor α1, α4, and β3 Subunit mRNA and Protein Expression in the Frontal Cortex of Human Alcoholics ⬇️

artículo científico publicado el 1 de junio de 1998

Gel-based mass spectrometric analysis of a strongly hydrophobic GABAA-receptor subunit containing four transmembrane domains

artículo científico publicado en 2009

Gel-based mass spectrometric analysis of recombinant GABA(A) receptor subunits representing strongly hydrophobic transmembrane proteins

artículo científico publicado en 2008

Genetic polymorphisms for drug metabolism (CYP2D6) and tardive dyskinesia in schizophrenia

scientific article published on 01 July 1998

Genome scan for susceptibility loci for schizophrenia

artículo científico publicado en 2000

Genome scan for susceptibility loci for schizophrenia and bipolar disorder

artículo científico publicado en 2002

Gephyrin, the enigmatic organizer at GABAergic synapses

artículo científico publicado en 2012

Glutamate-Stimulated Phosphorylation of a Specific Protein in P2Fractions of Rat Cerebral Cortex ⬇️

artículo científico publicado el 1 de noviembre de 1981

Heterogeneity of GABAA receptors

artículo científico publicado el 1 de enero de 1992

Heterogeneity of GABAA-benzodiazepine receptors ⬇️

artículo científico publicado el 1 de febrero de 1991

Histaminergic pharmacology of homo-oligomeric β3 γ-aminobutyric acid type A receptors characterized by surface plasmon resonance biosensor technology.

artículo científico publicado en 2012

Homologous sites of GABA(A) receptor alpha(1), beta(3) and gamma(2) subunits are important for assembly.

artículo científico publicado en 2002

Identification of amino acid residues important for assembly of GABA receptor alpha1 and gamma2 subunits.

artículo científico publicado en 2006

Identification of amino acid residues of GABA(A) receptor subunits contributing to the formation and affinity of the tert-butylbicyclophosphorothionate binding site.

artículo científico publicado en 2000

Identification of an amino acid sequence within GABA(A) receptor beta3 subunits that is important for receptor assembly.

artículo científico publicado en 2003

Identification of novel positive allosteric modulators and null modulators at the GABAA receptor α+β- interface

artículo científico publicado en 2013

Identification of the cyclic AMP-dependent protein kinase responsible for endogenous phosphorylation of substrate proteins in synaptic membrane fraction from rat brain ⬇️

artículo científico publicado el 10 de diciembre de 1979

Immunoaffinity purification of gamma-aminobutyric acidA (GABAA) receptors containing gamma 1-subunits. Evidence for the presence of a single type of gamma-subunit in GABAA receptors

artículo científico publicado en 1994

Immunocytochemical localization of the alpha 1 and beta 2/3 subunits of the GABAA receptor in relation to specific GABAergic synapses in the dentate gyrus

scientific article published on 01 April 1995

Immunohistochemical and neurochemical evidence for GABAA receptor heterogeneity between the hypothalamus and cortex.

artículo científico publicado en 1994

Improved radioimmunoassay of melatonin in serum

artículo científico publicado en 1987

In vivo and in vitro evaluation of [18F]FETO with respect to the adrenocortical and GABAergic system in rats.

artículo científico publicado en 2003

Increased Expression of GABAAReceptor β-Subunits in the Hippocampus of Patients with Temporal Lobe Epilepsy ⬇️

artículo científico publicado el 1 de agosto de 2003

Initially expressed early rat embryonic GABA(A) receptor Cl- ion channels exhibit heterogeneous channel properties.

artículo científico publicado en 1998

Insights into functional pharmacology of α₁ GABA(A) receptors: how much does partial activation at the benzodiazepine site matter?

artículo científico publicado en 2013

Interaction between serotonin 5-HT2A receptor gene and dopamine transporter (DAT1) gene polymorphisms influences personality trait of persistence in Austrian Caucasians

artículo científico publicado en 2010

Interaction of allosteric ligands with GABAA receptors containing one, two, or three different subunits

artículo científico publicado en 1996

Interaction of benzodiazepine agonists and antagonists with different benzodiazepine receptors

artículo científico publicado el 1 de enero de 1983

International Union of Pharmacology. XV. Subtypes of gamma-aminobutyric acidA receptors: classification on the basis of subunit structure and receptor function ⬇️

artículo científico publicado el 1 de junio de 1998

Investigation of the abundance and subunit composition of GABAA receptor subtypes in the cerebellum of alpha1-subunit-deficient mice.

artículo científico publicado en 2005

Irreversible Binding of [3H]Flunitrazepam to Different Proteins in Various Brain Regions ⬇️

artículo científico publicado el 1 de julio de 1983

Ligand-gated ion channel subunit partnerships: GABAA receptor alpha6 subunit gene inactivation inhibits delta subunit expression.

artículo científico publicado en 1997

Localization of GABA‐A receptor alpha subunits on neurochemically distinct cell types in the rat locus coeruleus ⬇️

artículo científico publicado el 21 de junio de 2011

Long-range interactions in neuronal gene expression: evidence from gene targeting in the GABA(A) receptor beta2-alpha6-alpha1-gamma2 subunit gene cluster

artículo científico publicado en 2000

Molecular basis of pharmacological heterogeneity of GABAA receptors

artículo científico publicado el 1 de mayo de 1992

Molecular basis of the γ-aminobutyric acid A receptor α3 subunit interaction with the clustering protein gephyrin

scientific journal article

Molecular heterogeneity of benzodiazepine receptors

artículo científico publicado en 1980

Multiplicity of GABAA--benzodiazepine receptors.

artículo científico publicado en 1989

Mutagenesis and computational docking studies support the existence of a histamine binding site at the extracellular β3+β3- interface of homooligomeric β3 GABAA receptors

artículo científico publicado en 2016

N-Deglycosylation and immunological identification indicates the existence of β-subunit isoforms of the rat GABAAreceptor ⬇️

artículo científico publicado el 5 de agosto de 1991

Neuronal localization of Ca2+-dependent protein phosphorylation in brain

scientific article published on 01 March 1980

Neuronal localization of specific brain phosphoproteins ⬇️

artículo científico publicado el 10 de noviembre de 1978

Neurosteroid Analog Photolabeling of a Site in the Third Transmembrane Domain of the β3 Subunit of the GABAA Receptor ⬇️

artículo científico publicado el 30 de mayo de 2012

Neurotoxins from snake venoms and α-conotoxin ImI inhibit functionally active ionotropic γ-aminobutyric acid (GABA) receptors

artículo científico publicado en 2015

No association of clock gene T3111C polymorphism and affective disorders

article

No association of the neuropeptide Y (Leu7Pro) and ghrelin gene (Arg51Gln, Leu72Met, Gln90Leu) single nucleotide polymorphisms with eating disorders

article

Non-association of dopamine D4 and D2 receptor genes with personality in healthy individuals

artículo científico publicado en 2000

Patterns of mRNA and protein expression for 12 GABAA receptor subunits in the mouse brain.

artículo científico publicado en 2013

Pentameric ligand-gated ion channel ELIC is activated by GABA and modulated by benzodiazepines

artículo científico publicado en 2012

Pharmacological properties of GABAA receptors containing gamma1 subunits.

artículo científico publicado en 2005

Phosphorylation of a single mast cell protein in response to drugs that inhibit secretion

artículo científico publicado en 1981

Photoaffinity labeling of benzodiazepine receptors with a partial inverse agonist ⬇️

artículo científico publicado el 15 de junio de 1984

Photoaffinity labeling of different benzodiazepine receptors at physiological temperature.

artículo científico publicado en 1984

Plasticity of GABAA receptors after ethanol pre-exposure in cultured hippocampal neurons.

artículo científico publicado en 2010

Possible association between childhood absence epilepsy and the gene encoding GABRB3

article

Possible linkage of schizophrenia and bipolar affective disorder to chromosome 3q29

artículo científico publicado en 2004

Postnatal development of proteins associated with different benzodiazepine receptors.

artículo científico publicado en 1986

Postnatal development of proteins irreversibly labeled by [3H]flunitrazepam.

artículo científico publicado en 1982

Potassium-evoked release of taurine from synaptosomal fractions of rat cerebral cortex.

artículo científico publicado en 1976

Potency of several type I-benzodiazepine receptor ligands for inhibition of [3H]flunitrazepam binding in different rat brain tissues ⬇️

artículo científico publicado el 2 de mayo de 1991

Properties of [3H]flunitrazepam binding to different benzodiazepine binding proteins

artículo científico publicado en 1983

Properties of [3H]taurine release from crude synaptosomal fractions of rat cerebral cortex ⬇️

artículo científico publicado el 1 de diciembre de 1979

Properties of a high affinity binding site for [3H]avermectin B1a.

artículo científico publicado en 1984

Protein kinase C phosphorylation regulates membrane insertion of GABAA receptor subtypes that mediate tonic inhibition.

artículo científico publicado en 2010

Quantitative localisation of synaptic and extrasynaptic GABAA receptor subunits on hippocampal pyramidal cells by freeze-fracture replica immunolabelling.

artículo científico publicado en 2010

Rat beta 3 subunits expressed in human embryonic kidney 293 cells form high affinity [35S]t-butylbicyclophosphorothionate binding sites modulated by several allosteric ligands of gamma-aminobutyric acid type A receptors

scientific article published on 01 September 1995

Regulation of GABA(A) receptor dynamics by interaction with purinergic P2X(2) receptors.

artículo científico publicado en 2011

Removal of GABA(A) receptor γ2 subunits from parvalbumin neurons causes wide-ranging behavioral alterations

artículo científico publicado en 2011

Response of thyrotropin to thyrotropin-releasing hormone as predictor of treatment outcome. Prediction of recovery and relapse in treatment with antidepressants and neuroleptics

scientific article published on 01 September 1986

Role of the GABAAreceptor γ2 subunit in the development of gonadotropin-releasing hormone neurons in vivo

article

Schizophrenia and the dopamine-beta-hydroxylase gene: results of a linkage and association study

article

Schizophrenia and the dopamine-β-hydroxylase gene

article

Search for α3β₂/₃γ2 subtype selective ligands that are stable on human liver microsomes

artículo científico publicado en 2012

Sedimentation and release properties of P2 fractions derived from rat cerebral cortex slices incubated with radiolabeled GABA for a short or long time period.

artículo científico publicado en 1981

Sedimentation and release properties of glial particles present in P2-fractions isolated from rat cerebral cortex

artículo científico publicado el 6 de julio de 1979

Sedimentation characteristics of subcellular vesicles derived from three glial systems

artículo científico publicado el 1 de junio de 1978

Segregation of different GABAA receptors to synaptic and extrasynaptic membranes of cerebellar granule cells

artículo científico publicado en 1998

Several new benzodiazepines selectively interact with a benzodiazepine receptor subtype

artículo científico publicado en 1983

Sh-I-048A, an in vitro non-selective super-agonist at the benzodiazepine site of GABAA receptors: the approximated activation of receptor subtypes may explain behavioral effects

artículo científico publicado en 2014

Somatostatin-induced phosphorylation of mast cell proteins

scientific article published on 01 October 1981

Spatio-temporal expression analysis of the calcium-binding protein calumenin in the rodent brain

artículo científico publicado en 2011

Spontaneous cross-link of mutated alpha1 subunits during GABA(A) receptor assembly.

artículo científico publicado en 2006

Stoichiometry and assembly of a recombinant GABAA receptor subtype.

artículo científico publicado en 1997

Striatal efferents preferentially innervate neurons in the ventral pallidum containing GABAA receptor alpha 1 subunit-like immunoreactivity

scientific article published on 01 June 1996

Structure and pharmacology of gamma-aminobutyric acidA receptor subtypes.

artículo científico publicado en 1995

Structure and subunit composition of GABA(A) receptors.

artículo científico publicado en 1999

Structure, pharmacology, and function of GABAA receptor subtypes.

artículo científico publicado en 2006

Subcellular distribution of dopamine-sensitive adenylate cyclase.

artículo científico publicado en 1976

Subtype selectivity of α+β- site ligands of GABAA receptors: identification of the first highly specific positive modulators at α6β2/3γ2 receptors.

artículo científico publicado en 2013

Subunit Compensation and Plasticity of Synaptic GABAA Receptors Induced by Ethanol in ?4 Subunit Knockout Mice ⬇️

artículo científico publicado el 23 de septiembre de 2011

Subunit composition and pharmacological characterization of gamma-aminobutyric acid type A receptors in frog pituitary melanotrophs

artículo científico publicado en 2000

Subunit composition and quantitative importance of hetero-oligomeric receptors: GABAA receptors containing alpha6 subunits.

artículo científico publicado en 1998

Synthesis and GABA(A) receptor activity of 6-oxa-analogs of neurosteroids

scientific article published on 01 June 2000

Synthesis, in vitro affinity, and efficacy of a bis 8-ethynyl-4H-imidazo[1,5a]- [1,4]benzodiazepine analogue, the first bivalent alpha5 subtype selective BzR/GABA(A) antagonist.

artículo científico publicado en 2003

Targeted disruption of the GABA(A) receptor delta subunit gene leads to an up-regulation of gamma 2 subunit-containing receptors in cerebellar granule cells

scientific journal article

The Cell Adhesion Molecule Neuroplastin-65 Is a Novel Interaction Partner of γ-Aminobutyric Acid Type A Receptors ⬇️

artículo científico publicado el 2 de marzo de 2012

The GABAA receptor alpha+beta- interface: a novel target for subtype selective drugs

artículo científico publicado en 2011

The alpha 6 subunit of the GABAA receptor is concentrated in both inhibitory and excitatory synapses on cerebellar granule cells

scientific journal article

The citalopram challenge test in patients with major depression and in healthy controls

artículo científico publicado en 1999

The gamma 2 subunit of the GABAA receptor is concentrated in synaptic junctions containing the alpha 1 and beta 2/3 subunits in hippocampus, cerebellum and globus pallidus

artículo científico publicado en 1996

The influence of phenotype on the outcome of linkage analysis of schizophrenia

artículo científico publicado en 1996

The parvalbumin-positive interneurons in the mouse dentate gyrus express GABAA receptor subunits α1, β2, and δ along their extrasynaptic cell membrane

artículo científico publicado en 2013

The α1, α2, α3, and γ2 subunits of GABAA receptors show characteristic spatial and temporal expression patterns in rhombencephalic structures during normal human brain development

artículo científico publicado en 2015

The α6 subunit-containing GABA receptor: A novel drug target for inhibition of trigeminal activation

scholarly article by Pi-Chuan Fan et al published 15 September 2018 in Neuropharmacology

Transient transfection coupled to baculovirus infection for rapid protein expression screening in insect cells

artículo científico publicado en 2012

Two novel residues in M2 of the gamma-aminobutyric acid type A receptor affecting gating by GABA and picrotoxin affinity.

artículo científico publicado en 2000

Understanding subtype-selective allosteric modulation of GABAA receptors.

artículo científico publicado en 2012

Unexpected Properties of δ-Containing GABAA Receptors in Response to Ligands Interacting with the α+ β- Site.

artículo científico publicado en 2013

Unraveling the function of GABA(A) receptor subtypes.

artículo científico publicado en 2000

Unravelling the role of GABAA receptor subtypes in distinct neurons and behaviour ⬇️

artículo científico publicado el 15 de mayo de 2012

Uptake of taurine into subcellular fractions of C-6 glioma cells

artículo científico publicado el 1 de mayo de 1976

Various proteins from rat brain, specifically and irreversibly labeled by [3H]flunitrazepam, are distinct alpha-subunits of the GABA-benzodiazepine receptor complex

scientific article published on 01 August 1988

[35S]tert.-butylbicyclophosphorothionate and avermectin bind to different sites associated with the gamma- aminobutyric acid-benzodiazepine receptor complex.

artículo científico publicado en 1984

[3H]propyl-6-azido-beta-carboline-3-carboxylate: a new photoaffinity label for the GABAA-benzodiazepine receptor.

artículo científico publicado en 1995

[Comparison of the bioavailability of two diazepam preparations. Clinical comparison between a new commercial preparation and a standard preparation after oral and intramuscular administration]

scientific article published on 01 April 1986

[Orally-administered taurine in therapy-resistant epilepsy (author's transl)]

scientific article published on 01 February 1977

gamma-Aminobutyric acid, acting through gamma -aminobutyric acid type A receptors, inhibits the biosynthesis of neurosteroids in the frog hypothalamus.

artículo científico publicado en 2000

gamma-Aminobutyric acidA receptors displaying association of gamma 3-subunits with beta 2/3 and different alpha-subunits exhibit unique pharmacological properties

artículo científico publicado en 1994

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