Lista de obras - Nicolas Inguimbert - Dominio Público Uruguay

Access to α,α-Disubstituted Disilylated Amino Acids and Their Use in Solid-Phase Peptide Synthesis

artículo científico publicado en 2015

Asp218 participates with Asp213 to bind a Ca2+ atom into the S1 subsite of aminopeptidase A: a key element for substrate specificity.

artículo científico publicado en 2008

Biochemical and structural analysis of the binding determinants of a vascular endothelial growth factor receptor peptidic antagonist

artículo científico publicado en 2010

Biological Activities of Cyclic and Acyclic B-Type Laxaphycins in SH-SY5Y Human Neuroblastoma Cells

artículo científico publicado en 2020

Biophysical Studies of the Induced Dimerization of Human VEGF Receptor 1 Binding Domain by Divalent Metals Competing with VEGF-A.

artículo científico publicado en 2016

Characterization of a new anticancer agent, EAPB0203, and its main metabolites: nuclear magnetic resonance and liquid chromatography-mass spectrometry studies

scientific article published on 31 October 2012

Chemiluminescence immunoassays for estradiol and ethinylestradiol based on new biotinylated estrogen derivatives.

artículo científico publicado en 2017

Cooperation and cheating orchestrate Vibrio assemblages and polymicrobial synergy in oysters infected with OsHV-1 virus

artículo científico publicado en 2023

Development and validation of LC-MS methods for peptaibol quantification in fungal extracts according to their lengths.

artículo científico publicado en 2015

Development of a chemiluminescent screening assay for detection of vascular endothelial growth factor receptor 1 ligands

artículo científico publicado en 2007

Disulfide and amide-bridged cyclic peptide analogues of the VEGF81–91 fragment: Synthesis, conformational analysis and biological evaluation

article

Efficient microwave-assisted one shot synthesis of peptaibols using inexpensive coupling reagents

artículo científico publicado en 2014

Enhancing the Antimicrobial Activity of Alamethicin F50/5 by Incorporating N-terminal Hydrophobic Triazole Substituents.

artículo científico publicado en 2017

Exploration of the S(')(1) subsite of neprilysin: a joined molecular modeling and site-directed mutagenesis study

scientific article published on 01 June 2000

First total synthesis and stereochemical revision of laxaphycin B and its extension to lyngbyacyclamide A ⬇️

artículo científico publicado en 2013

Helical peptides from VEGF and Vammin hotspots for modulating the VEGF-VEGFR interaction.

artículo científico publicado en 2013

How are 1,2,3-triazoles accommodated in helical secondary structures?

artículo científico publicado en 2018

Immunosensors for estradiol and ethinylestradiol based on new synthetic estrogen derivatives: application to wastewater analysis.

artículo científico publicado en 2013

Isolation and Synthesis of Laxaphycin B-Type Peptides: A Case Study and Clues to Their Biosynthesis. ⬇️

artículo científico publicado en 2015

NI956/QGC006, a Potent Orally Active, Brain-Penetrating Aminopeptidase A Inhibitor for Treating Hypertension

artículo científico publicado en 2019

On-resin cyclization of peptide ligands of the Vascular Endothelial Growth Factor Receptor 1 by copper(I)-catalyzed 1,3-dipolar azide-alkyne cycloaddition

scientific article published on 22 August 2007

Oxovanadium-salen and -salan complexes as effective labels for electrochemical immunosensing: a case study for estradiol detection

artículo científico publicado en 2014

Parallel solid-phase synthesis of a small library of linear and hydrocarbon-bridged analogues of VEGF(81-91): potential biological tools for studying the VEGF/VEGFR-1 interaction.

artículo científico publicado en 2011

Peptaibols as a model for the insertions of chemical modifications

scientific article published on 20 September 2018

Photodegradation of Myrigalone A, an Allelochemical from Myrica gale: Photoproducts and Effect of Terpenes

artículo científico publicado en 2019

Rational design, structure, and biological evaluation of cyclic peptides mimicking the vascular endothelial growth factor.

artículo científico publicado en 2007

Salen/salan metallic complexes as redox labels for electrochemical aptasensors

scientific article published on 09 October 2019

Soluble fms-like tyrosine kinase-1 antibody for diagnosis purposes (WO2010075475)

scientific article published on 21 April 2011

Straightforward strategy to substitute amide bonds by 1,2,3-triazoles in peptaibols analogs using Aibψ[Tz]-Xaa dipeptides

artículo científico publicado en 2015

Structure and biological evaluation of new cyclic and acyclic laxaphycin-A type peptides ⬇️

scientific article published on 26 March 2019

Structure-based design of a bicyclic peptide antagonist of the vascular endothelial growth factor receptors.

artículo científico publicado en 2008

Synthesis and in vitro activities of new non-peptidic APA inhibitors.

artículo científico publicado en 2005

Targeting VEGFR1 on endothelial progenitors modulates their differentiation potential.

artículo científico publicado en 2014

Towards the total synthesis of trichormamide A, a cyclic undecapeptide

artículo científico publicado en 2018

Trichormamide C Structural Confirmation through Total Synthesis and Extension to Analogs

scientific article published on 19 December 2019

Lista de obras de Nicolas Inguimbert

Access to α,α-Disubstituted Disilylated Amino Acids and Their Use in Solid-Phase Peptide Synthesis

Asp218 participates with Asp213 to bind a Ca2+ atom into the S1 subsite of aminopeptidase A: a key element for substrate specificity.

Biochemical and structural analysis of the binding determinants of a vascular endothelial growth factor receptor peptidic antagonist

Biological Activities of Cyclic and Acyclic B-Type Laxaphycins in SH-SY5Y Human Neuroblastoma Cells

Biophysical Studies of the Induced Dimerization of Human VEGF Receptor 1 Binding Domain by Divalent Metals Competing with VEGF-A.

Characterization of a new anticancer agent, EAPB0203, and its main metabolites: nuclear magnetic resonance and liquid chromatography-mass spectrometry studies

Chemiluminescence immunoassays for estradiol and ethinylestradiol based on new biotinylated estrogen derivatives.

Cooperation and cheating orchestrate Vibrio assemblages and polymicrobial synergy in oysters infected with OsHV-1 virus

Development and validation of LC-MS methods for peptaibol quantification in fungal extracts according to their lengths.

Development of a chemiluminescent screening assay for detection of vascular endothelial growth factor receptor 1 ligands

Disulfide and amide-bridged cyclic peptide analogues of the VEGF81–91 fragment: Synthesis, conformational analysis and biological evaluation

Efficient microwave-assisted one shot synthesis of peptaibols using inexpensive coupling reagents

Enhancing the Antimicrobial Activity of Alamethicin F50/5 by Incorporating N-terminal Hydrophobic Triazole Substituents.

Exploration of the S(')(1) subsite of neprilysin: a joined molecular modeling and site-directed mutagenesis study

First total synthesis and stereochemical revision of laxaphycin B and its extension to lyngbyacyclamide A ⬇️

Helical peptides from VEGF and Vammin hotspots for modulating the VEGF-VEGFR interaction.

How are 1,2,3-triazoles accommodated in helical secondary structures?

Immunosensors for estradiol and ethinylestradiol based on new synthetic estrogen derivatives: application to wastewater analysis.

Isolation and Synthesis of Laxaphycin B-Type Peptides: A Case Study and Clues to Their Biosynthesis. ⬇️

NI956/QGC006, a Potent Orally Active, Brain-Penetrating Aminopeptidase A Inhibitor for Treating Hypertension

On-resin cyclization of peptide ligands of the Vascular Endothelial Growth Factor Receptor 1 by copper(I)-catalyzed 1,3-dipolar azide-alkyne cycloaddition

Oxovanadium-salen and -salan complexes as effective labels for electrochemical immunosensing: a case study for estradiol detection

Parallel solid-phase synthesis of a small library of linear and hydrocarbon-bridged analogues of VEGF(81-91): potential biological tools for studying the VEGF/VEGFR-1 interaction.

Peptaibols as a model for the insertions of chemical modifications

Photodegradation of Myrigalone A, an Allelochemical from Myrica gale: Photoproducts and Effect of Terpenes

Rational design, structure, and biological evaluation of cyclic peptides mimicking the vascular endothelial growth factor.

Salen/salan metallic complexes as redox labels for electrochemical aptasensors

Soluble fms-like tyrosine kinase-1 antibody for diagnosis purposes (WO2010075475)

Straightforward strategy to substitute amide bonds by 1,2,3-triazoles in peptaibols analogs using Aibψ[Tz]-Xaa dipeptides

Structure and biological evaluation of new cyclic and acyclic laxaphycin-A type peptides ⬇️

Structure-based design of a bicyclic peptide antagonist of the vascular endothelial growth factor receptors.

Synthesis and in vitro activities of new non-peptidic APA inhibitors.

Targeting VEGFR1 on endothelial progenitors modulates their differentiation potential.

Towards the total synthesis of trichormamide A, a cyclic undecapeptide

Trichormamide C Structural Confirmation through Total Synthesis and Extension to Analogs