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Lista de obras de Tristan A. Reekie

A Raney-cobalt-mediated tandem reductive cyclization route to the 1,5-methanoazocino[4,3-b]indole framework of the uleine and Strychnos alkaloids

scientific article published on 20 November 2012

A Three-Step Synthesis of Tetrasubstituted NH-Pyrroles

artículo científico publicado en 2016

A systematic exploration of the effects of flexibility and basicity on sigma (σ) receptor binding in a series of substituted diamines.

artículo científico publicado en 2016

Application of a Raney-cobalt-mediated tandem reductive cyclization protocol to total syntheses of the Aspidosperma alkaloids (±)-limaspermidine and (±)-1-acetylaspidoalbidine

artículo científico publicado en 2012

Body temperature and cardiac changes induced by peripherally administered oxytocin, vasopressin and the non-peptide oxytocin receptor agonist WAY 267,464: a biotelemetry study in rats.

artículo científico publicado en 2014

Comparative Evaluation of Three TSPO PET Radiotracers in a LPS-Induced Model of Mild Neuroinflammation in Rats

artículo científico publicado en 2016

Conformationally rigid derivatives of WAY-267,464: Synthesis and pharmacology at the human oxytocin and vasopressin-1a receptors.

artículo científico publicado en 2017

Determination and reduction of translocator protein (TSPO) ligand rs6971 discrimination

scientific article published on 15 November 2016

Discovery and pharmacological evaluation of a novel series of adamantyl cyanoguanidines as P2X7 receptor antagonists.

artículo científico publicado en 2017

Flexible analogues of WAY-267,464: Synthesis and pharmacology at the human oxytocin and vasopressin 1a receptors

scientific article published on 13 December 2015

Intramolecular cycloaddition reactions of cis-1,2-dihydrocatechol derivatives incorporating C3-tethered diazoketones, nitrile oxides, and azides: stereocontrolled routes to enantiomerically pure spiro[5.5]undecanes and related systems

artículo científico publicado en 2013

Investigation of pyrazolo-sulfonamides as putative small molecule oxytocin receptor agonists

artículo científico publicado en 2017

Investigations of amide bond variation and biaryl modification in analogues of α7 nAChR agonist SEN12333.

artículo científico publicado en 2014

Low intrinsic efficacy for G protein activation can explain the improved side effect profiles of new opioid agonists

scientific article published on 31 March 2020

Pharmacological evaluation of a novel series of urea, thiourea and guanidine derivatives as P2X7 receptor antagonists

artículo científico publicado en 2017

RANEY® cobalt--an underutilised reagent for the selective cleavage of C-X and N-O bonds

artículo científico publicado en 2014

Rapid Antibacterial Activity of Cannabichromenic Acid against Methicillin-Resistant Staphylococcus aureus

scientific article published on 16 August 2020

Rapid access to N-(indol-2-yl)amides and N-(indol-3-yl)amides as unexplored pharmacophores

artículo científico publicado en 2016

Ring-opened aminothienopyridazines as novel tau aggregation inhibitors

artículo científico publicado en 2017

Structural Optimization and Pharmacological Evaluation of Inhibitors Targeting Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases (DYRK) and CDC-like kinases (CLK) in Glioblastoma.

artículo científico publicado en 2017

Structure-activity relationship studies of SEN12333 analogues: determination of the optimal requirements for binding affinities at α7 nAChRs through incorporation of known structural motifs.

artículo científico publicado en 2015

The Formation of Seven-Membered Heterocycles under Mild Pictet-Spengler Conditions: A Route to Pyrazolo[3,4]benzodiazepines

artículo científico publicado en 2016

WAY 267,464, a non-peptide oxytocin receptor agonist, impairs social recognition memory in rats through a vasopressin 1A receptor antagonist action.

artículo científico publicado en 2015