Lista de obras - Terry W. Moore - Dominio Público Uruguay

A "cross-stitched" peptide with improved helicity and proteolytic stability

artículo científico publicado en 2018

A Cell-Permeable Stapled Peptide Inhibitor of the Estrogen Receptor/Coactivator Interaction.

artículo científico publicado en 2018

A set of time-resolved fluorescence resonance energy transfer assays for the discovery of inhibitors of estrogen receptor-coactivator binding

artículo científico publicado en 2009

Antiviral atropisomers: conformational energy surfaces by NMR for host-directed myxovirus blockers

artículo científico publicado en 2014

Asymmetric synthesis of host-directed inhibitors of myxoviruses.

artículo científico publicado en 2013

Curcumin analogue UBS109 prevents bone loss in breast cancer bone metastasis mouse model: involvement in osteoblastogenesis and osteoclastogenesis

artículo científico publicado en 2014

Discovering Small‐Molecule Estrogen Receptor α/Coactivator Binding Inhibitors: High‐Throughput Screening, Ligand Development, and Models for Enhanced Potency ⬇️

artículo científico publicado el 4 de abril de 2011

Estrogen receptor alpha/co-activator interaction assay: TR-FRET

artículo científico publicado en 2015

Inhibition of the NF-κB signaling pathway by the curcumin analog, 3,5-Bis(2-pyridinylmethylidene)-4-piperidone (EF31): anti-inflammatory and anti-cancer properties.

artículo científico publicado en 2011

Isoquinoline Kelch-like ECH-Associated Protein 1-Nuclear Factor (Erythroid-Derived 2)-like 2 (KEAP1-NRF2) Inhibitors with High Metabolic Stability

artículo científico publicado en 2019

Liver S9 Fraction-Derived Metabolites of Curcumin Analogue UBS109.

artículo científico publicado en 2014

Minireview: Not picking pockets: nuclear receptor alternate-site modulators (NRAMs)

artículo científico publicado en 2009

N-Substituted Pyrrole-Based Heterocycles as Broad-Spectrum Filoviral Entry Inhibitors

artículo científico publicado en 2024

Non-electrophilic modulators of the canonical Keap1/Nrf2 pathway

artículo científico publicado en 2015

Novel curcumin analogue UBS109 potently stimulates osteoblastogenesis and suppresses osteoclastogenesis: involvement in Smad activation and NF-κB inhibition.

artículo científico publicado en 2012

Probing the Topological Tolerance of Multimeric Protein Interactions: Evaluation of an Estrogen/Synthetic Ligand for FK506 Binding Protein Conjugate ⬇️

artículo científico publicado el 20 de octubre de 2010

Probing the structural requirements of non-electrophilic naphthalene-based Nrf2 activators.

artículo científico publicado en 2015

Recent structural advances in constrained helical peptides

artículo científico publicado en 2018

Replacement of a Naphthalene Scaffold in Kelch-like ECH-Associated Protein 1 (KEAP1)/Nuclear Factor (Erythroid-derived 2)-like 2 (NRF2) Inhibitors

scientific article published on 31 August 2018

SAR Study on Estrogen Receptor α/β Activity of (Iso)flavonoids: Importance of Prenylation, C-Ring (Un)Saturation, and Hydroxyl Substituents

scientific article published on 18 September 2020

Selective Human Estrogen Receptor Partial Agonists (ShERPAs) for Tamoxifen-Resistant Breast Cancer

artículo científico publicado en 2015

Stapled Peptides with γ-Methylated Hydrocarbon Chains for the Estrogen Receptor/Coactivator Interaction

artículo científico publicado en 2016

Steroid receptor/coactivator binding inhibitors: An update

scientific article published on 01 June 2019

Synthetic curcumin analog EF31 inhibits the growth of head and neck squamous cell carcinoma xenografts

artículo científico publicado en 2012

Synthetic curcumin analog UBS109 inhibits the growth of head and neck squamous cell carcinoma xenografts.

artículo científico publicado en 2014

Time-Gated Detection of Cystathionine γ-Lyase Activity and Inhibition with a Selective, Luminogenic Hydrogen Sulfide Sensor.

artículo científico publicado en 2016

Time-Gated Luminescence Detection of Enzymatically Produced Hydrogen Sulfide: Design, Synthesis, and Application of a Lanthanide-Based Probe.

artículo científico publicado en 2017

Using Tumor Explants for Imaging Mass Spectrometry Visualization of Unlabeled Peptides and Small Molecules

artículo científico publicado en 2018

Visualizing cancer and response to therapy in vivo using Cy5.5-labeled factor VIIa and anti-tissue factor antibody

artículo científico publicado en 2014

Lista de obras de Terry W. Moore

A "cross-stitched" peptide with improved helicity and proteolytic stability

A Cell-Permeable Stapled Peptide Inhibitor of the Estrogen Receptor/Coactivator Interaction.

A set of time-resolved fluorescence resonance energy transfer assays for the discovery of inhibitors of estrogen receptor-coactivator binding

Antiviral atropisomers: conformational energy surfaces by NMR for host-directed myxovirus blockers

Asymmetric synthesis of host-directed inhibitors of myxoviruses.

Curcumin analogue UBS109 prevents bone loss in breast cancer bone metastasis mouse model: involvement in osteoblastogenesis and osteoclastogenesis

Discovering Small‐Molecule Estrogen Receptor α/Coactivator Binding Inhibitors: High‐Throughput Screening, Ligand Development, and Models for Enhanced Potency ⬇️

Estrogen receptor alpha/co-activator interaction assay: TR-FRET

Inhibition of the NF-κB signaling pathway by the curcumin analog, 3,5-Bis(2-pyridinylmethylidene)-4-piperidone (EF31): anti-inflammatory and anti-cancer properties.

Isoquinoline Kelch-like ECH-Associated Protein 1-Nuclear Factor (Erythroid-Derived 2)-like 2 (KEAP1-NRF2) Inhibitors with High Metabolic Stability

Liver S9 Fraction-Derived Metabolites of Curcumin Analogue UBS109.

Minireview: Not picking pockets: nuclear receptor alternate-site modulators (NRAMs)

N-Substituted Pyrrole-Based Heterocycles as Broad-Spectrum Filoviral Entry Inhibitors

Non-electrophilic modulators of the canonical Keap1/Nrf2 pathway

Novel curcumin analogue UBS109 potently stimulates osteoblastogenesis and suppresses osteoclastogenesis: involvement in Smad activation and NF-κB inhibition.

Probing the Topological Tolerance of Multimeric Protein Interactions: Evaluation of an Estrogen/Synthetic Ligand for FK506 Binding Protein Conjugate ⬇️

Probing the structural requirements of non-electrophilic naphthalene-based Nrf2 activators.

Recent structural advances in constrained helical peptides

Replacement of a Naphthalene Scaffold in Kelch-like ECH-Associated Protein 1 (KEAP1)/Nuclear Factor (Erythroid-derived 2)-like 2 (NRF2) Inhibitors

SAR Study on Estrogen Receptor α/β Activity of (Iso)flavonoids: Importance of Prenylation, C-Ring (Un)Saturation, and Hydroxyl Substituents

Selective Human Estrogen Receptor Partial Agonists (ShERPAs) for Tamoxifen-Resistant Breast Cancer

Stapled Peptides with γ-Methylated Hydrocarbon Chains for the Estrogen Receptor/Coactivator Interaction

Steroid receptor/coactivator binding inhibitors: An update

Synthetic curcumin analog EF31 inhibits the growth of head and neck squamous cell carcinoma xenografts

Synthetic curcumin analog UBS109 inhibits the growth of head and neck squamous cell carcinoma xenografts.

Time-Gated Detection of Cystathionine γ-Lyase Activity and Inhibition with a Selective, Luminogenic Hydrogen Sulfide Sensor.

Time-Gated Luminescence Detection of Enzymatically Produced Hydrogen Sulfide: Design, Synthesis, and Application of a Lanthanide-Based Probe.

Using Tumor Explants for Imaging Mass Spectrometry Visualization of Unlabeled Peptides and Small Molecules

Visualizing cancer and response to therapy in vivo using Cy5.5-labeled factor VIIa and anti-tissue factor antibody