Lista de obras -

1-Phenyl-3H-2,3-benzodiazepin-4(5H)-one

artículo científico publicado en 2012

A Yeast/Drosophila Screen to Identify New Compounds Overcoming Frataxin Deficiency

artículo científico publicado en 2015

CMTX Disorder and CamKinase

artículo científico publicado en 2016

CamKII inhibitors reduce mitotic instability, connexon anomalies and progression of the in vivo behavioral phenotype in transgenic animals expressing a mutated Gjb1 gene

artículo científico publicado en 2014

Development of a peptidomimetic antagonist of neuropeptide FF receptors for the prevention of opioid-induced hyperalgesia

artículo científico publicado en 2015

Endogenous mammalian RF-amide peptides, including PrRP, kisspeptin and 26RFa, modulate nociception and morphine analgesia via NPFF receptors

artículo científico publicado en 2013

Fully regiocontrolled polyarylation of pyridine

artículo científico publicado en 2014

N-Heteroarylation of chiral α-aminoesters by means of palladium-catalyzed Buchwald-Hartwig reaction

artículo científico publicado en 2013

N-acyl substituted 7-amino-4-chloroisocoumarin: a peptide degradation model via an imide mechanism

artículo científico publicado en 2004

New 2-bromomethyl-8-substituted-benzo[c]chromen-6-ones. Synthesis and biological properties

artículo científico publicado en 2005

New beta-strand macrocyclic peptidomimetic analogues containing alpha-(O-, S- or NH-)aryl substituted glycine residues: synthesis, chemical and enzymatic properties

artículo científico publicado en 2003

Novel synthesis of 3,4-dihydro-5-bromo[1,4]oxazin-2-one derivatives, new protease inhibitor scaffold

artículo científico publicado en 2003

Opioid adjuvant strategy: improving opioid effectiveness

artículo científico publicado en 2016

RF-amide neuropeptides and their receptors in Mammals: Pharmacological properties, drug development and main physiological functions

artículo científico publicado en 2016

RF313, an orally bioavailable neuropeptide FF receptor antagonist, opposes effects of RF-amide-related peptide-3 and opioid-induced hyperalgesia in rodents

artículo científico publicado en 2017

Rapid and scalable synthesis of innovative unnatural α,β or γ-amino acids functionalized with tertiary amines on their side-chains

artículo científico publicado en 2015

Reactivity studies of 3-alkoxy-7-amino-4-chloroisocoumarins (beta-amyloid peptide inhibitors) versus different classes of amines

artículo científico publicado en 2003

Structure-activity relationship study around guanabenz identifies two derivatives retaining antiprion activity but having lost α2-adrenergic receptor agonistic activity

artículo científico publicado en 2014

Synthesis and antiviral activity of new anti-HIV amprenavir bioisosteres

artículo científico publicado en 2002

Synthesis of new 3-alkoxy-7-amino-4-chloro-isocoumarin derivatives as new beta-amyloid peptide production inhibitors and their activities on various classes of protease

artículo científico publicado en 2003

The initial substrate-binding site of gamma-secretase is located on presenilin near the active site

artículo científico publicado en 2005

The long-lasting love affair between the budding yeast Saccharomyces cerevisiae and the Epstein-Barr virus

artículo científico

The neuroprotector kynurenic acid increases neuronal cell survival through neprilysin induction

artículo científico publicado en 2013

Lista de obras de

1-Phenyl-3H-2,3-benzodiazepin-4(5H)-one

A Yeast/Drosophila Screen to Identify New Compounds Overcoming Frataxin Deficiency

CMTX Disorder and CamKinase

CamKII inhibitors reduce mitotic instability, connexon anomalies and progression of the in vivo behavioral phenotype in transgenic animals expressing a mutated Gjb1 gene

Development of a peptidomimetic antagonist of neuropeptide FF receptors for the prevention of opioid-induced hyperalgesia

Endogenous mammalian RF-amide peptides, including PrRP, kisspeptin and 26RFa, modulate nociception and morphine analgesia via NPFF receptors

Fully regiocontrolled polyarylation of pyridine

N-Heteroarylation of chiral α-aminoesters by means of palladium-catalyzed Buchwald-Hartwig reaction

N-acyl substituted 7-amino-4-chloroisocoumarin: a peptide degradation model via an imide mechanism

New 2-bromomethyl-8-substituted-benzo[c]chromen-6-ones. Synthesis and biological properties

New beta-strand macrocyclic peptidomimetic analogues containing alpha-(O-, S- or NH-)aryl substituted glycine residues: synthesis, chemical and enzymatic properties

Novel synthesis of 3,4-dihydro-5-bromo[1,4]oxazin-2-one derivatives, new protease inhibitor scaffold

Opioid adjuvant strategy: improving opioid effectiveness

RF-amide neuropeptides and their receptors in Mammals: Pharmacological properties, drug development and main physiological functions

RF313, an orally bioavailable neuropeptide FF receptor antagonist, opposes effects of RF-amide-related peptide-3 and opioid-induced hyperalgesia in rodents

Rapid and scalable synthesis of innovative unnatural α,β or γ-amino acids functionalized with tertiary amines on their side-chains

Reactivity studies of 3-alkoxy-7-amino-4-chloroisocoumarins (beta-amyloid peptide inhibitors) versus different classes of amines

Structure-activity relationship study around guanabenz identifies two derivatives retaining antiprion activity but having lost α2-adrenergic receptor agonistic activity

Synthesis and antiviral activity of new anti-HIV amprenavir bioisosteres

Synthesis of new 3-alkoxy-7-amino-4-chloro-isocoumarin derivatives as new beta-amyloid peptide production inhibitors and their activities on various classes of protease

The initial substrate-binding site of gamma-secretase is located on presenilin near the active site

The long-lasting love affair between the budding yeast Saccharomyces cerevisiae and the Epstein-Barr virus

The neuroprotector kynurenic acid increases neuronal cell survival through neprilysin induction